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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3180 products of "Endocrinology/Hormones"

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  • Ralaniten

    CAS:
    <p>Ralaniten (EPI-002), a potent AR-NTD antagonist, inhibits AR with IC50 of 7.4 μM, for CRPC study.</p>
    Formula:C21H27ClO5
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:394.89
  • Fludrocortisone

    CAS:
    <p>Fludrocortisone (Florinef) is a synthetic corticosteroid with moderate glucocorticoid potency and greater mineralocorticoid potency.Cost-effective and quality-assured.</p>
    Formula:C21H29FO5
    Purity:98.56% - 98.66%
    Color and Shape:White Solid
    Molecular weight:380.45
  • ALB-127158

    CAS:
    <p>ALB-127158(a): Potent MCH1 receptor antagonist, potential IBD treatment.</p>
    Formula:C23H21FN4O2
    Color and Shape:Solid
    Molecular weight:404.44
  • L 364918

    CAS:
    <p>L 364918 is an oxytocin antagonist.</p>
    Formula:C40H54N8O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:742.91
  • AZD3514

    CAS:
    <p>AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM and has ability of reducing AR protein expression.Phase 1.</p>
    Formula:C25H32F3N7O2
    Purity:98.09%
    Color and Shape:Solid
    Molecular weight:519.56
  • Loperamide oxide

    CAS:
    <p>Loperamide oxide (R 58425) is a secreted antidiarrheal agent that increases peristalsis and inhibits intestinal absorption of water and ions.</p>
    Formula:C29H33ClN2O3
    Color and Shape:Solid
    Molecular weight:493.04
  • AR antagonist 2

    CAS:
    <p>AR antagonist 2 (compound 58) is a potent inhibitor of the androgen receptor (AR) (IC50: 0.95 μM).</p>
    Formula:C22H17ClFN5O2S
    Color and Shape:Solid
    Molecular weight:469.92
  • Tranilast Sodium

    CAS:
    <p>Tranilast Sodium has been used for the treatment of bronchial asthma. Tranilast is also used to autoimmune diseases, atopic and fibrotic pat.</p>
    Formula:C18H17NNaO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:350.32
  • SQ 30774

    CAS:
    <p>SQ 30774 is a representative of the imidazole alcohols-a novel class of renin inhibitors.</p>
    Formula:C32H45N7O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:607.74
  • GPR40 Activator 1

    CAS:
    GPR40 Activator 1 is a potent GPR40 activator for treatment of type 2 diabetes.
    Formula:C31H31NO3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:497.65
  • AS-1669058 free base

    CAS:
    <p>AS-1669058 free base is a G-protein-coupled receptor 119 (GPR119) agonist used to as new drug to treat type 2 diabetes.</p>
    Formula:C18H15BrF2N4O
    Color and Shape:Solid
    Molecular weight:421.24
  • AMG-076

    CAS:
    <p>AMG-076 is an antagonist of melanin-concentrating hormone receptor 1. It also reduced hERG inhibition.</p>
    Formula:C32H39F3N2O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:620.72
  • Acolbifene Hydrochloride

    CAS:
    <p>Acolbifene hydrochloride binds to estrogen receptors in the body. It is a type of selective estrogen receptor modulator</p>
    Formula:C29H32ClNO4
    Color and Shape:Solid
    Molecular weight:494.02
  • DS20362725

    CAS:
    <p>DS20362725 is a selective estrogen-related receptor alpha (ERRα) agonist, commonly used in the study of metabolic disorders.</p>
    Formula:C19H22N2O2
    Purity:99.34%
    Color and Shape:Solid
    Molecular weight:310.39
  • CRTh2 antagonist 1

    CAS:
    <p>CRTh2 antagonist 1 is a CRTh2 antagonist (IC50: 89 nM).</p>
    Formula:C23H25N3O5S
    Purity:97.24%
    Color and Shape:Solid
    Molecular weight:455.53
  • (R)-Viloxazine Hydrochloride

    CAS:
    <p>(R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.</p>
    Formula:C13H20ClNO3
    Purity:99.88% - 99.94%
    Color and Shape:Solid
    Molecular weight:273.76
  • Cholesterol-d6

