Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
KPT185
CAS:1333151-73-7
KPT185 (KPT 185) is a selective CRM1 inhibitor, inducing apoptosis, cell-cycle arrest.
Formula:
C16H16F3N3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
355.31
Ref: TM-T2425
| 2mg | 35.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
(R)-Lansoprazole
CAS:138530-94-6
(R)-Lansoprazole (T 168390) is the R-isomer of lansoprazole and a substituted benzimidazole prodrug with selective …
Formula:
C16H14F3N3O2S
Purity:
98.09% - 98.99%
Color and Shape:
Brown Solid
Molecular weight:
369.36
Ref: TM-T1021
| 50mg | 39.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 63.00 € | ||
| 500mg | 89.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
PF-05186462
CAS:1235406-03-7
PF-05186462 (PF-05150122) is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, …
Formula:
C19H10ClF4N5O3S2
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
531.89
Ref: TM-T8711
| 1mg | 129.00 € | ||
| 5mg | 281.00 € | ||
| 10mg | 421.00 € | ||
| 25mg | 694.00 € | ||
| 50mg | 979.00 € | ||
| 1mL*10mM (DMSO) | 366.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
α-Asarone
CAS:2883-98-9
alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.
Formula:
C12H16O3
Purity:
99.59%
Color and Shape:
Monoclinic Needles From Water Monoclinic Needles From Water
Molecular weight:
208.25
Ref: TM-T3698
| 100mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Ralfinamide mesylate
CAS:202825-45-4
Ralfinamide mesylate (FCE-26742A (mesylate)) is an orally available Na+ channel blocker.
Formula:
C18H23FN2O5S
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
398.45
Ref: TM-T7547
| 1mg | 76.00 € | ||
| 5mg | 164.00 € | ||
| 10mg | 248.00 € | ||
| 25mg | 408.00 € | ||
| 50mg | 543.00 € | ||
| 100mg | 763.00 € | ||
| 200mg | 1,026.00 € | ||
| 1mL*10mM (DMSO) | 250.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
LY 303511 hydrochloride
CAS:2070014-90-1
LY 303511 hydrochloride is a potent mTOR inhibitor
Formula:
C19H19ClN2O2
Purity:
97.44%
Color and Shape:
Solid
Molecular weight:
342.82
Ref: TM-T4423
| 1mg | 39.00 € | ||
| 2mg | 35.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 468.00 € | ||
| 100mg | 681.00 € | ||
| 200mg | 566.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
(-)-Blebbistatin
CAS:856925-71-8
(-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin …
Formula:
C18H16N2O2
Purity:
99.38% - 99.59%
Color and Shape:
Solid
Molecular weight:
292.33
Ref: TM-T6038
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 176.00 € | ||
| 50mg | 276.00 € | ||
| 100mg | 447.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
AER-271
CAS:634913-39-6
AER-271 is an inhibitor of aquaporin-4.
Formula:
C15H9ClF6NO5P
Purity:
99.03%
Color and Shape:
Solid
Molecular weight:
463.65
Ref: TM-T7946
| 2mg | 44.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 214.00 € | ||
| 50mg | 325.00 € | ||
| 100mg | 487.00 € | ||
| 1mL*10mM (DMSO) | 66.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
TKIM
CAS:326921-25-9
TKIM is a TWIK-related potassium channel 1 (TREK-1) inhibitor, binding to the pocket of the …
Formula:
C18H14ClN3O2S
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
371.84
Ref: TM-T8700
| 1mg | 62.00 € | ||
| 5mg | 137.00 € | ||
| 10mg | 206.00 € | ||
| 25mg | 363.00 € | ||
| 50mg | 509.00 € | ||
| 100mg | 682.00 € | ||
| 200mg | 918.00 € | ||
| 1mL*10mM (DMSO) | 149.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
ICA-069673
CAS:582323-16-8
ICA-069673 is an activator of KCNQ2/Q3 potassium channel (IC50: 0.69 μM).
