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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2293 products of "Membrane Transporter/Ion Channel"

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  • TRPV4 antagonist 3

    CAS:
    <p>TRPV4 antagonist 3 is a TRPV4 antagonist (p IC 50 = 8.4).</p>
    Formula:C20H18F4N4O3S
    Color and Shape:Solid
    Molecular weight:470.44
  • 17(R)-Resolvin D1

    CAS:
    <p>Resolvins are anti-inflammatory lipids from EPA and DHA. Resolvin D1, made from DHA, and its aspirin-triggered epimer 17(R)-RvD1, inhibit acute inflammation.</p>
    Formula:C22H32O5
    Color and Shape:Solid
    Molecular weight:376.493
  • Charybdotoxin

    CAS:
    <p>Specific inhibitor of the big conductance Ca2+-activated K+ channel.</p>
    Formula:C176H277N57O55S7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4295.95
  • Calcium Ionophore I

    CAS:
    <p>Calcium Ionophore I has a wide range of applications in life science related research.</p>
    Formula:C38H72N2O8
    Color and Shape:Solid
    Molecular weight:685.0
  • JTS-653

    CAS:
    <p>JTS-653 is a potent TRPV1 antagonist, effective in reducing chronic pain unresponsive to NSAIDs.</p>
    Formula:C23H21F3N4O4
    Color and Shape:Solid
    Molecular weight:474.44
  • 8-Azido-ATP

    CAS:
    <p>8-Azido-ATP is a nucleotide analog that demonstrates photo-reactivity properties.</p>
    Formula:C10H15N8O13P3
    Color and Shape:Solid
    Molecular weight:548.19
  • Fipronil sulfone

    CAS:
    Fipronil sulfone is an insecticide fipronil. Its metabolite fipronil sulphone is an inhibitor of rat ɑ1β2γ2L GABA(A) receptor.
    Formula:C12H4Cl2F6N4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:453.14
  • Bendroflumethiazide

    CAS:
    <p>Bendroflumethiazide (Naturetin) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE. It has been used in the treatment of familial hyperkalemia, hypertension, edema, and urinary tract disorders. (From Martindale, The Extra Pharmacopoeia, 30th ed, p810)</p>
    Formula:C15H14F3N3O4S2
    Purity:98% - >99.99%
    Color and Shape:Crystals From Dioxane Solid
    Molecular weight:421.41
  • 3-Aminopropylphosphonic Acid

    CAS:
    <p>3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand binding</p>
    Formula:C3H10NO3P
    Purity:99.84%
    Color and Shape:Light Yellow Liquid
    Molecular weight:139.09
  • P2X4 antagonist-3


    <p>P2X4 antagonist-3 (Compound 14c) is a P2X4 inhibitor with an IC50 value of 1.2 μM. It holds potential for research into neuroinflammation, chronic pain, and cancer progression.</p>
    Formula:C19H20FN3O4
    Color and Shape:Solid
    Molecular weight:373.38
  • Chrodrimanin B

    CAS:
    <p>Chrodrimanin B is a useful organic compound for research related to life sciences. The catalog number is T126052 and the CAS number is 132196-54-4.</p>
    Formula:C27H32O8
    Color and Shape:Solid
    Molecular weight:484.545
  • Crocetin meglumine


    <p>Crocetin (Transcrocetin) meglumine, sourced from Crocus sativus L. (saffron), functions as a high-affinity antagonist of the NMDA receptor.</p>
    Formula:C34H58N2O14
    Color and Shape:Solid
    Molecular weight:718.83
  • Idactamab

    CAS:
    <p>Idactamab (INT-001) is a monoclonal antibody to the human amino acid transport protein ASCT2.</p>
    Purity:> 95%
    Color and Shape:Liquid
    Molecular weight:146.2 kDa
  • Concanamycin B

    CAS:
    Concanamycin B, a macrolide, inhibits V-ATPases (IC50 = 5 nM), blocks vacuole acidification, affects bone resorption, CD8 T cells, and MHC II in B cells.
    Formula:C45H73NO14
    Color and Shape:Solid
    Molecular weight:852.072
  • rac-trans-4-hydroxy Glyburide