    CAS:
    <p>Cholesterol-d6 is a deuterated chlosterol that can be used to study lipid membrane flow and chlosterol metabolism in vivo.</p>
    Formula:C27H40D6O
    Color and Shape:Solid
    Molecular weight:392.69
  • VPC-14449

    CAS:
    <p>VPC-14449 is a selective androgen receptor DNA-binding domain (AR-DBD) inhibitor, useful in prostate cancer research.</p>
    Formula:C10H10Br2N4OS
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:394.09
  • Norbinaltorphimine

    CAS:
    <p>nor-Binaltorphimine dihydrochloride is a long-acting potent and highly selective kappa opioid receptor antagonist.</p>
    Formula:C40H43N3O6
    Color and Shape:Solid
    Molecular weight:661.79
  • AZ12216052

    CAS:
    <p>AZ12216052 is a GRP8 antagonist with anxiolytic and anti-inflammatory activity and can be used to study obesity and metabolic disorders.</p>
    Formula:C19H22BrNOS
    Purity:99.29%
    Color and Shape:Solid
    Molecular weight:392.35
  • LY 43578

    CAS:
    <p>LY 43578 is an orally active aromatase inhibitor.</p>
    Formula:C17H12Cl2N2O
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:331.2
  • Estrogen receptor α antagonist 1

    CAS:
    <p>Estrogen receptor α antagonist 1 (compound 35) is a highly selective estrogen receptor α antagonist that acts on estrogen receptor α (IC50: 0.02 μM), estrogen</p>
    Formula:C26H32N2O5
    Color and Shape:Solid
    Molecular weight:452.54
  • SR8993

    CAS:
    <p>SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.</p>
    Formula:C25H37FN4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:412.59
  • Embusartan

    CAS:
    <p>Embusartan (BAY 10-6734) is a potent, orally active angiotensin II receptor antagonist used as an antihypertensive agent.</p>
    Formula:C25H24FN5O3
    Color and Shape:Solid
    Molecular weight:461.49
  • GPR84 antagonist 2

    CAS:
    <p>Potent, selective oral GPR84 antagonist with IC50 of 8.95 nM, inhibits neutrophil/macrophage chemotaxis, potential in ulcerative colitis research.</p>
    Formula:C28H16Cl2NaO4PS2
    Color and Shape:Solid
    Molecular weight:605.42
  • Demegestone

    CAS:
    <p>Demegestone: synthetic progestogen, progesterone receptor agonist, treats luteal insufficiency, no androgenic activity.</p>
    Formula:C21H28O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:312.45
  • L-751788

    CAS:
    <p>L-751788 is an inhibits of type 1 5alpha-reductase.</p>
    Formula:C26H36ClNO2
    Color and Shape:Solid
    Molecular weight:430.02
  • σ1 Receptor/μ Opioid receptor modulator 1

    CAS:
    <p>σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM).</p>
    Formula:C24H31FN2O2
    Color and Shape:Solid
    Molecular weight:398.51
  • ERRγ Inverse Agonist 1

    CAS:
    <p>ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1].</p>
    Formula:C30H38Cl2N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:529.54
  • ASN06917370

    CAS:
    <p>ASN06917370 (Compound V) is a specific modulator of the orphan receptor GPR17 (Uracil Nucleotide/Cysteinyl Leukotriene Receptor), neuroprotective</p>
    Formula:C24H21ClF3N7O2
    Color and Shape:Solid
    Molecular weight:531.92
  • Bopindolol

    CAS:
    <p>Bopindolol: oral β1/β2-ARs antagonist and partial agonist; prodrug of pindolol for hypertension research.</p>
    Formula:C23H28N2O3
    Color and Shape:Solid
    Molecular weight:380.48
  • Aldose reductase-IN-2

    CAS:
    <p>Aldose reductase-IN-2 (5f) inhibits AR with antioxidant effects; potential anti-diabetic drug.</p>
    Formula:C25H28N4O5
    Color and Shape:Solid
    Molecular weight:464.51
  • Ono-3805 sodium

    CAS:
    <p>Ono-3805 is an inhibitor of nonsteroidal 5 alpha-reductase.</p>
    Formula:C31H37NNaO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:526.629
  • CAY10595

