Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(100 products)
- Adiponectin receptor(5 products)
- CFTR(66 products)
- CGRP Receptor(54 products)
- Calcium Channel(545 products)
- Chloride channel(53 products)
- GABA Receptor(369 products)
- Monoamine Transporter(30 products)
- Monocarboxylate transporter(18 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(10 products)
- OAT(32 products)
- OCT(7 products)
- P-gp(55 products)
- Potassium Channel(283 products)
- Proton pump(41 products)
- SGLT(31 products)
- Sodium Channel(219 products)
- TRP/TRPV Channel(96 products)
Show 13 more subcategories
Found 2586 products of "Membrane Transporter/Ion Channel"
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RS 30026
CAS:RS 30026 is a potent calcium channel agonist.Formula:C23H21NO4SColor and Shape:SolidMolecular weight:407.48(S)-Propafenone
CAS:(S)-Propafenone, or (S)-SA-79, is an S-enantiomer with beta-blocking effects and sodium channel blocking class 1 antiarrhythmic properties.Formula:C21H27NO3Purity:98%Color and Shape:SolidMolecular weight:341.44GYKI-52466
CAS:GYKI-52466: non-competitive AMPA antagonist, IC50: 10-20 μM for AMPA. Also relaxes muscles, treats seizures, neuroprotects, reduces anxiety.Formula:C17H15N3O2Purity:98%Color and Shape:SolidMolecular weight:293.32Taplucainium chloride
CAS:Taplucainium chloride is a sodium channel blocker with applications as a pain reliever.Formula:C23H31ClN2OColor and Shape:SolidMolecular weight:386.96SX-3228
CAS:SX-3228 is a selective agonist of benzodiazepine1 (BZ1) receptor(IC50 of 17 nM).Formula:C18H18N4O3Purity:98%Color and Shape:SolidMolecular weight:338.36GX-936
CAS:GX-936, Selective Nav1.7 inhibitor, binds activated VSD4 to oppose inactivation, for pain perception research.Formula:C24H20F3N7O3S2Purity:98%Color and Shape:SolidMolecular weight:575.59LY 97241
CAS:LY 97241 is an inhibitor of hEAG1 and hERG1 potassium channel.Formula:C19H32N2O2Color and Shape:SolidMolecular weight:320.47RPR104632
CAS:RPR104632 is a novel and potent antagonist located at the NMDA glycine site with neuroprotective activity.Formula:C15H11BrCl2N2O4SPurity:99.06%Color and Shape:SolidMolecular weight:466.13ITH-12575
CAS:ITH-12575 is an inhibitor of Mitochondrial Na+/Ca2+ exchange (mNCX). ITH12575 reduces Ca(2+) influx through CALHM1 at low micromolar concentrations.Formula:C18H18ClNOSColor and Shape:SolidMolecular weight:331.86ML218 hydrochloride
CAS:ML218 hydrochloride inhibits T-type Ca2+ channels Cav3.1-3.3; most effective on Cav3.2 and Cav3.3 (IC50s: 310 nM, 270 nM).Formula:C19H27Cl3N2OPurity:98%Color and Shape:SolidMolecular weight:405.79N-Methyl Duloxetine hydrochloride
CAS:N-Methyl Duloxetine hydrochloride elicits both tonic and use-dependent block of neuronal Na+ channels. N-Methyl Duloxetine hydrochloride is an analgesic.Formula:C19H22ClNOSPurity:98%Color and Shape:SolidMolecular weight:347.9Cyprodenate
CAS:Cyprodenate (Actebral) is a potent orally active brain-activating agent with appetite-suppressing properties, useful in studying metabolic.Formula:C13H25NO2Color and Shape:SolidMolecular weight:227.34Ref: TM-T72977
1mg38.00€5mg75.00€10mg105.00€25mg172.00€50mg242.00€100mg337.00€200mg498.00€1mL*10mM (DMSO)84.00€AZSMO-23
CAS:AZSMO-23 activates hERG K+ channels; blocks hKv4.3-hKChIP2.2, hCav3.2, hKv1.5; activates hCav1.2/β2/α2δ.Formula:C19H13ClN4OPurity:98%Color and Shape:SolidMolecular weight:348.79Halofantrine
