Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(99 products)
- Adiponectin receptor(5 products)
- CFTR(65 products)
- CGRP Receptor(54 products)
- Calcium Channel(546 products)
- Chloride channel(53 products)
- GABA Receptor(369 products)
- Monoamine Transporter(30 products)
- Monocarboxylate transporter(18 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(10 products)
- OAT(32 products)
- OCT(7 products)
- P-gp(55 products)
- Potassium Channel(289 products)
- Proton pump(41 products)
- SGLT(31 products)
- Sodium Channel(226 products)
- TRP/TRPV Channel(96 products)
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Found 2631 products of "Membrane Transporter/Ion Channel"
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P-gp modulator 2
P-gp modulator 2 (Compound 27) is a potent competitive and metabotropic P-glycoprotein (P-gp) modulator.Formula:C22H20BrN3O4Color and Shape:SolidMolecular weight:470.32hURAT1 inhibitor 2
CAS:hURAT1 inhibitor 2 (Compound 5) is an inhibitor of hURAT1 (uric acid transporter 1, SLC22A12) with an IC50 of 18 nM. It also exhibits some inhibitory activity against OATP1B1, with an IC50 of 0.73 μM. hURAT1 inhibitor 2 can be used in research related to hyperuricemia, gout, and other diseases associated with abnormal uric acid metabolism.Formula:C17H11Br2FO3Color and Shape:SolidMolecular weight:442.074CFTR corrector 17
CAS:CFTRcorrector 17 (example 17) is a regulator of the cystic fibrosis transmembrane conductance regulator (CFTR). It is utilized in the study of diseases mediated by CFTR.Formula:C18H15FN2O2Color and Shape:SolidMolecular weight:310.32DAD
DAD is an ion channel blocker (blocks voltage-gated potassium channels) and is a third generation photoelectric switch that responds to visible light.Formula:C26H40N6OColor and Shape:SolidMolecular weight:452.64BGT1-IN-1
CAS:BGT1-IN-1 (compound 9) is an effective inhibitor of BGT1, demonstrating IC50 values of 13.9 µM for hBGT1 and 58.3 µM for GAT3. It exhibits no cytotoxic effects and possesses neuroprotective activity.Formula:C6H9NO2Color and Shape:SolidMolecular weight:127.14P-gp/BCRP-IN-1
CAS:P-gp/BCRP-IN-1, safe and oral, inhibits P-gp/BCRP transporters, enhancing Paclitaxel bioavailability.Formula:C27H25ClN4O3Color and Shape:SolidMolecular weight:488.97SDZ 220-040
CAS:SDZ 220-040 是一种选择性哺乳动物 NMDA 受体拮抗剂，可诱导根系生长的部分无重力模式 。Formula:C16H16Cl2NO6PPurity:98.13%Color and Shape:SolidMolecular weight:420.18Odevixibat
CAS:Odevixibat (A4250) is a selective oral inhibitor for ileal bile acid transport, potentially treating primary biliary cirrhosis.Formula:C37H48N4O8S2Purity:99.53% - 99.83%Color and Shape:SolidMolecular weight:740.93BDZ-g
CAS:BDZ-g: potent, selective AMPA receptor antagonist; useful for researching neurological disorders.Formula:C21H21N5O2SPurity:99.97%Color and Shape:SolidMolecular weight:407.49SYM2206
CAS:SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 μM.SYM2206 exhibits anticancer activity by blocking Nav1.6-mediatedFormula:C20H22N4O3Purity:99.8%Color and Shape:SolidMolecular weight:366.41Suzetrigine
CAS:Suzetrigine (VX-548) is an oral NaV1.8 inhibitor with analgesic properties for acute pain research.Formula:C21H20F5N3O4Purity:98.08% - 99.27%Color and Shape:SolidMolecular weight:473.39Ref: TM-T69552
1mg58.00€5mg114.00€10mg170.00€25mg266.00€300g129,112.00€50mg457.00€100mg747.00€200mg1,026.00€1mL*10mM (DMSO)118.00€(+)-Tetrabenazine
CAS:(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-foldFormula:C19H27NO3Purity:98.69%Color and Shape:SolidMolecular weight:317.42(-)-Bicuculline methobromide
CAS:(-)-Bicuculline methobromide is a potent antagonist of GABAA receptor .Formula:C21H20BrNO6Color and Shape:WhiteMolecular weight:462.29A-887826
CAS:A-887826 is a selective, orally bioavailable, and voltage-dependent Na(v1.8) channel blocker (IC50: 11 nM). It attenuates neuropathic tactile allodynia in vivo.Formula:C26H29ClN4O3Color and Shape:SolidMolecular weight:480.99Umbellulone
CAS:Umbellulone is a natural product isolated from Umbellularia californica, and stimulates the TRPA1 channel in a subset of peptidergic, nociceptive neurons, activating the trigeminovascular system via this mechanism.Formula:C10H14OPurity:98%Color and Shape:SolidMolecular weight:150.225-Hydroxylansoprazole
CAS:5-Hydroxylansoprazole (AG1908) is the active metabolite of plasma Lansoprazole, inhibits the proton pump, and is used in the study of peptic ulcers.Formula:C16H14F3N3O3SPurity:99.00%Color and Shape:SolidMolecular weight:385.36Indoxacarb
CAS:Indoxacarb is an Oxadiazine insecticide.Formula:C22H17ClF3N3O7Purity:98%Color and Shape:SolidMolecular weight:527.83Apcin A HCL
CAS:Apcin A HCL is an Apcin derivative. Apcin A HCL is an anaphase-promoting complex (APC) inhibitor. Apcin-A HCL interacts strongly with Cdc20, and inhibits the ubiquitination of Cdc20 substrates. Apcin-A HCL can be used to synthesize the PROTAC CP5V [1].
Formula:C10H15Cl4N5O2Purity:99.30%Color and Shape:SolidMolecular weight:379.073-Methylglutaconic acid
CAS:3-Methylglutaconic acid, a primary metabolite accumulating in 3-Methylglutaconic aciduria (MGTA), induces lipid and protein oxidation, while diminishing non-enzymatic antioxidant defenses in cerebral cortex supernatants, thereby promoting oxidative stress in the cerebral cortex. This compound is utilized in research concerning brain damage diseases [1].Formula:C6H8O4Purity:98%Color and Shape:SolidMolecular weight:144.132-AEMP TFA
CAS:2-AEMP TFA is a potent and rapidly acting antagonist of GABA(A)-ρ1 receptors. 2-AEMP is an analog of GABA.Formula:C3H10NO3PPurity:98%Color and Shape:SolidMolecular weight:139.091
