Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(229 products)
- Annexin A(16 products)
- Aromatase(23 products)
- Estrogen/progestogen Receptor(66 products)
- GPR(1 products)
- Glucocorticoid Receptor(165 products)
- LHRH(2 products)
- Opioid Receptor(327 products)
- Prostaglandin Receptor(122 products)
- RAAS(89 products)
- Reductase(51 products)
- Somatostatin(57 products)
- Thyroid hormone receptor(THR)(33 products)
- Vasopressin Receptor(48 products)
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Found 3420 products of "Endocrinology/Hormones"
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RU 58841
CAS:RU 58841 (PSK-3841) is a specific androgen receptor antagonist or anti-androgen; RU 58841(PSK-3841) has a significant effect on hair regrowth.Formula:C17H18F3N3O3Purity:99.31% - 99.70%Color and Shape:SolidMolecular weight:369.34Ref: TM-T2236
5mg40.00€10mg63.00€25mg99.00€50mg130.00€100mg177.00€200mg245.00€500mg371.00€1mL*10mM (DMSO)48.00€DSRM-3716
CAS:Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery ofFormula:C9H6INPurity:97.28% - 99.785%Color and Shape:SolidMolecular weight:255.06Fluorometholone
CAS:Fluorometholone (Fluoromethalone) is a corticosteroid, most often used after laser-based refractive surgery.Formula:C22H29FO4Purity:99% - 99.15%Color and Shape:SolidMolecular weight:376.46Clascoterone
CAS:Clascoterone (CB-03-01) is a new topical and peripherally selective androgen antagonist.Formula:C24H34O5Purity:99.2% - 99.72%Color and Shape:SolidMolecular weight:402.52PROTAC ERRα ligand 2
CAS:PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)Formula:C20H13F6NO4Purity:≥95%Color and Shape:SolidMolecular weight:445.31Ref: TM-T5835
1mg43.00€5mg96.00€10mg116.00€25mg198.00€50mg299.00€100mg449.00€200mg627.00€1mL*10mM (DMSO)96.00€Osilodrostat
CAS:Osilodrostat (LCI699) is a potent inhibitor of human 11β-hydroxylase (CYP11B1) and aldosterone synthase (CYP11B2).Cost-effective and quality-assured.Formula:C13H10FN3Purity:99.10% - 99.36%Color and Shape:SolidMolecular weight:227.24Ref: TM-T4277
1mg34.00€5mg71.00€10mg99.00€25mg160.00€50mg234.00€100mg356.00€150mg772.00€1mL*10mM (DMSO)77.00€Endoxifen
CAS:(E/Z)-Endoxifen, an active tamoxifen metabolite via CYP2D6, binds estrogen receptors 100x better than tamoxifen. CYP2D6 variations affect its efficacy.Formula:C25H27NO2Purity:98.55% - >99.99%Color and Shape:SolidMolecular weight:373.49Zofenopril calcium
CAS:Zofenopril calcium (SQ26991) is an antioxidant that acts as an angiotensin-converting enzyme inhibitor.
