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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2507 products of "Membrane Transporter/Ion Channel"

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  • CymitQuimica logo
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    (3R,6S)-Bassiatin

    CAS:
    (3R,6S)-Bassiatin represents the enantiomeric form of the fungal metabolite known as bassiatin.
    Formula:C15H19NO3
    Molecular weight:261.32

    Ref: TM-TYD-02564

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    DFBTA

    DFBTA inhibits ANO1 with IC50 of 24 nM, effectively treating inflammatory pain orally.
    Formula:C18H10ClF2NO3S
    Color and Shape:Solid
    Molecular weight:393.79

    Ref: TM-T61818

  • ZK 93426 hydrochloride
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    ZK 93426 hydrochloride

    CAS:
    benzodiazepine receptor antagonist,competitive
    Formula:C18H21ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.82

    Ref: TM-T23562

  • Olorigliflozin
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    Olorigliflozin

    CAS:
    Olorigliflozin is a sodium glucose co-transporter (SGLT) inhibitor with antihyperglycemic properties.
    Formula:C23H27ClO7
    Color and Shape:Solid
    Molecular weight:450.909

    Ref: TM-T205428

  • Coleon-U-quinone
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    Coleon-U-quinone

    CAS:
    Coleon-U-quinone, a P-gp inhibitor, reduces cancer cell viability and enhances Doxorubicin sensitivity in resistant cells.
    Formula:C20H24O5
    Color and Shape:Solid
    Molecular weight:344.4

    Ref: TM-T72735

  • SP100030 analogue 1
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    SP100030 analogue 1

    CAS:
    SP100030 analogue 1 (compound 11) is a selective transcription activation (SITA) inhibitor within the SP100030 class, capable of inhibiting XPO1-dependent upregulation of IL2 in a Jurkat-based IL2-Luc reporter assay, with an EC50 of 137 nM.
    Formula:C13H5ClF7N3O
    Color and Shape:Solid
    Molecular weight:387.64

    Ref: TM-T89990

  • H052
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    H052

    CAS:
    <p>H052 is a selective inhibitor of Staphylococcus aureus α-hemolysin (Hla). It binds to the Hla monomer, disrupting its interaction with the host cell membrane, thereby blocking pore formation and inhibiting calcium influx, cytotoxicity, and inflammatory response. H052 exhibits inhibitory activity against Hla-induced calcium influx (EC50 = 30 nM in U937 cells) and holds potential for research into lung infections caused by S. aureus.</p>
    Formula:C21H15ClFN3O4S
    Color and Shape:Solid
    Molecular weight:459.88

    Ref: TM-T207113

  • Cyproflanilide
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    Cyproflanilide

    CAS:
    Cyproflanilide is a GABAR antagonist that exhibits high activity against a variety of pests, including those from the Lepidoptera, Coleoptera, and Thysanoptera orders.
    Formula:C28H17BrF12N2O2
    Color and Shape:Solid
    Molecular weight:721.33

    Ref: TM-T201028

  • O4I4
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    O4I4

    CAS:
    O4I4 is an OCT4-inducing compound capable of activating endogenous OCT4 and its associated signaling pathways, shown anti-aging effects.
    Formula:C15H20N2S
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:260.4

    Ref: TM-T87051

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    WS-898

    <p>WS-898 boosts paclitaxel efficacy in resistant cells by inhibiting ABCB1; IC50: SW620/Ad300 - 5.0 nM, KB-C2 - 3.67 nM, HEK293/ABCB1 - 3.68 nM.</p>
    Formula:C33H25N7OS
    Color and Shape:Solid
    Molecular weight:567.66

    Ref: TM-T64016

  • CFTR corrector 16
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    CFTR corrector 16

    CAS:
    CFTRcorrector 16 (Compound 39) is a corrector of the cystic fibrosis transmembrane conductance regulator (CFTR), utilized in the research of cystic fibrosis disease.
    Formula:C27H26ClN5O2S
    Color and Shape:Solid
    Molecular weight:520.05