    CAS:
    <p>rac-trans-4-hydroxy Glyburide, a metabolite of glyburide, inhibits binding at SUR1/Kir6.2 sites with IC50 values of 0.95 and 100 nM.</p>
    Formula:C23H28ClN3O6S
    Color and Shape:Solid
    Molecular weight:510.0
  • ATP Synthesis-IN-1


    <p>ATP Synthesis-IN-1 (Compound 4), a quinoline derivative, potently inhibits PA ATP synthesis with an IC50 of 11.1μg/mL and exhibits antibacterial properties.</p>
    Color and Shape:Odour Solid
  • NF279

    CAS:
    <p>P2X1 antagonist</p>
    Formula:C49H36N6Na6O23S6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1407.17
  • TNP-ATP triethylammonium salt

    CAS:
    <p>P2X receptor antagonist</p>
    Formula:C40H77N12O19P3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1123.042
  • AChE/Aβ-IN-2


    <p>AChE/Aβ-IN-2 (compound 33) is a powerful, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 135 nM.</p>
    Formula:C20H25ClN4
    Color and Shape:Solid
    Molecular weight:356.89
  • Margatoxin

    CAS:
    <p>KV1.3 channel blocker, IC50 36 pM, no effect on calcium-activated channels, hinders VEGF-induced Ca++ influx &amp; NO in endothelial cells.</p>
    Formula:C178H286N52O50S7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4178.96
  • Cevadine


    <p>Cevadine is a natural product that can be used as a reference standard.</p>
    Formula:C32H49NO9
    Color and Shape:Solid
    Molecular weight:591.742
  • Brevetoxin B

    CAS:
    <p>Brevetoxin B, a polyketide neurotoxin from Karenia, affects sodium channels causing neurotoxic shellfish poisoning. IC50=15nM.</p>
    Formula:C50H70O14
    Color and Shape:Solid
    Molecular weight:895.096
  • GYKI-47261 dihydrochloride

    CAS:
    <p>GYKI-47261 dihydrochloride is an AMPA receptor antagonist and CYP2E1 inducer, demonstrating broad-spectrum anticonvulsant and neuroprotective activities.</p>
    Formula:C18H17Cl3N4
    Purity:98.32% - 99.14%
    Color and Shape:Solid
    Molecular weight:395.71
  • (2R,3S,11bS)-Dihydrotetrabenazine

    CAS:
    <p>(2R,3S,11bS)-Tetrabenazine impurity, VMAT inhibitor for movement disorders.</p>
    Formula:C19H29NO3
    Purity:99.29%
    Color and Shape:Solid
    Molecular weight:319.44
  • PDDHV

    CAS:
    <p>PDDHV: a capsaicin-like vanilloid selective for rat TRPV1; induces Ca2+ uptake in neurons, EC50 of 70 nM.</p>
    Formula:C49H72O11
    Color and Shape:Solid
    Molecular weight:837.09
  • Vanzacaftor

    CAS:
    <p>Vanzacaftor is a CFTR modulator improving protein processing and surface trafficking, restoring chloride transport and aiding cystic fibrosis therapy research.</p>
    Formula:C32H39N7O4S
    Purity:99.14%
    Color and Shape:Solid
    Molecular weight:617.76
  • Flufiprole

    CAS:
    <p>Flufiprole is used as a phenylpyrazole pesticide. It has enantioselective metabolism in human and rat liver microsomes.</p>
    Formula:C16H10Cl2F6N4OS
    Color and Shape:Solid
    Molecular weight:491.24
  • CHET3

    CAS:
    <p>CHET3 is a highly selective allosteric activator for TASK-3-containing K2P channels. CHET3 has shown potent in vivo analgesic effects. Cost-effective and quality-assured.</p>
    Formula:C21H21N5O3S
    Purity:99.64% - >99.99%
    Color and Shape:Soild
    Molecular weight:423.49
  • AHN-683

    CAS:
    AHN-683 is a fluorescent ligand. It was used for peripheral-type benzodiazepine receptors.
    Formula:C42H32FN3O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:709.72
  • RuBi-GABA

