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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2293 products of "Membrane Transporter/Ion Channel"

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  • Repaglinide D5

    CAS:
    <p>Repaglinide D5 is deuterium labeled Repaglinide. Repaglinide is an insulin secretagogue for treatment type-2 diabetes mellitus.</p>
    Formula:C27H36N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:457.62
  • Bumetanide-d5

    CAS:
    Bumetanide D5 is a deuterium-labeled Bumetanide. Bumetanide is a Na+-K+-Cl- (NKCC1) inhibitor (IC50s: 0.68 and 4.0 μM for hNKCC1A and hNKCC2A).
    Formula:C17H20N2O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:369.45
  • Propafenone D7 hydrochloride

    CAS:
    <p>Propafenone D7 hydrochloride is the deuterium labeled Propafenone, and is a classic anti-arrhythmic medication.</p>
    Formula:C21H28ClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:384.95
  • Nifedipine-d6

    CAS:
    <p>Nifedipine D6 is deuterium labeled nifedipine which is a potent blocker of calcium channel.</p>
    Formula:C17H18N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.37
  • Methocarbamol D5

    CAS:
    <p>Methocarbamol is a central muscle relaxant. Methocarbamol D5 is deuterium labeled Methocarbamol.</p>
    Formula:C11H15NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:246.27
  • MNI-caged-NMDA

    CAS:
    <p>NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group</p>
    Formula:C14H17N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:323.30
  • A-317491 sodium salt hydrate


    <p>A-317491 sodium salt hydrate is a non-nucleotide P2X3 and P2X2/3 receptor antagonist, which inhibits calcium flux mediated by the receptors.</p>
    Formula:C33H29NNaO9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:606.57
  • DL-AP7

    CAS:
    <p>DL-AP7: competitive NMDA antagonist, anticonvulsant, inhibits NMDA convulsions, impairs mice learning.</p>
    Formula:C7H16NO5P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:225.18
  • N-Acetylglycyl-D-glutamic acid

    CAS:
    <p>Excitatory peptide that induces seizures</p>
    Formula:C9H14N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:246.22
  • S1647

    CAS:
    S1647 is a dual inhibitor targeting both ASBT and SOAT. It is utilized in research focused on intrahepatic cholestasis, cholestatic pruritus, and constipation.
    Formula:C19H13Cl2N3O5S
    Molecular weight:466.30
  • R-(-)-Niguldipine hydrochloride

    CAS:
    <p>R-(-)-Niguldipine HCl: L-type Ca2+ blocker, K+ agonist, α1A antagonist; lowers blood pressure; weaker enantiomer.</p>
    Formula:C36H40ClN3O6
    Color and Shape:Solid
    Molecular weight:646.17
  • Pradigastat

    CAS:
    Pradigastat (LCQ-908) is a diacylglycerol acyltransferase 1 (DGAT1) inhibitor for the treatment of constipation and can be used in the study of obesity
    Formula:C25H24F3N3O2
    Purity:95.21% - 95.21%
    Color and Shape:Solid
    Molecular weight:455.47
  • LY 303511

    CAS:
    <p>LY303511, an inactive analogue of LY294002, is a mTOR inhibitor and no inhibition for PI3-K.</p>
    Formula:C19H18N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:306.36
  • Tetradifon

    CAS:
    <p>Tetradifon is a broad-spectrum organochlorine acaricide that inhibits mitochondrial OSCP, blocking energy production (IC50=4.5-27nmoL/mg) with oligomycin-like effects.</p>
    Formula:C12H6Cl4O2S
    Purity:99.84%
    Color and Shape:Yellowish Odorless Oil
    Molecular weight:356.05
  • 8-Pcpt-cGMP sodium

    CAS:
    <p>8-Pcpt-cGMP sodium, with an EC50 of 0.5 μM, acts as an agonist for cyclic nucleotide-gated (CNG) channels and demonstrates effective membrane permeability. This compound is utilized in research focused on the role of CNG channels in visual and olfactory signal transduction.</p>
    Formula:C16H14ClN5NaO7PS
    Color and Shape:Solid
    Molecular weight:509.79
  • ORM-10103

