Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(209 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(49 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(298 products)
- Prostaglandin Receptor(120 products)
- RAAS(87 products)
- Reductase(52 products)
- Somatostatin(49 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
Show 6 more subcategories
Found 3184 products of "Endocrinology/Hormones"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
NCG21
CAS:<p>NCG21, a GPR120 agonist, boosts ERK, Ca²⁺ responses, and GLP-1 in GPR120-expressing cells; raises GLP-1 in mice.</p>Formula:C23H24N2O3Purity:98%Color and Shape:SolidMolecular weight:376.45ADL-5859 HCl
CAS:<p>ADL-5859 is a delta-opioid receptor agonist.</p>Formula:C24H28N2O3Purity:98%Color and Shape:SolidMolecular weight:392.49EM-800
CAS:<p>EM-800, an ERα ligand & prodrug of EM-652, inhibits E1-stimulated ZR-75-1 tumor growth in mice.</p>Formula:C39H47NO6Color and Shape:SolidMolecular weight:625.79(R)-Bicalutamide
CAS:<p>(R)-Bicalutamide, an AR antagonist with antitumor properties, is crucial in prostate cancer research.</p>Formula:C18H14F4N2O4SColor and Shape:SolidMolecular weight:430.37BMS 183920
CAS:<p>BMS 183920 is a potent Angiotensin II Receptor antagonist that improves improves Caco-2 cell permeability in vivo.</p>Formula:C26H19N5O3Purity:98.92%Color and Shape:SolidMolecular weight:449.46OT antagonist 3
CAS:<p>OT antagonist 3 is an antagonist of oxytocin (OT).</p>Formula:C21H20N6O2Purity:98%Color and Shape:SolidMolecular weight:388.42TUG-905
CAS:<p>TUG-905 is an agonist for free fatty acid receptor 4 (FFA4/GPR120), and TUG-905 has the potential to treat agitation.</p>Formula:C27H30FNO5SColor and Shape:SolidMolecular weight:499.59MK181
CAS:<p>MK181 is an inhibitor of AKR1B10, a tumor marker and promising antineoplastic target.</p>Formula:C16H13BrClNO4Purity:98%Color and Shape:SolidMolecular weight:398.64DIPPA hydrochloride
CAS:<p>κ receptor antagonist</p>Formula:C22H24Cl3N3OSPurity:98%Color and Shape:SolidMolecular weight:484.87Methylprednisolone Aceponate
CAS:<p>Methylprednisolone Aceponate (SH 440), a non-halogenated corticosteroid, is a potent anti-inflammatory agent.</p>Formula:C27H36O7Purity:99.00% - 99.61%Color and Shape:SolidMolecular weight:472.57D-Methionine sulfoxide
CAS:<p>D-Methionine sulfoxide inhibits peptide methionine sulfoxide reductase and can be used to inhibit ochre mites.D-Methionine sulfoxide can be added to chicken</p>Formula:C5H11NO3SPurity:99.54%Color and Shape:SolidMolecular weight:165.21LY117018
CAS:<p>LY117018 shows antiproliferative effects on breast cancer cell lines. LY117018 is a Raloxifene analog and is a selective estrogen receptor modulator.</p>Formula:C27H25NO4SPurity:98%Color and Shape:SolidMolecular weight:459.56SB 611812
CAS:<p>SB 611812 is an antagonist of urotensin-II (UT) and can be used in studies about the treatment of cardiovascular disease.</p>Formula:C17H16Cl3F3N2O3SPurity:99.34%Color and Shape:SolidMolecular weight:491.74OBHS
CAS:<p>OBHS is an inhibitor of estrogen receptor alpha (ERα).</p>Formula:C24H20O6SColor and Shape:SolidMolecular weight:436.48A 81282
CAS:<p>A 81282 is a selective antagonist of angiotensin receptors. It has the activity of lowering blood pressure.</p>Formula:C23H23N7O2Purity:98%Color and Shape:SolidMolecular weight:429.47(±)-AC 7954 hydrochloride
