Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(98 products)
- Adiponectin receptor(5 products)
- CFTR(66 products)
- CGRP Receptor(55 products)
- Calcium Channel(574 products)
- Chloride channel(54 products)
- GABA Receptor(372 products)
- Monoamine Transporter(30 products)
- Monocarboxylate transporter(18 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(10 products)
- OAT(32 products)
- OCT(7 products)
- P-gp(55 products)
- Potassium Channel(304 products)
- Proton pump(42 products)
- SGLT(31 products)
- Sodium Channel(257 products)
- TRP/TRPV Channel(95 products)
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Found 2738 products of "Membrane Transporter/Ion Channel"
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Levamlodipine besylate Hemipentahydrate
CAS:Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.Formula:C20H25ClN2O5·C6H6O3SH2OColor and Shape:SolidMolecular weight:1224.18Isotachysterol 3
CAS:Isotachysterol 3 boosts calcium transport in gut and bone mobilization in kidneyless rats.Formula:C27H44OColor and Shape:SolidMolecular weight:384.64GaTx2
CAS:High-affinity ClC-2 blocker (KD ~50 pM), selective over other ClCs/CFTR/GABAC/CaCC/KV1.2; slows activation, no effect on open channels.Formula:C125H199N39O47S6Purity:98%Color and Shape:SolidMolecular weight:3192.54GDC-0334
CAS:GDC-0334 is a TRPA1 antagonist useful in treatment TRPA1-mediated diseases, such as pain or asthma.Formula:C24H19F8N5O3SColor and Shape:SolidMolecular weight:609.5FD 12-9
CAS:FD 12-9, Anti-glioblastoma activity. is a flavonoid dimer, acts as a dual inhibitor of P-gp and BCRP, with EC50s of 285 nM and 0.9 nM, respectively.Formula:C51H47N3O11Purity:98%Color and Shape:SolidMolecular weight:877.93UK-59811 hydrochloride
CAS:UK-59811 hydrochloride, Br-dihydropyridine derivative, blocks Ca V Ab channels in bacteria, IC50: 194 nM.Formula:C22H30BrClN2O5Color and Shape:SolidMolecular weight:517.85TRPV1 activator-1
CAS:TRPV1 Activator-1 (Compound 8), a capsaicin analog featuring a modified neck structure, specifically interacts with the T551 residue [1].Formula:C18H27NO2SColor and Shape:SolidMolecular weight:321.48ω-Conotoxin MVIIC TFA
ω-Conotoxin MVIIC TFA is a peptide and neurotoxin blocks P-type and q-type voltage-sensitive neuronal Ca ++ channels (VGCCs) radiolabel immunoprecipitation.Formula:C106H178N40O32S7·C2HF3O2Color and Shape:SolidMolecular weight:2863.27(±)8(9)-EpETE
CAS:(±)8(9)-EpETE ((±)8,9-EEQ) is an epoxide of arachidonic acid biosynthesized by CYP450 epoxygenase.1.2 In rat and rabbit liver microsomes.Formula:C20H30O3Color and Shape:SolidMolecular weight:318.45Prilocaine acetate
Prilocaine acetate, an amino amide compound, functions as a Na/K-ATPase inhibitor, exhibiting neurotoxic effects [1] [2].Formula:C15H24N2O3Color and Shape:SolidMolecular weight:280.36Cyclocreatine
CAS:Cyclocreatine, a creatine analogue and substrate for creatine kinase, inhibits creatine metabolism and prostate cancer cell proliferation.Formula:C5H9N3O2Purity:99.864%Color and Shape:SolidMolecular weight:143.14(R)-IDHP
CAS:(R)-IDHP, a salvia derivative, relaxes blood vessels by blocking calcium channels, aiding cardiovascular research.Formula:C12H16O5Color and Shape:SolidMolecular weight:240.25CALP3
