Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
Subcategories of "Chromatin/Epigenetics"
Found 2677 products for "Chromatin/Epigenetics".
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BRD 4354
CAS:BRD 4354 is an inhibitor of HDAC5 and HDAC9. For HDAC5 and HDAC9, the IC50s values are 0.85 and 1.88 μM, respectively.Formula:C21H23ClN4OPurity:99.86%Color and Shape:SolidMolecular weight:382.89Ref: TM-T10602L
1mg34.00€2mg44.00€5mg66.00€1mL*10mM (DMSO)73.00€10mg92.00€25mg178.00€50mg308.00€100mg512.00€500mg1,071.00€Abexinostat
CAS:Abexinostat (PCI-24781) is a pan-HDAC inhibitor, strongest on HDAC1; less so on HDACs 2, 3, 6, 10. Very select for HDAC8. In Phase 1/2 trials.Formula:C21H23N3O5Purity:98.19% - 98.43%Color and Shape:White SolidMolecular weight:397.42SIRT-IN-2
CAS:SIRT-IN-2 is a potent SIRT1/2/3 inhibitor(IC50s of 4, 1, 7 μM, respectively).Formula:C15H21N5O3S2Purity:98.26%Color and Shape:SolidMolecular weight:383.49Ref: TM-T12919
1mg92.00€5mg215.00€1mL*10mM (DMSO)236.00€10mg344.00€25mg587.00€50mg803.00€100mg1,099.00€200mg1,468.00€SNDX-5613
CAS:Revumenib (SNDX-5613) is a potent and selective oral inhibitor of menin-KMT2A interaction.Cost-effective and quality-assured.Formula:C32H47FN6O4SPurity:99.12% - 99.97%Color and Shape:Yellow SolidMolecular weight:630.82Ref: TM-T12943
1mg70.00€2mg92.00€5mg152.00€1mL*10mM (DMSO)207.00€10mg259.00€25mg513.00€50mg737.00€100mg1,018.00€AES-135
CAS:AES-135 is a potent HDAC inhibitor, inhibits HDAC3, HDAC6, HDAC11 (IC50s: 654, 190, and 636 nM) with anti-tumor activity.Formula:C33H29F6N3O5SPurity:97.72%Color and Shape:SolidMolecular weight:693.66Ref: TM-T10255
1mg79.00€5mg152.00€1mL*10mM (DMSO)225.00€10mg250.00€25mg424.00€50mg583.00€100mg803.00€A-3 hydrochloride
CAS:A-3 hydrochloride: potent, reversible kinase antagonist; permeable; inhibits PKC, CKI, PKA, CKII, MLCK; Ki: 4.3-80 μM.Formula:C12H14Cl2N2O2SPurity:99.32%Color and Shape:SolidMolecular weight:321.22Pulrodemstat benzenesulfonate
CAS:Pulrodemstat benzenesulfonate (CC-90011 benzenesulfonate) is a potent and orally inhibitor of lysine specific demethylase-1 (LSD1) with anticancer effect.Formula:C30H29F2N5O5SPurity:97.67%Color and Shape:White SolidMolecular weight:609.64Ref: TM-T11882
1mg57.00€2mg81.00€5mg117.00€1mL*10mM (DMSO)167.00€10mg178.00€25mg313.00€50mg464.00€100mg672.00€HDAC-IN-40
CAS:HDAC-IN-40 is a potent alkoxyamide-based HDAC inhibitor with Ki of 60 nM and 30 nM for HDAC2 and HDAC6, respectively. HDAC-IN-40 had antitumor effectsFormula:C15H22N2O6Purity:99.04%Color and Shape:SolidMolecular weight:326.35Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formula:C21H24ClNOPurity:99.77% - 99.99%Color and Shape:White SolidMolecular weight:341.88Ilginatinib
CAS:Ilginatinib (NS-018) is a highly active and orally bioavailable inhibitor of JAK2.Formula:C21H20FN7Purity:98.4% - 99.01%Color and Shape:SolidMolecular weight:389.43Ref: TM-T12266
1mg60.00€1mL*10mM (DMSO)126.00€5mg131.00€10mg177.00€25mg259.00€50mg371.00€100mg532.00€200mg705.00€Lin28-let-7a antagonist 1
CAS:Lin28-let-7a antagonist 1, with an IC50 of 4.03 μM for Lin28A-let-7a-1 interaction，and shows a clear antagonistic effect against the Lin28-let-7a interaction.Formula:C31H29N5O7Purity:99.44%Color and Shape:SolidMolecular weight:583.59Ref: TM-T11851
1mg96.00€5mg205.00€1mL*10mM (DMSO)266.00€10mg313.00€25mg562.00€50mg845.00€100mg1,243.00€Fenbendazole
CAS:Fenbendazole (Fenbendazol) is an antinematodal benzimidazole used in veterinary medicine.Formula:C15H13N3O2SPurity:99.74%Color and Shape:SolidMolecular weight:299.35Tranylcypromine (2-PCPA) hydrochloride
CAS:Tranylcypromine (2-PCPA) HCl, a MAO inhibitor, treats major, dysthymic, and atypical depression.Formula:C9H11N·HClPurity:99.48% - 99.86%Color and Shape:SolidMolecular weight:169.66EBI-2511
CAS:EBI-2511 is a highly potent and orally active inhibitor of EZH2 (IC50: 6 nM in Pfeffiera cell lines).Formula:C34H48N4O4Purity:99.74%Color and Shape:SolidMolecular weight:576.77Decitabine
CAS:Decitabine (Deoxycytidine) is a deoxycytidine analog, a DNA methyltransferase inhibitor with oral activity.Formula:C8H12N4O4Purity:98.06% - 99.87%Color and Shape:SolidMolecular weight:228.21M-89
CAS:M-89, a potent menin inhibitor (Kd 1.4 nM), disrupts Menin-MLL interaction, offering possible MLL leukemia treatment.Formula:C37H47N5O4SPurity:98.38%Color and Shape:SolidMolecular weight:657.87Ref: TM-T11925
1mg158.00€5mg385.00€10mg532.00€1mL*10mM (DMSO)538.00€25mg782.00€50mg1,063.00€100mg1,468.00€MAT2A inhibitor 2
CAS:MAT2A inhibitor 2 is an inhibitor of methionine adenosyltransferase 2A (MAT2A).Formula:C18H24ClN3O3Purity:99.52%Color and Shape:White SolidMolecular weight:365.85PBRM1-BD2-IN-3
CAS:PBRM1-BD2-IN-3 (compound 12) is a potent inhibitor of PBRM1-BD2, exhibiting an IC50 value of 1.1 μM, and is utilized in anticancer research.Formula:C14H11ClN2OPurity:99.77%Color and Shape:SolidMolecular weight:258.7Ref: TM-T60158
1mg73.00€1mL*10mM (DMSO)133.00€5mg149.00€10mg213.00€25mg319.00€50mg450.00€100mg605.00€SW2_110A
CAS:SW2_110A: Cell-permeable, CBX8 ChD inhibitor, Kd 800 nM; 5x selective over other CBXs in vitro.Formula:C42H60N6O7Purity:98%Color and Shape:SolidMolecular weight:760.96Inobrodib
CAS:Inobrodib (CBP-IN-1) is a potent inhibitor of p300/CBP bromodomain.Formula:C30H32F2N4O3Purity:98.91% - 99.18%Color and Shape:SolidMolecular weight:534.6Ref: TM-T10717
1mg66.00€2mg96.00€5mg144.00€1mL*10mM (DMSO)170.00€10mg250.00€25mg528.00€50mg755.00€100mg1,018.00€
