Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(101 products)
- Adiponectin receptor(5 products)
- CFTR(65 products)
- CGRP Receptor(54 products)
- Calcium Channel(541 products)
- Chloride channel(53 products)
- GABA Receptor(365 products)
- Monoamine Transporter(30 products)
- Monocarboxylate transporter(18 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(10 products)
- OAT(32 products)
- OCT(7 products)
- P-gp(54 products)
- Potassium Channel(280 products)
- Proton pump(42 products)
- SGLT(31 products)
- Sodium Channel(209 products)
- TRP/TRPV Channel(95 products)
Show 13 more subcategories
Found 2512 products of "Membrane Transporter/Ion Channel"
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Lesogaberan napadisylate
CAS:Lesogaberan (AZD-3355) is a selective GABAB agonist with EC50 of 8.6 nM, Ki of 5.1 nM in rats, and acts peripherally on the esophageal sphincter.Formula:C13H17FNO5PSColor and Shape:SolidMolecular weight:349.31ABCB1-IN-1
ABCB1-IN-1 (compound 3) is a potent inhibitor of ABCB1 that promotes cell apoptosis.Formula:C36H33F3FeN2O4PSColor and Shape:SolidMolecular weight:733.54Phrixotoxin-1
CAS:Phrixotoxin 1, a specific peptide inhibitor of Kv4 potassium channels, originates from the venom of the theraphosid spider Phrixotrichus auratus [1] [2].Formula:C156H246N44O37S7Purity:98%Color and Shape:SolidMolecular weight:3554.35Camegliptin
CAS:Cameglipti, a dipeptidyl peptidase IV (DPP-4) inhibitor, is used potentially for the treatment of type 2 diabetes.Formula:C20H28FN3O3Color and Shape:SolidMolecular weight:377.4524-Hydroxycholesterol
CAS:24-Hydroxycholesterol (Cholest-5-ene-3beta,24-diol) is an activator of the LXR and can be used to study cardiogenesis and pancreatic cancer.Formula:C27H46O2Purity:99.8%Color and Shape:SolidMolecular weight:402.65Aglafoline
CAS:Aglafoline inhibits in a concentration-dependent manner the aggregation and ATP release reaction induced in washed rabbit platelets by PAF (platelet-activatingFormula:C28H28O8Color and Shape:SolidMolecular weight:492.52Aam-KTX
Aam-KTX, a toxic peptide sourced from Mesobuthus eupeus scorpion venom, acts as a selective K_v channel inhibitor, exhibiting IC_50 values of 1.1 nM for K_v1.3Formula:C174H288N58O48S7Purity:98%Color and Shape:SolidMolecular weight:4184.96Atelopidtoxin
CAS:Atelopidtoxin is a biochemical.Formula:C16H24N8O12SColor and Shape:SolidMolecular weight:552.47ShK toxin
CAS:ShK toxin, isolated from the Caribbean sea anemone (Stichodactyla helianthus), is an inhibitor of the voltage-dependent potassium channel (Kv1.3 channel).Formula:C169H274N54O48S7Purity:98%Color and Shape:SolidMolecular weight:4054.8Lyso-Globotriaosylceramide (d18:1)
CAS:Lyso-Gb3, lacking fatty acyl, binds Stx1 with cholesterol and phosphatidylcholine, not Stx2; lowers neutrophil viability; accumulates in Fabry disease.Formula:C36H67NO17Color and Shape:SolidMolecular weight:785.922µ-Conotoxin BuIIIC
CAS:μ-Conotoxin BuIIIC (Mu-Conotoxin BuIIIC) effectively inhibits the NaV1.4 sodium channel [1].Formula:C116H189N49O34S6Purity:98%Color and Shape:SolidMolecular weight:3006.44Mesoridazine free base
CAS:Mesoridazine (thioridazine EP impurity B) is a phenothiazine antipsychotic with effects similar to chlorpromazine.Formula:C21H26N2OS2Color and Shape:SolidMolecular weight:386.57MRK-016
CAS:MRK-016 is a selective GABAA α5 receptor inverse agonist/ negative allosteric modulator, orally available and penetrating the BBB. MRK-016 is antidepressant.Formula:C17H20N8O2Purity:99.76%Color and Shape:SolidMolecular weight:368.39Ethacizine hydrochloride
CAS:Ethacizine hydrochloride (NIK-244) has antiarrhythmic activity and can be used to study arrhythmias and myocardial infarction.Formula:C22H28ClN3O3SPurity:98.08% - 98.08%Color and Shape:SolidMolecular weight:449.99Halofantrine hydrochloride
CAS:Halofantrine hydrochloride (SKF-102886) is an orally administered antimalarial drug effective against drug-resistant P. falciparum and P. vivax. SKF-102886 has cardiac toxicity, inhibiting hERG and delayed rectifier potassium channel I Kr, leading to prolonged QTc and PR intervals.Formula:C26H31Cl3F3NOPurity:98%Color and Shape:SolidMolecular weight:536.89KCNQ1 activator-1
CAS:<p>N-[4-(4-Methoxyphenyl)-2-thiazolyl]-2-piperidinecarboxamide is a potent KCNQ1 activator for LQTS research.</p>Formula:C22H23N3O4S2Purity:99.71%Color and Shape:SolidMolecular weight:457.57Nicardipine-d3 hydrochloride
CAS:Nicardipine D3 hydrochloride is the deuterium labeled Nicardipine hydrochloride.Formula:C26H30ClN3O6Purity:98%Color and Shape:SolidMolecular weight:519(S)-Nicardipine
CAS:(S)-Nicardipine is the less active S enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).Formula:C26H29N3O6Color and Shape:SolidMolecular weight:479.535-Hydroxydecanoic acid
CAS:5-Hydroxydecanoic acid is a selective ATP-sensitive K+ (KATP) channel blocker (IC50 of ~30 μM). 5-Hydroxydecanoic acid is a substrate for mitochondrial outer membrane acyl-CoA synthetase and has antioxidant activity.Formula:C10H20O3Purity:99.24%Color and Shape:SolidMolecular weight:188.26MDL 105519
CAS:MDL 105519 is a selective, non-competitive antagonist of NMDA receptors. It inhibits cyclic GMP accumulation in brain slices, anxiolytic in rat models.Formula:C18H11Cl2NO4Purity:99.67%Color and Shape:SolidMolecular weight:376.19
