Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
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Subcategories of "Chromatin/Epigenetics"
Products of "Chromatin/Epigenetics"
GSK8573
CAS:1693766-04-9
GSK8573 is an inactive control compound for GSK2801. GSK8573 has binding activity to BRD9 (Kd …
Formula:
C20H21NO3
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
323.39
Ref: TM-T15441
| 1mg | 46.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 338.00 € | ||
| 100mg | 500.00 € | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
CM-579 trihydrochloride (1846570-40-8 free base)
CM-579 trihydrochloride is a first-in-class reversible and dual inhibitor of G9a and DNMT (IC50s: 16 …
Formula:
C29H43Cl3N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
602.04
Ref: TM-T10840
| 5mg | 211.00 € | ||
| 10mg | 327.00 € | ||
| 50mg | 917.00 € | ||
| 100mg | 1,249.00 € | ||
| 200mg | To inquire | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 279.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
WDR5-47
CAS:1422389-91-0
WDR5-47 is a potent small molecule to disturb the interaction of MLL1-WDR5 with IC50 value …
Formula:
C19H20ClFN4O3
Purity:
98.08%
Color and Shape:
Soild
Molecular weight:
406.84
Ref: TM-T67697
| 1mg | 112.00 € | ||
| 5mg | 249.00 € | ||
| 10mg | 365.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 765.00 € | ||
| 100mg | 1,044.00 € | ||
| 200mg | 1,404.00 € | ||
| 1mL*10mM (DMSO) | 271.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
PROTAC BRD4 Degrader-2
CAS:2185795-53-1
PROTAC BRD4 Degrader-2 is an efficacious degrader of PROTAC BRD4(BRD4 BD1,IC50 of 14.2 nM).
Formula:
C40H39N9O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
757.79
Ref: TM-T13834
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Wednesday 6 Nov 2024
PBRM1-BD2-IN-5
CAS:2819989-61-0
PBRM1-BD2-IN-5 is a potent inhibitor of the PBRM1 Bromodomain, demonstrating dissociation constant (Kd) values of …
Formula:
C15H13ClN2O
Purity:
99.55%
Color and Shape:
Soild
Molecular weight:
272.73
Ref: TM-T60159
| 1mg | 95.00 € | ||
| 2mg | 122.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 295.00 € | ||
| 25mg | 443.00 € | ||
| 50mg | 591.00 € | ||
| 100mg | 819.00 € | ||
| 500mg | 1,643.00 € | ||
| 1mL*10mM (DMSO) | 178.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
FKBP12 PROTAC dTAG-7
CAS:2064175-32-0
dTAG-7 selectively degrades BRD4 and FKBP12F36V by linking BET bromodomains to E3 ligase CRBN; it's …
Formula:
C63H79N5O19
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1210.32
Ref: TM-T11292
| 5mg | 1,214.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
FHD-286
CAS:2671128-05-3
FHD-286 is an inhibitor of BRM/BRG1 ATPase and can be used for studies on the …
Formula:
C24H30N6O6S2
Purity:
98.7%
Color and Shape:
Solid
Molecular weight:
562.66
Ref: TM-T9749
| 1mg | 144.00 € | ||
| 5mg | 346.00 € | ||
| 10mg | 539.00 € | ||
| 25mg | 730.00 € | ||
| 50mg | 915.00 € | ||
| 100mg | 1,261.00 € | ||
| 500mg | 2,531.00 € | ||
| 1mL*10mM (DMSO) | 373.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
CARM1 degrader-2
PROTAC CARM1 degrader-2 (compound 3e), with a DC50 value of 8.8 nM, is a VHL- …
Formula:
C72H100N12O7S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1277.71
Ref: TM-T79742
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 6 Nov 2024
OTS186935 FA
OTS186935 FA is a protein methyltransferase SUV39H2 inhibitor.OTS186935 FA inhibits tumor growth in MDA-MB-231 breast …
Formula:
C26H28ClN5O4
Purity:
98.16%
Color and Shape:
Soild
Molecular weight:
509.98
Ref: TM-T12344L1
| 1mg | 94.00 € | ||
| 5mg | 229.00 € | ||
| 10mg | 382.00 € | ||
| 25mg | 692.00 € | ||
| 50mg | 1,072.00 € | ||
| 100mg | 1,497.00 € | ||
| 500mg | 2,985.00 € | ||
| 1mL*10mM (DMSO) | 265.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
Sageone
CAS:142546-15-4
Sageone represents a promising anticancer agent against gastric cancer that warrants further study, it synergizes …
Formula:
C19H24O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
300.39
Ref: TM-TN4932
| 5mg | 3,028.00 € | ||
| 1mL*10mM (DMSO) | 3,028.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
5-Hydroxy-7-acetoxy-8-methoxyflavone
CAS:95480-80-1
5-Hydroxy-7-acetoxy-8-methoxyflavone is a flavonoid compound that inhibits lipid peroxidation and may have anti-influenza virus activity.