    CAS:
    <p>Ruthenium-bipyridine-triphenylphosphine caged GABA</p>
    Formula:C42H39F6N5O2P2Ru
    Purity:98%
    Color and Shape:Solid
    Molecular weight:922.8
  • WAY-326766

    CAS:
    WAY-326766 increases ion transport through mutant CFTR and can be used to alter the lifespan of eukaryotes.WAY-326766 can be used to treat cystic fibrosis (CF).
    Formula:C21H23N3O5
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:397.42
  • Dalazatide HCl


    <p>Dalazatide HCl is a peptide and specific Kv1.3 inhibitor that suppresses the activation and proliferation of memory effector T cells,</p>
    Color and Shape:Solid
    Molecular weight:4317.53 (Free base)
  • Neurotransmitter Receptor Compound Library


    <p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>
    Color and Shape:Odour Solid
  • GpTx-1 TFA


    <p>GpTx-1 TFA is a polypeptide NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. It exhibits potent inhibitory activity on the NaV1.7 channel with an IC50 value of 10 nM, demonstrating excellent selectivity over NaV1.4 (IC50 = 0.301 μM) and NaV1.5 (IC50 = 4.20 μM) with &gt;20-fold and &gt;950-fold selectivity, respectively.</p>
    Color and Shape:Odour Solid
  • (Rac)-Tezacaftor

    CAS:
    <p>(Rac)-Tezacaftor, a racemate, corrects F508del CFTR for cystic fibrosis research.</p>
    Formula:C26H27F3N2O6
    Color and Shape:Solid
    Molecular weight:520.5
  • CALP3

    CAS:
    <p>Cell-permeable CaM agonist, binds EF-hand, activates phosphodiesterase without Ca2+, inhibits Ca2+ toxicity, IC50=33μM.</p>
    Formula:C44H68N10O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:881.08
  • Kurtoxin


    <p>Kurtoxin is a selective Cav3 (T-type) voltage-gated Ca2+ channel gating inhibitor, exhibiting a dissociation constant (Kd) of 15 nM for the Cav3.1 (α1G T-type)</p>
    Formula:C324H478N94O90S8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:7386.36
  • SG-094

    CAS:
    <p>SG-094 inhibits TPC2, halts RIL175 cell growth, IC50: 3.7 μM for cancer research.</p>
    Formula:C30H29NO3
    Purity:97.06%
    Color and Shape:Soild
    Molecular weight:451.56
  • Phe-Met-Arg-Phe amide trifluoroacetate

    CAS:
    Phe-met-arg-phe amide trifluoroacetate is an activator of K+ current with an ED50 of 23nm on the fundus nerve.
    Formula:C33H44F6N8O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:826.81
  • ω-Agatoxin IVA

    CAS:
    Selective blocker of P-type calcium channels (IC50 < 1 - 3 nM). Also inhibits N-type channels at micromolar concentrations.
    Formula:C217H360N68O60S10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:5202.25
  • (1S,3R)-3-Aminocyclopentane carboxylic acid

    CAS:
    <p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>
    Formula:C6H11NO2
    Color and Shape:Solid
    Molecular weight:129.16
  • 17R(18S)-EpETE

    CAS:
    <p>17R(18S)-EpETE: Oxylipin, eicosapentaenoic acid metabolite, activates BKCa channels, has negative chronotropic effects.</p>
    Formula:C20H30O3
    Color and Shape:Solid
    Molecular weight:318.457
  • P2X4 antagonist-4


    <p>P2X4 antagonist-4 (compound 64) is a potent P2X4R antagonist with an IC50 value of 8 µM. It can inhibit ATP-induced activation of the NLRP3 inflammasome and the subsequent release of IL-1β.</p>
    Formula:C27H22FN3O4S
    Color and Shape:Solid
    Molecular weight:503.545
  • (±)8(9)-EpETE

    CAS:
    <p>(±)8(9)-EpETE ((±)8,9-EEQ) is an epoxide of arachidonic acid biosynthesized by CYP450 epoxygenase.1.2 In rat and rabbit liver microsomes.</p>
    Formula:C20H30O3
    Color and Shape:Solid
    Molecular weight:318.45
  • Tacrine hydrochloride