Formula:
C11H6ClF2N3O
Purity:
98.97% - 99.66%
Color and Shape:
Solid
Molecular weight:
269.63
Ref: TM-T3959
| 5mg | 45.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 249.00 € | ||
| 100mg | 362.00 € | ||
| 200mg | 525.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
L-DABA
CAS:1758-80-1
L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 >500 μM).
Formula:
C4H10N2O2
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
118.13
Ref: TM-T7595
| 25mg | 34.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
SB-705498
CAS:501951-42-4
SB705498 is a TRPV1 antagonist for hTRPV1. SB-705498 has been investigated for the treatment of …
Formula:
C17H16BrF3N4O
Purity:
98% - ≥95%
Color and Shape:
Solid
Molecular weight:
429.23
Ref: TM-T6660
| 5mg | 47.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 293.00 € | ||
| 100mg | 423.00 € | ||
| 200mg | 589.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Lorediplon
CAS:917393-39-6
Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at …
Formula:
C20H15FN4O2S
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
394.42
Ref: TM-TQ0023
| 10mg | 46.00 € | ||
| 25mg | 86.00 € | ||
| 50mg | 149.00 € | ||
| 100mg | 226.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
O4I2
CAS:165682-93-9
O4I2 is an effective Oct3/4 inducer in various human cell lines including human fibroblasts.
Formula:
C12H11ClN2O2S
Purity:
99.12% - 99.25%
Color and Shape:
Solid
Molecular weight:
282.75
Ref: TM-T2437
| 5mg | 51.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 115.00 € | ||
| 50mg | 186.00 € | ||
| 100mg | 347.00 € | ||
| 200mg | 301.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
M8-B Hydrochloride
CAS:883976-12-3
M8-B Hydrochloride is a selective transient receptor potential melastatin-8 (TRPM8) channel antagonist.
Formula:
C22H25ClN2O3S
Purity:
99.33%
Color and Shape:
Solid
Molecular weight:
432.96
Ref: TM-T8442
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 218.00 € | ||
| 100mg | 324.00 € | ||
| 200mg | 452.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
DHQ
CAS:15804-19-0
DHQ (2,3-dihydroxy-quinoxalin) is an inducer of ATPase activity that of Herpes Simplex Virus thymidine kinase.
Formula:
C8H6N2O2
Purity:
100.00%
Color and Shape:
Solid
Molecular weight:
162.15
Ref: TM-T20436
| 50mg | 44.00 € | ||
| 100mg | 63.00 € | ||
| 200mg | 88.00 € | ||
| 500mg | 149.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
CL 218872
CAS:66548-69-4
CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less …
Formula:
C13H9F3N4
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
278.23
Ref: TM-T8572
| 25mg | 53.00 € | ||
| 50mg | 93.00 € | ||
| 100mg | 141.00 € | ||
| 200mg | 201.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Vonoprazan fumarate
CAS:1260141-27-2
Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.
Formula:
C17H16FN3O2S·C4H4O4
Purity:
100% - 99.16%
Color and Shape:
Solid
Molecular weight:
461.46
Ref: TM-T2404
| 500mg | 47.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Nav1.8-IN-1
CAS:1026822-49-0
Nav1.8-IN-1 (CHEMBL1270208) is an inhibitor of human NaV1.8
Formula:
C20H15ClF3N3O2
Purity:
97.59%
Color and Shape:
Solid
Molecular weight:
421.8
Ref: TM-T8579
| 1mg | 84.00 € | ||
| 5mg | 168.00 € | ||
| 10mg | 248.00 € | ||
| 25mg | 408.00 € | ||
| 50mg | 574.00 € | ||
| 100mg | 776.00 € | ||
| 200mg | 1,029.00 € | ||
| 1mL*10mM (DMSO) | 190.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
SB-366791
CAS:472981-92-3
SB-366791 is a new and selective cinnamide TRPV1 antagonist.
Formula:
C16H14ClNO2
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
287.74
Ref: TM-T6977
| 5mg | 35.00 € | ||
| 10mg | 44.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 123.00 € | ||
| 100mg | 196.00 € | ||
| 200mg | 291.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