Formula:
C18H14O6
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
326.3
Ref: TM-TN3120
| 1mg | 231.00 € | ||
| 5mg | 578.00 € | ||
| 10mg | 819.00 € | ||
| 25mg | 1,235.00 € | ||
| 50mg | 1,653.00 € | ||
| 1mL*10mM (DMSO) | 595.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
Pim-1 kinase inhibitor 8
CAS:916038-47-6
Pim-1 kinase inhibitor 8 is a Pim-1 kinase inhibitor with anticancer activity that inhibits cell …
Formula:
C14H17N3O3
Purity:
99.81%
Color and Shape:
Soild
Molecular weight:
275.3
Ref: TM-T83627
| 1mg | 61.00 € | ||
| 5mg | 133.00 € | ||
| 10mg | 206.00 € | ||
| 25mg | 414.00 € | ||
| 50mg | 664.00 € | ||
| 100mg | 1,045.00 € | ||
| 500mg | 2,116.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
LSD1-IN-27
CAS:2904571-94-2
LSD1-IN-27 inhibits LSD1 (IC50=13 nM), blocks gastric cancer cell stemness/migration, reduces PD-L1, and boosts T-cell …
Formula:
C24H25N3
Purity:
98.65%
Color and Shape:
Soild
Molecular weight:
355.48
Ref: TM-T77635
| 1mg | 152.00 € | ||
| 5mg | 351.00 € | ||
| 10mg | 500.00 € | ||
| 25mg | 829.00 € | ||
| 50mg | 1,095.00 € | ||
| 100mg | 1,503.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
PBRM1-BD2-IN-7
CAS:2819989-68-7
PBRM1-BD2-IN-7, a PBRM1 bromodomain inhibitor with an IC50 of 0.29 μM, is used in cancer …
Formula:
C16H15ClN2O
Purity:
99% - 99.86%
Color and Shape:
Soild
Molecular weight:
286.76
Ref: TM-T60155
| 1mg | 113.00 € | ||
| 5mg | 251.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 551.00 € | ||
| 50mg | 776.00 € | ||
| 100mg | 1,043.00 € | ||
| 500mg | 2,103.00 € | ||
| 1mL*10mM (DMSO) | 238.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
HIV-IN-7
Axl-IN-16 (Compound 4), an Axl inhibitor, not only suppresses Axl expression and HIF activity but …
Formula:
C32H61N3O10P2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
709.79
Ref: TM-T78834
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 6 Nov 2024
3',4'-Dimethoxyflavone
CAS:4143-62-8
3',4'-Dimethoxyflavone is a standard compound of flavonoids with numerous medicinal activities.
Formula:
C17H14O4
Purity:
98.05%
Color and Shape:
Solid
Molecular weight:
282.29
Ref: TM-TN2883
| 5mg | 64.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 184.00 € | ||
| 100mg | 278.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
IV-275
IV-275 is a dual inhibitor targeting the bromodomains of both BRG1 and BRM.
Formula:
C19H18F2N2O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
360.35
Ref: TM-T79642
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 6 Nov 2024
PROTAC BRD4 Degrader-1
CAS:2133360-00-4
PROTAC BRD4 Degrader-1 is an efficacious degrader of BRD4(BRD4 BD1,IC50 of 41.8 nM).
Formula:
C40H37N9O8
Purity:
98%
Color and Shape:
Solid
Molecular weight:
771.78
Ref: TM-T13833
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Wednesday 6 Nov 2024
EEDi-5285
CAS:2488952-40-3
EEDi-5285: potent EED inhibitor, orally active, IC50=0.2nM, targets EED protein, anti-cancer properties.
Formula:
C24H22FN5O3S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
479.53
Ref: TM-T22322
| 1mg | To inquire | ||
| 5mg | 1,546.00 € | ||
| 10mg | 1,859.00 € | ||
| 25mg | 2,377.00 € | ||
| 50mg | 3,128.00 € | ||
| 1mL*10mM (DMSO) | 527.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
GXF-111
GXF-111, a proteolysis targeting chimera (PROTAC) molecule, efficiently induces the selective degradation of the BRD3 …
Formula:
C42H42ClN7O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
728.28
Ref: TM-T79034
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 6 Nov 2024