    CAS:
    <p>Tacrine: a cholinergic agonist, anticholinesterase; inhibits AChE/BChE with IC50s of 31/25.6 nM.</p>
    Formula:C13H15ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:234.73
  • Jingzhaotoxin-XII TFA


    <p>Jingzhaotoxin-XII (JzTx-XII) TFA is a specific inhibitor of the Kv4.1 channel, exhibiting an IC50 of 0.363 μM. It interacts with the channel by altering gating behavior.</p>
    Color and Shape:Odour Solid
  • LRRK2-IN-15


    <p>LRRK2-IN-15 is an inhibitor of LRRK2. It exhibits an IC50 value of 5 nM in PBMC cells and 1.5 μM for BCRP. This compound is utilized in the research of Parkinson's disease.</p>
    Color and Shape:Odour Solid
  • Nitrazolam

    CAS:
    <p>Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.</p>
    Formula:C17H13N5O2
    Color and Shape:Solid
    Molecular weight:319.32
  • Sinapine hydroxide

    CAS:
    <p>Sinapine hydroxide from crucifer seeds has anti-inflammatory, anti-oxidant, anti-tumor properties, and inhibits AChE, aiding neurodegenerative research.</p>
    Formula:C16H25NO6
    Color and Shape:Solid
    Molecular weight:327.377
  • Tertiapin LQ


    <p>Kir1.1 channel blocker, 250x selective; Kd: Kir1.1 (1.1 nM), Kir3.1/3.2 (274 nM), Kir3.1/3.4 (361 nM). Tertiapin-Q derivative.</p>
    Formula:C106H179N33O24S4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2428.03
  • Leptomycin A

    CAS:
    <p>Leptomycin A from Streptomyces inhibits CRM1, reducing HIV-1 replication, less potent than Leptomycin B, blocks protein nuclear export.</p>
    Formula:C32H46O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:526.7
  • A-317567

    CAS:
    A-317567 is a potent acid-sensing ion channel 3 (ASIC-3) inhibitor with an IC50 of 1.025 μM, and it has antidepressant and antinociception effects[1][2].
    Formula:C27H31N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:397.56
  • Oleoyl-D-lysine

    CAS:
    <p>Oleoyl-D-lysine: lipid-based GlyT2 inhibitor, eases neuropathic pain in mice, safe, non-sedative, no respiratory depression.</p>
    Formula:C24H46N2O3
    Color and Shape:Solid
    Molecular weight:410.63
  • ω-Conotoxin GVIA

    CAS:
    <p>Peptide neurotoxin; selectively and reversibly blocks N-type calcium channels (IC50 = 0.15 nM). Reduces (RS)-3,5-DHPG -induced long term depression in vivo.</p>
    Formula:C120H182N38O43S6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3037
  • BKCa activator-1


    <p>BKCa activator-1 (Compound 51b) is an orally active activator of BKCa calcium-activated potassium channels with an EC50 of 2.82 μM. It promotes K+ efflux, leading to cell membrane hyperpolarization and inhibition of smooth muscle contraction. In a spontaneous hypertensive rat (SHR) model, it alleviates urinary incontinence and exhibits antitussive effects in a guinea pig cough model.</p>
    Formula:C22H23F7N2O3
    Color and Shape:Solid
    Molecular weight:496.418
  • Nipecotic acid

    CAS:
    <p>Compound PDK0243, with CAS No. 498-95-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0243 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>
    Formula:C6H11NO2
    Color and Shape:Off-White To Pale Yellow-Beige Powder
    Molecular weight:129.16
  • ABCB1-IN-1


    <p>ABCB1-IN-1 (compound 3) is a potent inhibitor of ABCB1 that promotes cell apoptosis.</p>
    Formula:C36H33F3FeN2O4PS
    Color and Shape:Solid
    Molecular weight:733.54
  • Tiludronate disodium hemihydrate

    CAS:
    <p>Tiludronate: an oral bisphosphonate for bone disorder research; inhibits osteoclasts and reduces inflammation.</p>
    Formula:C14H16Cl2Na4O13P4S2
    Color and Shape:Solid
    Molecular weight:743.16
  • GSK2332255B

