Vasopressin Receptor
Vasopressin receptors are a family of G protein-coupled receptors that mediate the effects of vasopressin, a hormone involved in regulating water balance, blood pressure, and kidney function. Vasopressin receptor agonists and antagonists are studied for their roles in treating conditions such as diabetes insipidus, hyponatremia, and heart failure. These receptors are also important targets in research on fluid balance and cardiovascular health. At CymitQuimica, we provide a selection of high-quality vasopressin receptor modulators to support your research in endocrinology, nephrology, and cardiovascular biology.
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Terlipressin Acetate
CAS:1884420-36-3
Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial …
Formula:
C56H82N16O19S2
Purity:
98.50% - 99.69%
Color and Shape:
Solid
Molecular weight:
1347.5
Ref: TM-T13920L
| 5mg | 48.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 103.00 € | ||
| 50mg | 136.00 € | ||
| 100mg | 207.00 € | ||
| 200mg | 310.00 € |
Estimated delivery in United States, on Tuesday 13 May 2025
Balovaptan
CAS:1228088-30-9
Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism …
Formula:
C22H24ClN5O
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
409.91
Ref: TM-T14494
| 5mg | 66.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 303.00 € | ||
| 100mg | 472.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Tuesday 13 May 2025
V1a/V2 antagonist 1
V1a/V2 antagonist 1 (Compound 18j) is an orally active dual-target antagonist of V1a and V2 …
Formula:
C25H26ClN5O3
Color and Shape:
Solid
Molecular weight:
479.96
Ref: TM-T203525
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 12 May 2025
Nelivaptan
CAS:439687-69-1
Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective …
Formula:
C30H32ClN3O8S
Purity:
98% - 98.39%
Color and Shape:
Solid
Molecular weight:
630.11
Ref: TM-T28153
| 1mg | 78.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 210.00 € | ||
| 25mg | 349.00 € | ||
| 50mg | 517.00 € | ||
| 100mg | 745.00 € | ||
| 500mg | 1,549.00 € |
Estimated delivery in United States, on Monday 12 May 2025
Fedovapagon
CAS:347887-36-9
Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder …
Formula:
C27H34N4O3
Purity:
99.33%
Color and Shape:
Solid
Molecular weight:
462.58
Ref: TM-T15273
| 5mg | 111.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 373.00 € | ||
| 50mg | 655.00 € | ||
| 100mg | 924.00 € | ||
| 1mL*10mM (DMSO) | 124.00 € |
Estimated delivery in United States, on Wednesday 14 May 2025
Argipressin
CAS:113-79-1
Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM …
Formula:
C46H65N15O12S2
Purity:
98%
Color and Shape:
White Powder
Molecular weight:
1084.23
Ref: TM-T7434
| 1mg | 50.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 118.00 € |
Estimated delivery in United States, on Wednesday 14 May 2025
Atosiban
CAS:90779-69-4
Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions …
Formula:
C43H67N11O12S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
994.19
Ref: TM-T4996
| 5mg | 67.00 € | ||
| 10mg | 90.00 € | ||
| 50mg | 205.00 € | ||
| 100mg | 299.00 € |
Estimated delivery in United States, on Wednesday 14 May 2025
LIXIVAPTAN
CAS:168079-32-1
Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
Formula:
C27H21ClFN3O2
Purity:
98.36%
Color and Shape:
Solid
Molecular weight:
473.93
Ref: TM-T7303
| 1mg | 43.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 81.00 € | ||
| 10mg | 127.00 € | ||
| 25mg | 249.00 € | ||
| 50mg | 424.00 € | ||
| 100mg | 625.00 € | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Tuesday 20 May 2025
Fuscoside
CAS:131631-89-5
Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value …
Formula:
C26H31N3O4
Purity:
97.98% - 99.66%
Color and Shape:
Solid
Molecular weight:
449.54
Ref: TM-T4355
| 2mg | 57.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 106.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 244.00 € | ||
| 100mg | 419.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Tuesday 20 May 2025
Felypressin
CAS:56-59-7
Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic …
Formula:
C46H65N13O11S2
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
1040.22
Ref: TM-T2568
| 2mg | 37.00 € | ||
| 5mg | 55.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 116.00 € | ||
| 50mg | 172.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 20 May 2025
RG7713
CAS:920022-47-5
RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.