CAS:Halofantrine: antimalarial, lipophilic, blocks HERG K+ channels, targets Chloroquine-resistant P. falciparum.Formula:C26H30Cl2F3NOColor and Shape:SolidMolecular weight:500.42Diltiazem malate
CAS:Diltiazem malate is an ACE inhibitor and non-dihydropyridine calcium channel blocker used in the treatment of hypertension.Formula:C26H32N2O9SColor and Shape:SolidMolecular weight:548.60(R)-Amlodipine
CAS:(R)-Amlodipine is the R-enantiomer of Amlodipine and functions as an orally active dihydropyridine calcium channel blocker with antianginal properties.Formula:C20H25ClN2O5Purity:99.977%Color and Shape:SolidMolecular weight:408.88U-7524
CAS:U-7524 (AOAA), an inhibitor of GABA-T and other PLP-dependent enzymes, disrupts the Schiff base linkage, forming oxime complexes.Formula:C2H5NO3Color and Shape:SolidMolecular weight:91.073-Methyl-GABA
CAS:3-Methyl-GABA activates GABA aminotransferase, fits GABAaR, stimulates GAD, and acts as an anticonvulsant.Formula:C20H30N2O10S2Purity:98%Color and Shape:SolidMolecular weight:522.59Ethyl dirazepate
CAS:Ethyl dirazepate has anxiolytic and hypnotic and possibly other characteristic benzodiazepine properties,is a drug which is a benzodiazepine derivative.Formula:C18H14Cl2N2O3Purity:98%Color and Shape:SolidMolecular weight:377.22UBP301
CAS:UBP301 is a kainate receptor antagonist.Formula:C15H14IN3O6Purity:98%Color and Shape:SolidMolecular weight:459.19Felbamate hydrate
CAS:Felbamate hydrate is an effective nonsedative anticonvulsant. It is a clinical effect that may be related to the inhibition of N-methyl-D-aspartate.Formula:C11H16N2O5Purity:98%Color and Shape:SolidMolecular weight:256.26Arbaclofen placarbil
CAS:Arbaclofen placarbil is a GABA(B) receptor agonist with better ADMET than R-baclofen, reducing postprandial reflux in GERD.Formula:C19H26ClNO6Color and Shape:SolidMolecular weight:399.87Carburazepam
CAS:Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.Formula:C17H16ClN3O2Purity:98%Color and Shape:SolidMolecular weight:329.78Cibenzoline
CAS:Cibenzoline: antiarrhythmic, blocks KATP channels, minimizes LVPG, useful in hypertrophic cardiomyopathy studies.Formula:C18H18N2Color and Shape:SolidMolecular weight:262.35URAT1&XO inhibitor 2
CAS:Compound BDEO (URAT1&XO inhibitor 2) serves as a dual-action inhibitor targeting both xanthine oxidase (XO) and URAT1, demonstrating an IC50 value of 3.3 μM forFormula:C14H12BrNO3Purity:98%Color and Shape:SolidMolecular weight:322.15TCS 1105
CAS:TCS 1105 is a GABAA BZR ligand, blocking Sema3A and altering mouse anxiety, aggression, and social dominance.Formula:C17H13FN2O2Purity:99.75%Color and Shape:SolidMolecular weight:296.3(R)-CPP
CAS:(R)-CPP is a NMDA antagonist.Formula:C8H17N2O5PPurity:98%Color and Shape:SolidMolecular weight:252.2PD-151307
CAS:PD-151307 is used as an N-type calcium channel blocker.Formula:C33H47N3O5Purity:98%Color and Shape:SolidMolecular weight:565.74SN05
CAS:SN05 inhibits AAT with Ki: ASCT1 (2.77μM), rASCT2 (0.73μM), hASCT2 (0.87μM), EAAT1-5 (3.7-7.25μM); used in cancer research.Formula:C18H17NO4Color and Shape:SolidMolecular weight:311.33RU 33965
CAS:RU 33965, a 3-cyclopropyl carbonyl imidazobenzodiazepine, act as a low-efficacy benzodiazepine receptor inverse agonist.Formula:C16H15N3O2Purity:98%Color and Shape:SolidMolecular weight:281.31Dihydrocapsiate
CAS:Dihydrocapsiate is a compound of capsinoid family that can be used in metabolism diseas research. Dihydrocapsiate is an orally active agonist of TRPV1 [1].Formula:C18H28O4Color and Shape:SolidMolecular weight:308.41BTG-1640