    Ref: TM-T200113

  • Vormatrigine
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    Vormatrigine

    CAS:
    Vormatrigine effectively inhibits sodium channels (sodium channel).
    Formula:C16H12F6N4O2
    Color and Shape:Solid
    Molecular weight:406.28

    Ref: TM-T201328

  • Kv7.2/Kv7.3 agonist 1
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    Kv7.2/Kv7.3 agonist 1

    CAS:
    Kv7.2/Kv7.3 agonist 1 (Compound 16) is an orally effective agonist for the KV7.2/7.3 channels (KV7.2/7.3 channel/KCNQ2/3) with an EC50 of 1.03 μM. This compound demonstrates analgesic effects in mouse models of chronic constriction injury (CCI) and Streptozotocin-induced diabetic peripheral neuropathy (DPNP), with ED50 values of 12.02 mg/kg and 9.63 mg/kg, respectively.
    Formula:C14H14FN3O2
    Color and Shape:Solid
    Molecular weight:275.28

    Ref: TM-T201063

  • LY503430
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    LY503430

    CAS:
    LY503430: Oral AMPA enhancer with nootropic, neuroprotective properties, mitigates 6-OHDA/MPTP brain damage.
    Formula:C20H25FN2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.49

    Ref: TM-T27959

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    Cav 3.2 inhibitor 1

    Cav 3.2 inhibitor 1 targets T-type calcium channels, weakly binds D2 receptors, and aids physical and visceral pain research.
    Formula:C32H39N3O
    Color and Shape:Solid
    Molecular weight:481.67

    Ref: TM-T63186

  • Perfluoroheptanesulfonic acid
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    Perfluoroheptanesulfonic acid

    CAS:
    Perfluoroheptanesulfonic acid (1-Perfluoroheptanesulfonic acid; Perfluoroheptanesulphonic acid) is a perfluoroalkyl substance (PFAS). This compound has been detected in landfill leachate and has been shown to induce deformities in zebrafish larvae (EC50=168.1 μM). Exposure to PFHpS in fetuses can lead to reduced birth weight.
    Formula:C7HF15O3S
    Color and Shape:Solid
    Molecular weight:450.12

    Ref: TM-T200995

  • Onfasprodil
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    Onfasprodil

    CAS:
    Onfasprodil, NR2B inhibitor & GABA regulator, potential for Alzheimer's research. (Patent CN111481543A)
    Formula:C20H23FN2O3
    Color and Shape:Solid
    Molecular weight:358.41

    Ref: TM-T61319

  • PF-05661014
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    PF-05661014

    CAS:
    PF-05661014, a demethylated analogue of PF-06526290, selectively inhibits Nav1.3 and Nav1.7 currents by stabilizing the inactivated state through interaction with the D4 VSD. This compound is utilized in research focused on sodium channel modulation.
    Formula:C17H16N4O3S2
    Color and Shape:Solid
    Molecular weight:388.46

    Ref: TM-T89885

  • S 0960
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    S 0960

    CAS:
    S 0960 is a dimeric bile acid analogue, a specific inhibitor of the sodium-dependent bile salt transporter in the ileum, used in metabolic disease research.
    Formula:C48H79NO8
    Purity:99.32% - >99.99%
    Color and Shape:Solid
    Molecular weight:798.14

    Ref: TM-T70688

  • ABCG2-IN-4
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    ABCG2-IN-4

    CAS:
    <p>ABCG2-IN-4 (Compound K31) is an orally active ABCG2 inhibitor that reduces the release of Protoporphyrin IX (PPIX) from red blood cells into the plasma and prevents phototoxicity. In mouse models, ABCG2-IN-4 also demonstrates anti-inflammatory and antioxidant properties.</p>
    Formula:C24H32N4O4
    Color and Shape:Solid
    Molecular weight:440.535

    Ref: TM-T204144