CAS:Cell-permeable CaM agonist, binds EF-hand, activates phosphodiesterase without Ca2+, inhibits Ca2+ toxicity, IC50=33μM.Formula:C44H68N10O9Purity:98%Color and Shape:SolidMolecular weight:881.08Iberiotoxin
CAS:Selective blocker of the big conductance Ca2+-activated K+ channel.Formula:C179H274N50O55S7Purity:98%Color and Shape:SolidMolecular weight:4230Kurtoxin
Kurtoxin is a selective Cav3 (T-type) voltage-gated Ca2+ channel gating inhibitor, exhibiting a dissociation constant (Kd) of 15 nM for the Cav3.1 (α1G T-type)Formula:C324H478N94O90S8Purity:98%Color and Shape:SolidMolecular weight:7386.36Anticonvulsant agent 9
Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.Formula:C22H24N4O2Color and Shape:SolidMolecular weight:376.45P-gp/BCRP-IN-2
P-gp/BCRP-IN-2 (compound 15), an oxadiazole derivative, functions as a dual inhibitor targeting both the ABC transporter P-glycoprotein (IC50: 1.6 nM) and BCRPFormula:C32H35N3O6Color and Shape:SolidMolecular weight:557.64OD1
Activates rat Nav1.7, human Nav1.4, rat Nav1.6 (EC50: 7, 10, 47 nM); minimal on Nav1.2, 1.3, 1.5 (EC50 >3 μM); blocks fast inactivation; triggers pain.Formula:C308H466N90O95S8Purity:98%Color and Shape:SolidMolecular weight:7206.1Ethacrynic acid D5
CAS:Ethacrynic acid: a diuretic, anti-inflammatory, inhibits calcium channels, GSTs, NF-kB pathway, and modulates leukotriene; has deuterium-labeled form.Formula:C13H12Cl2O4Purity:98%Color and Shape:SolidMolecular weight:308.17Way 125971
CAS:Way 125971 is a bioactive chemcial.Formula:C22H28N4O5S2Color and Shape:SolidMolecular weight:492.61Apamin
CAS:Apamin: 18-amino acid bee venom peptide, blocks SK channels, anti-inflammatory, anti-fibrotic, strongly basic.Formula:C79H131N31O24S4Purity:98%Color and Shape:SolidMolecular weight:2027.34GpTx-1 TFA
GpTx-1 TFA is a polypeptide NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. It exhibits potent inhibitory activity on the NaV1.7 channel with an IC50 value of 10 nM, demonstrating excellent selectivity over NaV1.4 (IC50 = 0.301 μM) and NaV1.5 (IC50 = 4.20 μM) with >20-fold and >950-fold selectivity, respectively.Color and Shape:Odour SolidVerruculogen
CAS:Verruculogen, a toxin from Penicillium/Aspergillus, blocks Ca2+-K+ channels and halts mammalian M phase.Formula:C27H33N3O7Purity:98%Color and Shape:White PowderMolecular weight:511.57Neurotransmitter Receptor Compound Library
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；
Color and Shape:Odour SolidLeptomycin A
CAS:Leptomycin A from Streptomyces inhibits CRM1, reducing HIV-1 replication, less potent than Leptomycin B, blocks protein nuclear export.Formula:C32H46O6Purity:98%Color and Shape:SolidMolecular weight:526.7(Rac)-Tezacaftor
CAS:(Rac)-Tezacaftor, a racemate, corrects F508del CFTR for cystic fibrosis research.Formula:C26H27F3N2O6Color and Shape:SolidMolecular weight:520.5(1S,3R)-3-Aminocyclopentane carboxylic acid
CAS:(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.Formula:C6H11NO2Color and Shape:SolidMolecular weight:129.16SG-094
CAS:SG-094 inhibits TPC2, halts RIL175 cell growth, IC50: 3.7 μM for cancer research.