CAS:<p>(±)-AC 7954 hydrochloride is a urotensin-II (UT) receptor activator.</p>Formula:C19H21Cl2NO2Purity:99.42%Color and Shape:White SolidMolecular weight:366.28SHR1653
CAS:<p>SHR1653 is a highly potent, selective and brain penetrated antagonist of oxytocin receptor (OTR)(IC50 of 15 nM for hOTR).</p>Formula:C21H21ClFN5O2Purity:98%Color and Shape:SolidMolecular weight:429.88Androgen receptor antagonist 1
CAS:<p>Androgen receptor antagonist 1, an oral full AR antagonist (IC50 59 nM), for PROTAC synthesis, reducing AR protein by 24–47% in LNCaP cells at 1–10 μM.</p>Formula:C21H25ClN4O3Purity:99.054%Color and Shape:SolidMolecular weight:416.9MCH-1 antagonist 1
CAS:<p>MCH-1 antagonist 1 also inhibits CYP3A4 (IC50: 10μM).MCH-1 antagonist 1 is a potent melanin concentrating hormone (MCH-1) antagonist (Ki: 2.6 nM).</p>Formula:C25H26N4O2Purity:98%Color and Shape:SolidMolecular weight:414.5L 366682
CAS:<p>L 366682 is an oxytocin antagonist.</p>Formula:C40H53N9O6Purity:98%Color and Shape:SolidMolecular weight:755.91OT antagonist 1
CAS:<p>OT antagonist 1 is a potent and selective antagonist of Oxytocin(Ki of 50 nM)</p>Formula:C22H22N4O3Purity:98%Color and Shape:SolidMolecular weight:390.44VPC-13789
CAS:<p>VPC-13789: potent, selective oral antiandrogen for CRPC with 0.19 μM IC50 in LNCaP cells.</p>Formula:C21H16F3N3OColor and Shape:SolidMolecular weight:383.37D36
CAS:<p>D36 is an androgen receptor allosteric antagonist. It also has inverse agonist properties.</p>Formula:C21H24N2O2Purity:98%Color and Shape:SolidMolecular weight:336.43BTI-A-404
CAS:<p>BTI-A-404 is a potent and selective competitive inverse agonist of human GPR43.</p>Formula:C22H26N4O2Color and Shape:SolidMolecular weight:378.47MK-4541
CAS:<p>MK-4541: oral, selective AR modulator, blocks 5α-reductase, curbs AR+ prostate cancer growth, effective in mouse model.</p>Formula:C22H31F3N2O3Color and Shape:SolidMolecular weight:428.49KB-130015
CAS:<p>KB-130015, a activator of hERG1 potassium channels, blocks native and recombinant hERG1 channels at high voltages.</p>Formula:C18H14I2O4Purity:98%Color and Shape:SolidMolecular weight:548.11RU 43044
CAS:<p>RU 43044 is a selective glucocorticoid receptor antagonist that has exhibited an antidepressant-like effect.</p>Formula:C29H34O2Purity:98%Color and Shape:SolidMolecular weight:414.58L-366509
CAS:<p>L-366,509 is an antagonist of oxytocin.</p>Formula:C25H33NO5SPurity:98%Color and Shape:SolidMolecular weight:459.6Androgen receptor antagonist 3
CAS:<p>Androgen receptor antagonist 3 (Compound C18) has anticancer activities that is an antagonist of androgen receptor (AR) (IC 50 = 2.4 μM) [1].</p>Formula:C22H18ClNColor and Shape:SolidMolecular weight:331.84BMS-819881
CAS:<p>BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM and it also is selective and potent for</p>Formula:C24H21ClN2O4SPurity:98%Color and Shape:SolidMolecular weight:468.95GPR40 agonist 1
CAS:<p>GPR40 agonist 1 is an effective new GPR40 agonist (EC50s: 17 nM and 2 nM for rGPR40 and hGPR40).</p>Formula:C27H30FN3O4Purity:98%Color and Shape:SolidMolecular weight:479.54Estrogen receptor-IN-1
CAS:<p>Estrogen receptor-IN-1 (compound 16) is an effective estrogen receptor (ER) inhibitor with IC 50 s of 13, 5μM for ERα and Erβ, respectively [1].</p>Formula:C14H16OSiColor and Shape:SolidMolecular weight:228.36SC 51316
