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Membrane Transporter/Ion Channel
Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
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Rapastinel
CAS:117928-94-6
Rapastinel (TPPT-amide) (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator.
Formula:
C18H31N5O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
413.47
Ref: TM-T3407
1mg | 47.00 € | ||
5mg | 87.00 € | ||
10mg | 114.00 € | ||
25mg | 226.00 € | ||
50mg | 336.00 € | ||
1ml*10 (DMSO) | 89.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Philanthotoxin 74 dihydrochloride
CAS:1227301-51-0
Philanthotoxin 74 dihydrochloride is an antagonist of AMPAR with IC50s of 263 and 296 nM …
Formula:
C24H44Cl2N4O3
Purity:
98.6%
Color and Shape:
Solid
Molecular weight:
507.54
Ref: TM-T16524
1mg | 51.00 € | ||
5mg | 144.00 € | ||
50mg | To inquire | ||
1ml*10 (DMSO) | 185.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Bamaquimast
CAS:135779-82-7
Bamaquimast (L 0042) is a proton pump inhibitor for the study of asthma-like immune system …
Formula:
C16H21N3O3
Purity:
98.40%
Color and Shape:
Solid
Molecular weight:
303.36
Ref: TM-T5449
1mg | 53.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Pandinotoxin Kα
CAS:185529-64-0
Pandinotoxin Kα, a chemical compound extracted from the emperor scorpion (Pandinus imperator) venom, functions as …
Formula:
C169H267N53O48S7
Purity:
98%
Molecular weight:
4033.71
Ref: TM-T80058
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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KT-362 fumarate
CAS:105394-80-7
KT-362 fumarate is a novel compound that acts as an antagonist of calcium channels, potassium …
Formula:
C26H32N2O7S
Purity:
99.90%
Color and Shape:
Solid
Molecular weight:
516.61
Ref: TM-T27753
1mg | 300.00 € | ||
5mg | 694.00 € | ||
10mg | 981.00 € | ||
25mg | 1,449.00 € | ||
50mg | 1,930.00 € | ||
100mg | 2,627.00 € | ||
1ml*10 (DMSO) | 833.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Bulleyaconitine A
CAS:107668-79-1
Bulleyaconitine A (Bulleyaconi cine A), an analgesic and antiinflammatory drug isolated from Aconitum plants, has …
Formula:
C35H49NO9
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
627.76
Ref: TM-T3021
20mg | 54.00 € | ||
1ml*10 (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Cytochalasin D
CAS:22144-77-0
Cytochalasin D is an actin inhibitor, the removal of actin stress fibers is crucial for …
Formula:
C30H37NO6
Color and Shape:
Needles From Acetone-Petroleum Ether Physical Description Needles Or Fluffy White Powder (Ntp 1992)
Molecular weight:
507.62
Ref: TM-T3229
1mg | 237.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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κM-Conotoxin RIIIJ
κM-Conotoxin RIIIJ (κM-RIIIJ) selectively inhibits Kv1.2 channels, exhibiting an IC50 value of 33 nM [1].
Formula:
C117H184N32O36S6
Purity:
98%
Molecular weight:
2807.3
Ref: TM-T80464
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Cirsimaritin
CAS:6601-62-3
Cirsimaritin exhibits antibacterial, anti-inflammation, anti-tumor, antioxidant properties and renal protection. Cirsimaritin binds weakly to the …
Formula:
C17H14O6
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
314.29
Ref: TM-TQ0119
1mg | 56.00 € | ||
5mg | 121.00 € | ||
10mg | 171.00 € | ||
25mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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ω-Conotoxin Bu8
ω-Conotoxin Bu8 is a 25-amino-acid-residue ω-conotoxin that features three disulfide bridges. It selectively and potently …
Formula:
C103H174N42O35S6
Purity:
98%
Molecular weight:
2753.13
Ref: TM-T80457
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Hongotoxin-1
Hongotoxin-1, a chemical compound isolated from the venom of Centruroides limbatus, functions as a potassium …
Formula:
C181H299N53O49S7
Purity:
98%
Molecular weight:
4226.13
Ref: TM-T80061
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Vocacapsaicin hydrochloride
CAS:1931116-92-5
Vocacapsaicin hydrochloride (CA-008 hydrochloride) is a non-opioid TRPV1 agonist, a raw material for capsaicin, and …
Formula:
C26H42ClN3O4
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
496.08
Ref: TM-T39349
1mg | 375.00 € | ||
5mg | 915.00 € | ||
10mg | 1,217.00 € | ||
25mg | 1,839.00 € | ||
50mg | 2,471.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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LY836
LY836 is an orally active, neuroprotective compound that effectively inhibits the PSD95-nNOS association in cortical …