Formula:C30H29NO3Purity:97.06%Color and Shape:SoildMolecular weight:451.56Ion Channel Targeted Library
A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;
Color and Shape:Odour SolidZiconotide
CAS:Ziconotide: analgesic from cone snail for severe, chronic pain; synthetic ω-conotoxin.Formula:C102H172N36O32S7Purity:98%Color and Shape:White PowderMolecular weight:2639.13WAY-326766
CAS:WAY-326766 increases ion transport through mutant CFTR and can be used to alter the lifespan of eukaryotes.WAY-326766 can be used to treat cystic fibrosis (CF).Formula:C21H23N3O5Purity:99.87%Color and Shape:SolidMolecular weight:397.42Sulcardine 2HCl
CAS:Sulcardine 2HCl is a multi-ion channel blocker that blocks the properties of hERG and hNav1.5 channels and can be used to study atrial fibrillation.Formula:C24H35Cl2N3O4SPurity:99.33% - 99.76%Color and Shape:SoildMolecular weight:532.523Nitrazolam
CAS:Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.Formula:C17H13N5O2Color and Shape:SolidMolecular weight:319.32Azocarnil
Azocarnil is a GABAergic agonist-enhancer used in neurological system research.Color and Shape:Odour SolidJingzhaotoxin-XII TFA
Jingzhaotoxin-XII (JzTx-XII) TFA is a specific inhibitor of the Kv4.1 channel, exhibiting an IC50 of 0.363 μM. It interacts with the channel by altering gating behavior.Color and Shape:Odour SolidPptT-IN-4
PptT-IN-4 (Compound 3a) is a PptT inhibitor exhibiting an IC50 of 0.71 μM.Formula:C17H23N3Purity:98%Color and Shape:SolidMolecular weight:269.38PDZ1 Domain inhibitor peptide
CAS:Novel cyclic peptide that disrupts interaction between GluR6 and PSD-95Formula:C38H61N9O11Purity:98%Color and Shape:SolidMolecular weight:819.94APETx2
CAS:ASIC3 inhibitor; IC50: 63 nM (rat), 175 nM (human). Blocks NaV1.8, NaV1.2; analgesic for acid/inflammatory pain.Formula:C196H280N54O61S6Purity:98%Color and Shape:SolidMolecular weight:4561.06GX 201
CAS:GX 201 is a selective NaV1.7 inhibitor, IC50 of < 3.2 nM for hNaV1.7.Formula:C25H27ClF4N2O4SPurity:99.81%Color and Shape:SolidMolecular weight:563Anticonvulsant agent 8
Anticonvulsant agent 8 (compound D4) is a chemical used in treating epilepsy by inhibiting GABAA currents. In mouse models, its ED50 values are 2.23 mg/kg for the maximal electroshock (MES) test and 24.60 mg/kg for the pentylenetetrazol (PTZ) test.Formula:C15H11N5OColor and Shape:SolidMolecular weight:277.28CHET3
CAS:CHET3 is a highly selective allosteric activator for TASK-3-containing K2P channels. CHET3 has shown potent in vivo analgesic effects. Cost-effective and quality-assured.Formula:C21H21N5O3SPurity:98.28% - 99.92%Color and Shape:SoildMolecular weight:423.49Ruzinurad
CAS:Ruzinurad (WO2020088641, compound I) is a potent URAT1 inhibitor, exhibiting high selectivity.Formula:C14H12BrNO2SColor and Shape:SolidMolecular weight:338.22Roquefortine C
CAS:Roquefortine C is a fungal cyclopeptide isolated from Penicillium roquefortii, activates P-gp and also inhibits P450-3A and other haemoproteinsFormula:C22H23N5O2Purity:98%Color and Shape:SolidMolecular weight:389.45P-gp inhibitor 15
P-gp Inhibitor 15 (compound 7a), a nonsubstrate inhibitor of P-glycoprotein (Pgp), inhibits Pgp-ATPase activity and interferes with Pgp-mediated Rhodamine123Formula:C35H60N2O4Color and Shape:SolidMolecular weight:572.86Fumitremorgin C
CAS:Fumitremorgin C (12α-Fumitremorgin C) is a mycotoxin and inhibits ABCG2/BRCP.Formula:C22H25N3O3Purity:98%Color and Shape:SolidMolecular weight:379.45Agitoxin-2
CAS:Potent Shaker K+ channel blocker (Ki = 0.64 nM). Also inhibits Kv1.3, Kv1.6 and Kv1.1 K+ channels (Ki values are 4, 37 and 44 pM respectively).Formula:C169H278N54O48S8Purity:98%Color and Shape:SolidMolecular weight:4090.87AQP4 (205-215)
CAS:AQP4 (205-215) is a fragment of the water channel protein Aquaporin-4 (AQP4). This protein is an autoimmune antigen in optic neuromyelitis and, upon binding with CD40, is upregulated and presented in B cells. AQP4 is associated with neuromyelitis optica (NMO), an autoimmune inflammatory disease of the central nervous system (CNS).Formula:C48H75N13O17SColor and Shape:SolidMolecular weight:1138.25(±)5(6)-DiHETE
CAS:Eicosapentaenoic acid is an ω-3 polyunsaturated fatty acid that is abundant in marine organisms and fish oils.Formula:C20H32O4Color and Shape:SolidMolecular weight:336.472JYL-79
CAS:JYL-79 is an agonist of the vanilloid receptor.Formula:C26H36N2O4SColor and Shape:SolidMolecular weight:472.64TRPV4 antagonist 4
CAS:Potent TRPV4 blocker with 22.65 nM IC50; inhibits current and aids acute lung injury.
