Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(209 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(49 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(297 products)
- Prostaglandin Receptor(120 products)
- RAAS(87 products)
- Reductase(52 products)
- Somatostatin(49 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
Show 6 more subcategories
Found 3183 products of "Endocrinology/Hormones"
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LP-471756
CAS:<p>LP-471756 is a specific antagonist of GPR139 and inhibits LP-360924-stimulated cAMP production (IC50 = 640 nM).</p>Formula:C19H23NO2SPurity:99.76%Color and Shape:SolidMolecular weight:329.46SSR126768A
CAS:<p>SSR126768A is an oxytocin receptor antagonist that inhibits uterine contractions and may be used to prevent preterm labor.</p>Formula:C33H31Cl2N3O4Purity:97.06%Color and Shape:SolidMolecular weight:604.52Acifran
CAS:<p>Acifran (AY 25712) is an HM74A/GPR109A and GPR109B agonist and displays antihyperlipidemic activity.</p>Formula:C12H10O4Purity:99.19%Color and Shape:SolidMolecular weight:218.21ICI 204,448
CAS:<p>ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of neurological diseases.</p>Formula:C23H27Cl3N2O4Purity:>99.99%Color and Shape:SolidMolecular weight:501.83NNC 63-0532
CAS:<p>NNC 63-0532 is a potentnociceptin receptor agonist, Ki=7.3 nM, EC50=305 nM.</p>Formula:C27H29N3O3Purity:99.53%Color and Shape:SolidMolecular weight:443.54CAY10786
CAS:<p>CAY10786 (GPR52 antagonist-1) is an antagonist of G protein-coupled receptor 52 (GPR52, IC50 = 0.63 μM).</p>Formula:C15H14OSPurity:99.82%Color and Shape:SolidMolecular weight:242.34AMG-009
CAS:<p>AMG-009 is a prostaglandin D2 antagonist. For CRTH2 and DP receptors, the IC50s are 3 nM and 12 nM, respectively.</p>Formula:C26H26Cl2N2O7SPurity:97.88%Color and Shape:SolidMolecular weight:581.47Faxeladol
CAS:<p>Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.</p>Formula:C15H23NOPurity:98.09% - 98.77%Color and Shape:SolidMolecular weight:233.35GPR40/FFAR1 modulator 1
CAS:<p>GPR40/FFAR1 modulator 1 is a Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1) agonist and allosteric modulator.</p>Formula:C21H19N5O3Purity:99.7%Color and Shape:SolidMolecular weight:389.41JNJ-20788560
CAS:<p>JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective for DOR than for mu opioid receptors (MOR).</p>Formula:C25H28N2O2Purity:98.02%Color and Shape:SolidMolecular weight:388.5ICI 199,441 hydrochloride
CAS:<p>ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.</p>Formula:C21H25Cl3N2OPurity:99.57%Color and Shape:SolidMolecular weight:427.8SCH-486757
CAS:<p>SCH-486757 is an agonist of nociceptin-1 (NOP1) and orphanin FQ peptide receptors and is used in the study of cough.</p>Formula:C24H23Cl2N3OPurity:99.53% - >99.99%Color and Shape:SolidMolecular weight:440.37Trimebutine CTB salt
CAS:<p>Trimebutine CTB salt (GIC-1001) is an opioid receptor agonist used in the study of pain.</p>Formula:C29H36N2O8S2Purity:99.85% - >99.99%Color and Shape:SolidMolecular weight:604.74IPAG
CAS:<p>IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.</p>Formula:C17H22IN3Purity:99.65%Color and Shape:SolidMolecular weight:395.28FPL-62129
CAS:<p>FPL-62129 is a calcium channel antagonist and a novel angiotensin-converting enzyme inhibitor with vasodilator activity for the study of cardiovascular disease.</p>Formula:C20H19ClF5NO4Purity:98.27% - 99.34%Color and Shape:SolidMolecular weight:467.81Fezagepras sodium