Purity:
98%
Ref: TM-T81899
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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CRM1-IN-1
CRM1-IN-1 (Compound KL1), a noncovalent inhibitor of CRM1, promotes nuclear degradation of CRM1 with an …
Formula:
C29H48N2O5
Purity:
98%
Molecular weight:
504.7
Ref: TM-T79654
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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VU 0240551
CAS:893990-34-6
VU 0240551 is a selective antagonist of neuronal K-Cl cotransporter KCC2 inhibitor with an IC50 …
Formula:
C16H14N4OS2
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
342.44
Ref: TM-TQ0139
1mg | 50.00 € | ||
2mg | 66.00 € | ||
5mg | 94.00 € | ||
10mg | 143.00 € | ||
25mg | 291.00 € | ||
50mg | 547.00 € | ||
100mg | 787.00 € | ||
200mg | 1,067.00 € | ||
500mg | 1,576.00 € | ||
1ml*10 (DMSO) | 108.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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JTV-519 fumarate
CAS:1883549-36-7
JTV-519 fumarate (K201 fumarate) is a SERCA blocker and partial agonist at the ryanodine receptor …
Formula:
C29H36N2O6S
Molecular weight:
540.67
Ref: TM-T37807
1mg | 141.00 € | ||
5mg | 335.00 € | ||
10mg | 497.00 € | ||
25mg | 805.00 € | ||
50mg | 1,109.00 € | ||
100mg | 1,473.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Heteropodatoxin-1
Heteropodatoxin-1 (HpTx1), a spider peptide toxin, acts as an inhibitor of the Kv4.2 current, while …
Formula:
C168H238N46O51S6
Purity:
98%
Molecular weight:
3910.35
Ref: TM-T80435
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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PF-04745637
CAS:1917294-46-2
PF-04745637 is a potent and selective TRPA1 antagonist with an IC50 of 17 nM[1].
Formula:
C27H32ClF3N2O2
Purity:
99.3%
Color and Shape:
Solid
Molecular weight:
509
Ref: TM-T64337
1mg | 108.00 € | ||
5mg | 230.00 € | ||
10mg | 321.00 € | ||
25mg | 545.00 € | ||
50mg | 776.00 € | ||
100mg | 1,068.00 € | ||
500mg | 2,133.00 € | ||
1ml*10 (DMSO) | 258.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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A 839977
CAS:870061-27-1
A 839977 is a selective P2X7 receptor antagonist with anti-inflammatory and analgesic activity that inhibits …
Formula:
C19H14Cl2N6O
Purity:
98.01%
Color and Shape:
Solid
Molecular weight:
413.26
Ref: TM-T14076
1mg | 44.00 € | ||
2mg | 57.00 € | ||
5mg | 92.00 € | ||
1ml*10 (DMSO) | 143.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Nav1.8-IN-4
CAS:1620846-16-3
Nav1.8-IN-4 is a potent Nav1.8 channel inhibitor with potential analgesic activity.Nav1.8-IN-4 can be used for …
Formula:
C20H14F4N2O3
Purity:
99.83%
Color and Shape:
Soild
Molecular weight:
406.33
Ref: TM-T77693
1mg | 59.00 € | ||
2mg | 84.00 € | ||
5mg | 124.00 € | ||
10mg | 187.00 € | ||
25mg | 374.00 € | ||
50mg | 608.00 € | ||
100mg | 931.00 € | ||
500mg | 1,866.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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MitTx
MitTx, a complex consisting of MitTx-α and MitTx-β, serves as an ASIC1 channel activator, demonstrating …
Formula:
C899H1331N259O271S23
Purity:
98%
Molecular weight:
20840.26
Ref: TM-T80182
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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3'-Methoxydaidzein
CAS:21913-98-4
3'-Methoxydaidzein is a dual isoflavone and Sodium Channel inhibitor. 3'-Methoxydaidzein inhibited NaV1.7, NaV1.8 and NaV1.3 …
Formula:
C16H12O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
284.26
Ref: TM-TN1254
1mg | 142.00 € | ||
5mg | 343.00 € | ||
10mg | 549.00 € | ||
25mg | 868.00 € | ||
50mg | 1,170.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Fargesone B
CAS:116424-70-5
Fargesone B inhibits the vascular smooth muscle contraction by suppressing the voltage- and receptor-activated calcium …
Formula:
C21H24O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
372.417
Ref: TM-TN4051
5mg | To inquire | ||
1ml*10 (DMSO) | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Gavestinel
CAS:153436-38-5
Gavestinel (GV 150526) is a non-competitive NMDA receptor antagonist that is potent, selective and orally …
Formula:
C18H12Cl2N2NaO3
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
398.2
Ref: TM-T22798
1mg | 45.00 € | ||
5mg | 96.00 € | ||
10mg | 142.00 € | ||
25mg | 231.00 € | ||
50mg | 343.00 € | ||
100mg | 507.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Tamolarizine
CAS:93035-32-6
Tamolarizine (Tamolarizine free base) free base is a novel calcium antagonist.