Formula:
C25H28ClN3O2
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
437.96
Ref: TM-T4141
| 1mg | 59.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 200.00 € | ||
| 25mg | 339.00 € | ||
| 50mg | 507.00 € | ||
| 100mg | 730.00 € |
Estimated delivery in United States, on Tuesday 20 May 2025
Tolvaptan
CAS:150683-30-0
Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that …
Formula:
C26H25ClN2O3
Purity:
97% - 99.91%
Color and Shape:
Solid
Molecular weight:
448.94
Ref: TM-T2326
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 81.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 364.00 € | ||
| 1mL*10mM (DMSO) | 127.00 € |
Estimated delivery in United States, on Tuesday 20 May 2025
Atosiban acetate
CAS:914453-95-5
Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin.
Formula:
C45H71N11O14S2
Purity:
99.15% - 99.84%
Color and Shape:
Solid
Molecular weight:
1054.24
Ref: TM-T5148
| 5mg | 73.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 207.00 € | ||
| 100mg | 268.00 € | ||
| 500mg | 660.00 € | ||
| 1mL*10mM (DMSO) | 134.00 € |
Estimated delivery in United States, on Tuesday 20 May 2025
Conivaptan hydrochloride
CAS:168626-94-6
Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in …
Formula:
C32H26N4O2·HCl
Purity:
98.33% - 99.86%
Color and Shape:
Solid
Molecular weight:
535.04
Ref: TM-T6453
| 5mg | 44.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 378.00 € | ||
| 200mg | 567.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Tuesday 20 May 2025
Mozavaptan
CAS:137975-06-5
Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with …
Formula:
C27H29N3O2
Purity:
98.98% - 99.12%
Color and Shape:
Solid
Molecular weight:
427.54
Ref: TM-T6288
| 10mg | 50.00 € | ||
| 25mg | 74.00 € | ||
| 50mg | 97.00 € | ||
| 100mg | 154.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 20 May 2025
Felypressin acetate
CAS:914453-97-7
Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin …
Formula:
C48H69N13O13S2
Purity:
97.06%
Color and Shape:
Solid
Molecular weight:
1100.27
Ref: TM-T2568L
| 5mg | 47.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 187.00 € | ||
| 100mg | 298.00 € | ||
| 200mg | 444.00 € | ||
| 500mg | 715.00 € |
Estimated delivery in United States, on Tuesday 1 Jul 2025
OPC-51803
CAS:192514-54-8
OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of …
Formula:
C26H32ClN3O2
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
454
Ref: TM-T28257
| 1mg | 333.00 € | ||
| 5mg | 787.00 € | ||
| 10mg | 1,074.00 € | ||
| 25mg | 1,510.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € | ||
| 500mg | 4,655.00 € |
Estimated delivery in United States, on Tuesday 1 Jul 2025
E-4177
CAS:135070-05-2
E-4177 is an angiotensin II type 1 receptor (AT1R) antagonist and can be used to …
Formula:
C24H21N3O2
Purity:
98.63% - 99.39%
Color and Shape:
Solid
Molecular weight:
383.44
Ref: TM-T27229
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 1 Jul 2025
TASP0390325
CAS:1642187-96-9
TASP0390325, a potent and orally active V1B receptor antagonist, has antidepressant and anxiolytic activities in …
Formula:
C25H30Cl2FN5O4
Purity:
98.62%
Color and Shape:
Solid
Molecular weight:
554.44
Ref: TM-T28926
| 1mg | 57.00 € | ||
| 5mg | 120.00 € | ||
| 10mg | 188.00 € | ||
| 25mg | 432.00 € | ||
| 50mg | 747.00 € | ||
| 100mg | 1,216.00 € |
Estimated delivery in United States, on Tuesday 1 Jul 2025