Formula:C28H32Cl2N6OColor and Shape:SolidMolecular weight:539.50RuBi-GABA
CAS:Ruthenium-bipyridine-triphenylphosphine caged GABAFormula:C42H39F6N5O2P2RuPurity:98%Color and Shape:SolidMolecular weight:922.812,14-Dichlorodehydroabietic acid
CAS:12,14-Dichlorodehydroabietic acid activates BK channels, blocks GABA A receptors, and increases calcium and neurotransmitter release.Formula:C20H26Cl2O2Color and Shape:SolidMolecular weight:369.33ADWX 1
Potent KV1.3 blocker, IC50: 0.0019 nM; less effective on KV1.1. Curbs CD4+ T cell activation; eases rat multiple sclerosis model.Formula:C169H281N57O46S7Purity:98%Color and Shape:SolidMolecular weight:4071.86ProTx II
CAS:Selective NaV1.7 inhibitor, alters activation, reduces current, 100x more selective for 1.7 over other Na+ channels.
Formula:C168H250N46O41S8Purity:98%Color and Shape:SolidMolecular weight:3826.59MRS4596
MRS4596: selective P2X4 blocker, IC50 1.38 μM, neuroprotective in stroke research.Formula:C21H14N5NaO3SColor and Shape:SolidMolecular weight:439.42AHN-683
CAS:AHN-683 is a fluorescent ligand. It was used for peripheral-type benzodiazepine receptors.Formula:C42H32FN3O7Purity:98%Color and Shape:SolidMolecular weight:709.7224-Hydroxycholesterol
CAS:24-Hydroxycholesterol (Cholest-5-ene-3beta,24-diol) is an activator of the LXR and can be used to study cardiogenesis and pancreatic cancer.Formula:C27H46O2Purity:99.8%Color and Shape:SolidMolecular weight:402.65Digoxigenin Monodigitoxoside
CAS:Digoxigenin monodigitoxoside is a cardiac glycoside metabolite of digoxin and a Na+/K+ ATPase inhibitor.Formula:C29H44O8Color and Shape:SolidMolecular weight:520.663NF864
CAS:NF864, a suramin analog, is a P2X1 receptor inhibitor.Formula:C57H28N6Na12O41S12Purity:98%Color and Shape:SolidMolecular weight:2113.5Sinapine hydroxide
CAS:Sinapine hydroxide from crucifer seeds has anti-inflammatory, anti-oxidant, anti-tumor properties, and inhibits AChE, aiding neurodegenerative research.Formula:C16H25NO6Color and Shape:SolidMolecular weight:327.377Guangxitoxin 1E
CAS:Guangxitoxin 1E acts as a gating modifier since it shifts the voltage-dependence of Kv2.1 K+ currents towards depolarized potentials.Formula:C178H248N44O45S7Purity:98%Color and Shape:SolidMolecular weight:3948.61Brevetoxin B
CAS:Brevetoxin B, a polyketide neurotoxin from Karenia, affects sodium channels causing neurotoxic shellfish poisoning. IC50=15nM.Formula:C50H70O14Color and Shape:SolidMolecular weight:895.096AChE/Aβ-IN-2
AChE/Aβ-IN-2 (compound 33) is a powerful, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 135 nM.Formula:C20H25ClN4Color and Shape:SolidMolecular weight:356.89S-Sulfo-L-cysteine sodium salt
CAS:S-Sulfo-L-cysteine sodium salt shows a weak affinity for mGluR1α and mGluR5a at high concentrations and has potential antioxidant activity.Formula:C3H6NNaO5S2Purity:99.59%Color and Shape:SolidMolecular weight:223.2S-Bioallethrin
CAS:S-Bioallethrin is a pure S-form of Bioallethrin.Formula:C19H26O3Purity:98%Molecular weight:302.41epi-Aszonalenin A
CAS:epi-Aszonalenin A: a psychoactive benzodiazepine from Aspergillus novofumigatus.Formula:C25H25N3O3Color and Shape:SolidMolecular weight:415.488-Bromo-ATP
CAS:8-Bromo-ATP (8-Bromoadenosine 5'-triphosphate) is a purinergic P2X receptor agonist and an ATP analogue.Formula:C10H15BrN5O13P3Color and Shape:SolidMolecular weight:586.077Brevetoxin-3