Formula:
C27H32N2O3
Purity:
97.46%
Color and Shape:
Soild
Molecular weight:
432.55
Ref: TM-T34782
1mg | 138.00 € | ||
5mg | 335.00 € | ||
10mg | 495.00 € | ||
25mg | 798.00 € | ||
50mg | 1,095.00 € | ||
100mg | 1,486.00 € | ||
500mg | 2,960.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Clopimozide
CAS:53179-12-7
Clopimozide (R-29764) acts as a calcium channel antagonist and inhibits [3H] nilandipine binding.Clopimozide is a …
Formula:
C28H28ClF2N3O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
495.99
Ref: TM-T25263
1mg | 138.00 € | ||
5mg | 336.00 € | ||
10mg | 493.00 € | ||
25mg | 797.00 € | ||
50mg | 1,096.00 € | ||
100mg | 1,476.00 € | ||
500mg | 2,960.00 € | ||
1ml*10 (DMSO) | 410.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Amlodipine maleate
CAS:88150-47-4
Amlodipine maleate (Amvaz) is an orally active dihydropyridine calcium channel blocker that inhibits calcium inward …
Formula:
C24H29ClN2O9
Purity:
99.4%
Color and Shape:
White To Pale Yellow Crystalline Powder
Molecular weight:
524.95
Ref: TM-T21263
1g | 74.00 € | ||
500mg | 49.00 € | ||
1ml*10 (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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ProTx-III
ProTx-III, a spider venom peptide derived from the Peruvian green velvet tarantula, functions as a …
Formula:
C162H246N52O43S6
Purity:
98%
Molecular weight:
3802.4
Ref: TM-T80169
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Cis-22a
CAS:1819366-84-1
Cis-22a is a TRPV6 inhibitor (IC50 = 0.32 μM), which exhibits selectivity against related TRPV …
Formula:
C24H30F3N3O2
Purity:
98.49%
Color and Shape:
Solid
Molecular weight:
449.51
Ref: TM-T41233
1mg | 125.00 € | ||
5mg | 293.00 € | ||
10mg | 543.00 € | ||
25mg | 871.00 € | ||
50mg | 1,180.00 € | ||
100mg | 1,597.00 € | ||
500mg | 3,184.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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1-Hydroxy-2,3,5-trimethoxyxanthone
CAS:22804-49-5
1-Hydroxy-2,3,5-trimethoxyxanthone (HM-1) has vasodilator action ,which involves both an endothelium-dependent mechanism involving NO and an …
Formula:
C16H14O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
302.28
Ref: TM-TN2534
5mg | To inquire | ||
1ml*10 (DMSO) | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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TASK-1-IN-1
CAS:600125-11-9
TASK-1-IN-1 is a potent and selective inhibitor of TASK-1 (Potassium Channel) (IC50: 148 nM).TASK-1-IN-1 has …
Formula:
C22H20N2O2
Purity:
100%
Color and Shape:
Soild
Molecular weight:
344.41
Ref: TM-T72064
1mg | 40.00 € | ||
5mg | 86.00 € | ||
10mg | 123.00 € | ||
25mg | 270.00 € | ||
50mg | 423.00 € | ||
100mg | 625.00 € | ||
500mg | 1,327.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Nerisopam
CAS:102771-12-0
Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.