Formula:C44H44CaN2O8S4Purity:98.37%Color and Shape:White Or Whitish Crystalline PowderMolecular weight:897.17AC-262536
CAS:AC-262536 is a selective androgen receptor (SAR) modulator and exhibits potent agonist activity at the androgen receptor.Formula:C18H18N2OPurity:99.88%Color and Shape:SolidMolecular weight:278.35Ref: TM-T26539
5mg46.00€10mg74.00€25mg145.00€50mg240.00€100mg359.00€200mg510.00€1mL*10mM (DMSO)49.00€Olodanrigan
CAS:Olodanrigan (EMA401), a highly selective AT2R antagonist, inhibition of augmented AngII/AT2R induced p38 and p42/p44 MAPK activation.Formula:C32H29NO5Purity:98.33%Color and Shape:SolidMolecular weight:507.58SR 19881
CAS:SR 19881 is a full agonist of ERRγ(EC50 value of 0.39 μM in a binding assay and an EC50 value of 4.7 μM in a cell-based assay).Formula:C19H24N2O2Purity:98.54%Color and Shape:SolidMolecular weight:312.41Ref: TM-T7904
1mg97.00€2mg149.00€5mg202.00€10mg324.00€25mg548.00€50mg785.00€100mg1,074.00€1mL*10mM (DMSO)220.00€Angiotensin (1-7)
CAS:Angiotensin (1-7) (ASP-ARG-VAL-TYR-ILE-HIS-PRO) is a synthetic heptapeptide, inhibits canine ACE activity with vasodilator and antiproliferative activities.Formula:C41H62N12O11Purity:>99.99%Color and Shape:White Lyophilised SolidMolecular weight:899TRV-120027 acetate (1234510-46-3 free base)
CAS:TRV-120027 acetate: a β-arrestin-1-biased AT1 receptor agonist that inhibits G-protein signaling.Formula:C45H71N13O12Purity:99.34%Color and Shape:SolidMolecular weight:986.14GSK5182
CAS:GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)Formula:C27H31NO3Purity:97.63% - 99.42%Color and Shape:SolidMolecular weight:417.54Ref: TM-T8370
1mg50.00€2mg71.00€5mg90.00€10mg144.00€25mg260.00€50mg394.00€100mg582.00€1mL*10mM (DMSO)108.00€Darolutamide
CAS:Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).Formula:C19H19ClN6O2Purity:97.36% - >99.99%Color and Shape:SolidMolecular weight:398.85Ref: TM-T6915
1mg50.00€2mg66.00€5mg100.00€10mg158.00€25mg250.00€50mg358.00€100mg512.00€200mg732.00€1mL*10mM (DMSO)101.00€TRV-120027 TFA
TRV-120027 TFA is an angiotensin II–mediated vasoconstriction inhibitor and increases cardiomyocyte contractility.Formula:C45H68F3N13O12Purity:97.45%Color and Shape:SolidMolecular weight:1040.1Ref: TM-TP2158
1mg43.00€5mg111.00€10mg170.00€25mg293.00€50mg423.00€100mg577.00€200mg778.00€1mL*10mM (DMSO)193.00€AZD9496
CAS:AZD9496 is an orally available selective estrogen receptor(ERα) antagonist, with potential antineoplastic activity.Formula:C25H25F3N2O2Purity:97.28% - 98.47%Color and Shape:SolidMolecular weight:442.47Ref: TM-T3975
1mg52.00€2mg73.00€5mg110.00€10mg178.00€25mg334.00€50mg494.00€100mg712.00€1mL*10mM (DMSO)105.00€Chlorotrianisene
CAS:Chlorotrianisene, a synthetic SERM, is orally active, lipophilic, and has estrogenic and antiestrogenic effects.Formula:C23H21ClO3Purity:98.88% - 99.03%Color and Shape:Crystals From Methanol Physical Description Small White Crystals Or White Powder Softens At 226°F Odorless (Ntp 1992)Molecular weight:380.86Ref: TM-T2569
1mg54.00€5mg114.00€10mg178.00€25mg313.00€50mg464.00€100mg660.00€200mg888.00€1mL*10mM (DMSO)126.00€BW-180C
CAS:BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.Formula:C29H39N5O7Purity:>99.99%Color and Shape:SolidMolecular weight:569.65Ref: TM-TP1905
2mg39.00€5mg58.00€10mg93.00€25mg145.00€50mg260.00€100mg462.00€200mg655.00€1mL*10mM (DMSO)73.00€Fevipiprant
CAS:Fevipiprant (NVP-QAW039) is a selective, potent, reversible competitive CRTh2 antagonist.Formula:C19H17F3N2O4SPurity:99.32% - 99.59%Color and Shape:SolidMolecular weight:426.41PZM21
CAS:PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).Formula:C19H27N3O2SPurity:99.93% - >99.99%Color and Shape:SolidMolecular weight:361.5Ref: TM-T4386
1mg44.00€2mg57.00€5mg93.00€10mg120.00€25mg193.00€50mg281.00€100mg447.00€1mL*10mM (DMSO)92.00€SNAP 94847 hydrochloride