    CAS:
    <p>CAY10595 is an antagonist of the CRTh2 (DP2) receptor with a Ki of 10 nM.</p>
    Formula:C20H13Cl2FN2O5
    Purity:99.95% - 99.97%
    Color and Shape:Solid
    Molecular weight:451.23
  • Aldose reductase-IN-3

    CAS:
    <p>Aldose reductase-IN-3 (Compound 5) is a moderately selective AR inhibitor with IC50 of 3.99 μM, potential for sepsis research.</p>
    Formula:C18H12ClN3O2S2
    Color and Shape:Solid
    Molecular weight:401.89
  • BHPI

    CAS:
    <p>BHPI is a potent ERα inhibitor, activating UPR and blocking protein synthesis with an IC50 value. It depletes EnR Ca(2+) via PLCγ in ERα(+) cancer cells.</p>
    Formula:C21H17NO3
    Color and Shape:Solid
    Molecular weight:331.36
  • FK-739 free acid

    CAS:
    <p>FK-739, an angiotensin II receptor blocker, inhibits rat aorta binding (IC50=8.6 nM) but not bovine cerebellum.</p>
    Formula:C24H23N7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:409.49
  • GPR120 modulator 1

    CAS:
    <p>GPR120 modulator 1 is useful for modulating GPR120.</p>
    Formula:C19H16ClNO4S
    Color and Shape:Solid
    Molecular weight:389.85
  • Prochloraz

    CAS:
    <p>Prochloraz: broad-spectrum imidazole fungicide; blocks placental aromatase (IC50=40nM), estrogen/androgen receptors; activates aryl hydrocarbon receptors.</p>
    Formula:C15H16Cl3N3O2
    Purity:99.75% - 99.79%
    Color and Shape:Colorless Solid
    Molecular weight:376.67
  • Acolbifene

    CAS:
    <p>Acolbifene (SCH 57068) is a selective antagonist of estrogen receptors with IC50s of 2 nM and 0.4 nM for estradiol-induced transcriptional activity of ERα and</p>
    Formula:C29H31NO4
    Purity:98.17%
    Color and Shape:Solid
    Molecular weight:457.56
  • PF-3882845

    CAS:
    <p>PF-3882845, a high affinity MR antagonist (IC50=2.7 nM) for hypertension, also targets progesterone receptor (IC50: 310 nM).</p>
    Formula:C24H22ClN3O2
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:419.9
  • AZD2906

    CAS:
    <p>AZD2906: selective GR agonist with human/rat IC50s - 2.2/0.3 nM (PBMC), 41.6/7.5 nM (blood); induces rat bone marrow micronuclei.</p>
    Formula:C26H25FN4O3
    Color and Shape:Solid
    Molecular weight:460.5
  • NNC45-0781

    CAS:
    <p>NNC45-0781 is a tissue-selective partial-agonist of estrogen.</p>
    Formula:C27H29NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:415.52
  • Prednisolone hemisuccinate

    CAS:
    <p>Prednisolone hemisuccinate is a soluble glucocorticoid and cortisol exerts anti-inflammatory, immunosuppressive, and antiallergic by binding to GR receptor.</p>
    Formula:C25H32O8
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:460.52
  • GPR35 agonist 3

    CAS:
    <p>GPR35 agonist 3 is a synthetic GPR35 agonist used in the study of cancer, type 2 diabetes and cardiovascular disease.</p>
    Formula:C12H9NO5S
    Purity:98.80%
    Color and Shape:Solid
    Molecular weight:279.27
  • RU 28318, potassium salt

    CAS:
    <p>mineralocorticoid receptor (MR) antagonist</p>
    Formula:C25H38KO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.67
  • THPN

    CAS:
    <p>THPN is a Nur77 agonist. It also induces autophagy in melanoma cell lines.</p>
    Formula:C15H22O4
    Color and Shape:Solid
    Molecular weight:266.33
  • Pivalopril

    CAS:
    <p>Pivalopril is a new orally active inhibitor of angiotensin-converting enzyme.</p>
    Formula:C16H27NO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.45
  • GSK706