Formula:
C18H19N3O2
Purity:
97.27%
Color and Shape:
Solid
Molecular weight:
309.36
Ref: TM-T28159
1mg | 138.00 € | ||
5mg | 327.00 € | ||
10mg | 496.00 € | ||
25mg | 798.00 € | ||
50mg | 1,096.00 € | ||
100mg | 1,477.00 € | ||
500mg | 2,960.00 € | ||
1ml*10 (DMSO) | 441.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Fengabine
CAS:80018-06-0
Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat …
Formula:
C17H17Cl2NO
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
322.23
Ref: TM-T27310
1mg | 82.00 € | ||
5mg | 170.00 € | ||
10mg | 242.00 € | ||
25mg | 470.00 € | ||
50mg | 643.00 € | ||
100mg | 912.00 € | ||
500mg | 1,829.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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6-Hydroxyflavanone
CAS:4250-77-5
6-Hydroxyflavanone, extracted from the leaves of Acorus calamus, exhibits anti-inflammatory and anti-neuropathic pain activity by …
Formula:
C15H12O3
Purity:
98%
Color and Shape:
Slightly Yellow-Cream Powder
Molecular weight:
240.25
Ref: TM-TN1308
100mg | 54.00 € | ||
1ml*10 (DMSO) | 49.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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FS-2
FS-2 is a potent, specific inhibitor of L-type CaV channels, effectively impeding high K+ or …
Formula:
C297H462N92O86S10
Purity:
98%
Molecular weight:
7018.06
Ref: TM-T80441
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Tuvatexib
CAS:2055404-90-3
Tuvatexib is a small molecule VDAC/HK2 dual modulator.
Formula:
C21H23NO3
Purity:
99.90%
Color and Shape:
Solid
Molecular weight:
337.41
Ref: TM-T68018
1mg | 93.00 € | ||
5mg | 186.00 € | ||
10mg | 280.00 € | ||
25mg | 545.00 € | ||
50mg | 743.00 € | ||
100mg | 1,012.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Vesnarinone HCl
Vesnarinone HCl (OPC-8212 HCl) is an orally active phosphodiesterase 3 (PDE3) inhibitor.Vesnarinone HCl modulates calcium …
Formula:
C22H26ClN3O4
Purity:
99.17%
Color and Shape:
Soild
Molecular weight:
431.91
Ref: TM-T3465L
1mg | 54.00 € | ||
5mg | 96.00 € | ||
10mg | 128.00 € | ||
25mg | 208.00 € | ||
50mg | 368.00 € | ||
1ml*10 (DMSO) | 83.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Pazinaclone
CAS:103255-66-9
Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.
Formula:
C25H23ClN4O4
Purity:
98.12%
Color and Shape:
Solid
Molecular weight:
478.93
Ref: TM-T28303
1mg | 138.00 € | ||
5mg | 325.00 € | ||
10mg | 492.00 € | ||
25mg | 797.00 € | ||
50mg | 1,100.00 € | ||
100mg | 1,476.00 € | ||
500mg | 2,980.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Pafenolol
CAS:75949-61-0
Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an …
Formula:
C18H31N3O3
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
337.46
Ref: TM-T68124
1mg | 93.00 € | ||
5mg | 186.00 € | ||
10mg | 279.00 € | ||
25mg | 544.00 € | ||
50mg | 743.00 € | ||
100mg | 1,019.00 € | ||
500mg | 2,070.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Oxodipine
CAS:90729-41-2
Oxodipine, a dihydropyridine-type calcium antagonist , inhibited KCl-induced aortic contraction in rabbits and reduced cardiac …
Formula:
C19H21NO6
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
359.37
Ref: TM-T68123
1mg | 82.00 € | ||
5mg | 171.00 € | ||
10mg | 242.00 € | ||
25mg | 470.00 € | ||
50mg | 645.00 € | ||
100mg | 918.00 € | ||
500mg | 1,830.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Bupivacaine hydrochloride monohydrate
CAS:73360-54-0
Bupivacaine hydrochloride monohydrate is a potent NMDA receptor inhibitor of sodium, L-calcium, and potassium channels.Bupivacaine …
Formula:
C18H31ClN2O2
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
342.9
Ref: TM-T80641
1mg | 181.00 € | ||
5mg | 449.00 € | ||
10mg | 643.00 € | ||
25mg | 1,003.00 € | ||
50mg | 1,383.00 € | ||
100mg | 1,828.00 € | ||
500mg | 3,647.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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µ-Conotoxin-CnIIIC acetate
µ-Conotoxin-CnIIIC acetate is a potent NaV1.4 sodium channel antagonist, a conotoxin peptide consisting of 22 …
Formula:
C92H139N35O28S6·xC2H4O2
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
2375.70 (free base)
Ref: TM-T78108
1mg | 46.00 € | ||
5mg | 118.00 € | ||
10mg | 185.00 € | ||
25mg | 312.00 € | ||
50mg | 465.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Ethacizine hydrochloride
CAS:57530-40-2
Ethacizine hydrochloride (NIK-244) has antiarrhythmic activity, and its effects are related to cardiac activity and …
Formula:
C22H28ClN3O3S
Purity:
98.08%
Color and Shape:
Solid
Molecular weight:
449.99
Ref: TM-T11239
1mg | 78.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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KCNQ1 activator-1
CAS:1008671-38-2
2-Piperidinecarboxamide, N-[4-(4-methoxyphenyl)-2-thiazolyl]-1-(phenylsulfonyl)- is a potent KCNQ1 channel activator that can be used in long QT …
Formula:
C22H23N3O4S2
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
457.57
Ref: TM-T9778
1mg | 92.00 € | ||
5mg | 221.00 € | ||
10mg | 333.00 € | ||
25mg | 663.00 € | ||
50mg | 886.00 € | ||
100mg | 1,207.00 € | ||
500mg | 2,423.00 € | ||
1ml*10 (DMSO) | 245.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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TTA-A8
CAS:1146395-46-1
TTA-A8 is an antagonist of T-type calcium channel.
