Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(93 products)
- Adiponectin receptor(5 products)
- CFTR(64 products)
- CGRP Receptor(52 products)
- Calcium Channel(496 products)
- Chloride channel(49 products)
- GABA Receptor(337 products)
- Monoamine Transporter(23 products)
- Monocarboxylate transporter(17 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(8 products)
- OAT(27 products)
- OCT(7 products)
- P-gp(53 products)
- Potassium Channel(277 products)
- Proton pump(39 products)
- SGLT(30 products)
- Sodium Channel(202 products)
- TRP/TRPV Channel(93 products)
Show 13 more subcategories
Found 2293 products of "Membrane Transporter/Ion Channel"
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Quadrol
CAS:<p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>Formula:C14H32N2O4Purity:99.91% - 99.92%Color and Shape:Viscous Liquid Liquid ViscousMolecular weight:292.41Parimifasor
CAS:<p>Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.</p>Formula:C18H11Cl2F4N5OPurity:96.77% - 98.97%Color and Shape:SolidMolecular weight:460.21TKIM
CAS:<p>TKIM is a TWIK-related potassium channel 1 (TREK-1) inhibitor, binding to the pocket of the intermediate (IM) state of TREK-1.</p>Formula:C18H14ClN3O2SPurity:99.47%Color and Shape:SolidMolecular weight:371.84Budipine
CAS:Budipine is a low affinity, N-methyl-D-aspartate receptor antagonist,is an antiparkinsonian agent.Formula:C21H27NPurity:99.64%Color and Shape:SolidMolecular weight:293.45Guan-fu base A hydrochloride(1394-48-5 free base)
CAS:<p>Guanfu base A HCl, an antiarrhythmic from Aconitum coreanum, inhibits CYP2D6 in humans, monkeys, and dogs.</p>Formula:C24H32NO6ClPurity:99.9%Color and Shape:SolidMolecular weight:465.972'-O-Methylisoliquiritigenin
CAS:<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Formula:C16H14O4Purity:98.75%Color and Shape:SolidMolecular weight:270.28Cis-ACBD
CAS:<p>Cis-ACBD (cis-1-aminocyclobutane-1,3-dicarboxylic acid) is a potent and selective N-methyl-D-aspartate receptor agonist.</p>Formula:C6H9NO4Purity:99.77%Color and Shape:SolidMolecular weight:159.14DL-Willardiine
CAS:<p>DL-Willardiine (2-amino-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoic acid) is an unnatural amino acid, a derivative of glutamate.</p>Formula:C7H9N3O4Purity:99.83%Color and Shape:SolidMolecular weight:199.16Esomeprazole Magnesium
CAS:<p>Esomeprazole Magnesium (NEXIUM) is the S-isomer of omeprazole, can reduce gastric acid secretion with selective and irreversible proton pump inhibitor activity.</p>Formula:C34H36MgN6O6S2Purity:98.76% - 99.73%Color and Shape:SolidMolecular weight:713.12Eperisone hydrochloride
CAS:<p>Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.</p>Formula:C17H26ClNOPurity:99.80%Color and Shape:White Or Similar To White Crystalline Powder With Peculiar Smell And Bitter TasteMolecular weight:295.85AER-271
CAS:<p>AER-271 is an inhibitor of aquaporin-4.</p>Formula:C15H9ClF6NO5PPurity:97.45%Color and Shape:SolidMolecular weight:463.65Ibutilide
CAS:<p>Ibutilide (U70226E) is an antiarrhythmic that prolongs action potential by blocking I Kr in AT-1 cells.</p>Formula:C20H36N2O3SColor and Shape:SolidMolecular weight:384.58A2793
CAS:<p>A2793 is a dual inhibitor of TWIK-associated acid-sensitive K+ channel 1 (TASK-1)/TRESK, with an IC50 for mTRESK of 6.8 μM.</p>Formula:C13H12ClNO3Purity:98.54%Color and Shape:SolidMolecular weight:265.69Pilsicainide
CAS:<p>Pilsicainide (SUN 1165 free acid) is a potent class Ic antiarrhythmic agent. Pilsicainide is a potent sodium channel blocker[1][2].</p>Formula:C17H24N2OColor and Shape:SolidMolecular weight:272.39Ilaprazole sodium