    CAS:
    <p>GSK706 is a novel effective agonist of the GPR119.</p>
    Formula:C23H29N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:471.57
  • BMS-564929

    CAS:
    <p>BMS-564929 is an AR agonist that upregulates the expression and activity of fat-producing enzymes, reducing VAT content and lipid levels.</p>
    Formula:C14H12ClN3O3
    Purity:98.17%
    Color and Shape:Solid
    Molecular weight:305.72
  • Lubabegron fumarate

    CAS:
    <p>Lubabegron (LY591281, LY488756 fumarate) is a beta-agonist approved in 2018 to lower ammonia in cattle waste, aiding environment and health.</p>
    Formula:C29H29N3O3SC4H4O4
    Color and Shape:Solid
    Molecular weight:557.66
  • ERRα antagonist-1

    CAS:
    <p>ERRα antagonist-1 (ERR+/- antagonist-1) is a high-affinity, selective antagonist of the estrogen-related receptor α (ERRα).</p>
    Formula:C21H19N3S2
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:377.53
  • Omapatrilat

    CAS:
    <p>Omapatrilat is a metalloprotease ACE and NEP dual inhibitor (Ki: 0.64 and 0.45 nM, respectively).</p>
    Formula:C19H24N2O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.53
  • (S)-Baxdrostat

    CAS:
    <p>(S)-Baxdrostat is an S-enantiomer of Baxdrostat, which functions as an inhibitor of aldosterone synthase [1].</p>
    Formula:C22H25N3O2
    Color and Shape:Solid
    Molecular weight:363.45
  • Rentiapril

    CAS:
    <p>Rentiapril is an orally active inhibitor of angiotensin converting enzyme (ACE), with antihypertensive activity.</p>
    Formula:C13H15NO4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:313.39
  • Zenarestat

    CAS:
    <p>Zenarestat is an orally active aldose reductase inhibitor capable of ameliorating diabetic peripheral neuropathy in rats with type 2 diabetes.</p>
    Formula:C17H11BrClFN2O4
    Purity:99.51% - 99.51%
    Color and Shape:Solid
    Molecular weight:441.64
  • TUG-424

    CAS:
    <p>TUG-424 boosts insulin secretion, is a selective FFAR1 agonist with an EC50 of 32 nM.</p>
    Formula:C18H16O2
    Purity:98.94%
    Color and Shape:Solid
    Molecular weight:264.32
  • NXT629

    CAS:
    <p>NXT629 is a PPAR-α antagonist with anticancer activity, inhibiting PPARδ, and can be used in ovarian cancer and melanoma research.</p>
    Formula:C35H39N5O3S
    Purity:99.07% - 99.07%
    Color and Shape:Solid
    Molecular weight:609.78
  • GSK9027

    CAS:
    <p>GSK9027, a nonsteroidal GR agonist, is a partial 2×GRE reporter gene activator, less potent than dexamethasone.</p>
    Formula:C27H19F4N3O2S
    Purity:99.36%
    Color and Shape:Solid
    Molecular weight:525.52
  • 6-Raloxifene-β-D-glucopyranoside

    CAS:
    <p>6-Raloxifene-β-D-glucopyranoside is a benzothiophene glucuronidated at the 6' position.</p>
    Formula:C34H37NO9S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:635.72
  • 5-bromo-3-phenyl Salicylic Acid

    CAS:
    <p>AKR1C1 inhibitor</p>
    Formula:C13H9BrO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:293.11
  • ALR1/2-IN-1

    CAS:
    <p>ALR1/2-IN-1 (Compound 6e) is an aldehyde reductase (ALR1) (IC50: 3.26 μM) and aldose reductase (ALR2) (IC50: 3.06 μM) inhibitor with anticancer effects.</p>
    Formula:C18H18N4O5S2
    Color and Shape:Solid
    Molecular weight:434.49
  • ES 6864

    CAS:
    <p>ES 6864 is an orally active inhibitor of renin.</p>
    Formula:C42H58N6O7S
    Color and Shape:Solid
    Molecular weight:791.01
  • Pipendoxifene hydrochloride

    CAS:
    <p>Pipendoxifene hydrochloride is a selective modulator of estrogen receptor.</p>
    Formula:C29H33ClN2O3
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:493.04
  • Erteberel