CAS:<p>Fezagepras sodium (Setogepram sodium salt) is an orally active GPR40 agonist and is an antagonist or inverse agonist for GPR84, with anti-fibrotic, anti-</p>Formula:C13H17NaO2Purity:99.49%Color and Shape:SolidMolecular weight:228.26GR 89696 fumarate
CAS:<p>GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.</p>Formula:C23H29Cl2N3O7Purity:99.84%Color and Shape:SolidMolecular weight:530.4ZD-6888 Hydrochloride
CAS:<p>ZD-6888 Hydrochloride, an angiotensin type 1 receptor antagonist, is used potentially for the treatment of hypertension.</p>Formula:C25H26ClN5OPurity:98.61% - 99.60%Color and Shape:SolidMolecular weight:447.96L-162,313
CAS:<p>L-162,313 is an ANG II receptor agonist, a nonpeptide that mimics the biological actions of angiotensin II and induces an increase in MAP.</p>Formula:C30H38N4O4S2Purity:99.56%Color and Shape:SolidMolecular weight:582.78TC-MCH 7c
CAS:<p>TC-MCH 7c is an oral, selectable and blood-brain barrier penetrating MCH1R antagonist with IC50 performance of 5.6 nM against hMCH1R, and TC-MCH 7c is a</p>Formula:C24H25FN2O3Purity:99.54%Color and Shape:SolidMolecular weight:408.47Posatirelin
CAS:<p>Posatirelin, a synthetic peptide, modulates and nourishes brain systems, aiding in vascular dementia research.</p>Formula:C17H28N4O4Purity:98.08% - 98.87%Color and Shape:SolidMolecular weight:352.43Estrogen receptor antagonist 8
CAS:<p>Estrogen Receptor Antagonist 8 is an ER antagonist with anti-uterine activity and may be used in the study of ovarian dysfunction.CASNETIN SODIUM (CasN)</p>Formula:C25H21N3O4Purity:98.48%Color and Shape:SolidMolecular weight:427.45Zindoxifene
CAS:<p>Zindoxifene (D 16726) is an anti-estrogenic compound with antitumor activity that can be used in studies of breast and prostate cancer.</p>Formula:C21H21NO4Purity:98.99%Color and Shape:SolidMolecular weight:351.4LY88074
CAS:<p>LY88074, a raloxifene analog sans basic side chain, is an ERβ agonist (EC50 = 232 nM) that promotes uterine cell growth.</p>Formula:C21H14O4SPurity:98.31%Color and Shape:SolidMolecular weight:362.4Indazole-Cl
CAS:<p>Indazole-Cl is a selective ERß agonist and a selective estrogen receptor modifier (SERM).</p>Formula:C13H9ClN2O2Purity:99.02% - 99.86%Color and Shape:SolidMolecular weight:260.68Orotirelin
CAS:<p>Orotirelin (CG 3509), a TRH analog, counters pentobarbital sleep; may aid in cerebral ischemia.</p>Formula:C16H19N7O5Purity:99.08%Color and Shape:SolidMolecular weight:389.37Terlakiren
CAS:<p>Terlakiren (CP-80,794) is a renin inhibitor that inhibits the potency of human renin and can be used to study neurological disorders of the hypertensive type.</p>Formula:C31H48N4O7SPurity:99.38%Color and Shape:SolidMolecular weight:620.8Moveltipril
CAS:<p>Moveltipril (Moveltipril calcium) is a potent angiotensin-converting enzyme (ACE) inhibitor.Moveltipril is converted to captopril in the body for action.</p>Formula:C19H30N2O5SPurity:97.55% - 98.28%Color and Shape:SolidMolecular weight:398.52ME-3221
CAS:<p>Apomine inhibits HMG-CoA-reductase, induces myeloma cell apoptosis, modulates myeloma, and boosts lovastatin's antitumor effects.</p>Formula:C22H21N5O2Purity:99.84% - 99.93%Color and Shape:SolidMolecular weight:387.43ONC1-13B
CAS:<p>ONC1-13B, an androgen receptor antagonist, is used potentially for the treatment of prostate cancer.</p>Formula:C22H16F4N4O3SPurity:99.36% - 99.85%Color and Shape:SolidMolecular weight:492.45Buloxibutid
CAS:<p>Buloxibutid: a novel AT2 receptor agonist, Ki=0.4 nM (AT2), 10 μM (AT1).</p>Formula:C23H29N3O4S2Purity:97.68% - 98.58%Color and Shape:SolidMolecular weight:475.62SB-657510
