Vasopressin Receptor
Vasopressin receptors are a family of G protein-coupled receptors that mediate the effects of vasopressin, a hormone involved in regulating water balance, blood pressure, and kidney function. Vasopressin receptor agonists and antagonists are studied for their roles in treating conditions such as diabetes insipidus, hyponatremia, and heart failure. These receptors are also important targets in research on fluid balance and cardiovascular health. At CymitQuimica, we provide a selection of high-quality vasopressin receptor modulators to support your research in endocrinology, nephrology, and cardiovascular biology.
Found 44 products of "Vasopressin Receptor"
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Terlipressin Acetate
CAS:<p>Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).</p>Formula:C56H82N16O19S2Purity:98.50% - 99.69%Color and Shape:SolidMolecular weight:1347.5Nelivaptan
CAS:<p>Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective and quality-assured.</p>Formula:C30H32ClN3O8SPurity:98.46% - 99.89%Color and Shape:SolidMolecular weight:630.11Balovaptan
CAS:<p>Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.</p>Formula:C22H24ClN5OPurity:99.88%Color and Shape:SolidMolecular weight:409.91(D-Arg8)-Inotocin
CAS:<p>'(D-Arg8)-Inotocin is a potent, selective, and competitive antagonist of the vasopressin receptor (V 1a R), exhibiting a binding affinity (K i) of 1.3 nM.</p>Formula:C39H68N14O11S2Purity:98%Color and Shape:SolidMolecular weight:973.17d[Cha4]-AVP
CAS:<p>Potent human V1B vasopressin receptor agonist; Ki: V1B=1.2 nM; increases ACTH, corticosterone; low vasopressor effect.</p>Formula:C50H71N13O11S2Purity:98%Color and Shape:SolidMolecular weight:1094.31(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
CAS:<p>V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.</p>Formula:C52H74N14O12S2Purity:98%Color and Shape:White Lyophilized PowderMolecular weight:1151.38d[Leu4,Lys8]-VP
CAS:<p>Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.</p>Formula:C47H67N11O11S2Purity:98%Color and Shape:SolidMolecular weight:1026.2d[Cha4]-AVP TFA
<p>d[Cha4]-AVP TFA: potent, selective V1b agonist, K i 1.2 nM, favors V1b over V1a, V2, oxytocin receptors.</p>Formula:C52H72F3N13O13S2Color and Shape:SolidMolecular weight:1208.33Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
CAS:<p>Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), acts as a weak agonist at the antidiuretic receptor but is a potent</p>Formula:C45H63N15O11S2Color and Shape:SolidMolecular weight:1054.21[Asu1,6-Arg8]Vasopressin
CAS:<p>[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.</p>Formula:C48H68N14O12Color and Shape:SolidMolecular weight:1033.14(Phe2,Orn8)-Oxytocin acetate
<p>(Phe2,Orn8)-Oxytocin acetate: V1 agonist with EC50 of 280 nM for rabbit epididymis contractility.</p>Formula:C44H69N13O13S2Color and Shape:SolidMolecular weight:1052.23Selepressin acetate
<p>Selepressin acetate is a useful organic compound for research related to life sciences and the catalog number is T73654.</p>Formula:C48H77N13O13S2Color and Shape:SolidMolecular weight:1108.33(Phe2,Orn8)-Oxytocin
CAS:<p>(Phe2,Orn8)-Oxytocin: Selective V1 agonist, induces rabbit epididymis contractility, EC50=280 nM.</p>Formula:C42H65N13O11S2Color and Shape:SolidMolecular weight:992.18D[LEU4,LYS8]-VP TFA
<p>D[LEU4,LYS8]-VP TFA: V1b receptor agonist; K_i: 0.16 nM (rat), 0.52 nM (human), 1.38 nM (mouse); weak antidiuretic/vasopressor/oxytocic.</p>Formula:C49H68F3N11O13S2Color and Shape:SolidMolecular weight:1140.25(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin
CAS:<p>Potent VP V1R antagonist, lowers rat MAP: '(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin'.</p>Formula:C54H76N14O11Color and Shape:SolidMolecular weight:1097.27[8-L-arginine] deaminovasopressin
CAS:<p>[8-L-arginine] deaminovasopressin (dAVP) is a vasopressin analog [1] .</p>Formula:C46H64N14O13S2Color and Shape:SolidMolecular weight:1085.22Endolide F
<p>Endolide F (Compound 2) is a proline-containing lactone that serves as a moderate antagonist of the arginine vasopressin V1A receptor.</p>Formula:C25H32N4O6Molecular weight:484.23218Velmupressin acetate
CAS:<p>Potent, selective, short-acting peptidic V2R agonist; EC50: 0.07 nM (hV2R), 0.02 nM (rV2R).</p>Formula:C44H64ClN11O10S2Purity:98%Color and Shape:SolidMolecular weight:1006.63d[Leu4,Lys8]-VP acetate
<p>d[Leu4,Lys8]-VP acetate: Vasopressin V1b agonist. Ki: rat 0.16 nM, human 0.52 nM, mouse 1.38 nM. Low antidiuretic/vasopressor effects.</p>Formula:C49H71N11O13S2Purity:98.86%Color and Shape:SolidMolecular weight:1086.28Dp[Tyr(methyl)2,Arg8]-Vasopressin
CAS:<p>Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].</p>Formula:C49H70N14O12S2Purity:98%Color and Shape:SolidMolecular weight:1111.3Invopressin
CAS:<p>Invopressin (Compound 42), a vasopressin V1A receptor partial agonist (EC50: 1.0 nM), is utilized in research related to cirrhosis conditions such as bacterial</p>Formula:C110H161N31O27S2Purity:98%Color and Shape:SolidMolecular weight:2413.78[Deamino-Pen1,Val4,D-Arg8]-vasopressin
