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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2293 products of "Membrane Transporter/Ion Channel"

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  • DS1
    Targetmol
    + Info

    DS1

    CAS:
    <p>DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.</p>
    Formula:C18H10Br2ClN3OS
    Color and Shape:Solid
    Molecular weight:511.62

    Ref: TM-T71848

  • Sodium Channel inhibitor 1
    Targetmol
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    Sodium Channel inhibitor 1

    CAS:
    Sodium Channel inhibitor1 is a novel and selective voltage-gated sodium channel for pain treatment.
    Formula:C24H19F4N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:473.42

    Ref: TM-T12948

  • VU625
    Targetmol
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    VU625

    CAS:
    <p>VU625 (VU007625) is an AeKir1 inhibitor (IC50: 96.8nM) that acts as a mosquito killer and inhibits AeKir1-mediated currents.</p>
    Formula:C19H22N2O4S
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:374.45

    Ref: TM-T24948

  • Terodiline
    Targetmol
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    Terodiline

    CAS:
    <p>Terodiline is an orally available selective muscarinic M1 receptor and calcium channel antagonist for the study of diseases caused by abnormal bladder function.</p>
    Formula:C20H27N
    Purity:98.20% - 99.59%
    Color and Shape:Solid
    Molecular weight:281.44

    Ref: TM-T60536

  • Asivatrep
    Targetmol
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    Asivatrep

    CAS:
    <p>Asivatrep (PAC14028) is a selective and potent antagonist of transient receptor potential vanilloid subtype 1 (TRPV1) for the study of atopic dermatitis.</p>
    Formula:C21H22F5N3O3S
    Purity:95.13%
    Color and Shape:Solid
    Molecular weight:491.48

    Ref: TM-T16426

  • AMG9678
    Targetmol
    + Info

    AMG9678

    CAS:
    <p>AMG9678 is a selective, potent, orally active TRPM8 antagonist (IC50: 31.2 nM).</p>
    Formula:C20H18F6N2O
    Color and Shape:Solid
    Molecular weight:416.36

    Ref: TM-T62158

  • Topiramate lithium
    Targetmol
    + Info

    Topiramate lithium

    CAS:
    <p>Topiramate lithium: antiepileptic, GluR5 antagonist, enhances GABA, inhibits kainate/AMPA, Na+/Ca2+ channels; ↑ K+ conductance; ↓ carbonic anhydrase.</p>
    Formula:C12H20LiNO8S
    Color and Shape:Solid
    Molecular weight:345.29

    Ref: TM-T61145

  • MC-70
    Targetmol
    + Info

    MC-70

    CAS:
    <p>MC-70 is a potent P-glycoprotein (P-gp) inhibitor (EC50 = 0.69 μM).</p>
    Formula:C24H25NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:375.46

    Ref: TM-T27985

  • ORM-10962
    Targetmol
    + Info

    ORM-10962

    CAS:
    ORM-10962 is a potent, highly selective inhibitor of sodium-calcium exchanger (NCX) (for the reverse and forward mode inhibition with IC50 values of 67 and 55
    Formula:C27H29N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:459.54

    Ref: TM-T12322

  • Caldaret
    Targetmol
    + Info

    Caldaret

    CAS:
    <p>Caldaret is an intracellular Ca2+ handling modulator that acts through reverse mode Na+/Ca2+ exchanger inhibition.</p>
    Formula:C11H16N2O3S
    Color and Shape:Solid
    Molecular weight:256.32

    Ref: TM-T14857

  • UBP 296
    Targetmol
    + Info

    UBP 296

    CAS:
    <p>GluR5-subunit containing kainate receptor antagonist</p>
    Formula:C15H15N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:333.3

    Ref: TM-T23488

  • Y 23684
    Targetmol
    + Info

    Y 23684

    CAS:
    <p>Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.</p>
    Formula:C18H13ClN2O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.83