    CAS:
    <p>GSK2332255B: potent TRPC3/6 antagonist; IC50 5 nM (TRPC3), 4 nM (TRPC6); over 100-fold selectivity vs other Ca2+ channels.</p>
    Formula:C18H19ClFN3O3S
    Color and Shape:Solid
    Molecular weight:411.88
  • N-Oleoyl Glutamine

    CAS:
    <p>N-Oleoyl Glutamine (Oleoyl-L-glutamine) antagonizes TRPV1 of the transient receptor potential (TRP) calcium channel.</p>
    Formula:C23H42N2O4
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:410.59
  • LTGO-33

    CAS:
    <p>LTGO-33 is a voltage-gated sodium channel NaV1.8 inhibitor that inhibits NaV1.8, NaV1.1-NaV1.7, and NaV1.9.</p>
    Formula:C21H17F4N3O3S
    Purity:97.6%
    Color and Shape:Soild
    Molecular weight:467.44
  • 5-Hydroxy-2′,3,4′,7-tetramethoxyflavone

    CAS:
    5-Hydroxy-2′,3,4′,7-tetramethoxyflavone shows weak ABCG2 inhibitory potency with IC50s of 3.27 and 3.89 µM in the Hoechst 33342 and pheophorbide A assays.
    Formula:C19H18O7
    Purity:98%
    Color and Shape:Soild
    Molecular weight:358.34
  • S-Sulfo-L-cysteine sodium salt

    CAS:
    <p>S-Sulfo-L-cysteine sodium salt shows a weak affinity for mGluR1α and mGluR5a at high concentrations and has potential antioxidant activity.</p>
    Formula:C3H6NNaO5S2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:223.2
  • NF864

    CAS:
    NF864, a suramin analog, is a P2X1 receptor inhibitor.
    Formula:C57H28N6Na12O41S12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2113.5
  • 18β-Glycyrrhetyl-3-O-sulfate

    CAS:
    <p>18β-Glycyrrhetyl-3-O-sulfate (Glycyrrhetic acid 3-O-(hydrogen sulfate)), a major metabolite of Glycyrrhetinic acid (GA), serves as a potent inhibitor of type 2</p>
    Formula:C30H46O7S
    Color and Shape:Solid
    Molecular weight:550.75
  • Phrixotoxin 3

    CAS:
    <p>Potent NaV blocker: IC50 - 0.6 nM (NaV1.2), 42 nM (NaV1.3), 72 nM (NaV1.5); voltage-dependent inhibition.</p>
    Formula:C176H269N51O48S6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4059.74
  • TRPA1-IN-1

    CAS:
    <p>TRPA1-IN-1 is a potent, selective antagonist of the TRPA1 channel, demonstrating significant oral bioavailability as a small molecule.</p>
    Formula:C19H17ClN6O3
    Color and Shape:Solid
    Molecular weight:412.83
  • 17α-Hydroxywithanolide D


    <p>17alpha-Hydroxywithanolide D is an allosteric modulator of the NMDA receptor, with an IC50 of 44.24 nM. This compound exhibits neuroprotective properties and can be utilized in Alzheimer's disease research.</p>
    Formula:C28H46O7
    Color and Shape:Solid
    Molecular weight:494.661
  • Apamin acetate


    <p>Apamin acetate: Selective Ca2+-activated K+ channel blocker, 18-amino acid bee venom peptide, promotes synapse repair, anti-inflammatory.</p>
    Purity:96.97%
    Color and Shape:Solid
  • Conantokin G TFA


    <p>Conantokin G TFA, a 17-aa peptide, blocks NMDA receptors with 480 nM IC50 and is neuroprotective.</p>
    Formula:C90H139F3N26O46
    Color and Shape:Solid
    Molecular weight:2378.21
  • GS-9191 PM


    <p>GS-9191 PM: novel antitumorviral bis-amide prodrug, inhibits MDR1/BCRP, has antiproliferative activity.</p>
    Formula:C11H16N6O
    Purity:99.79%
    Color and Shape:Soild
    Molecular weight:248.28
  • LY-466195

    CAS:
    <p>LY-466195 is a competitive antagonist of GLUK5 receptor.</p>
    Formula:C16H24F2N2O4
    Color and Shape:Solid
    Molecular weight:346.37
  • ProTx II

