Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
UCCF-853
CAS:625458-06-2
UCCF-853 is a small-molecule CFTR modulator that can be used to study cystic fibrosis.
Formula:
C14H8ClF3N2O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
312.67
Ref: TM-T29041
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 179.00 € | ||
| 50mg | 267.00 € | ||
| 100mg | 396.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
R 56865
CAS:104606-13-5
R 56865 is a weak potential-operated channel inhibitor that inhibits the late sodium current in …
Formula:
C23H28FN3OS
Purity:
99.08%
Color and Shape:
Solid
Molecular weight:
413.55
Ref: TM-T26016
| 1mg | 278.00 € | ||
| 5mg | 684.00 € | ||
| 10mg | 935.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
GAL-021 sulfate
CAS:1380342-00-6
GAL-021 sulfate is a BKCa channel blocker that inhibits the analgesic effects of opioids and …
Formula:
C11H24N6O5S
Purity:
99.68%
Color and Shape:
Liquid
Molecular weight:
352.41
Ref: TM-T61239
| 1mg | 75.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 225.00 € | ||
| 25mg | 378.00 € | ||
| 50mg | 563.00 € | ||
| 100mg | 803.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Istaroxime hydrochloride
CAS:374559-48-5
Istaroxime hydrochloride (PST2744 hydrochloride) is a Na+/K+-ATPase inhibitor and SERCA 2 activator, and is a …
Formula:
C21H33ClN2O3
Color and Shape:
Solid
Molecular weight:
396.95
Ref: TM-T15599
| 2mg | 129.00 € | ||
| 5mg | 215.00 € | ||
| 10mg | 352.00 € | ||
| 50mg | 739.00 € | ||
| 100mg | 1,105.00 € | ||
| 1mL*10mM (DMSO) | 238.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Bamocaftor
CAS:2204245-48-5
Bamocaftor corrects CFTR in CF, restoring F508del-CFTR function, used with tezacaftor and VX-561 for F508del/MF …
Formula:
C28H32F3N5O4S
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
591.65
Ref: TM-T30293
| 1mg | 347.00 € | ||
| 5mg | 828.00 € | ||
| 10mg | 1,138.00 € | ||
| 25mg | 1,662.00 € | ||
| 50mg | 2,270.00 € | ||
| 100mg | 3,047.00 € | ||
| 1mL*10mM (DMSO) | 1,218.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
CFTR corrector 8
CAS:1918142-35-4
CFTR corrector 8: potent for cystic fibrosis research, modulates CFTR protein.
Formula:
C29H27F2NO7
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
539.52
Ref: TM-T63806
| 1mg | 80.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 258.00 € | ||
| 25mg | 522.00 € | ||
| 50mg | 820.00 € | ||
| 100mg | 1,345.00 € | ||
| 1mL*10mM (DMSO) | 216.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
VRT-532
CAS:38214-71-0
VRT-532 (CFpot-532) is an effective modulator of CFTR and is commonly used in studies of …
Formula:
C16H14N2O
Purity:
100% - 99.89%
Color and Shape:
Solid
Molecular weight:
250.3
Ref: TM-T29114
| 1mg | 150.00 € | ||
| 5mg | 363.00 € | ||
| 10mg | 546.00 € | ||
| 25mg | 904.00 € | ||
| 50mg | 1,235.00 € | ||
| 100mg | 1,625.00 € | ||
| 1mL*10mM (DMSO) | 327.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
NaV1.2/1.6 channel blocker-1
CAS:1199944-04-1
NaV1.2/1.6 channel blocker-1 is a NaV1.2/1.6 channel blocker that inhibits rNaV1.6 and can be used …
Formula:
C14H14N2OS
Purity:
99.54%
Color and Shape:
Liquid
Molecular weight:
258.34
Ref: TM-T72170
| 1mg | 40.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 116.00 € | ||
| 25mg | 225.00 € | ||
| 50mg | 333.00 € | ||
| 100mg | 495.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
ELB-139
CAS:188116-08-7
ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal …
Formula:
C14H16ClN3O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
277.75
Ref: TM-T27252
| 1mg | 274.00 € | ||
| 2mg | 408.00 € | ||
| 5mg | 675.00 € | ||
| 10mg | 922.00 € | ||
| 25mg | 1,417.00 € | ||
| 50mg | 1,846.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Pinacidil
CAS:60560-33-0
Pinacidil (P 1134) is a guanidine that opens potassium channels and directly dilates peripheral blood …
Formula:
C13H19N5
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
245.32
Ref: TM-T12478L
| 5mg | 49.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 161.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Picrotin
CAS:21416-53-5
Picrotin is an inhibitor of glycine receptors. Picrotin blocks α2 GlyR, α1 GlyR, and α3 …
Formula:
C15H18O7
Purity:
97.11%
Color and Shape:
Solid
Molecular weight:
310.3
Ref: TM-T16533
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 74.00 € | ||
| 50mg | 93.00 € | ||
| 100mg | 140.00 € | ||
| 500mg | 343.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Pazinaclone
CAS:103255-66-9
Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.