    CAS:
    ORM-10103 is a novel potent and selective inhibitor of the Na+/Ca2+ exchanger (NCX).ORM-10103 inhibited NCX currents with estimated IC50 values of 55 and 67 nM
    Formula:C20H16N2O4
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:348.35
  • FFN 511 hydrochloride

    CAS:
    <p>FFN 511 hydrochloride is a fluorescent pseudo-neurotransmitter (FFNs) targeting VMA T2 that can be used to label baraminergic nerve endings.</p>
    Formula:C17H21ClN2O2
    Purity:99.83%
    Color and Shape:Soild
    Molecular weight:320.81
  • Diphenidol

    CAS:
    <p>Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.</p>
    Formula:C21H27NO
    Color and Shape:Needles From Petroleum Ether Solid
    Molecular weight:309.45
  • IEM 1754 2HBr

    CAS:
    <p>IEM 1754 2HBr (IEM 1754 dihydrobromide) is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM.</p>
    Formula:C16H30N2·2HBr
    Purity:99.71% - 99.72%
    Color and Shape:Solid
    Molecular weight:412.25
  • Verapamil

    CAS:
    <p>Verapamil (CP-16533-1), an oral calcium channel blocker, inhibits P-gp and CYP3A4, used for hypertension, arrhythmias, and angina research.</p>
    Formula:C27H38N2O4
    Purity:99.61% - 99.93%
    Color and Shape:Oil
    Molecular weight:454.6
  • Clopamide

    CAS:
    <p>Clopamide (Brinaldix) is a piperidine and sulfamoylbenzamide-based diuretic with thiazide-like diuretic activity.</p>
    Formula:C14H20ClN3O3S
    Purity:99.71%
    Color and Shape:White To Yellowish Crystalline Powder
    Molecular weight:345.84
  • Aprikalim

    CAS:
    <p>Aprikalim opens KATP channels, protects the heart, and at high doses, dilates blood vessels.</p>
    Formula:C12H16N2OS2
    Purity:99.42% - 99.90%
    Color and Shape:Solid
    Molecular weight:268.4
  • SCH 50911 hydrochloride

    CAS:
    <p>SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).</p>
    Formula:C8H16ClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:209.67
  • PPNDS

    CAS:
    <p>P2X1 receptor antagonist</p>
    Formula:C18H15N4NaO14PS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:629.42
  • NO 711

    CAS:
    <p>NO 711(NNC-711 free acid) is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.</p>
    Formula:C21H22N2O3
    Purity:99.70%
    Color and Shape:Solid
    Molecular weight:350.41
  • (±)-Homoproline Hydrochloride

    CAS:
    <p>(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can Trust</p>
    Formula:C6H12ClNO2
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:165.62
  • VU0405601

    CAS:
    <p>VU0405601 is a hERG channel activator that protects against drug-induced cardiac arrhythmias.</p>
    Formula:C17H13BrN2O2
    Purity:99.16%
    Color and Shape:Solid
    Molecular weight:357.2
  • JTV-519 hemifumarate

    CAS:
    <p>JTV-519 hemifumarate: Ca2+ blocker, SERCA inhibitor, ryanodine receptor partial agonist; antiarrhythmic, cardioprotective.</p>
    Formula:C54H68N4O8S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:965.28
  • HN37

    CAS:
    <p>HN37, KCNQ2 activator (EC50=37 nM). Affordable Excellence: Reliable Quality You Can Trust</p>
    Formula:C20H21FN2O2
    Purity:99.27%
    Color and Shape:Solid
    Molecular weight:340.39
  • ICA

    CAS:
    ICA (N-[4-(2-Pyridinyl)-2-thiazolyl]-2-pyridinamine) is a SK channel inhibitor and exhibits antileishmanial activity (IC50: 2.1 µM).
    Formula:C13H10N4S
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:254.31
  • Benzamil hydrochloride

    CAS:
    <p>Benzamil hydrochloride is a specific and potent sodium channel (ENaC) blocker.</p>
    Formula:C13H15Cl2N7O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.21
  • V-9302