    CAS:
    <p>Selective NaV1.7 inhibitor, alters activation, reduces current, 100x more selective for 1.7 over other Na+ channels.</p>
    Formula:C168H250N46O41S8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3826.59
  • Conantokin G

    CAS:
    GluN2B-specific NMDA receptor blocker; IC50=480 nM in neurons, ~300 nM in oocytes; neuroprotective.
    Formula:C88H138N26O44
    Purity:98%
    Color and Shape:White Lyophilised Solid
    Molecular weight:2264.21
  • NSC265473

    CAS:
    <p>NSC265473 is an ABCG2 substrate.</p>
    Formula:C21H35N3O4S
    Color and Shape:Solid
    Molecular weight:425.58
  • Linoleic Acid Amide

    CAS:
    <p>Linoleic Acid Amide (Linoleamide) is derived from linoleic acid and regulates Ca2+ flux by inhibiting the sarco/endoplasmic reticulum Ca2+-ATPase.</p>
    Formula:C18H33NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:279.46
  • α,β-Methylene-ATP dilithium

    CAS:
    <p>α,β-Methylene ATP dilithium, a phosphonic analog of ATP, serves as a ligand for P2X3 and P2X7 receptors.</p>
    Formula:C11H16Li2N5O12P3
    Color and Shape:Solid
    Molecular weight:517.07
  • MIDD0301

    CAS:
    <p>MIDD0301 is a potent positive allosteric α5β3γ selective GABAA receptor (GABAAR) ligand with EC50 of 17 nM.</p>
    Formula:C19H13BrFN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.23
  • Anisatin


    <p>Anisatin is a useful organic compound for research related to life sciences and the catalog number is T124719.</p>
    Formula:C15H20O8
    Color and Shape:Solid
    Molecular weight:328.317
  • Lyso-Globotriaosylceramide (d18:1)

    CAS:
    <p>Lyso-Gb3, lacking fatty acyl, binds Stx1 with cholesterol and phosphatidylcholine, not Stx2; lowers neutrophil viability; accumulates in Fabry disease.</p>
    Formula:C36H67NO17
    Color and Shape:Solid
    Molecular weight:785.922
  • 4-oxo-2-Nonenal

    CAS:
    <p>4-Hydroxy Nonenal and 4-oxo-2-Nonenal are lipid peroxidation byproducts, signaling oxidative stress and possibly causing mutagenesis.</p>
    Formula:C9H14O2
    Color and Shape:Solid
    Molecular weight:154.209
  • Mesoridazine free base

    CAS:
    <p>Mesoridazine (thioridazine EP impurity B) is a phenothiazine antipsychotic with effects similar to chlorpromazine.</p>
    Formula:C21H26N2OS2
    Color and Shape:Solid
    Molecular weight:386.57
  • Furosemide sodium

    CAS:
    <p>Furosemide sodium: potent NKCC inhibitor, loop diuretic, treats heart failure, hypertension, edema, selective GABAA antagonist.</p>
    Formula:C12H10ClN2NaO5S
    Purity:99.52% - >99.99%
    Color and Shape:Solid
    Molecular weight:352.73
  • Resolvin D2 methyl ester

    CAS:
    <p>RvD2 is an anti-inflammatory lipid made from docosahexaenoic acid by 15- and 5-lipoxygenase. Its methyl ester may serve as a prodrug.</p>
    Formula:C23H34O5
    Color and Shape:Solid
    Molecular weight:390.52
  • (+)-Lycoctonine

    CAS:
    Compound TJS1874 is a useful organic compound for research related to life sciences. The catalog number is TJS1874 and the CAS number is 26000-17-9.
    Formula:C25H41NO7
    Color and Shape:Solid
    Molecular weight:467.6
  • PtdIns-(1,2-dioctanoyl) (sodium salt)

    CAS:
    <p>PtdIns phosphates, a minor membrane lipid fraction, are vital for cell signaling. Synthetic PtdIns-(1,2-dioctanoyl) has C8:0 fatty acids and high solubility.</p>
    Formula:C25H47NaO13P
    Color and Shape:Solid
    Molecular weight:609.602
  • Tariquidar dimesylate