CAS:<p>Ilaprazole sodium (IY-81149 sodium) , a substituted benzimidazole prodrug, is a selective and irreversible proton pump inhibitor.</p>Formula:C19H17N4NaO2SPurity:99.06%Color and Shape:SolidMolecular weight:388.42Mitiglinide calcium hydrate
CAS:<p>Mitiglinide calcium hydrate (S-21403 calcium hydrate) is a drug for the treatment of type 2 diabetes.</p>Formula:C38H52CaN2O8Purity:98.97% - 99.96%Color and Shape:White SolidMolecular weight:704.91Tiagabine
CAS:<p>Tiagabine (NO050328) is an Anti-epileptic Agent.</p>Formula:C20H25NO2S2Purity:99.25%Color and Shape:White To Off-White Crystalline SolidMolecular weight:375.55Ocinaplon
CAS:<p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>Formula:C17H11N5OPurity:99.81%Color and Shape:SolidMolecular weight:301.37-Chlorokynurenic acid sodium salt
CAS:<p>7-CKA sodium salt: NMDA receptor antagonist, glycine B site (IC50: 0.56 μM), blocks glutamate reuptake (Ki: 0.59 μM).</p>Formula:C10H6ClNNaO3Color and Shape:SolidMolecular weight:246.6(-)-Blebbistatin
CAS:<p>(-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin II inhibitor with IC50 ranging from 0.5 to 5 μM.</p>Formula:C18H16N2O2Purity:99.38% - 99.61%Color and Shape:SolidMolecular weight:292.33Metaflumizone
CAS:<p>Metaflumizone (BAS-320I) is a sodium channel blocker insecticide.</p>Formula:C24H16F6N4O2Purity:98.73%Color and Shape:SolidMolecular weight:506.40LY 303511 hydrochloride
CAS:<p>LY 303511 hydrochloride is a potent mTOR inhibitor</p>Formula:C19H19ClN2O2Purity:98.47%Color and Shape:SolidMolecular weight:342.82NBI-98782
CAS:<p>NBI-98782 ((+)-α-DHTBZ) is an inhibtior of vesicular monoamine transporter (VMAT2) (Ki: 0.97 nM)</p>Formula:C19H29NO3Purity:99.29%Color and Shape:SolidMolecular weight:319.44SG-209
CAS:<p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>Formula:C10H12N2O3Purity:99.84%Color and Shape:SolidMolecular weight:208.21Ropivacaine hydrochloride monohydrate
CAS:<p>Ropivacaine hydrochloride monohydrate (LEA-103 HCl) is an anaesthetic agent and blocks impulse conduction through inhibiting sodium ion influx reversibly.</p>Formula:C17H29ClN2O2Purity:99.94% - 99.95%Color and Shape:White SolidMolecular weight:328.88Arecaidine hydrochloride
CAS:Arecaidine hydrochloride may have carcinogenesis.Formula:C7H12ClNO2Purity:99.69% - ≥95%Color and Shape:SolidMolecular weight:177.63AZ194
CAS:<p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>Formula:C34H31F2N3O3Purity:99.61%Color and Shape:SolidMolecular weight:567.62Neboglamine
CAS:<p>Neboglamine, a glycine NMDA-associated agonist, is used potentially for the treatment of schizophrenia.</p>Formula:C13H24N2O3Purity:98%Color and Shape:SolidMolecular weight:256.34Lansoprazole sulfone
CAS:<p>Lansoprazole sulfone is a metabolite of the gastric pump inhibitor Lansoprazole.</p>Formula:C16H14F3N3O3SPurity:99.67%Color and Shape:SolidMolecular weight:385.36Ralfinamide mesylate
CAS:<p>Ralfinamide mesylate (FCE-26742A (mesylate)) is an orally available Na+ channel blocker.</p>Formula:C18H23FN2O5SPurity:99.83%Color and Shape:SolidMolecular weight:398.45DAAO inhibitor-1
CAS:<p>DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor (IC50: 0.12 μM).</p>Formula:C7H5FN2OPurity:97.84%Color and Shape:SolidMolecular weight:152.13MDR-652
CAS:<p>MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1) with Ki value of 11.4 nM and 23.8 nM for</p>Formula:C22H23ClFN3O2SPurity:99.96%Color and Shape:SolidMolecular weight:447.95Kv2-IN-A1