CAS:SNAP 94847 hydrochloride is a melanin-concentrating hormonereceptor1 (MCHR1) antagonist(Ki= 2.2 nM)Formula:C29H33ClF2N2O2Purity:99.85% - >99.99%Color and Shape:SolidMolecular weight:515.03BigLEN (mouse) acetate
BigLEN (mouse) acetate is a potent and selective agonist of orphan G protein-coupled receptor 171 (GPR171), with a Kd of ∼0.5 nM.Formula:C80H134N24O24Purity:>99.99%Color and Shape:SolidMolecular weight:1816.07Fasiglifam
CAS:Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.Formula:C29H32O7SPurity:99.82% - 99.9%Color and Shape:SolidMolecular weight:524.63Ref: TM-T2351
1mg49.00€5mg90.00€10mg141.00€25mg236.00€50mg356.00€100mg522.00€200mg713.00€1mL*10mM (DMSO)116.00€Deltorphin I
CAS:Deltorphin I is an agonist of δ-opioid receptor.Formula:C37H52N8O10Purity:>99.99%Color and Shape:SolidMolecular weight:768.86AR 231453
CAS:Azenosertib (ZN-c3) is an orally active, specific GPR119 agonist. Cost-effective and quality-assured.Formula:C21H24FN7O5SPurity:99.31% - 99.34%Color and Shape:SolidMolecular weight:505.52MK-6892
CAS:MK-6892 is a selective and full agonist for the high-affinity nicotinic acid receptor GPR109A (Ki: 4 nM; GTPγS EC50: 16 nM).Formula:C19H22N4O5Purity:99.01% - 99.67%Color and Shape:SolidMolecular weight:386.4Ref: TM-TQ0108
1mg92.00€5mg178.00€10mg268.00€25mg447.00€50mg620.00€100mg888.00€200mg1,198.00€1mL*10mM (DMSO)203.00€VPC-13566
CAS:VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the
Formula:C18H14N2Purity:99.55%Color and Shape:SolidMolecular weight:258.32GW9508
CAS:GW9508(GW 9508) is a potent and selective agonist for FFA1 (GPR40), stimulates insulin secretion in a glucose-sensitive manner.
Formula:C22H21NO3Purity:97.89% - 99.19%Color and Shape:SolidMolecular weight:347.41BMS986188
CAS:BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.Formula:C30H31BrO4Purity:98.76%Color and Shape:SolidMolecular weight:535.476-OAU
CAS:6-OAU is a GPR84 agonist, activates it in HEK293 cells with a 105 nM EC50.Formula:C12H21N3O2Purity:98.14% - 99.01%Color and Shape:SolidMolecular weight:239.31Ref: TM-T2036
1mg152.00€2mg203.00€5mg313.00€10mg447.00€25mg713.00€50mg1,018.00€100mg1,369.00€1mL*10mM (DMSO)285.00€N-terminally acetylated Leu-enkephalin
Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.Formula:C30H39N5O8Purity:>99.99%Color and Shape:SolidMolecular weight:597.66Nociceptin (1-7) acetate
Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.Formula:C31H41N7O9Purity:98.92%Color and Shape:SoildMolecular weight:655.7Ref: TM-T23076L
1mg294.00€2mg439.00€5mg660.00€10mg999.00€25mg1,468.00€50mg1,998.00€100mg2,692.00€1mL*10mM (DMSO)897.00€[Leu5]-Enkephalin, amide acetate
[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.Formula:C30H42N6O8Purity:99.36%Color and Shape:SolidMolecular weight:614.69Orphanin FQ(1-11) acetate(178249-41-7 free base)
Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.Formula:C51H79N15O16Purity:95.54%Color and Shape:SolidMolecular weight:1158.26Dynorphin A 1-10 acetate(79994-24-4 free base)
Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.Formula:C59H95N19O14Purity:99.88%Color and Shape:SolidMolecular weight:1294.53Urotensin II, mouse acetate (9047-55-6 free base)
Urotensin II, mouse acetate (9047-55-6 free base) is an endogenous ligand for the orphan GPR14 or SENR. It is a potent vasoconstrictor.Formula:C64H88N14O19S2Purity:97.86%Color and Shape:SolidMolecular weight:1421.61Hemorphin-7 acetate(152685-85-3 free base)
Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.Formula:C51H68N12O13Purity:99.66%Color and Shape:SolidMolecular weight:1057.16Ac-RYYRWK-NH2 acetate
Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.Formula:C51H73N15O11Purity:98.59%Color and Shape:SolidMolecular weight:1072.22AH-7614
CAS:AH-7614 (AH 7614) is a selective and potent free fatty acid receptor 4 (FFA4/GPR120) antagonist.Formula:C20H17NO3SPurity:98.05%Color and Shape:SolidMolecular weight:351.42Ref: TM-T22027