    CAS:
    <p>Tariquidar, a non-competitive P-glycoprotein inhibitor, may help combat cancer drug resistance.</p>
    Formula:C80H94N8O25S4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1695.9
  • Resolvin D2

    CAS:
    <p>Resolvin D2 (RvD2) is a TRPV1 inhibitor and pro-ablative mediator with anti-inflammatory, anti-infective and pro-ablative effects.</p>
    Formula:C22H32O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.49
  • BMS 199264

    CAS:
    <p>BMS 199264 hydrochlorid a inhibitor of mitochondrial F1F0 ATP hydrolase, thus preventing ATP reduction to ameliorate cardiac necrosis during ischemia.</p>
    Formula:C26H31ClN4O4S
    Purity:99.83%
    Color and Shape:Soild
    Molecular weight:531.07
  • Venturicidin A

    CAS:
    <p>Venturicidin A is a macrolide antibiotic.</p>
    Formula:C41H67NO11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:749.97
  • Foslevcromakalim

    CAS:
    <p>Foslevcromakalim (QLS-101), an ATP-sensitive potassium channel opener, serves as a proagent for ocular hypotensive effects [1] [2].</p>
    Formula:C16H19N2O6P
    Color and Shape:Solid
    Molecular weight:366.31
  • α-Casozepine

    CAS:
    <p>α-Casozepine,Bioactive peptide from milk α-S1 casein. Binds GABA receptors. Anti-anxiety effects.</p>
    Formula:C60H94N14O16
    Color and Shape:Solid
    Molecular weight:1267.47
  • P-gp inhibitor 13


    <p>P-gp Inhibitor 13, a P-glycoprotein antagonist, can counteract paclitaxel resistance in A2780/T cells, proving valuable for advanced acute myeloid leukemia</p>
    Formula:C32H34O8
    Color and Shape:Solid
    Molecular weight:546.61
  • NT 13

    CAS:
    <p>NT 13 is a partial N-methyl-D-aspartate receptor (NMDAR) agonist used in the study of depression, anxiety, and other related diseases.</p>
    Formula:C18H30N4O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.45
  • 3-Aminopropylphosphinic acid

    CAS:
    <p>3-Aminopropylphosphinic acid (3-APPA) is a phosphonic analog of gamma-aminobutyric acid (GABA).</p>
    Formula:C3H10NO2P
    Color and Shape:Solid
    Molecular weight:123.092
  • Vedroprevir

    CAS:
    <p>Vedroprevir (GS9451), a selective HCV NS3 protease inhibitor, targets genotype 1 HCV.</p>
    Formula:C45H60ClN7O9S
    Color and Shape:Solid
    Molecular weight:910.53
  • A 80915A

    CAS:
    <p>A80915A: Semi-naphthoquinone antibiotic, blocks gastric (H(+)-K+)-ATPase; potency varies with enzyme conformation; K+ reduces binding rate.</p>
    Formula:C26H31Cl3O5
    Color and Shape:Solid
    Molecular weight:529.88
  • (±)5(6)-DiHETE

    CAS:
    <p>Eicosapentaenoic acid is an ω-3 polyunsaturated fatty acid that is abundant in marine organisms and fish oils.</p>
    Formula:C20H32O4
    Color and Shape:Solid
    Molecular weight:336.472
  • 6-FAM-AEEAC-SHK TFA


    <p>6-FAM-AEEAC-SHK TFA, a peptide neurotoxin derived from Stichodactyla helianthus and conjugated with a fluorescent marker, selectively blocks voltage-gated potassium channels (kv1.1 and kv1.2). By prolonging action potentials, it interferes with neural signal conduction, making it valuable in neuroscience research.</p>
    Formula:C196H295N55O57S7·xCHF3O2
    Color and Shape:Solid
    Molecular weight:4558.23 (free acid)
  • ω-Conotoxin MVIIC

    CAS:
    <p>Peptide neurotoxin; wide spectrum blocker of N, P and Q type calcium channels.</p>
    Formula:C106H178N40O32S7
    Purity:98%
    Color and Shape:White Lyophilised Solid
    Molecular weight:2749