    Ref: TM-T24367

  • Nav1.7-IN-3
    Targetmol
    + Info

    Nav1.7-IN-3

    CAS:
    <p>Nav1.7-IN-3 is a selective and orally bioavailable inhibitor of voltage-gated sodium channel Nav1.7(IC50 of 8 nM).</p>
    Formula:C17H20ClFN4O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.95

    Ref: TM-T12183

  • CGP 46381
    Targetmol
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    CGP 46381

    CAS:
    <p>CGP 46381 is a GABAB receptor antagonist.</p>
    Formula:C10H22NO2P
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:219.26

    Ref: TM-T22649

  • YS-201
    Targetmol
    + Info

    YS-201

    CAS:
    <p>YS-201 is an antagonist of dihydropyridine-type calcium channel.</p>
    Formula:C24H31N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:457.52

    Ref: TM-T17277

  • IEM 1460
    Targetmol
    + Info

    IEM 1460

    CAS:
    <p>AMPA receptors blocker</p>
    Formula:C19H38Br2N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.33

    Ref: TM-T22854

  • (S)-ML753286
    Targetmol
    + Info

    (S)-ML753286

    CAS:
    (S)-ML753286 is a breast cancer resistance protein (BCRP) inhibitor (IC50: 0.6 μM on BCRP efflux transporter).
    Formula:C20H25N3O3
    Color and Shape:Solid
    Molecular weight:355.43

    Ref: TM-T10490

  • Indantadol HCl
    Targetmol
    + Info

    Indantadol HCl

    CAS:
    Indantadol HCl (CHF-3381) is a NMDA antagonist and nonselective MAO inhibitor.
    Formula:C11H15ClN2O
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:226.7

    Ref: TM-T27606

  • GABAA receptor agent 5
    Targetmol
    + Info

    GABAA receptor agent 5

    CAS:
    <p>Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.</p>
    Formula:C21H25N3O2S
    Color and Shape:Solid
    Molecular weight:383.51

    Ref: TM-T61668

  • CP-409092 hydrochloride
    Targetmol
    + Info

    CP-409092 hydrochloride

    CAS:
    <p>CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.</p>
    Formula:C17H20ClN3O2
    Color and Shape:Solid
    Molecular weight:333.81

    Ref: TM-T10869

  • BGT1-IN-9
    Targetmol
    + Info

    BGT1-IN-9

    CAS:
    <p>BGT1-IN-9 is an M1 muscarinic agonist.</p>
    Formula:C5H10ClN3O2
    Color and Shape:Solid
    Molecular weight:179.605

    Ref: TM-T23787

  • Atomoxetine
    Targetmol
    + Info

    Atomoxetine

    CAS:
    <p>Atomoxetine (HSDB 7352) is a selective norepinephrine inhibitor that may cause an increase in blood pressure by increasing norepinephrine concentrations in</p>
    Formula:C17H21NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:255.35

    Ref: TM-T20886

  • Flordipine
    Targetmol
    + Info

    Flordipine

    CAS:
    <p>Flordipine is used as a calcium channel blocker.</p>
    Formula:C26H33F3N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:510.55

    Ref: TM-T25425

  • Omeprazole magnesium
    Targetmol
    + Info

    Omeprazole magnesium

    CAS:
    <p>Omeprazole magnesium: oral PPI that reduces stomach acid, treats acid reflux and heartburn.</p>
    Formula:C34H36MgN6O6S2
    Color and Shape:Solid
    Molecular weight:713.12

    Ref: TM-T68250

  • Ro 04-5595 hydrochloride
    Targetmol
    + Info

    Ro 04-5595 hydrochloride

    CAS:
    NR2B-containing NMDA receptors antagonist
    Formula:C19H23Cl2NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:368.3

    Ref: TM-T23239

  • TTA-Q6(isomer)
    Targetmol
    + Info

    TTA-Q6(isomer)

    CAS:
    TTA-Q6(isomer) is an isomer of TTA-Q6. TTA-Q6 is a selective antagonist of the T-type Ca2+ channel.
    Formula:C20H15ClF3N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:405.8