CAS:Brevetoxin-3 activates Na+ channels, binding strongly to site 5, preventing their inactivation.Formula:C50H72O14Purity:98%Color and Shape:SolidMolecular weight:897.112TNP-ATP triethylammonium salt
CAS:P2X receptor antagonistFormula:C40H77N12O19P3Purity:98%Color and Shape:SolidMolecular weight:1123.042LY393615
LY393615 (NCC1048) is a novel blocker of both neuronal Ca²⁺ (calcium) and Na⁺ (sodium) channels, exhibiting half-maximal inhibitory concentrations (IC₅₀) of 1.9Purity:98%Color and Shape:Odour SolidNSC156529
CAS:NSC156529 suppresses AKT1, reduces cancer cell growth in vitro, and inhibits prostate tumors in vivo.Formula:C28H21ClS2Purity:98%Color and Shape:SolidMolecular weight:457.05Calcium Ionophore I
CAS:Calcium Ionophore I has a wide range of applications in life science related research.Formula:C38H72N2O8Color and Shape:SolidMolecular weight:685.0L-Palmitoylcarnitine TFA
L-Palmitoylcarnitine TFA: long-chain fat metabolite that disrupts membranes in ischaemia & inhibits KATP channels via Kir6.2 interaction.
Formula:C25H46F3NO6Color and Shape:SolidMolecular weight:513.63Idactamab
CAS:Idactamab (INT-001) is a monoclonal antibody to the human amino acid transport protein ASCT2.Purity:> 95%Color and Shape:LiquidMolecular weight:146.2 kDaConcanamycin B
CAS:Concanamycin B, a macrolide, inhibits V-ATPases (IC50 = 5 nM), blocks vacuole acidification, affects bone resorption, CD8 T cells, and MHC II in B cells.Formula:C45H73NO14Color and Shape:SolidMolecular weight:852.072ML353
ML353 activates TREK-1/2, binds mGlu5 SAM (Ki=18.2 nM), surpasses 5mpep, may address SAM activity/blocking.Formula:C19H15FN2OPurity:99.98% - 99.98%Color and Shape:SoildMolecular weight:306.33Ref: TM-T67917
5mg50.00€1mL*10mM (DMSO)50.00€10mg74.00€25mg114.00€50mg156.00€100mg219.00€200mg298.00€17(R)-Resolvin D1
CAS:Resolvins are anti-inflammatory lipids from EPA and DHA. Resolvin D1, made from DHA, and its aspirin-triggered epimer 17(R)-RvD1, inhibit acute inflammation.Formula:C22H32O5Color and Shape:SolidMolecular weight:376.493Charybdotoxin
CAS:Specific inhibitor of the big conductance Ca2+-activated K+ channel.Formula:C176H277N57O55S7Purity:98%Color and Shape:SolidMolecular weight:4295.95Nav1.7-IN-8
CAS:Nav1.7-IN-8 selectively inhibits NaV1.7 over hNaV1.1/1.5, affects CYP2C9/3A4 (IC50: 0.17/0.077 μM), and provides rodent pain relief.Formula:C21H12ClF2N5O4S2Color and Shape:SolidMolecular weight:535.93JTS-653
CAS:JTS-653 is a potent TRPV1 antagonist, effective in reducing chronic pain unresponsive to NSAIDs.Formula:C23H21F3N4O4Color and Shape:SolidMolecular weight:474.443-Aminopropylphosphonic Acid
CAS:3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand binding
Formula:C3H10NO3PPurity:99.84%Color and Shape:Light Yellow LiquidMolecular weight:139.09Fipronil sulfone
CAS:Fipronil sulfone is an insecticide fipronil. Its metabolite fipronil sulphone is an inhibitor of rat ɑ1β2γ2L GABA(A) receptor.Formula:C12H4Cl2F6N4O2SPurity:98%Color and Shape:SolidMolecular weight:453.14Bendroflumethiazide
CAS:Bendroflumethiazide (Naturetin) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE. It has been used in the treatment of familial hyperkalemia, hypertension, edema, and urinary tract disorders. (From Martindale, The Extra Pharmacopoeia, 30th ed, p810)Formula:C15H14F3N3O4S2Purity:98% - >99.99%Color and Shape:Crystals From Dioxane SolidMolecular weight:421.41ABCB1-IN-1