    CAS:
    <p>V-9302 (V9302) is a competitive antagonist of transmembrane glutamine flux that selectively and potently targets the amino acid transporter ASCT2 (IC50: 9.6 uM</p>
    Formula:C34H38N2O4
    Purity:98% - 99.54%
    Color and Shape:Solid
    Molecular weight:538.68
  • Nifekalant hydrochloride

    CAS:
    Nifekalant hydrochloride is an IKr potassium channel blocker with an IC50 of 10 µM.
    Formula:C19H28ClN5O5
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:441.91
  • CFTR corrector 9

    CAS:
    <p>CFTR corrector 9 is a CF modulator used to research cystic fibrosis and related disorders.</p>
    Formula:C16H14N2O4
    Purity:98.24%
    Color and Shape:Solid
    Molecular weight:298.29
  • L-4FPG

    CAS:
    <p>L-4FPG is a Glycine derivative, inhibits the neutral amino acid transporters ASCT1 and ASCT2.</p>
    Formula:C8H8FNO2
    Purity:99.26%
    Color and Shape:Solid
    Molecular weight:169.15
  • TRPC6-PAM-C20

    CAS:
    <p>TRPC6-PAM-C20, a selective enhancer for TRPC6, boosts calcium in HEK cells and OAG-related platelet clumping, EC50: 2.37μM.</p>
    Formula:C22H21NO4
    Purity:98.16%
    Color and Shape:Solid
    Molecular weight:363.41
  • CP-100356 hydrochloride

    CAS:
    <p>CP-100356 hydrochloride is an MDR1 (P-gp) and BCRP inhibitor, a nucleotide-derived substrate analog that induces stomatal opening in the dark.</p>
    Formula:C31H37ClN4O6
    Purity:99.19%
    Color and Shape:Solid
    Molecular weight:597.1
  • Nav1.7 inhibitor

    CAS:
    <p>Nav1.7 inhibitor is a Nav1.7 inhibitor for research in the field of pain and anesthesia.</p>
    Formula:C15H11Cl3FNO4S
    Purity:97.52%
    Color and Shape:Solid
    Molecular weight:426.68
  • CP-457920

    CAS:
    <p>CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.</p>
    Formula:C18H17N3O3
    Purity:99.06% - 99.74%
    Color and Shape:Solid
    Molecular weight:323.35
  • FSBA hydrochloride

    CAS:
    <p>FSBA hydrochloride(5'-p-Fluorosulfonylbenzoyladenosine) is an ATP analogue serving as an affinity probe for the ATP site of Na/K-ATPase.</p>
    Formula:C17H17ClFN5O7S
    Purity:97.96%
    Color and Shape:Solid
    Molecular weight:489.86
  • Sodium Channel inhibitor 2

    CAS:
    <p>Sodium Channel inhibitor 2 is a blocker of sodium channel.</p>
    Formula:C26H25Cl2N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:466.4
  • Cilobradine hydrochloride

    CAS:
    <p>Cilobradine hydrochloride (DK-AH 269) is an HCN Channel blocker and an open channel blocker of neuronal Ih and related cardiac If channels.</p>
    Formula:C28H39ClN2O5
    Purity:98.40%
    Color and Shape:Solid
    Molecular weight:519.07
  • TC-AQP1-1

    CAS:
    TC-AQP1-1 blocks aquaporin 1; found via virtual screening; hinders water flux in Xenopus oocytes at low µM.
    Formula:C12H10O4
    Purity:97.59%
    Color and Shape:Solid
    Molecular weight:218.21
  • Bamaluzole

    CAS:
    <p>Bamaluzole is an agonist of GABA receptor.</p>
    Formula:C14H12ClN3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:273.72
  • BK 129

    CAS:
    BK 129 is a local anesthetic with relaxant properties. BK 129 inhibits Ca2+ entry into the smooth muscle cell and Ca2+ release from sarcoplasmic reticulum.
    Formula:C22H36N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.53
  • Almokalant

    CAS:
    <p>Almokalant: Class III antiarrhythmic, K+ channel blocker, inhibits Ikr current.</p>
    Formula:C18H28N2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.49
  • V116517

    CAS:
    <p>V-116517, a TRPV1 antagonist, is used potentially for the treatment of severe pain due to osteoarthritis and chronic pain due postherpetic neuralgia (PHN).</p>
    Formula:C19H18ClF3N4O3
    Color and Shape:Solid
    Molecular weight:442.82
  • AMG8788