Formula:
C22H21F3N4O2
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
430.42
Ref: TM-T71990
1mg | 377.00 € | ||
5mg | 900.00 € | ||
10mg | 1,119.00 € | ||
25mg | 1,499.00 € | ||
50mg | 1,838.00 € | ||
100mg | 2,320.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Adenosine 5'-diphosphoribose sodium
CAS:68414-18-6
Adenosine 5'-diphosphoribose sodium (ADP ribose sodium) is a metabolite of nicotinamide adenine nucleotide (NAD+), which …
Formula:
C15H22N5NaO14P2
Purity:
99.38%
Color and Shape:
Solid
Molecular weight:
581.3
Ref: TM-T10247
5mg | 66.00 € | ||
10mg | 94.00 € | ||
25mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Transcainide
CAS:88296-62-2
Transcainide(R 54718), a new lidocaine analog, is an orally active antiarrhythmic agent.Transcainide blocks the open …
Formula:
C22H35N3O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
373.53
Ref: TM-T26287
1mg | 250.00 € | ||
5mg | 616.00 € | ||
10mg | 879.00 € | ||
25mg | 1,299.00 € | ||
50mg | 1,746.00 € | ||
100mg | 2,378.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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RN9893
CAS:1803003-68-0
RN9893 is a selective and potent TRPV4 receptor antagonist with IC50 values of 320, 420 …
Formula:
C21H23F3N4O5S
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
500.49
Ref: TM-T28548
1mg | 46.00 € | ||
5mg | 96.00 € | ||
10mg | 141.00 € | ||
25mg | 268.00 € | ||
50mg | 397.00 € | ||
100mg | 578.00 € | ||
500mg | 1,187.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Suzetrigine
CAS:2649467-58-1
Suzetrigine(VX-548) is an orally active and specific NaV1.8 inhibitor. Suzetrigine has analgesic activity and can …
Formula:
C21H20F5N3O4
Purity:
98.08%
Color and Shape:
Solid
Molecular weight:
473.39
Ref: TM-T69552
1mg | 444.00 € | ||
5mg | 1,096.00 € | ||
10mg | 1,466.00 € | ||
25mg | 2,191.00 € | ||
50mg | 2,952.00 € |
Estimated delivery in United States, on Monday 8 Jul 2024
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Imperatoxin A
CAS:172451-37-5
Imperatoxin A, a peptide toxin sourced from the African scorpion Pandinus imperator, functions as an …
Formula:
C148H254N58O45S6
Purity:
98%
Molecular weight:
3758.35
Ref: TM-T80063
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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KV1.3-IN-1
KV1.3-IN-1 (Compound trans-18), a selective KV1.3 channel inhibitor with IC50 values of 230 nM in …
Formula:
C23H30N2O4S
Purity:
98%
Molecular weight:
430.56
Ref: TM-T79445
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Anthopleurin-C
Anthopleurin-C (APE 2-1) is a cardiotonic polypeptide exhibiting a potent positive inotropic effect [1].
Formula:
C210H316N62O61S6
Purity:
98%
Molecular weight:
4877.52
Ref: TM-T80461
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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γ-Glutamylserine TFA
γ-Glutamylserine TFA (γ-Glu-Ser TFA) serves as a calcium receptor activator and is utilized in research …
Formula:
C10H15F3N2O8
Purity:
98%
Molecular weight:
348.23
Ref: TM-T80681
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Jingzhaotoxin-X
Jingzhaotoxin-X (JZTX-X) selectively inhibits Kv4.2 and Kv4.3 potassium channels, resulting in prolonged mechanical hyperalgesia [1].
