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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2290 products of "Membrane Transporter/Ion Channel"

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  • mGAT3/4-IN-2
    Targetmol
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    mGAT3/4-IN-2

    CAS:
    <p>mGAT3/4-IN-2 are potent inhibitors of mGAT3/mGAT4 with their pIC50 values of 5.44 and 5.25, respectively.</p>
    Formula:C26H32ClN3OS2
    Color and Shape:Solid
    Molecular weight:502.13

    Ref: TM-T63408

  • GDC-6599
    Targetmol
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    GDC-6599

    CAS:
    <p>GDC-6599 (Example 8) is an orally active inhibitor of the TRPA1 channel, potentially useful for researching TRPA1-mediated conditions, including pain [1].</p>
    Formula:C20H19ClN6O3
    Color and Shape:Solid
    Molecular weight:426.86

    Ref: TM-T79875

  • M084 hydrochloride
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    M084 hydrochloride

    CAS:
    <p>M084 hydrochloride, a TRPC4/5 channel blocker, exhibits IC50 values of 10.3 μM and 8.2 μM, respectively. This compound is noted for its antidepressant and anxiolytic effects [1] [2].</p>
    Formula:C11H16ClN3
    Color and Shape:Solid
    Molecular weight:225.72

    Ref: TM-T84900

  • MONIRO-1
    Targetmol
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    MONIRO-1

    CAS:
    <p>MONIRO-1 blocks T/N-type Ca²⁺ channels: hCav2.2 (IC50: 34μM), hCav3.1 (3.3μM), hCav3.2 (1.7μM), hCav3.3 (7.2μM).</p>
    Formula:C23H24ClFN4O3
    Color and Shape:Solid
    Molecular weight:458.92

    Ref: TM-T62876

  • NMDA receptor modulator 6
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    NMDA receptor modulator 6

    CAS:
    <p>NMDA receptor regulator 6 (Compound 183) is an effective NMDA receptor regulator and has research value in neurological disorders.</p>
    Formula:C20H17FN2O4S
    Color and Shape:Solid
    Molecular weight:400.42

    Ref: TM-T61924

  • Clobutinol hydrochloride
    Targetmol
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    Clobutinol hydrochloride

    CAS:
    <p>Clobutinol hydrochloride, an antitussive agent, influences heart rate and blood pressure, and is utilized in cough-related research [1] [2] [3].</p>
    Formula:C14H23Cl2NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:292.25

    Ref: TM-T78523

  • CFTR corrector 12
    Targetmol
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    CFTR corrector 12

    CAS:
    <p>CFTR corrector 12 is a CFTR corrector that rescues all mutant proteins except M760R ABCA3 and can be used to study cystic fibrosis.</p>
    Formula:C19H21ClN4O2S2
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:436.98

    Ref: TM-T79578

  • CFTR corrector 6
    Targetmol
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    CFTR corrector 6

    CAS:
    <p>CFTR corrector 6, a potent CFTR potentiator, aids cystic fibrosis research and related disorders.</p>
    Formula:C22H13F4N9
    Color and Shape:Solid
    Molecular weight:479.39

    Ref: TM-T37686

  • LG 83-6-05
    Targetmol
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    LG 83-6-05

    CAS:
    <p>LG 83-6-05 is a novel kind of sodium channel blocking agent.</p>
    Formula:C21H30ClNO3S
    Color and Shape:Solid
    Molecular weight:411.99

    Ref: TM-T32731

  • TRPC5 modulator-1
    Targetmol
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    TRPC5 modulator-1

    CAS:
    <p>TRPC5 modulator-1 (Compound 9) is a TRPC5 modulator (IC50&lt;1 nM) that can be used to study neuropsychiatric disorders.</p>
    Formula:C23H27FN2O4
    Color and Shape:Solid
    Molecular weight:414.47

    Ref: TM-T62133

  • ROMK-IN-32
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    ROMK-IN-32

    CAS:
    <p>ROMK-IN-32 is an inhibitor of the extra-renal medullary potassium channel (ROMK) (IC50: 35 nM) and also inhibits hERG (IC50: 22 μM).</p>
    Formula:C24H28N4O5
    Color and Shape:Solid
    Molecular weight:452.5

    Ref: TM-T62760

  • Dibutyryl-cGMP sodium
    Targetmol
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    Dibutyryl-cGMP sodium

    CAS:
    Bt2cGMP sodium is a cGMP analog, activates PKG, inhibits platelet [3H]-arachidonate, and induces analgesia via K+ channels.
    Formula:C18H24N5NaO9P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:508.38

    Ref: TM-T11038

  • CGP-54626 free base
    Targetmol
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    CGP-54626 free base

    CAS:
    CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).
    Formula:C18H28Cl2NO3P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.3

    Ref: TM-T26998

  • GSK3395879
    Targetmol
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    GSK3395879

    CAS:
    <p>GSK3395879 is a selective and orally bioavailable antagonist of transient receptor potential vanilloid-4 (TRPV4) (IC50: 1 nM for hTRPV4).</p>
    Formula:C20H15F4N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:485.41

    Ref: TM-T15439

  • SN40 hydrochloride
    Targetmol
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    SN40 hydrochloride

    CAS:
    <p>SN40 hydrochloride is a potent inhibitor of amino acid transport (AAT), exhibiting inhibitory constants (Kis) of 7.29 μM, 2.42 μM, 2.94 μM, 5.55 μM, 24.43 μM, and 5.55 μM for rat ASCT2, human ASCT2, EAAT1, EAAT2, EAAC1, and EAAT5, respectively. It is utilized in cancer research. [1]</p>
    Formula:C18H21ClN2O2
    Color and Shape:Solid
    Molecular weight:332.82

    Ref: TM-T84754

  • AMPA-IN-1
    Targetmol
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    AMPA-IN-1

    CAS:
    <p>AMPA-IN-1: Potent AMPA receptor inhibitor; key in regulating brain excitatory transmission and plasticity.</p>
    Formula:C23H12F2N4O2
    Color and Shape:Solid
    Molecular weight:414.36

    Ref: TM-T62127

  • L-822179
    Targetmol
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    L-822179

    CAS:
    <p>L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.</p>
    Formula:C17H14N8O2
    Purity:98.5% - 99.61%
    Color and Shape:Solid
    Molecular weight:362.35

    Ref: TM-T24381

  • KCa1.1 channel activator-1
    Targetmol
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    KCa1.1 channel activator-1

    <p>A selective vascular KCa1.1 channel stimulator with CaV1.2 blocking ability and mild myorelaxant effects.</p>
    Formula:C25H16O10
    Color and Shape:Solid
    Molecular weight:476.39

    Ref: TM-T72194

  • Afizagabar
    Targetmol
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    Afizagabar

    CAS:
    <p>Afizagabar, a first-in-class α5-GABAAR antagonist, IC50: 585 nM, Ki: 66 nM, may boost memory.</p>
    Formula:C19H12FN3O2S
    Color and Shape:Solid
    Molecular weight:365.38

    Ref: TM-T37388

  • JM-1232
    Targetmol
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    JM-1232

    CAS:
    <p>JM-1232 is a sedative and hypnotic drug being researched as a potential anesthetic.</p>
    Formula:C24H27N3O2
    Color and Shape:Solid
    Molecular weight:389.49

    Ref: TM-T24201