2mg35.00€5mg49.00€10mg86.00€25mg170.00€50mg264.00€100mg401.00€200mg522.00€1mL*10mM (DMSO)60.00€EST73502 HCl
CAS:EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.Formula:C19H27ClF2N2O2Purity:99.96%Color and Shape:SolidMolecular weight:388.88Ref: TM-T39284
1mg96.00€5mg172.00€10mg244.00€25mg403.00€50mg567.00€100mg750.00€200mg1,018.00€1mL*10mM (DMSO)187.00€Methylnaltrexone bromide
CAS:Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.Formula:C21H26BrNO4Purity:99.02%Color and Shape:SolidMolecular weight:436.35[D-Ala2]leucine-enkephalin
CAS:[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.Formula:C29H39N5O7Purity:98.06%Color and Shape:SolidMolecular weight:569.65PW0787
CAS:PW0787 is a potent, selective, orally active, and brain-penetrant GPR52 agonist (EC50=135 nM).Formula:C23H20F4N4O2Purity:98.42%Color and Shape:SolidMolecular weight:460.42Ref: TM-T9452
1mg34.00€5mg75.00€10mg111.00€25mg224.00€50mg334.00€100mg475.00€200mg653.00€1mL*10mM (DMSO)92.00€Adrenorphin 3TFA(88377-68-8(free base))
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).Formula:C50H72N15O15SPurity:>99.99%Color and Shape:SolidMolecular weight:1326.26MBX-2982
CAS:MBX-2982 is a selective, orally-available GPR119 agonist, used for the treatment of diabetes.Formula:C22H24N8OSPurity:98% - 99.96%Color and Shape:SolidMolecular weight:448.54Ref: TM-T1793
1mg34.00€2mg44.00€5mg67.00€10mg104.00€25mg182.00€50mg278.00€100mg414.00€200mg567.00€1mL*10mM (DMSO)73.00€AS1269574
CAS:AS1269574 is a potent, orally available GPR119 agonist. AS1269574(AS 1269574) has the potential for the research of type 2 diabetes.Formula:C13H14BrN3OPurity:99.99%Color and Shape:SolidMolecular weight:308.17Ref: TM-T21623
2mg37.00€5mg54.00€10mg92.00€25mg165.00€50mg256.00€100mg385.00€200mg560.00€1mL*10mM (DMSO)63.00€Urotensin II (114-124), human acetate
Urotensin II (114-124), human acetate is an 11-amino acid residue peptide, is a potent vasoconstrictor and agonist for the orphan receptor GPR14.Formula:C66H89N13O20S2Purity:>99.99%Color and Shape:SolidMolecular weight:1448.63Palosuran hydrochloride 540769-28-6(free base)
Palosuran hydrochloride 540769-28-6(free base)(ACT-058362 hydrochloride) is a new potent and specific antagonist of the human UT receptor with an IC50 of 3.6±0.Formula:C25H31ClN4O2Purity:99.75%Color and Shape:SolidMolecular weight:454.99MS21570
CAS:MS21570 as a GPR171 antagonist based on its ability to block,with an IC50 of 220 Nm,that reduces anxiety-like behavior and fear conditioning in mice.Formula:C10H11N3S2Purity:97.79%Color and Shape:SolidMolecular weight:237.34DAMGO
CAS:DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.Formula:C26H35N5O6Purity:98.83% - 99.92%Color and Shape:SolidMolecular weight:513.59Ref: TM-T4351
1mg50.00€2mg60.00€5mg87.00€10mg140.00€25mg283.00€50mg423.00€100mg623.00€1mL*10mM (DMSO)88.00€b-Casomorphin (1-3) Acetate
b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.Formula:C25H31N3O7Purity:98.99%Color and Shape:SolidMolecular weight:485.53Ref: TM-T21660L
5mg42.00€10mg57.00€25mg87.00€50mg131.00€100mg190.00€200mg285.00€1mL*10mM (DMSO)55.00€4-CMTB
CAS:4-CMTB is a selective agonist of FFA2 and GPR43.It also is a positive allosteric modulator (pEC50=6.38).Formula:C14H15ClN2OSPurity:99.59%Color and Shape:SolidMolecular weight:294.8Ref: TM-T8642
1mg46.00€2mg62.00€5mg92.00€10mg131.00€25mg219.00€50mg324.00€100mg480.00€1mL*10mM (DMSO)96.00€TC-O 9311
CAS:TC-O 9311 (TCO-9311) is an effective agonist of GPR139 (EC50 = 39 nM in CHO-K1 cells expressing human GPR139).Formula:C20H19N3O4Purity:99.24% - 99.84%Color and Shape:SolidMolecular weight:365.38AZD1981
CAS:AZD1981: selective CRTh2 antagonist, IC50 4 nM, 1000x specificity over 340+ enzymes/receptors, tested in asthma and other trials.Formula:C19H17ClN2O3SPurity:98.87% - 99.67%Color and Shape:SolidMolecular weight:388.87Timapiprant
CAS:Timapiprant (OC000459) is a potent and selective D prostanoid receptor 2 (DP2) antagonist (IC50: 13 nM).