CAS:<p>SB-657510: UT antagonist, Ki (nM) - human 61, monkey 17, cat 30, rat 65, mouse 56; reduces UII-induced inflammation, aids diabetic atherosclerosis.</p>Formula:C19H22BrClN2O5SPurity:98.06%Color and Shape:SolidMolecular weight:505.81Endoxifen hydrochloride
CAS:<p>Endoxifen HCl, a Tamoxifen metabolite, targets estrogen receptors more effectively and blocks aromatase, showing promise for breast cancer research.</p>Formula:C25H28ClNO2Purity:99.08%Color and Shape:SolidMolecular weight:409.95Ralaniten triacetate
CAS:<p>Ralaniten triacetate (EPI-506) is a precursor of Ralaniten, an AR-NTD inhibitor, which can be used in the study of prostate and breast cancer.</p>Formula:C27H33ClO8Purity:98.69%Color and Shape:SolidMolecular weight:521.00BMS-641988
CAS:<p>BMS-641988 is a novel nonsteroidal androgen receptor antagonist for the treatment of prostate cancer.</p>Formula:C20H20F3N3O5SPurity:99.57% - 99.92%Color and Shape:SoildMolecular weight:471.45Ripisartan
CAS:<p>Ripisartan (UP-269-6) is a potent and specific angiotensin II receptor antagonist that inhibits angiotensin II-mediated sympathetic tachycardia responses.</p>Formula:C23H22N8OPurity:98.86%Color and Shape:SolidMolecular weight:426.47Glucocorticoid receptor agonist-1
CAS:<p>Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM[1].</p>Formula:C35H39NO6Purity:99.68%Color and Shape:SolidMolecular weight:569.69Palazestrant
CAS:<p>Palazestrant, an antiestrogen and antineoplastic agent, effectively targets ER+/HER2+ cancer when used in conjunction with a HER2 inhibitor.</p>Formula:C28H36FN3OPurity:97.55%Color and Shape:SolidMolecular weight:449.6SQ 32970
CAS:<p>SQ 32970 is a potent Endothia aspartic proteinase inhibitor.</p>Formula:C33H51N5O4SColor and Shape:SolidMolecular weight:613.85PD 125754
CAS:<p>PD 125754 is a Renin inhibitor, which represents a group of pharmaceutical drugs used primarily to treat essential hypertension.</p>Formula:C42H65N5O7Purity:98%Color and Shape:SolidMolecular weight:751.99Nur77 modulator 2
CAS:<p>Nur77 modulator 2: Kd of 0.35 μM, oral anti-inflammatory, affects Nur77/mitochondria localization.</p>Formula:C26H25NO5Color and Shape:SolidMolecular weight:431.48PF 00277343
CAS:<p>PF 00277343, a thyroid receptor agonist, is used for the treatment of androgenetic alopecia.</p>Formula:C24H20FN3O4Purity:98%Color and Shape:SolidMolecular weight:433.43ADL-08-0011
CAS:<p>ADL-08-0011 is an metabolite of alvimopan.</p>Formula:C23H29NO3Color and Shape:SolidMolecular weight:367.49L 681176
CAS:<p>L 681176 is an inhibitor of the angiotensin-converting enzyme.</p>Formula:C12H23N5O7Color and Shape:SolidMolecular weight:349.34Frakefamide
CAS:<p>Frakefamide: potent analgesic, μ-selective agonist, non-CNS penetrating.</p>Formula:C30H34FN5O5Purity:98%Color and Shape:SolidMolecular weight:563.62JNJ-17148066
CAS:<p>JNJ-17148066 is an agonist of estrogen receptor ESR1.</p>Formula:C30H31NO5Purity:98%Color and Shape:SolidMolecular weight:485.57Estrogen receptor antagonist 5
CAS:<p>Compound 165: Potent estrogen receptor antagonist; useful for metastatic disease research.</p>Formula:C25H31F3N2O3Color and Shape:SolidMolecular weight:464.52Estrogen receptor modulator 7
CAS:<p>Estrogen Receptor Modulator 7 is a potent modulator of estrogen receptors, utilized in cancer research [1].</p>Formula:C30H31BCl2FNO3Purity:98%Color and Shape:SolidMolecular weight:554.29Mu opioid receptor antagonist 7
CAS:<p>Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (</p>Formula:C22H27ClN2O2Purity:98%Color and Shape:SolidMolecular weight:386.91CITFA
CAS:<p>CITFA, a GPER agonist, enhances neurite outgrowth in rat embryonic (E18) hippocampal neurons [1].</p>Formula:C25H35NO2Color and Shape:SolidMolecular weight:381.55
