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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2280 products of "Membrane Transporter/Ion Channel"

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  • CymitQuimica logo
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    Jingzhaotoxin III

    CAS:
    <p>NaV1.5 channels blocker</p>
    Formula:C174H241N47O46S6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3919.47

    Ref: TM-TP2263

  • P2X4 antagonist-4
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    P2X4 antagonist-4

    <p>P2X4 antagonist-4 (compound 64) is a potent P2X4R antagonist with an IC50 value of 8 µM. It can inhibit ATP-induced activation of the NLRP3 inflammasome and the subsequent release of IL-1β.</p>
    Formula:C27H22FN3O4S
    Color and Shape:Solid
    Molecular weight:503.545

    Ref: TM-T204441

  • Hyp9
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    Hyp9

    CAS:
    <p>Hyp9, a specific agonist for the transient receptor potential canonical 6 (TRPC6) channel, is utilized in spinal cord injury (SCI) research [1].</p>
    Formula:C18H26O5
    Color and Shape:Solid
    Molecular weight:322.40

    Ref: TM-T75550

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    Chlorotoxin TFA

    <p>Chlorotoxin TFA, a scorpion venom peptide, blocks chloride channels and has anti-cancer properties.</p>
    Formula:C160H250F3N53O49S11
    Color and Shape:Solid
    Molecular weight:4109.74

    Ref: TM-T75722

  • JAMI1001A
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    JAMI1001A

    CAS:
    <p>JAMI1001A enhances AMPA receptor signaling, slows deactivation/desensitization for flip/flop isoforms.</p>
    Formula:C16H17F3N4O3S
    Color and Shape:Solid
    Molecular weight:402.39

    Ref: TM-T38392

  • SLC26A3-IN-2
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    SLC26A3-IN-2

    CAS:
    <p>Vilobelimab (CaCP-29) is a human-mouse chimeric IgG antibody targeting human complement component 5a, a C5a inhibitor that inhibits neutrophil activation.</p>
    Formula:C19H13ClN2O2S
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:368.84

    Ref: TM-T74815

  • Homocarnosine
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    Homocarnosine

    CAS:
    <p>Homocarnosine is an endogenous dipeptide in cerebral regions and cerebrospinal fluid.</p>
    Formula:C10H16N4O3
    Color and Shape:Solid
    Molecular weight:240.26

    Ref: TM-T32098

  • Bendroflumethiazide
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    Bendroflumethiazide

    CAS:
    <p>Bendroflumethiazide (Naturetin) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE. It has been used in the treatment of familial hyperkalemia, hypertension, edema, and urinary tract disorders. (From Martindale, The Extra Pharmacopoeia, 30th ed, p810)</p>
    Formula:C15H14F3N3O4S2
    Purity:98% - >99.99%
    Color and Shape:Crystals From Dioxane Solid
    Molecular weight:421.41

    Ref: TM-T1204

  • TP-050
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    TP-050

    CAS:
    <p>TP-050: potent, selective NMDAR agonist, EC50 0.51 µM (GluN2A), 9.6 µM (GluN2D), BBB permeable, boosts hippocampal LTP.</p>
    Formula:C16H15ClF2N6O
    Color and Shape:Solid
    Molecular weight:380.78

    Ref: TM-T73491

  • Trans (2,3)-Dihydrotetrabenazine
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    Trans (2,3)-Dihydrotetrabenazine

    CAS:
    <p>Trans (2,3)-Dihydrotetrabenazine is a Tetrabenazine metabolite, shows inhibition activity on vesicular monoamine transporter (VMAT2).</p>
    Formula:C19H29NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:319.44

    Ref: TM-T12190

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    Anticonvulsant agent 9

    <p>Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.</p>
    Formula:C22H24N4O2
    Color and Shape:Solid
    Molecular weight:376.45

    Ref: TM-T205256

  • Levamlodipine besylate Hemipentahydrate
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    Levamlodipine besylate Hemipentahydrate

    CAS:
    <p>Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.</p>
    Formula:C20H25ClN2O5·C6H6O3SH2O
    Color and Shape:Solid
    Molecular weight:1224.18

    Ref: TM-T204904

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    Idactamab

    CAS:
    <p>Idactamab (INT-001) is a monoclonal antibody to the human amino acid transport protein ASCT2.</p>
    Purity:> 95%
    Color and Shape:Liquid
    Molecular weight:146.2 kDa

    Ref: TM-T77385

  • BeKm-1
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    BeKm-1

    CAS:
    <p>Potent, selective hERG (KV11.1) blocker; doesn't affect 14 other K+ channels; extends QTc in rabbit heart dose-dependently.</p>
    Formula:C174H261N51O52S6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4091.65

    Ref: TM-TP2072

  • Cevadine
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    Cevadine

    <p>Cevadine is a natural product that can be used as a reference standard.</p>
    Formula:C32H49NO9
    Color and Shape:Solid
    Molecular weight:591.742

    Ref: TM-T124525

  • Sulcardine 2HCl
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    Sulcardine 2HCl

    CAS:
    <p>Sulcardine 2HCl is a multi-ion channel blocker that blocks the properties of hERG and hNav1.5 channels and can be used to study atrial fibrillation.</p>
    Formula:C24H35Cl2N3O4S
    Purity:99.33% - 99.76%
    Color and Shape:Soild
    Molecular weight:532.523

    Ref: TM-T83979

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    Crofelemer

    CAS:
    <p>Crofelemer (Provir) is an orally active antidiarrheal agent. It targets the cystic fibrosis transmembrane conductance regulator (CFTR) and calcium-activated chloride channels (CACC), which are responsible for chloride and fluid secretion in the gastrointestinal tract. Crofelemer is applicable for research in diarrhea-related conditions.</p>
    Color and Shape:Solid

    Ref: TM-T205474

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    EVT-401

    <p>EVT-401 (P2X7 receptor antagonist-1), a purinergic P2X7 receptor antagonist, demonstrates efficacy in combating neuroinflammation [1].</p>
    Formula:C22H20F4N2O3
    Color and Shape:Solid
    Molecular weight:436.4

    Ref: TM-T74409

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    AChE/Aβ-IN-2

    <p>AChE/Aβ-IN-2 (compound 33) is a powerful, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 135 nM.</p>
    Formula:C20H25ClN4
    Color and Shape:Solid
    Molecular weight:356.89

    Ref: TM-T79571

  • 1-(1-Methyl-1h-pyrazol-4-yl)-ethanone
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    1-(1-Methyl-1h-pyrazol-4-yl)-ethanone

    CAS:
    <p>1-(1-Methyl-1h-pyrazol-4-yl)-ethanone is a high purity biochemical reagent that can be used in research related to life sciences.</p>
    Formula:C6H8N2O
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:124.14

    Ref: TM-TN9428