Formula:C21H17FN2O2Purity:97.44% - 99.51%Color and Shape:SolidMolecular weight:348.37Tyr-Gly-Gly-Phe-Met-OH
CAS:Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.
Formula:C27H35N5O7SPurity:≥95%Color and Shape:White Lyophilised SolidMolecular weight:573.66CVN424
CAS:CVN424 is a selective and novel GPR6 Inverse agonist effective in models of Parkinson Disease.Formula:C24H29F2N5O3Purity:99.02%Color and Shape:SolidMolecular weight:473.52Ref: TM-T9346
1mg90.00€5mg224.00€10mg356.00€25mg587.00€50mg848.00€100mg1,108.00€1mL*10mM (DMSO)235.00€JTC-801
CAS:JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.Formula:C26H25N3O2·HClPurity:99.27% - 99.59%Color and Shape:SolidMolecular weight:447.962-(pentylsulfanyl)pyrimidine-4,6-diol
CAS:2-(pentylsulfanyl)pyrimidine-4,6-diol 是一种新型 GRP84 激动剂。Formula:C9H14N2O2SPurity:97.58%Color and Shape:SolidMolecular weight:214.28Gluten Exorphin C
CAS:Gluten exorphin C is an opioid peptide derived from wheat gluten.Formula:C29H45N5O8Purity:99.39%Color and Shape:SolidMolecular weight:591.7Kisspeptin-10, human (TFA)(374675-21-5,FREE)
Kisspeptin-10 TFA: vasoconstrictor, inhibits angiogenesis & metastasis; key in kidney development & osteoblast differentiation via GPR54 & NFATc4/BMP2.Formula:C63H83N17O14·C2HF3O2Purity:>99.99%Color and Shape:SolidMolecular weight:1416.46JNJ-63533054
CAS:JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.Formula:C17H17ClN2O2Purity:99.71% - 99.88%Color and Shape:SolidMolecular weight:316.78Ref: TM-T3119
1mg34.00€5mg63.00€10mg93.00€25mg167.00€50mg259.00€100mg420.00€200mg602.00€1mL*10mM (DMSO)71.00€Carbetocin acetate
CAS:Carbetocin acetate is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth.Formula:C47H73N11O14SPurity:98.16% - 99.22%Color and Shape:SolidMolecular weight:1048.22GSK1292263
CAS:GSK1292263 is a GPR119 agonist and has been investigated for the treatment of DIABETES MELLITUS, TYPE 2.Formula:C23H28N4O4SPurity:98.34% - 99.53%Color and Shape:SolidMolecular weight:456.56PSN 375963
CAS:PSN 375963 (PSN 375963 hydrochloride) hydrochloride is a synthetic agonist of the endogenous ligand for GPR119.Formula:C17H23N3OPurity:99.63%Color and Shape:SolidMolecular weight:285.38Ref: TM-T23204
5mg43.00€10mg62.00€25mg110.00€50mg177.00€100mg290.00€200mg414.00€1mL*10mM (DMSO)60.00€DJ-V-159
CAS:DJ-V-159 is a GPRC6A agonist, targeting the G protein-coupled receptor family C group 6 member A (GPRC6A).