CAS:<p>SC 51316 is a nonpeptidic angiotensin II (AII) receptor antagonist.</p>Formula:C24H29N7OColor and Shape:SolidMolecular weight:431.53LGD-2226
CAS:<p>LGD-2226: selective oral androgen receptor modulator, EC50: 0.2nM, Ki: 1.5nM. Treats muscle loss, osteoporosis, sexual issues.</p>Formula:C14H9F9N2OPurity:98%Color and Shape:SolidMolecular weight:392.22LY191704
CAS:<p>LY 191704 is a 5α-reductase type 1 inhibitor.</p>Formula:C14H16ClNOColor and Shape:SolidMolecular weight:249.74DK1
CAS:<p>DK1: potent ERRα modulator, lowers blood glucose, promising for diabetes research.</p>Formula:C16H13ClN2O2Color and Shape:SolidMolecular weight:300.74AT2R antagonist 1
CAS:<p>AT2R antagonist 1: potent, selective ligand, Ki 29 nM, inhibits CYP enzymes, stable in liver microsomes.</p>Formula:C23H30N4O4S2Color and Shape:SolidMolecular weight:490.64NNC45-0781
CAS:<p>NNC45-0781 is a tissue-selective partial-agonist of estrogen.</p>Formula:C27H29NO3Purity:98%Color and Shape:SolidMolecular weight:415.52AZD2906
CAS:<p>AZD2906: selective GR agonist with human/rat IC50s - 2.2/0.3 nM (PBMC), 41.6/7.5 nM (blood); induces rat bone marrow micronuclei.</p>Formula:C26H25FN4O3Color and Shape:SolidMolecular weight:460.5PF-3882845
CAS:<p>PF-3882845, a high affinity MR antagonist (IC50=2.7 nM) for hypertension, also targets progesterone receptor (IC50: 310 nM).</p>Formula:C24H22ClN3O2Purity:99.63%Color and Shape:SolidMolecular weight:419.9(R)-Viloxazine Hydrochloride
CAS:<p>(R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.</p>Formula:C13H20ClNO3Purity:99.88% - 99.94%Color and Shape:SolidMolecular weight:273.76L 364918
CAS:<p>L 364918 is an oxytocin antagonist.</p>Formula:C40H54N8O6Purity:98%Color and Shape:SolidMolecular weight:742.91(1R,2R)-2-PCCA hydrochloride
CAS:<p>(1R,2R)-2-PCCA HCl: Potent, selective GPR88 agonist, crosses BBB, EC50 1140 nM in mouse striatum. Useful for CNS research.</p>Formula:C30H39Cl2N3OPurity:98.75% - 99.67%Color and Shape:SolidMolecular weight:528.56Bopindolol fumarate
CAS:<p>Bopindolol fumarate: non-selective β1/β2-adrenoceptor blocker, partial agonist, low β3 affinity, treats hypertension.</p>Formula:C27H32N2O7Color and Shape:SolidMolecular weight:496.56Fispemifene
CAS:<p>Fispemifene (HM-101) is an estrogen receptor modulator (SERM) used to treat genitourinary syndromes and vaginal atrophy.</p>Formula:C26H27ClO3Purity:98.74% - 99.67%Color and Shape:SolidMolecular weight:422.94Renin inhibitor-1
CAS:<p>Renin inhibitor-1 (compound 26) is a potent, orally active renin inhibitor capable of acting on rh-renin (IC50: 0.9 nM) and hPRA (IC50: 1.8 nM). renal disease.</p>Formula:C22H30N4O4Color and Shape:SolidMolecular weight:414.5Prednisolone Tebutate
CAS:<p>Prednisolone Tebutate is a synthetic glucocorticoid, and is an antiinflammatory and immunosuppressant.</p>Formula:C27H38O6Purity:98%Color and Shape:SolidMolecular weight:458.59ICI 154,129
CAS:<p>Selective δ opioid antagonist</p>Formula:C34H46N4O6SPurity:98%Color and Shape:SolidMolecular weight:638.82GW7604
CAS:<p>GW7604 is an antiestrogen and it also is the metabolite of GW5638. GW5638 is an antagonist of high-affinity estrogen receptor (ER).</p>Formula:C25H22O3Purity:98%Color and Shape:SolidMolecular weight:370.44Org-34517
CAS:<p>Org-34517, a glucocorticoid receptor (GR) antagonist, is used potentially for the treatment of depression.</p>Formula:C28H30O4Purity:98%Color and Shape:SolidMolecular weight:430.54