    CAS:
    <p>AMG8788 is a selective, potent and orally active TRPM8 antagonist (IC50: 63.2 nM).</p>
    Formula:C23H18F4N2O
    Color and Shape:Solid
    Molecular weight:414.4
  • JTV-519 fumarate

    CAS:
    Ryanodine receptor (RyR) inhibitor; stabilizes RyR2 in a closed conformation. Exhibits antiarrhythmic and cardioprotective properties in vivo.
    Formula:C29H36N2O6S
    Color and Shape:Solid
    Molecular weight:540.67
  • PD 122860

    CAS:
    <p>PD 122860 is a dihydropyridine enhancing heart contractility, altering ECG, and relaxing aortic rings.</p>
    Formula:C23H20F3N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:491.48
  • DS1

    CAS:
    <p>DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.</p>
    Formula:C18H10Br2ClN3OS
    Color and Shape:Solid
    Molecular weight:511.62
  • Sodium Channel inhibitor 1

    CAS:
    Sodium Channel inhibitor1 is a novel and selective voltage-gated sodium channel for pain treatment.
    Formula:C24H19F4N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:473.42
  • VU625

    CAS:
    <p>VU625 (VU007625) is an AeKir1 inhibitor (IC50: 96.8nM) that acts as a mosquito killer and inhibits AeKir1-mediated currents.</p>
    Formula:C19H22N2O4S
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:374.45
  • Terodiline

    CAS:
    <p>Terodiline is an orally available selective muscarinic M1 receptor and calcium channel antagonist for the study of diseases caused by abnormal bladder function.</p>
    Formula:C20H27N
    Purity:98.20% - 99.59%
    Color and Shape:Solid
    Molecular weight:281.44
  • Asivatrep

    CAS:
    <p>Asivatrep (PAC14028) is a selective and potent antagonist of transient receptor potential vanilloid subtype 1 (TRPV1) for the study of atopic dermatitis.</p>
    Formula:C21H22F5N3O3S
    Purity:95.13%
    Color and Shape:Solid
    Molecular weight:491.48
  • AMG9678

    CAS:
    <p>AMG9678 is a selective, potent, orally active TRPM8 antagonist (IC50: 31.2 nM).</p>
    Formula:C20H18F6N2O
    Color and Shape:Solid
    Molecular weight:416.36
  • Topiramate lithium

    CAS:
    <p>Topiramate lithium: antiepileptic, GluR5 antagonist, enhances GABA, inhibits kainate/AMPA, Na+/Ca2+ channels; ↑ K+ conductance; ↓ carbonic anhydrase.</p>
    Formula:C12H20LiNO8S
    Color and Shape:Solid
    Molecular weight:345.29
  • MC-70

    CAS:
    <p>MC-70 is a potent P-glycoprotein (P-gp) inhibitor (EC50 = 0.69 μM).</p>
    Formula:C24H25NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:375.46
  • ORM-10962

    CAS:
    ORM-10962 is a potent, highly selective inhibitor of sodium-calcium exchanger (NCX) (for the reverse and forward mode inhibition with IC50 values of 67 and 55
    Formula:C27H29N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:459.54
  • Caldaret

    CAS:
    <p>Caldaret is an intracellular Ca2+ handling modulator that acts through reverse mode Na+/Ca2+ exchanger inhibition.</p>
    Formula:C11H16N2O3S
    Color and Shape:Solid
    Molecular weight:256.32
  • UBP 296

    CAS:
    <p>GluR5-subunit containing kainate receptor antagonist</p>
    Formula:C15H15N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:333.3
  • Y 23684

    CAS:
    <p>Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.</p>
    Formula:C18H13ClN2O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.83
  • Nav1.7-IN-3

    CAS:
    <p>Nav1.7-IN-3 is a selective and orally bioavailable inhibitor of voltage-gated sodium channel Nav1.7(IC50 of 8 nM).</p>
    Formula:C17H20ClFN4O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.95
  • CGP 46381

    CAS:
    <p>CGP 46381 is a GABAB receptor antagonist.</p>
    Formula:C10H22NO2P
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:219.26
  • YS-201