    CAS:
    <p>Erteberel (LY500307) is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2.</p>
    Formula:C18H18O3
    Purity:99.46%
    Color and Shape:Solid
    Molecular weight:282.33
  • Bromopropylate

    CAS:
    <p>Bromopropylate is an insecticide. Bromopropylate is the active substance in fumigant strips for mites.</p>
    Formula:C17H16Br2O3
    Purity:98%
    Color and Shape:White Crystalline Solid Yellowish Crystals
    Molecular weight:428.11
  • WAY-267464

    CAS:
    <p>oxytocin receptor (OTR) agonist</p>
    Formula:C32H35N7O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:581.66
  • TRβ agonist 2

    CAS:
    <p>TRβ agonist 2 (Compound 1) is a highly potent agonist of TRβ.</p>
    Formula:C22H27NO4
    Color and Shape:Solid
    Molecular weight:369.45
  • KB-141

    CAS:
    <p>KB-141 is an agonist of thyroid hormone receptor.</p>
    Formula:C17H16Cl2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:355.21
  • TIPP

    CAS:
    <p>TIPP is an agent of delta opioid antagonist.</p>
    Formula:C37H38N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:634.72
  • Milfasartan

    CAS:
    <p>Milfasartan: Potent AT1 antagonist, oral, effectively reduces blood pressure in hypertensive rats.</p>
    Formula:C30H30N6O3S
    Color and Shape:Solid
    Molecular weight:554.66
  • 27-Hydroxycholesterol

    CAS:
    <p>27-Hydroxycholesterol (25(R)-27-hydroxy Cholesterol) is a selective modulator of estrogen receptor and an agonist of the liver X receptor.</p>
    Formula:C27H46O2
    Purity:99.45% - 99.82%
    Color and Shape:Solid
    Molecular weight:402.65
  • Anordiol

    CAS:
    <p>Anordiol is an antiestrogen with estrogenic activity. It also is known to inhibit fertility.</p>
    Formula:C22H30O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:326.47
  • (Rac)-Acolbifene

    CAS:
    <p>(Rac)-Acolbifene (EM-343) is the racemic form of Acolbifene.</p>
    Formula:C29H31NO4
    Purity:99.7%
    Color and Shape:Solid
    Molecular weight:457.56
  • LY88074 Trimethyl ether

    CAS:
    <p>LY88074 Trimethyl ether inhibits conditions like osteoporosis and hyperlipidemia caused by low estrogen.</p>
    Formula:C24H20O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:404.48
  • AM-4668

    CAS:
    <p>AM-4668, a GPR40 (FFA1) agonist with oral availability, was optimized to reduce central nervous system (CNS) permeability, and reduced blood glucose level.</p>
    Formula:C24H19F3N2O4S
    Purity:99.32% - 99.92%
    Color and Shape:Solid
    Molecular weight:488.48
  • AS-1669058 oxalate

    CAS:
    <p>AS-1669058 is a G-protein-coupled receptor 119 (GPR119) agonist for the treatment of type 2 diabetes mellitus.</p>
    Formula:C20H17BrF2N4O5
    Color and Shape:Solid
    Molecular weight:511.27
  • SC 46944

    CAS:
    <p>SC 46944 is a highly potent human renin inhibitor.</p>
    Formula:C34H55N3O7
    Color and Shape:Solid
    Molecular weight:617.82
  • Honokiol DCA

    CAS:
    <p>Honokiol DCA inhibits DRP1, enhances respiration via mitochondrial repair, and is active against Vemurafenib-resistant melanoma.</p>
    Formula:C22H18Cl4O4
    Color and Shape:Solid
    Molecular weight:488.19
  • Diallyl G

    CAS:
    <p>Diallyl G is a delta-opioid receptor antagonist agent.</p>
    Formula:C38H53N5O8
    Color and Shape:Solid
    Molecular weight:707.86
  • GSK 1562590 hydrochloride

    CAS:
    <p>urotensin II (UT) receptor antagonist</p>
    Formula:C30H31Cl3N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:617.95
  • Alrestatin Sodium