ABCB1-IN-1 (compound 3) is a potent inhibitor of ABCB1 that promotes cell apoptosis.Formula:C36H33F3FeN2O4PSColor and Shape:SolidMolecular weight:733.54Chrodrimanin B
CAS:Chrodrimanin B is a useful organic compound for research related to life sciences. The catalog number is T126052 and the CAS number is 132196-54-4.Formula:C27H32O8Color and Shape:SolidMolecular weight:484.545Margatoxin
CAS:KV1.3 channel blocker, IC50 36 pM, no effect on calcium-activated channels, hinders VEGF-induced Ca++ influx & NO in endothelial cells.Formula:C178H286N52O50S7Purity:98%Color and Shape:SolidMolecular weight:4178.96(S)-PF-03716556
CAS:(S)-PF-03716556 can be used as an acid pump inhibitor for the treatment of disease conditions mediated by acid pump inhibitory activity.Formula:C22H26N4O3Purity:99.75% - 99.91%Color and Shape:SoildMolecular weight:394.47ω-Agatoxin IVA
CAS:Selective blocker of P-type calcium channels (IC50 < 1 - 3 nM). Also inhibits N-type channels at micromolar concentrations.Formula:C217H360N68O60S10Purity:98%Color and Shape:SolidMolecular weight:5202.25ProTx-I
CAS:Selective blocker for CaV3.1 (IC50 = 0.2 μM), CaV3.2 (31.8 μM), also inhibits NaV1.8 and blocks KV2.1 channels.Formula:C171H245N53O47S6Purity:98%Color and Shape:SolidMolecular weight:3987.51Lifastuzumab
CAS:Sulfamethoxazole-NO (SMX-NO) is a SMX-NO derivative and is the primary immunogen for sulfonamide hypersensitivity reactions.Purity:97% (SDS-PAGE); 99.5% (SEC-HPLC) - 97% (SDS-PAGE); 99.5% (SEC-HPLC)Color and Shape:LiquidMolecular weight:145.5 kDa(±)16-HETE
CAS:Electrolyte and fluid transport in the kidney are regulated in part by arachidonic acid and its metabolites.Formula:C20H32O3Color and Shape:SolidMolecular weight:320.473Transdermal Peptide Disulfide
CAS:TD 1 peptide, an 11-amino acid, binds ATP1B1's C-terminus, enhancing transdermal drug delivery.Formula:C40H64N14O16S2Purity:98%Color and Shape:SolidMolecular weight:1061.15GluN2B-NMDAR antagonist-1
Orally active GluN2B-NMDAR antagonist with neuroprotective properties for ischemic injury research.Formula:C26H23BrN2O2Color and Shape:SolidMolecular weight:475.38PNU-140975
CAS:PNU-140975 is a bio-active chemical.Formula:C3H9N5O2Color and Shape:SolidMolecular weight:147.138Tacrine hydrochloride
CAS:Tacrine: a cholinergic agonist, anticholinesterase; inhibits AChE/BChE with IC50s of 31/25.6 nM.Formula:C13H15ClN2Purity:98%Color and Shape:SolidMolecular weight:234.73Conantokin-T
CAS:Non-competitive NMDA receptor antagonistFormula:C110H175N31O45SPurity:98%Color and Shape:SolidMolecular weight:2683.81P2X4 antagonist-4
P2X4 antagonist-4 (compound 64) is a potent P2X4R antagonist with an IC50 value of 8 µM. It can inhibit ATP-induced activation of the NLRP3 inflammasome and the subsequent release of IL-1β.Formula:C27H22FN3O4SColor and Shape:SolidMolecular weight:503.545Dalazatide HCl
Dalazatide HCl is a peptide and specific Kv1.3 inhibitor that suppresses the activation and proliferation of memory effector T cells,Color and Shape:SolidMolecular weight:4317.53 (Free base)H-Lys-Tyr-OH TFA
Lysyltyrosine TFA is a dipeptide that may enhance brain function by boosting noradrenaline and tyrosine release.Formula:C17H24F3N3O6Color and Shape:SolidMolecular weight:423.38Nipecotic acid
CAS:Compound PDK0243, with CAS No. 498-95-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0243 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formula:C6H11NO2Color and Shape:Off-White To Pale Yellow-Beige PowderMolecular weight:129.16