Formula:
C164H242N46O41S6
Purity:
98%
Molecular weight:
3706.35
Ref: TM-T80500
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Myr-TAT-CBD3
Myr-TAT-CBD3, a CRMP2-CaV2.2 interaction inhibitor, has been shown to significantly attenuate carrageenan-induced thermal hypersensitivity and …
Formula:
C148H269N59O33
Purity:
98%
Molecular weight:
3403.09
Ref: TM-T80501
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Pe1b
Pe1b (μ-TrTx-Pe1b) is a selective inhibitor of the NaV1.7 channel, exhibiting an inhibitory concentration 50 …
Formula:
C175H237N47O49S6
Purity:
98%
Molecular weight:
3975.43
Ref: TM-T80450
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Jingzhaotoxin-IX
Jingzhaotoxin-IX is a C-terminally amidated peptide neurotoxin consisting of 35 amino acid residues. It inhibits …
Formula:
C171H251N49O48S6
Purity:
98%
Molecular weight:
3953.51
Ref: TM-T80426
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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GABA receptor Antagonist 1
GABA receptor Antagonist 1 (compound 7w) effectively inhibits the Px RDL1 GABAR at an IC50 …
Purity:
98%
Ref: TM-T82357
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Nav1.3 channel inhibitor 1
Nav1.3 Channel Inhibitor 1 (Compound 15b) is a state-dependent inhibitor of the voltage-gated sodium channel …
Formula:
C19H15F2N3O3S2
Purity:
98%
Molecular weight:
435.47
Ref: TM-T79280
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Lactate transportor 1
Lactate Transporter 1 (Compound 1) serves as an active lactate transporter within living cells and …
Purity:
98%
Ref: TM-T81962
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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MmTx1 toxin
Micrurotoxin 1 (MmTx1 toxin) acts as an allosteric modulator of GABA A receptors, enhancing the …
Formula:
C295H455N95O97S10
Purity:
98%
Molecular weight:
7205
Ref: TM-T80489
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Tamapin
Tamapin, a venom peptide isolated from the Indian red scorpion (Mesobuthus tamulus) [1], selectively targets …
Formula:
C146H238N44O41S6
Purity:
98%
Molecular weight:
3458.11
Ref: TM-T80170
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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CFTR corrector 12
CAS:958941-60-1
CFTR Corrector 12 (Compound 17C), a bithiazole derivative, functions as a CFTR corrector by remedying …
Formula:
C19H21ClN4O2S2
Purity:
98%
Molecular weight:
436.98
Ref: TM-T79578
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Phrixotoxin-1
CAS:221872-97-5
Phrixotoxin 1, a specific peptide inhibitor of Kv4 potassium channels, originates from the venom of …
Formula:
C156H246N44O37S7
Purity:
98%
Molecular weight:
3554.35
Ref: TM-T80053
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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(Rac)-PD0299685
CAS:313651-02-4
(Rac)-PD0299685 is a potent voltage-dependent calcium channel inhibitor for the study of retina-related diseases.
Formula:
C10H21NO2
Purity:
97.20%
Color and Shape:
Solid
Molecular weight:
187.28
Ref: TM-T68125
Undefined size | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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CRM1-IN-2
CRM1-IN-2 (Compound KL2) is a noncovalent inhibitor that targets CRM1, localizing it to the nuclear …
Formula:
C29H48N2O5
Purity:
98%
Molecular weight:
504.7
Ref: TM-T79655
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Ancistrotecine B
Ancistrotecine B (Compound 2), a Nav1.7 channel inhibitor (IC50: 0.73 μM), has been shown to …
Formula:
C26H31NO4
Purity:
98%
Molecular weight:
421.53
Ref: TM-T79398
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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6-Hydroxykynurenic acid
CAS:3778-29-8
6-Hydroxykynurenic acid (6-HKA), a kynurenic acid (KYNA) derivative isolated from Ginkgo leaves, functions as a …
Formula:
C10H7NO4
Purity:
98%
Molecular weight:
205.17
Ref: TM-T79959
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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PptT-IN-4
PptT-IN-4 (Compound 3a) is a PptT inhibitor exhibiting an IC50 of 0.71 μM. It also …
Formula:
C17H23N3
Purity:
98%
Molecular weight:
269.38
Ref: TM-T78714
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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BBT
CAS:445000-45-3
BBT enhances glucose-stimulated insulin secretion (GSIS) in compromised conditions, demonstrates anti-hyperglycemia effects, and shields β-cells …
Formula:
C18H12BrNO2S
Purity:
98%
Molecular weight:
386.26
Ref: TM-T78066
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Mambalgin-2
Mambalgin-2 (Mamb-2), a venom peptide sourced from the African black mamba, acts as an inhibitor …
Formula:
C272H431N85O83S10
Purity:
