CymitQuimica logo
Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

Show 13 more subcategories

Found 2293 products of "Membrane Transporter/Ion Channel"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • NMDA agonist 2


    <p>NMDA agonist 2 (compound 8d) effectively inhibits NMDA receptors, exhibiting an EC50 of 0.034 μM for GluN1/2C. It plays a significant role in neurological and psychiatric disorders.</p>
    Formula:C14H12BrFN2O3S
    Color and Shape:Solid
    Molecular weight:387.224
  • Ion Channel Targeted Library


    <p>A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;</p>
    Color and Shape:Odour Solid
  • (1S,3R)-3-Aminocyclopentane carboxylic acid

    CAS:
    <p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>
    Formula:C6H11NO2
    Color and Shape:Solid
    Molecular weight:129.16
  • Volixibat

    CAS:
    <p>Volixibat, a selective inhibitor of the bile acid transporter, may treat non-alcoholic steatohepatitis.</p>
    Formula:C38H51N3O12S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:805.95
  • CALP3

    CAS:
    <p>Cell-permeable CaM agonist, binds EF-hand, activates phosphodiesterase without Ca2+, inhibits Ca2+ toxicity, IC50=33μM.</p>
    Formula:C44H68N10O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:881.08
  • Cyclic ADP-ribose ammonium


    <p>cADPR ammonium is a second messenger that boosts cytosolic calcium via Ryanodine receptors and TRPM2 channels.</p>
    Color and Shape:Liquid
  • Homocarnosine TFA


    <p>Homocarnosine TFA: brain-exclusive GABA-histidine dipeptide, neuronal, anticonvulsant, antioxidant, anti-inflammatory.</p>
    Formula:C12H17F3N4O5
    Color and Shape:Solid
    Molecular weight:354.28
  • Rapastinel acetate

    CAS:
    Rapastinel acetate is a modulator of N-methyl-D-aspartate (NMDA) receptor and a partial agonist of glycine site long-lasting antidepressant effects.
    Formula:C20H35N5O8
    Purity:99.6%
    Color and Shape:Soild
    Molecular weight:473.52
  • (±)8(9)-EpETE

    CAS:
    <p>(±)8(9)-EpETE ((±)8,9-EEQ) is an epoxide of arachidonic acid biosynthesized by CYP450 epoxygenase.1.2 In rat and rabbit liver microsomes.</p>
    Formula:C20H30O3
    Color and Shape:Solid
    Molecular weight:318.45
  • ShK-Dap22

    CAS:
    Potent KV1.3 channel blocker; Kd 23 pM; selective; inhibits T cell activation; IC50 < 500 pM for mKV1.3.
    Formula:C166H268N54O48S7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4012.7
  • Withasomniferolide B

    CAS:
    <p>Withasomniferolide B, a withanolide from Withania somnifera root, activates GABAA receptors.</p>
    Formula:C28H36O4
    Color and Shape:Solid
    Molecular weight:436.58
  • ML353


    <p>ML353 activates TREK-1/2, binds mGlu5 SAM (Ki=18.2 nM), surpasses 5mpep, may address SAM activity/blocking.</p>
    Formula:C19H15FN2O
    Purity:99.98% - 99.98%
    Color and Shape:Soild
    Molecular weight:306.33
  • Sinapine hydroxide

    CAS:
    <p>Sinapine hydroxide from crucifer seeds has anti-inflammatory, anti-oxidant, anti-tumor properties, and inhibits AChE, aiding neurodegenerative research.</p>
    Formula:C16H25NO6
    Color and Shape:Solid
    Molecular weight:327.377
  • Guangxitoxin 1E

    CAS:
    <p>Guangxitoxin 1E acts as a gating modifier since it shifts the voltage-dependence of Kv2.1 K+ currents towards depolarized potentials.</p>
    Formula:C178H248N44O45S7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3948.61
  • GeX-2

    CAS:
    <p>GeX-2 is a truncated analogue of αO-conotoxin. It has the ability to activate GABAB receptors and inhibit α9α10nAChR as well as CaV2.2 channels. Additionally, GeX-2 is effective in alleviating pain in a rat model of chronic constriction injury.</p>
    Formula:C103H169N43O27
    Color and Shape:Solid
    Molecular weight:2441.72
  • Albanin A


    <p>Albanin A is a useful organic compound for research related to life sciences and the catalog number is T124310.</p>
    Formula:C20H18O6
    Color and Shape:Solid
    Molecular weight:354.358
  • Nitrazolam

    CAS:
    <p>Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.</p>
    Formula:C17H13N5O2
    Color and Shape:Solid
    Molecular weight:319.32
  • Digoxigenin Monodigitoxoside

    CAS:
    <p>Digoxigenin monodigitoxoside is a cardiac glycoside metabolite of digoxin and a Na+/K+ ATPase inhibitor.</p>
    Formula:C29H44O8
    Color and Shape:Solid
    Molecular weight:520.663
  • L-689560

    CAS:
    L-689560, a radiolabeled ligand, studies NMDA receptors, is an antagonist at GluN1 glycine site.
    Formula:C17H15Cl2N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:380.23
  • Conantokin G TFA


    <p>Conantokin G TFA, a 17-aa peptide, blocks NMDA receptors with 480 nM IC50 and is neuroprotective.</p>
    Formula:C90H139F3N26O46
    Color and Shape:Solid
    Molecular weight:2378.21