    CAS:
    <p>YS-201 is an antagonist of dihydropyridine-type calcium channel.</p>
    Formula:C24H31N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:457.52
  • IEM 1460

    CAS:
    <p>AMPA receptors blocker</p>
    Formula:C19H38Br2N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.33
  • (S)-ML753286

    CAS:
    (S)-ML753286 is a breast cancer resistance protein (BCRP) inhibitor (IC50: 0.6 μM on BCRP efflux transporter).
    Formula:C20H25N3O3
    Color and Shape:Solid
    Molecular weight:355.43
  • Indantadol HCl

    CAS:
    Indantadol HCl (CHF-3381) is a NMDA antagonist and nonselective MAO inhibitor.
    Formula:C11H15ClN2O
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:226.7
  • GABAA receptor agent 5

    CAS:
    <p>Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.</p>
    Formula:C21H25N3O2S
    Color and Shape:Solid
    Molecular weight:383.51
  • CP-409092 hydrochloride

    CAS:
    <p>CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.</p>
    Formula:C17H20ClN3O2
    Color and Shape:Solid
    Molecular weight:333.81
  • BGT1-IN-9

    CAS:
    <p>BGT1-IN-9 is an M1 muscarinic agonist.</p>
    Formula:C5H10ClN3O2
    Color and Shape:Solid
    Molecular weight:179.605
  • Atomoxetine

    CAS:
    <p>Atomoxetine (HSDB 7352) is a selective norepinephrine inhibitor that may cause an increase in blood pressure by increasing norepinephrine concentrations in</p>
    Formula:C17H21NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:255.35
  • Flordipine

    CAS:
    <p>Flordipine is used as a calcium channel blocker.</p>
    Formula:C26H33F3N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:510.55
  • Omeprazole magnesium

    CAS:
    <p>Omeprazole magnesium: oral PPI that reduces stomach acid, treats acid reflux and heartburn.</p>
    Formula:C34H36MgN6O6S2
    Color and Shape:Solid
    Molecular weight:713.12
  • Ro 04-5595 hydrochloride

    CAS:
    NR2B-containing NMDA receptors antagonist
    Formula:C19H23Cl2NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:368.3
  • TTA-Q6(isomer)

    CAS:
    TTA-Q6(isomer) is an isomer of TTA-Q6. TTA-Q6 is a selective antagonist of the T-type Ca2+ channel.
    Formula:C20H15ClF3N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:405.8
  • Apimostinel

    CAS:
    <p>Apimostinel (NRX-1074; AGN-241660) is a partial agonist of NMDA receptor.</p>
    Formula:C25H37N5O6
    Color and Shape:Solid
    Molecular weight:503.59
  • NMDA receptor antagonist 4

    CAS:
    <p>NMDA antagonist 4 (IIc) is an oral, voltage-dependent blocker with IC50 of 1.93 μM and may penetrate the BBB, useful in Alzheimer's research.</p>
    Formula:C15H18FN
    Color and Shape:Solid
    Molecular weight:231.31
  • Istaroxime

    CAS:
    <p>Istaroxime is an effective inhibitor of Na+, K+-ATPase (IC50: 0.11 μM).</p>
    Formula:C21H32N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:360.49
  • JNJ-56022486

    CAS:
    <p>JNJ-56022486 is a selective TARP γ‑8 AMPA receptor modulator.</p>
    Formula:C15H10ClN3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:283.71
  • KCa1.1 channel activator-2


    <p>KCa1.1 channel activator-2, a Quercetin hybrid, selectively stimulates vascular KCa1.1 channel, with strong myorelaxant effects.</p>
    Formula:C23H22O8S2
    Color and Shape:Solid
    Molecular weight:490.55
  • PPDA

    CAS:
    <p>Subtype-selective NMDA receptor antagonist</p>
    Formula:C21H18N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:378.38
  • (R)-3C4HPG

    CAS:
    <p>NMDA and AMPA/kainate receptor antagonist</p>
    Formula:C9H9NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:211.17
  • GoSlo-SR-5-69