CAS:<p>[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an antagonist of arginine-vasopressin (AVP).</p>Formula:C48H69N13O11S2Purity:98%Color and Shape:SolidMolecular weight:1068.27Val9-Oxytocin
CAS:<p>Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor.</p>Formula:C46H72N12O12S2Purity:98%Color and Shape:SolidMolecular weight:1049.27(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS:<p>(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].</p>Formula:C52H76N14O11S2Purity:98%Color and Shape:SolidMolecular weight:1137.38V1a/V2 antagonist 1
<p>V1a/V2 antagonist 1 (Compound 18j) is an orally active dual-target antagonist of V1a and V2 receptors, exhibiting high binding affinity toward these receptors [Ki values are hV1a: 0.13 nM, hV2: 0.53 nM, and mV1a: 0.5 nM; IC50 for hV1a is 2.2 nM]. This compound can inhibit oxytocin-induced scratching behavior in mice.</p>Formula:C25H26ClN5O3Color and Shape:SolidMolecular weight:479.96Fedovapagon
CAS:<p>Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.</p>Formula:C27H34N4O3Purity:99.33%Color and Shape:SolidMolecular weight:462.58Argipressin
CAS:<p>Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.</p>Formula:C46H65N15O12S2Purity:98%Color and Shape:White PowderMolecular weight:1084.23Atosiban
CAS:<p>Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions rapidly.</p>Formula:C43H67N11O12S2Purity:98%Color and Shape:SolidMolecular weight:994.19Fuscoside
CAS:<p>Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.</p>Formula:C26H31N3O4Purity:98.13% - 99.66%Color and Shape:SolidMolecular weight:449.54d[Cha4]-AVP acetate(500170-27-4 free base)
<p>'d[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'</p>Formula:C52H75N13O13S2Purity:99.86%Color and Shape:SolidMolecular weight:1154.37Atosiban acetate
CAS:<p>Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin.</p>Formula:C45H71N11O14S2Purity:99.84% - 99.92%Color and Shape:SolidMolecular weight:1054.24Conopressin S acetate(111317-90-9 free base)
<p>Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b</p>Formula:C43H77N17O12S2Purity:99.79%Color and Shape:SolidMolecular weight:1088.32LIXIVAPTAN
CAS:<p>Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)</p>Formula:C27H21ClFN3O2Purity:98.36%Color and Shape:SolidMolecular weight:473.93Desmopressin acetate (16679-58-6 free base)
CAS:<p>Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine production.</p>Formula:C48H68N14O14S2Purity:98.84% - >99.99%Color and Shape:SolidMolecular weight:1129.26Tolvaptan
CAS:<p>Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.</p>Formula:C26H25ClN2O3Purity:99.78% - >99.99%Color and Shape:SolidMolecular weight:448.94Conivaptan hydrochloride
CAS:<p>Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and</p>Formula:C32H26N4O2·HClPurity:98.33% - 99.86%Color and Shape:SolidMolecular weight:535.04RG7713
CAS:<p>RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.</p>Formula:C25H28ClN3O2Purity:99.74%Color and Shape:SolidMolecular weight:437.96Mozavaptan
CAS:<p>Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.</p>Formula:C27H29N3O2Purity:98.98% - 99.12%Color and Shape:SolidMolecular weight:427.54Felypressin
CAS:<p>Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.</p>Formula:C46H65N13O11S2Purity:99.65%Color and Shape:SolidMolecular weight:1040.22Felypressin acetate
CAS:<p>Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS.</p>Formula:C48H69N13O13S2Purity:97.06%Color and Shape:SolidMolecular weight:1100.27OPC-51803
CAS:<p>OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.</p>Formula:C26H32ClN3O2Purity:98.93% - >99.99%Color and Shape:SolidMolecular weight:454TASP0390325
CAS:<p>TASP0390325, a potent and orally active V1B receptor antagonist, has antidepressant and anxiolytic activities in rodents.</p>Formula:C25H30Cl2FN5O4Purity:98.62%Color and Shape:SolidMolecular weight:554.44RGH-122
CAS:<p>RGH-122 (compound 43), characterized as an orally active, potent, and selective hV1a receptor antagonist, demonstrates significant affinity with a K i value of 0.3 nM and an IC 50 of 0.9 nM. It exhibits microsomal stability, indicated by a CL int value of 13/28/25 μL/min/mg [1].</p>Formula:C24H25ClN4O3Color and Shape:SolidMolecular weight:452.93Elsovaptan
CAS:<p>Elsovaptan is an antagonist of the vasopressin receptor and is applicable for research in Alzheimer's disease.</p>Formula:C19H20ClN5O2Color and Shape:SolidMolecular weight:385.847
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![[Asu1,6-Arg8]Vasopressin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT76510.webp&w=3840&q=75)
![[8-L-arginine] deaminovasopressin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT76573.webp&w=3840&q=75)
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![Dp[Tyr(methyl)2,Arg8]-Vasopressin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT80073.webp&w=3840&q=75)
![[Deamino-Pen1,Val4,D-Arg8]-vasopressin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT83501.webp&w=3840&q=75)
![d[Cha4]-AVP acetate(500170-27-4 free base)](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP2082L.webp&w=3840&q=75)