Formula:C24H12F6N4O2Purity:99.85% - 99.96%Color and Shape:SolidMolecular weight:502.37Myristyl nicotinate
CAS:Myristyl nicotinate (Tetradecyl nicotinate) is an ester prodrug being developed for delivery of nicotinic acid (NIC) into the skin for prevention of actinicFormula:C20H33NO2Purity:99.65%Color and Shape:SolidMolecular weight:319.48AM251
CAS:AM251: potent CB1 blocker (IC50: 8 nM), 306x CB2 selective; GPR55 activator (EC50: 39 nM).Formula:C22H21Cl2IN4OPurity:97.43% - 98.79%Color and Shape:A Crystalline SolidMolecular weight:555.24Kisspeptin 234 acetate(1145998-81-7 free base)
Kisspeptin receptor (KISS1/GPR54) blocker; analog to kisspeptin-10. Curbs IP activation (IC50=7nM) & GnRH release.Formula:C65H82N18O15Purity:99.34%Color and Shape:SolidMolecular weight:1355.46Asimadoline hydrochloride
CAS:Asimadoline HCl (EMD-61753) is a kappa-opioid receptor agonist for pruritus and IBS treatment.Formula:C27H31ClN2O2Purity:98.94% - 99.32%Color and Shape:SolidMolecular weight:451.01Ref: TM-T4691
1mg35.00€5mg73.00€10mg111.00€25mg227.00€50mg338.00€100mg500.00€500mg1,074.00€1mL*10mM (DMSO)81.00€BAM 22P acetate
BAM 22P acetate is a potent opioid agonist.Formula:C132H188N38O33S2Purity:99.87%Color and Shape:SoildMolecular weight:2899.27Ref: TM-TP1211L
1mg100.00€5mg376.00€10mg565.00€25mg1,009.00€50mg1,359.00€100mg1,845.00€200mg2,485.00€Ac-RYYRIK-NH2 acetate
Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.Formula:C46H74N14O11Purity:99.84%Color and Shape:SolidMolecular weight:999.17APD668
CAS:APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119, respectively.Formula:C21H24FN5O5SPurity:99.74% - 99.97%Color and Shape:SolidMolecular weight:477.51β-Neoendorphin acetate(77739-21-0 free base)
CAS:beta-Neoendorphin acetate is an agonist of κ-opioid receptorFormula:C56H81N13O14Purity:99.91%Color and Shape:SolidMolecular weight:1160.34AF64394
CAS:AF64394 is a selective inverse agonist of GPR3(pIC50 : 7.3)Formula:C21H20ClN5OPurity:97.22%Color and Shape:SolidMolecular weight:393.87Lasofoxifene Tartrate
CAS:Lasofoxifene Tartrate (CP-336156) is a third-generation, non-steroidal selective estrogen receptor modulator.Formula:C32H37NO8Purity:98.53%Color and Shape:SolidMolecular weight:563.64TUG-891
CAS:TUG-891 is a G protein-coupled receptor expressed in intestine, adipocytes, and pro-inflammatory macrophages that is activated by long chain free fatty acids.Formula:C23H21FO3Purity:98.18 - 99.21%Color and Shape:SolidMolecular weight:364.41Ref: TM-T3433
1mg40.00€2mg51.00€5mg85.00€10mg115.00€25mg225.00€50mg378.00€100mg552.00€500mg1,169.00€1mL*10mM (DMSO)93.00€Carbetocin
CAS:Carbetocin is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth.Formula:C45H69N11O12SPurity:99.96%Color and Shape:SolidMolecular weight:988.16CID 2745687
CAS:CID 2745687 blocks human GPR35, countering cromolyn disodium & zaprinast effects.Formula:C17H19F2N5O2SPurity:98.9% - 99.11%Color and Shape:SolidMolecular weight:395.43Ref: TM-T21874
1mg38.00€2mg50.00€5mg84.00€10mg119.00€25mg260.00€50mg409.00€100mg605.00€1mL*10mM (DMSO)93.00€IBC 293
CAS:IBC 293: Selective GPR109B agonist, favoring it over GPR109A; targets receptor in fat cells.Formula:C10H11N3O2Purity:99.63%Color and Shape:SolidMolecular weight:205.21Aticaprant
CAS:Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.Formula:C26H27FN2O2Purity:99.9% - 99.97%Color and Shape:SolidMolecular weight:418.5Ref: TM-TQ0082
1mg40.00€2mg52.00€5mg88.00€10mg126.00€25mg259.00€50mg406.00€100mg607.00€1mL*10mM (DMSO)87.00€Difelikefalin acetate