    CAS:
    <p>BK channel activator (EC50 = 251 nM). Shifts the voltage required for half maximal negatively (DV1/2 = -104 mV).</p>
    Formula:C24H20N2NaO5S
    Color and Shape:Solid
    Molecular weight:471.48
  • Hyperforin dicyclohexylammonium salt

    CAS:
    Hyperforin dicyclohexylammonium is a TRPC6 activator and antidepressant that modulates Ca2+ levels.
    Formula:C47H75NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:718.10
  • TRPC6-IN-2

    CAS:
    <p>TRPC6-IN-2 is a TRPC protein inhibitor, specifically inhibiting TRPC6 protein.</p>
    Formula:C19H17Cl2FN6
    Color and Shape:Solid
    Molecular weight:419.28
  • Metapramine

    CAS:
    Metapramine, a tricyclic antidepressant, blocks norepinephrine reuptake and is a low-affinity NMDA antagonist.
    Formula:C16H18N2
    Purity:99.03% - 99.67%
    Color and Shape:Solid
    Molecular weight:238.33
  • SB-237376 HCl

    CAS:
    <p>SB-237376 HCl (SB-237376 hydrochloride) is a calcium and potassium channel antagonist used in the treatment of cardiac arrhythmias.</p>
    Formula:C20H26ClN3O5
    Purity:98.70%
    Color and Shape:Solid
    Molecular weight:423.89
  • GNE-5729

    CAS:
    <p>GNE-5729 is a positive allosteric modulator of NMDAR blood-brain barrier orally available, GluN2A, GluN2C and GluN2D, neurological and psychiatric disorders.</p>
    Formula:C17H10Cl2F3N5O
    Purity:99.40% - 99.85%
    Color and Shape:Solid
    Molecular weight:428.2
  • JNc-440

    CAS:
    <p>JNc-440, a strong anti-hypertensive, boosts TRPV4-KCa2.3 interaction and vasodilation, lowering blood pressure in mice.</p>
    Formula:C26H24N4O3
    Color and Shape:Solid
    Molecular weight:440.49
  • ML252

    CAS:
    <p>ML252 selectively inhibits KCNQ2 (IC50=69nM) and Cytochrome P450 isoforms CYP1A2, CYP2C9, CYP3A4, CYP2D6 with low nanomolar IC50s.</p>
    Formula:C20H24N2O
    Color and Shape:Solid
    Molecular weight:308.42
  • XPC-6444

    CAS:
    <p>XPC-6444 is a isoform-selective, and CNS-penetrant inhibitor of NaV1.6 with IC50 of41 nM for hNaV1.6,with anticonvulsant activity.</p>
    Formula:C22H25F3N4O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:498.58
  • (BrMT)2

    CAS:
    <p>(BrMT)2 is an activator of the Kv1.1 potassium ion channel.</p>
    Formula:C20H20Br2N4S2
    Color and Shape:Solid
    Molecular weight:540.34
  • RPR-260243

    CAS:
    <p>RPR-260243 is a novel activator of HERG and modifies HERG currents inhibited by dofetilide (IC50 = 58 nM).</p>
    Formula:C28H25F3N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:510.5
  • β-CCB

    CAS:
    <p>benzodiazepine receptor ligand</p>
    Formula:C16H16N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:268.31
  • UCL-1848 trifluoroacetate salt

    CAS:
    <p>UCL-1848 trifluoroacetate salt is a selective Ca2+-activated, SK potassium channel blocker.</p>
    Formula:C32H34F6N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:652.638
  • UBP714

    CAS:
    UBP714, derived from UBP608, boosts NMDAR in CA1 hippocampus, promising for schizophrenia and cognitive deficits treatment.
    Formula:C11H7BrO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:283.07
  • ZD-9379

    CAS:
    <p>ZD-9379 is a NMDA receptor antagonist.</p>
    Formula:C19H14ClN3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:383.79
  • Ro 8-4304 hydrochloride

    CAS:
    <p>Ro 8-4304 hydrochloride is a NMDA receptor antagonist.</p>
    Formula:C21H24ClFN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:406.88
  • YM 244769 hydrochloride

    CAS:
    <p>inhibitor of the reverse mode of Na+/Ca2+ exchange (NCX)</p>
    Formula:C26H23ClFN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:479.93