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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2290 products of "Membrane Transporter/Ion Channel"

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  • Adjudin

    CAS:
    <p>Adjudin (AF-2364) is a small molecule compound known to possess antispermatogenic function, attenuates microglia activation by suppression of the NF-κB pathway.</p>
    Formula:C15H12Cl2N4O
    Purity:96.51% - ≥95%
    Color and Shape:Solid
    Molecular weight:335.19
  • SG-209

    CAS:
    <p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>
    Formula:C10H12N2O3
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:208.21
  • Almitrine mesylate

    CAS:
    <p>Almitrine mesylate targets Ca2+-dependent K+ channels in rat cells, used for chronic lung hypoxemia.</p>
    Formula:C28H37F2N7O6S2
    Purity:99.96%
    Color and Shape:Coa
    Molecular weight:669.76
  • AZ194

    CAS:
    <p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>
    Formula:C34H31F2N3O3
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:567.62
  • Tetrabenazine methanesulfonate

    CAS:
    <p>Tetrabenazine methanesulfonate: ex-antipsychotic/therapy for movement disorders, blocks neurotransmitter uptake, labels vesicle transport.</p>
    Formula:C20H31NO6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:413.53
  • Miltirone

    CAS:
    <p>Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.</p>
    Formula:C19H22O2
    Purity:99.22% - 99.66%
    Color and Shape:Solid
    Molecular weight:282.38
  • α-Asarone

    CAS:
    <p>alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.</p>
    Formula:C12H16O3
    Purity:99.64% - 99.64%
    Color and Shape:Monoclinic Needles From Water Monoclinic Needles From Water
    Molecular weight:208.25
  • Raxatrigine

    CAS:
    Raxatrigine (CNV 1014802) has been investigated for the treatment of Bipolar Disorder and Bipolar Depression.
    Formula:C18H19FN2O2
    Purity:98% - 99.43%
    Color and Shape:Solid
    Molecular weight:314.35
  • Baclofen hydrochloride

    CAS:
    Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.
    Formula:C10H13Cl2NO2
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:250.122
  • Zosuquidar trihydrochloride

    CAS:
    <p>Zosuquidar trihydrochloride (LY-335979 trihydrochloride) is a potent modulator of P-glycoprotein-mediated multi-drug resistance with Ki of 60 nM. Phase 3.</p>
    Formula:C32H31F2N3O2·3HCl
    Purity:99.49% - >99.99%
    Color and Shape:Solid
    Molecular weight:636.99
  • Raxatrigine hydrochloride

    CAS:
    Raxatrigine hydrochloride is a state-dependent sodium channel blocker and a Nav1.7 sodium channel inhibitor.
    Formula:C18H20ClFN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:350.82
  • Ataluren

    CAS:
    <p>Ataluren (PTC124) is a novel, orally administered drug that targets nonsense mutations.</p>
    Formula:C15H9FN2O3
    Purity:99.16% - 99.84%
    Color and Shape:Solid
    Molecular weight:284.24
  • Cyclothiazide

    CAS:
    <p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>
    Formula:C14H16ClN3O4S2
    Purity:98.23% - 99.49%
    Color and Shape:Crystals From Dilute Alcohol Solid
    Molecular weight:389.88
  • PF-05186462

    CAS:
    <p>PF-05186462 (PF-05150122) is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5.</p>
    Formula:C19H10ClF4N5O3S2
    Purity:99.10% - 99.37%
    Color and Shape:Solid
    Molecular weight:531.89
  • Guanosine 5'-diphosphate disodium salt

    CAS:
    <p>5'-GDP-Na2: a nucleoside diphosphate, iron mobilizer, blocks hepcidin-ferroportin, affects IL-6/stat-3.</p>
    Formula:C10H13N5Na2O11P2
    Purity:99.40%
    Color and Shape:White Powder
    Molecular weight:487.16
  • AM92016

    CAS:
    <p>AM92016 is a specific blocker of the time dependent delayed rectifier potassium current. AM92016 does not show any β-adrenoceptor blocking activity.</p>
    Formula:C26H30Cl2N2O6S
    Color and Shape:Solid
    Molecular weight:569.49
  • SAR7334 hydrochloride

    CAS:
    <p>SAR7334 hydrochloride is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).</p>
    Formula:C21H24Cl3N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.79
  • Ivacaftor

    CAS:
    <p>Ivacaftor (VX-770) (VX-770) is a potentiator of CFTR targeting G551D-CFTR (EC50: 100 nM) and F508del-CFTR (EC50: 25 nM) in Fisher rat thyroid cells,</p>
    Formula:C24H28N2O3
    Purity:99% - 99.98%
    Color and Shape:Solid
    Molecular weight:392.49
  • Tiagabine hydrochloride hydrate

    CAS:
    <p>Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.</p>
    Formula:C20H28ClNO3S2
    Color and Shape:Solid
    Molecular weight:430.02
  • Rbin-1

    CAS:
    <p>Rbin-1 (Ribozinoindole-1) is a potent,specific inhibitor of eukaryotic ribosome biogenesis.</p>
    Formula:C13H12N4S
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:256.33