    CAS:
    <p>Alrestatin is a specific inhibitor of the aldose reductase enzyme.</p>
    Formula:C14H9NNaO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:278.219
  • μ opioid receptor agonist 2

    CAS:
    <p>μ opioid receptor agonist 2 (Compound H-3)is a MOR receptor agonist. μ opioid receptor agonist 2 can be used for the research of pain and pain related diseases.</p>
    Formula:C25H34N4O
    Color and Shape:Solid
    Molecular weight:406.56
  • Glutaurine aceate


    <p>Glutaurine aceate containing glutamine and taurine residues is an orally active hormone of the parathyroid.</p>
    Formula:C9H18N2O8S
    Purity:98%
    Color and Shape:Soild
    Molecular weight:314.31
  • Viminol

    CAS:
    <p>Viminol is an opioid analgesic. Viminol is based on the α-pyrryl-2-aminoethanol structure, unlike any other class of opioids.</p>
    Formula:C21H31ClN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:362.94
  • LG-121071

    CAS:
    <p>LG-121071: oral SARM, high-affinity AR full agonist, Ki=17 nM.</p>
    Formula:C15H15F3N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:296.29
  • ATC0065

    CAS:
    <p>ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.</p>
    Formula:C25H29BrF3N5O
    Color and Shape:Solid
    Molecular weight:552.43
  • AS1907417

    CAS:
    <p>AS1907417 is a GPR119 agonist.</p>
    Formula:C19H27N3O4S
    Color and Shape:Solid
    Molecular weight:393.5
  • ALR2-IN-3


    <p>ALR2-IN-2 inhibits ALR2 strongly (IC50: 22 nM) and ALR1 less (IC50: 116 nM), used in diabetes complication studies.</p>
    Formula:C17H12N2O3S2
    Color and Shape:Solid
    Molecular weight:356.42
  • EMD 66684

    CAS:
    <p>angiotensin AT1 receptor antagonist</p>
    Formula:C28H31ClN8O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:547.06
  • TCS 3035

    CAS:
    <p>GPR35 agonist 4 (compound 10), pEC50 5.86, potent in human/rat but inactive with R3.36 mutation.</p>
    Formula:C12H9NO5S
    Color and Shape:Solid
    Molecular weight:279.27
  • Liothyronine HCl

    CAS:
    <p>Liothyronine is a T3 thyroid hormone normally synthesized and secreted by the thyroid gland in much smaller quantities than thyroxine.</p>
    Formula:C15H13ClI3NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:687.43
  • Androgen receptor antagonist 4

    CAS:
    <p>Compound AT2 is an AR inhibitor with anticancer effects, blocking DHT action and AR nuclear translocation (IC50=0.15μM).</p>
    Formula:C22H18ClN
    Color and Shape:Solid
    Molecular weight:331.84
  • L162441

    CAS:
    <p>L162441 is an antagonist of Angiotensin type 1 receptor.</p>
    Formula:C34H43N5O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:633.8
  • RU 752

    CAS:
    <p>RU 752 is an antagonist of mineralocorticoid receptor that inhibits aldosterone synthesis.</p>
    Formula:C22H30O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:358.47
  • TFM-4AS-1

    CAS:
    <p>androgen receptor modulator</p>
    Formula:C27H33F3N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:474.56
  • NCG21

    CAS:
    <p>NCG21, a GPR120 agonist, boosts ERK, Ca²⁺ responses, and GLP-1 in GPR120-expressing cells; raises GLP-1 in mice.</p>
    Formula:C23H24N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.45
  • ADL-5859 HCl

    CAS:
    <p>ADL-5859 is a delta-opioid receptor agonist.</p>
    Formula:C24H28N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.49
  • FFA1 agonist-1

    CAS:
    <p>FFA1 agonist-1 (Compound 17a) is an orally active fatty acid receptor (FFA1) agonist (EC50: 0.75 μM).</p>
    Formula:C27H36ClNO3
    Color and Shape:Solid
    Molecular weight:458.04
  • GPR4 antagonist 1

    CAS:
    <p>GPR4 antagonist 1 is a GPR4 antagonist (IC50: 189 nM).</p>
    Formula:C27H37N5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.62