Formula:
C25H23ClN4O4
Purity:
98.12% - 99%
Color and Shape:
Solid
Molecular weight:
478.93
Ref: TM-T28303
| 1mg | 138.00 € | ||
| 5mg | 325.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 797.00 € | ||
| 50mg | 1,100.00 € | ||
| 100mg | 1,476.00 € | ||
| 500mg | 2,980.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Amsacrine
CAS:51264-14-3
Amsacrine (AMSA) (mAMSA) an antineoplastic agent which can intercalate into the DNA of tumor cells.
Formula:
C21H19N3O3S
Purity:
98.59%
Color and Shape:
Yellow Crystalline Powder Solid
Molecular weight:
393.46
Ref: TM-T1206
| 10mg | 51.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Vernakalant
CAS:794466-70-9
Vernakalant (RSD-1235) is a mixed ion channel blocker.
Formula:
C20H31NO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
349.46
Ref: TM-TQ0307
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
(R)-Baclofen hydrochloride
CAS:63701-55-3
Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.
Formula:
C10H13Cl2NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
250.12
Ref: TM-T17306
| 10mg | 87.00 € | ||
| 25mg | 200.00 € | ||
| 50mg | 328.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Transcainide
CAS:88296-62-2
Transcainide (R 54718), an oral lidocaine-like antiarrhythmic, blocks BTX-activated Na+ channels in heart/muscle.
Formula:
C22H35N3O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
373.53
Ref: TM-T26287
| 1mg | 250.00 € | ||
| 5mg | 616.00 € | ||
| 10mg | 879.00 € | ||
| 25mg | 1,299.00 € | ||
| 50mg | 1,746.00 € | ||
| 100mg | 2,378.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
RN9893
CAS:1803003-68-0
RN9893 is a selective and potent TRPV4 receptor antagonist with IC50 values of 320, 420 …
Formula:
C21H23F3N4O5S
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
500.49
Ref: TM-T28548
| 1mg | 46.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 141.00 € | ||
| 25mg | 268.00 € | ||
| 50mg | 397.00 € | ||
| 100mg | 578.00 € | ||
| 500mg | 1,187.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Sipatrigine
CAS:130800-90-7
Sipatrigine (619C89) is an inhibitor of glutamate release, TREK ion channels, TRESK channels, sodium channels, …
Formula:
C15H16Cl3N5
Purity:
100% - 99.49%
Color and Shape:
Solid
Molecular weight:
372.68
Ref: TM-T16887
| 1mg | 96.00 € | ||
| 2mg | 124.00 € | ||
| 5mg | 201.00 € | ||
| 10mg | 300.00 € | ||
| 25mg | 503.00 € | ||
| 1mL*10mM (DMSO) | 222.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
BMS-919373
CAS:1272353-82-8
BMS-919373 is a potassium channel Kv1.5 (KCNA5) inhibitor for atrial fibrillation and acute coronary syndrome.
Formula:
C25H20N6O2S
Purity:
98.51%
Color and Shape:
Solid
Molecular weight:
468.53
Ref: TM-T30544
| 1mg | 237.00 € | ||
| 5mg | 581.00 € | ||
| 10mg | 817.00 € | ||
| 25mg | 1,207.00 € | ||
| 50mg | 1,628.00 € | ||
| 100mg | 2,185.00 € | ||
| 1mL*10mM (DMSO) | 632.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Bifenazate
CAS:149877-41-8
Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls …
Formula:
C17H20N2O3
Purity:
99.44%
Color and Shape:
Solid Crystalline
Molecular weight:
300.35
Ref: TM-T14571
| 25mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