CAS:<p>Kv2-IN-A1 is an inhibitor of Kv2.1 and Kv2.2.</p>Formula:C20H17ClN4OSPurity:98.83%Color and Shape:SolidMolecular weight:396.89Esomeprazole hemistrontium
CAS:<p>Esomeprazole hemistrontium, potent oral proton pump inhibitor, reduces gastric acid by blocking H+, K+-ATPase.</p>Formula:C34H36N6O6S2SrColor and Shape:SolidMolecular weight:776.44Adjudin
CAS:<p>Adjudin (AF-2364) is a small molecule compound known to possess antispermatogenic function, attenuates microglia activation by suppression of the NF-κB pathway.</p>Formula:C15H12Cl2N4OPurity:96.51% - ≥95%Color and Shape:SolidMolecular weight:335.19Almitrine mesylate
CAS:<p>Almitrine mesylate targets Ca2+-dependent K+ channels in rat cells, used for chronic lung hypoxemia.</p>Formula:C28H37F2N7O6S2Purity:99.96%Color and Shape:CoaMolecular weight:669.76Miltirone
CAS:<p>Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.</p>Formula:C19H22O2Purity:99.22% - 99.66%Color and Shape:SolidMolecular weight:282.38WS-12
CAS:WS-12 is a potent TRPM8 agonist that acts as a cooling agent (EC50 : 193 nM)Formula:C18H27NO2Purity:99.99%Color and Shape:Whitish To White Solid CrystallineMolecular weight:289.41α-Asarone
CAS:<p>alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.</p>Formula:C12H16O3Purity:99.64% - 99.64%Color and Shape:Monoclinic Needles From Water Monoclinic Needles From WaterMolecular weight:208.254-Acetamidobutanoic acid
CAS:<p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>Formula:C6H11NO3Purity:98.51%Color and Shape:SolidMolecular weight:145.16Baclofen hydrochloride
CAS:Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.Formula:C10H13Cl2NO2Purity:99.55%Color and Shape:SolidMolecular weight:250.122Raxatrigine hydrochloride
CAS:Raxatrigine hydrochloride is a state-dependent sodium channel blocker and a Nav1.7 sodium channel inhibitor.Formula:C18H20ClFN2O2Purity:98%Color and Shape:SolidMolecular weight:350.82Ataluren
CAS:<p>Ataluren (PTC124) is a novel, orally administered drug that targets nonsense mutations.</p>Formula:C15H9FN2O3Purity:99.16% - 99.84%Color and Shape:SolidMolecular weight:284.24Cyclothiazide
CAS:<p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>Formula:C14H16ClN3O4S2Purity:98.23% - 99.49%Color and Shape:Crystals From Dilute Alcohol SolidMolecular weight:389.88Flecainide hydrochloride
CAS:<p>Flecainide is a medication used to prevent and treat abnormally fast heart rates. This includes ventricular and supraventricular tachycardias.</p>Formula:C17H21ClF6N2O3Purity:97.79%Color and Shape:SolidMolecular weight:450.81PF-05186462
CAS:<p>PF-05186462 (PF-05150122) is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5.</p>Formula:C19H10ClF4N5O3S2Purity:99.10% - 99.37%Color and Shape:SolidMolecular weight:531.89Guanosine 5'-diphosphate disodium salt
CAS:<p>5'-GDP-Na2: a nucleoside diphosphate, iron mobilizer, blocks hepcidin-ferroportin, affects IL-6/stat-3.</p>Formula:C10H13N5Na2O11P2Purity:99.40%Color and Shape:White PowderMolecular weight:487.16Trofinetide
CAS:Trofinetide (NNZ-2566) is a synthetic analog of the endogenous N-terminus tripeptide. It has been shown to be neuroprotective in animal models of brain injury.Formula:C13H21N3O6Purity:98.70% - 99.50%Color and Shape:SolidMolecular weight:315.326-Methylflavone
CAS:6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.Formula:C16H12O2Purity:99.69%Color and Shape:SolidMolecular weight:236.27Nateglinide
CAS:<p>Nateglinide is an oral drug for type 2 diabetes, stimulating insulin release; may cause rare acute liver injury.</p>Formula:C19H27NO3Purity:99.93% - 99.94%Color and Shape:White Crystalline PowderMolecular weight:317.42