98%
Molecular weight:
6540.5
Ref: TM-T80492
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Jingzhaotoxin XI
Jingzhaotoxin XI (JZTX-XI) is a potent inhibitor of sodium conductance, exhibiting an IC50 value of …
Formula:
C158H234N44O47S7
Purity:
98%
Molecular weight:
3726.27
Ref: TM-T80499
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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µ-Conotoxin BuIIIB
CAS:1400096-06-1
μ-Conotoxin BuIIIB (Mu-Conotoxin BuIIIB), a selective blocker of mammalian neuronal voltage-gated sodium channels (VGSC), is …
Formula:
C106H172N46O30S6
Purity:
98%
Molecular weight:
2763.18
Ref: TM-T80491
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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wt hMLN
Wild-type human myoregulin (wt hMLN) is a microprotein that inhibits the sarcoplasmic reticulum Ca²⁺ pump …
Formula:
C245H404N54O66S
Purity:
98%
Molecular weight:
5194.22
Ref: TM-T80556
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Arecaidine hydrobromide
CAS:6013-57-6
Arecaidine hydrobromide, a pyridine alkaloid, functions as a potent GABA uptake inhibitor and acts as …
Formula:
C7H12BrNO2
Purity:
98%
Molecular weight:
222.08
Ref: TM-T80013
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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ω-Conotoxin FVIA
ω-Conotoxin FVIA is an inhibitor of N-type Ca²⁺ channels (Caᵥ2.2), shown to alleviate mechanical and …
Formula:
C98H164N36O33S6
Purity:
98%
Molecular weight:
2566.96
Ref: TM-T80446
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Aah II
Aah II, a sodium channel modulator, is a toxin derived from the venom of the …
Formula:
C313H457N89O95S8
Purity:
98%
Molecular weight:
7243.04
Ref: TM-T80162
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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D-GsMTx4 TFA
D-GsMTx4 TFA, a selective spider venom peptide, is a TRPC1/6 and Piezo2 inhibitor that inhibits …
Formula:
C187H279F3N48O48S6
Purity:
98%
Color and Shape:
Soild
Molecular weight:
4217
Ref: TM-T37697L
Undefined size | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Phlo1b
Phlo1b (μ-TrTx-Phlo1b), a 35-amino acid peptide toxin, selectively inhibits Nav1.7 channels with minimal inhibition of …
Formula:
C181H260N52O49S6
Purity:
98%
Molecular weight:
4140.71
Ref: TM-T80444
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Aam-KTX
Aam-KTX, a toxic peptide sourced from Mesobuthus eupeus scorpion venom, acts as a selective K_v …
Formula:
C174H288N58O48S7
Purity:
98%
Molecular weight:
4184.96
Ref: TM-T80483
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Vm24-toxin
CAS:1373890-79-9
Vm24-toxin, a peptide toxin isolated from the Mexican scorpion Vaejovis mexicanus smithi, serves as an …
Formula:
C157H253N51O45S9
Purity:
98%
Molecular weight:
3863.59
Ref: TM-T80524
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Ssm spooky toxin
Ssm Spooky Toxin, derived from Scolopendra mutilans, exhibits potent lethality affecting both hematological and respiratory …
Formula:
C270H413N69O79S4
Purity:
98%
Molecular weight:
6017.84
Ref: TM-T80528
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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LFS-1107
CAS:1799330-91-8
LFS-1107, a reversible CRM1 inhibitor (Kd: 12.5 pM), selectively targets and eliminates ENKTL cells, offering …
Formula:
C12H11N5OS2
Purity:
98%
Molecular weight:
305.38
Ref: TM-T81936
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Phlotoxin-1
Phlotoxin-1 (PhlTx1), a 34-amino acid peptide featuring three disulfide bridges, is derived from the Phlogiellus …
Formula:
C183H254N46O48S6
Purity:
98%
Molecular weight:
4058.64
Ref: TM-T80177
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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NMDA receptor antagonist 7
Compound (S)-10a, a GluN2B subunit-selective NMDA receptor antagonist, exhibits a K i of 93 nM …
Formula:
C22H27N3O
Purity:
98%
Molecular weight:
349.47
Ref: TM-T79374
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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ω-Conotoxin SO3
CAS:441284-32-8
ω-Conotoxin SO3 is an analgesic peptide that functions as an antagonist to N-type voltage-sensitive calcium …
Formula:
C100H166N36O31S6
Purity:
98%
Molecular weight:
2561
Ref: TM-T80161
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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μ-Conotoxin SxIIIC
μ-Conotoxin SxIIIC, an irreversible NaV channel inhibitor, is derived from Conus striolatus and is useful …
Formula:
C90H142N42O27S6
Purity:
98%
Molecular weight:
2436.75
Ref: TM-T80485
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Pterinotoxin-2
Pterinotoxin-2 is a peptide toxin that acts as a sodium channel inhibitor [1].