CAS:Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.Formula:C38H57N7O8Purity:99.55%Color and Shape:SolidMolecular weight:739.9ADL-5859
CAS:ADL-5859 HCl is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for theFormula:C24H28N2O3·HClPurity:98.78% - 99.11%Color and Shape:SolidMolecular weight:428.95Ref: TM-T6175
1mg49.00€2mg66.00€5mg90.00€10mg166.00€25mg319.00€50mg492.00€100mg710.00€500mg1,468.00€1mL*10mM (DMSO)108.00€GSK137647A
CAS:GSK137647A (GSK 137647) is a selective FFA4 agonist.Formula:C16H19NO3SPurity:99.26% - >99.99%Color and Shape:SolidMolecular weight:305.39Ref: TM-T3171
2mg34.00€5mg49.00€10mg80.00€25mg146.00€50mg231.00€100mg403.00€200mg582.00€500mg888.00€1mL*10mM (DMSO)54.00€Benzyl nicotinate
CAS:Benzyl nicotinate (Pycaril) is a agonist of GPR109A receptor and GPR109B receptorFormula:C13H11NO2Purity:98.22%Color and Shape:Yellow LiquidMolecular weight:213.23SNAP 94847
CAS:SNAP 94847 (SNAP-94847) is a selective and competitive MCH1 receptor (MCH1-R) antagonist (Ki: 2.2 nM).Formula:C29H32F2N2O2Purity:98%Color and Shape:SolidMolecular weight:478.57BRL 52537 hydrochloride
CAS:BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.Formula:C18H25Cl3N2OPurity:99.04%Color and Shape:SolidMolecular weight:391.76Leuphasyl TFA
CAS:Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.Formula:C31H40F3N5O9Purity:98.79%Color and Shape:SolidMolecular weight:683.67[Met5]-Enkephalin, amide TFA
[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.Formula:C29H37F3N6O8SPurity:99.81%Color and Shape:SolidMolecular weight:686.7Endomorphin 2
CAS:EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.Formula:C32H37N5O5Purity:99.64%Color and Shape:SolidMolecular weight:571.67CAY10471 Racemate
CAS:CAY10471 Racemate is a potent CRTH2/DP2 antagonist with Ki of 0.6 nM; less active on DP1 and TP.Formula:C21H21FN2O4SPurity:99.08%Color and Shape:SolidMolecular weight:416.47LY2795050
CAS:LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).Formula:C23H22ClN3O2Purity:97.77%Color and Shape:SolidMolecular weight:407.89Ref: TM-TQ0091
1mg50.00€2mg71.00€5mg110.00€10mg172.00€25mg281.00€50mgTo inquire1mL*10mM (DMSO)120.00€BMS-986122
CAS:BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1Formula:C16H15BrClNO3S2Purity:98.42%Color and Shape:SolidMolecular weight:448.78Ref: TM-T26869
1mg46.00€5mg90.00€10mg152.00€25mg295.00€50mg447.00€100mg623.00€200mg880.00€1mL*10mM (DMSO)90.00€Kisspeptin-10, rat acetate(478507-53-8 free base)
Kisspeptin-10, rat acetate is an endogenous ligand for the rodent kisspeptin receptor (KISS1, GPR54).Formula:C65H87N17O17Purity:99.92%Color and Shape:SolidMolecular weight:1378.45Nociceptin (1-13) amide TFA
Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat forebrain binding).Formula:C63H101F3N22O17Purity:97.64%Color and Shape:SolidMolecular weight:1495.61Setipiprant
CAS:Setipiprant (ACT-129968) is an oral CRTH2 antagonist for asthma/allergy, targeting PGD2-induced inflammation (IC50: 6.0 nM).Formula:C24H19FN2O3Purity:99.16%Color and Shape:SolidMolecular weight:402.42CTAP(TFA) (103429-32-9 free base)
CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM.Formula:C53H70F3N13O13S2Purity:99.62%Color and Shape:SolidMolecular weight:1218.33Dynorphin B (1-13) acetate(83335-41-5 free base)
Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.Formula:C76H119N21O19Purity:99.72%Color and Shape:SolidMolecular weight:1630.89CID1231538
CAS:CID1231538 is a potent GPR35 antagonist.Formula:C26H22ClN3O3S2Purity:98.79%Color and Shape:SolidMolecular weight:524.05
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