    Ref: TM-T13220

  • Apimostinel
    Targetmol
    + Info

    Apimostinel

    CAS:
    <p>Apimostinel (NRX-1074; AGN-241660) is a partial agonist of NMDA receptor.</p>
    Formula:C25H37N5O6
    Color and Shape:Solid
    Molecular weight:503.59

    Ref: TM-T14306

  • NMDA receptor antagonist 4
    Targetmol
    + Info

    NMDA receptor antagonist 4

    CAS:
    <p>NMDA antagonist 4 (IIc) is an oral, voltage-dependent blocker with IC50 of 1.93 μM and may penetrate the BBB, useful in Alzheimer's research.</p>
    Formula:C15H18FN
    Color and Shape:Solid
    Molecular weight:231.31

    Ref: TM-T60306

  • Istaroxime
    Targetmol
    + Info

    Istaroxime

    CAS:
    <p>Istaroxime is an effective inhibitor of Na+, K+-ATPase (IC50: 0.11 μM).</p>
    Formula:C21H32N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:360.49

    Ref: TM-T15600

  • JNJ-56022486
    Targetmol
    + Info

    JNJ-56022486

    CAS:
    <p>JNJ-56022486 is a selective TARP γ‑8 AMPA receptor modulator.</p>
    Formula:C15H10ClN3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:283.71

    Ref: TM-T25559

  • KCa1.1 channel activator-2
    Targetmol
    + Info

    KCa1.1 channel activator-2

    <p>KCa1.1 channel activator-2, a Quercetin hybrid, selectively stimulates vascular KCa1.1 channel, with strong myorelaxant effects.</p>
    Formula:C23H22O8S2
    Color and Shape:Solid
    Molecular weight:490.55

    Ref: TM-T72195

  • PPDA
    Targetmol
    + Info

    PPDA

    CAS:
    <p>Subtype-selective NMDA receptor antagonist</p>
    Formula:C21H18N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:378.38

    Ref: TM-T23179

  • (R)-3C4HPG
    Targetmol
    + Info

    (R)-3C4HPG

    CAS:
    <p>NMDA and AMPA/kainate receptor antagonist</p>
    Formula:C9H9NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:211.17

    Ref: TM-T23216

  • GoSlo-SR-5-69
    Targetmol
    + Info

    GoSlo-SR-5-69

    CAS:
    <p>BK channel activator (EC50 = 251 nM). Shifts the voltage required for half maximal negatively (DV1/2 = -104 mV).</p>
    Formula:C24H20N2NaO5S
    Color and Shape:Solid
    Molecular weight:471.48

    Ref: TM-T37294

  • Hyperforin dicyclohexylammonium salt
    Targetmol
    + Info

    Hyperforin dicyclohexylammonium salt

    CAS:
    Hyperforin dicyclohexylammonium is a TRPC6 activator and antidepressant that modulates Ca2+ levels.
    Formula:C47H75NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:718.10

    Ref: TM-T15541

  • TRPC6-IN-2
    Targetmol
    + Info

    TRPC6-IN-2

    CAS:
    <p>TRPC6-IN-2 is a TRPC protein inhibitor, specifically inhibiting TRPC6 protein.</p>
    Formula:C19H17Cl2FN6
    Color and Shape:Solid
    Molecular weight:419.28

    Ref: TM-T62201

  • Metapramine
    Targetmol
    + Info

    Metapramine

    CAS:
    Metapramine, a tricyclic antidepressant, blocks norepinephrine reuptake and is a low-affinity NMDA antagonist.
    Formula:C16H18N2
    Purity:99.03% - 99.67%
    Color and Shape:Solid
    Molecular weight:238.33

    Ref: TM-T60330

  • SB-237376 HCl
    Targetmol
    + Info

    SB-237376 HCl

    CAS:
    <p>SB-237376 HCl (SB-237376 hydrochloride) is a calcium and potassium channel antagonist used in the treatment of cardiac arrhythmias.</p>
    Formula:C20H26ClN3O5
    Purity:98.70%
    Color and Shape:Solid
    Molecular weight:423.89