Formula:
C156H237N45O42S7
Purity:
98%
Molecular weight:
3639.28
Ref: TM-T80533
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Mambalgin-3
Mambalgin-3, an acid-sensitive ion channel 1 (ASIC1) inhibitor, has potential applications in analgesia research [1].
Formula:
C274H433N85O83S10
Purity:
98%
Molecular weight:
6566.54
Ref: TM-T80518
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Calcicludine
CAS:178036-64-1
Calcicludine, a protein toxin derived from the green mamba (Dendroaspis angusticeps) venom, selectively inhibits high-voltage-activated, …
Formula:
C321H476N86O78S6
Purity:
98%
Molecular weight:
6980.13
Ref: TM-T80065
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Caloxin 3A1
Caloxin 3A1, a biologically active peptide, is a member of the caloxins, which are inhibitors …
Formula:
C83H126N22O30
Purity:
98%
Molecular weight:
1912.02
Ref: TM-T80247
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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δ-Theraphotoxin-Hm1b
δ-Theraphotoxin-Hm1b, a 42-amino acid peptide derived from the Togo starburst tarantula (Heteroscodra maculata) venom, selectively …
Formula:
C169H241N45O50S6
Purity:
98%
Molecular weight:
3895.38
Ref: TM-T80430
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Jingzhaotoxin-II
Jingzhaotoxin-II, a neurotoxin composed of 32 amino acid residues featuring two acidic and two basic …
Formula:
C154H219N39O45S7
Purity:
98%
Molecular weight:
3561.08
Ref: TM-T80427
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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ω-Conotoxin CVIF
ω-Conotoxin CVIF is a selective inhibitor of Ca v 2.2 channels, demonstrating an IC50 value …
Formula:
C101H170N40O33S6
Purity:
98%
Molecular weight:
2665.07
Ref: TM-T80448
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50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Aa1 toxin
Aa1 toxin, sourced from Androctonus australis Garzoni venom, is a neurotoxic peptide that specifically blocks …
Formula:
C156H260N54O49S6
Purity:
98%
Molecular weight:
3868.46
Ref: TM-T80484
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Estimated delivery in United States, on Monday 8 Jul 2024
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δ-Buthitoxin-Hj1a
δ-Buthitoxin-Hj1a, a scorpion-venom peptide, functions as a potent agonist for the NaV1.1 channel, exhibiting an …
Formula:
C326H482N92O96S8
Purity:
98%
Molecular weight:
7482.39
Ref: TM-T80433
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Estimated delivery in United States, on Monday 8 Jul 2024
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GAD65(247-266) epitope TFA
GAD65(247-266) epitope TFA, a T cell epitope derived from islet antigens, exhibits competitive binding to …
Formula:
C111H174F3N27O29S4
Purity:
98%
Molecular weight:
2535.99
Ref: TM-T80218
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Estimated delivery in United States, on Monday 8 Jul 2024
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Hemitoxin
Hemitoxin, a scorpion-venom peptide, functions as a K+ channel blocker and selectively inhibits rat Kv1.1, …
Formula:
C159H259N49O49S8
Purity:
98%
Molecular weight:
3897.58
Ref: TM-T80436
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50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Phlo1a
Phlo1a (μ-TrTx-Phlo1a), a 35-amino acid peptide toxin, demonstrates a weak inhibitory effect on Nav1.2 and …
Formula:
C178H262N52O49S6
Purity:
98%
Molecular weight:
4106.69
Ref: TM-T80445
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50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024
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Sodium Channel inhibitor 4
CAS:587843-16-1
Sodium Channel Inhibitor 4 is a compound that functions as a sodium channel inhibitor [1].
Formula:
C19H18ClN3O4S2
Purity:
98%
Molecular weight:
451.95
Ref: TM-T81134
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50mg | To inquire |
Estimated delivery in United States, on Monday 8 Jul 2024