CAS:BTG-1640 is used potentially for the treatment of anxiety and panic disorder.Formula:C15H19NO2Color and Shape:SolidMolecular weight:245.32MCC-134
CAS:MCC-134 is an inverse agonist for the pancreatic-type ATP-sensitive K(+) channel. It also used as a vascular relaxing agent.Formula:C16H17N3OSColor and Shape:SolidMolecular weight:299.39(Rac)-MEM 1003
CAS:MEM-1003, a calcium channel blocker, is used potentially for the treatment of bipolar disorders.Formula:C22H25ClN2O5Color and Shape:SolidMolecular weight:432.9(S)-AMPA
CAS:(S)-AMPA is an active isomer of AMPA and a selective agonist of AMPA.Formula:C7H10N2O4Color and Shape:SolidMolecular weight:186.17DDO-02005 free base
CAS:DDO-02005 is a potent Kv1.5 inhibitor with IC50 of 0.72μM, showing strong anti-arrhythmic and anti-AF effects in rat models.Formula:C21H25N3O2Color and Shape:SolidMolecular weight:351.44NS-8
CAS:NS-8, a pyrrole, activates Ca2+-sensitive K+ channels, reducing urinary frequency by inhibiting pelvic nerve activity.Formula:C12H10FN3Color and Shape:SolidMolecular weight:215.23Sadopine
CAS:Sadopine is a high-affinity radioligand for DHP receptor in L-type Ca2+ channels, suitable for tissue and membrane labeling.Formula:C30H40F3N3O7SColor and Shape:SolidMolecular weight:643.71P2X7 receptor antagonist-2
CAS:P2X7 receptor antagonist-2: potent, pIC50 6.5-7.5, reduces neuroinflammation.Formula:C19H18Cl2N2O2Color and Shape:SolidMolecular weight:377.26Bts 39542
CAS:Bts 39542 is a diuretic that plays a major role in the Henle circulation and increases renal blood flow without affecting glomerular filtration rate.Formula:C16H11ClN4O3SColor and Shape:SolidMolecular weight:374.8UBP646
CAS:UBP646 is a GluN1/GluN2 receptors potentiator.Formula:C21H22O2Purity:98%Color and Shape:SolidMolecular weight:306.4NMDA receptor modulator 2
CAS:NMDA receptor modulator 2 (Compound 1) is a potent modulator of the NMDA receptor that can be used for neurological disorder research [1].Formula:C13H11F3N2O2Color and Shape:SolidMolecular weight:284.23NAP-1
CAS:NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).Formula:C20H18ClNO2Color and Shape:SolidMolecular weight:339.82TRPC5-IN-2
CAS:TRPC5-IN-2 is a potent inhibitor of TRPC5.Formula:C17H14ClF3N6OColor and Shape:SolidMolecular weight:410.78CGP 39551
CAS:CGP 39551 is a NMDA antagonist.Formula:C8H16NO5PPurity:98%Color and Shape:White SolidMolecular weight:237.19bis(7)-Tacrine
CAS:Bis(7)-tacrine dihydrochloride: dimeric AChE inhibitor; may treat Alzheimer's; blocks NMDA, antagonizes GABA A.Formula:C33H42Cl2N4Color and Shape:SolidMolecular weight:565.63AS1928370
CAS:AS1928370 is an antagonist of transient receptor potential vanilloid 1 (TRPV1).Formula:C29H31N3O2Color and Shape:SolidMolecular weight:453.58NAB-14
CAS:NAB-14: non-competitive GluN2C/D antagonist, IC50 580 nM for GluN1/2D, >800x selectivity over GluN2A/B, blood-brain-barrier penetrant.Formula:C20H21N3O3Color and Shape:SolidMolecular weight:351.4Ac32Az19
CAS:Ac32Az19 is a potent, non-toxic, and highly selective inhibitor of Breast Cancer Resistance Protein (BCRP), demonstrating an EC50 of 13 nM in BCRP-overexpressedFormula:C37H33N3O6Color and Shape:SolidMolecular weight:615.67GABAA receptor agent 7
CAS:Compound 5c, a GABAA receptor modulator with anticonvulsant properties and low neurotoxicity, is promising for epilepsy research.Formula:C18H13ClN4OColor and Shape:SolidMolecular weight:336.77