    Ref: TM-T28686

  • GNE-5729
    Targetmol
    + Info

    GNE-5729

    CAS:
    <p>GNE-5729 is a positive allosteric modulator of NMDAR blood-brain barrier orally available, GluN2A, GluN2C and GluN2D, neurological and psychiatric disorders.</p>
    Formula:C17H10Cl2F3N5O
    Purity:99.40% - 99.85%
    Color and Shape:Solid
    Molecular weight:428.2

    Ref: TM-T15408

  • JNc-440
    Targetmol
    + Info

    JNc-440

    CAS:
    <p>JNc-440, a strong anti-hypertensive, boosts TRPV4-KCa2.3 interaction and vasodilation, lowering blood pressure in mice.</p>
    Formula:C26H24N4O3
    Color and Shape:Solid
    Molecular weight:440.49

    Ref: TM-T62543

  • ML252
    Targetmol
    + Info

    ML252

    CAS:
    <p>ML252 selectively inhibits KCNQ2 (IC50=69nM) and Cytochrome P450 isoforms CYP1A2, CYP2C9, CYP3A4, CYP2D6 with low nanomolar IC50s.</p>
    Formula:C20H24N2O
    Color and Shape:Solid
    Molecular weight:308.42

    Ref: TM-T70786

  • XPC-6444
    Targetmol
    + Info

    XPC-6444

    CAS:
    <p>XPC-6444 is a isoform-selective, and CNS-penetrant inhibitor of NaV1.6 with IC50 of41 nM for hNaV1.6,with anticonvulsant activity.</p>
    Formula:C22H25F3N4O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:498.58

    Ref: TM-T13359

  • (BrMT)2
    Targetmol
    + Info

    (BrMT)2

    CAS:
    <p>(BrMT)2 is an activator of the Kv1.1 potassium ion channel.</p>
    Formula:C20H20Br2N4S2
    Color and Shape:Solid
    Molecular weight:540.34

    Ref: TM-T26372

  • RPR-260243
    Targetmol
    + Info

    RPR-260243

    CAS:
    <p>RPR-260243 is a novel activator of HERG and modifies HERG currents inhibited by dofetilide (IC50 = 58 nM).</p>
    Formula:C28H25F3N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:510.5

    Ref: TM-T16796

  • β-CCB
    Targetmol
    + Info

    β-CCB

    CAS:
    <p>benzodiazepine receptor ligand</p>
    Formula:C16H16N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:268.31

    Ref: TM-T22602

  • UCL-1848 trifluoroacetate salt
    Targetmol
    + Info

    UCL-1848 trifluoroacetate salt

    CAS:
    <p>UCL-1848 trifluoroacetate salt is a selective Ca2+-activated, SK potassium channel blocker.</p>
    Formula:C32H34F6N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:652.638

    Ref: TM-T29042

  • UBP714
    Targetmol
    + Info

    UBP714

    CAS:
    UBP714, derived from UBP608, boosts NMDAR in CA1 hippocampus, promising for schizophrenia and cognitive deficits treatment.
    Formula:C11H7BrO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:283.07

    Ref: TM-T24919

  • ZD-9379
    Targetmol
    + Info

    ZD-9379

    CAS:
    <p>ZD-9379 is a NMDA receptor antagonist.</p>
    Formula:C19H14ClN3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:383.79

    Ref: TM-T23559

  • Ro 8-4304 hydrochloride
    Targetmol
    + Info

    Ro 8-4304 hydrochloride

    CAS:
    <p>Ro 8-4304 hydrochloride is a NMDA receptor antagonist.</p>
    Formula:C21H24ClFN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:406.88

    Ref: TM-T23249

  • YM 244769 hydrochloride
    Targetmol
    + Info

    YM 244769 hydrochloride

    CAS:
    <p>inhibitor of the reverse mode of Na+/Ca2+ exchange (NCX)</p>
    Formula:C26H23ClFN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:479.93

    Ref: TM-T23546