Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
ABT 102
CAS:808756-71-0
ABT 102 (CHEMBL398338) is a selective antagonist of transient receptor potential vanilloid 1 (TRPV1) receptor.
Formula:
C21H24N4O
Purity:
98.38% - 99.72%
Color and Shape:
Solid
Molecular weight:
348.44
Ref: TM-T29522
| 1mg | 112.00 € | ||
| 5mg | 242.00 € | ||
| 10mg | 359.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 765.00 € | ||
| 100mg | 1,026.00 € | ||
| 200mg | 1,367.00 € | ||
| 1mL*10mM (DMSO) | 252.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
ML402
CAS:298684-44-3
ML402 (ZINC3671497) is an activator of TREK-1 and TREK-2 with EC50s of 13.7 μM and …
Formula:
C14H14ClNO2S
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
295.78
Ref: TM-T16109
| 1mg | 37.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 232.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 553.00 € | ||
| 200mg | 451.00 € | ||
| 500mg | 1,188.00 € | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Panadiplon
CAS:124423-84-3
Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, …
Formula:
C18H17N5O2
Purity:
100% - 99.75%
Color and Shape:
Solid
Molecular weight:
335.36
Ref: TM-T28294
| 1mg | 138.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 797.00 € | ||
| 50mg | 1,095.00 € | ||
| 100mg | 1,477.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Losigamone
CAS:112856-44-7
Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about …
Formula:
C12H11ClO4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
254.67
Ref: TM-T27845
| 1mg | 81.00 € | ||
| 5mg | 168.00 € | ||
| 10mg | 253.00 € | ||
| 25mg | 470.00 € | ||
| 50mg | 631.00 € | ||
| 100mg | 920.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Rilmakalim
CAS:132014-21-2
Rilmakalim is a potassium channel opener. Rilmakalim shows antivasoconstrictor effect.
Formula:
C21H23NO5S
Purity:
100% - 99.63%
Color and Shape:
Solid
Molecular weight:
401.48
Ref: TM-T26086
| 1mg | 126.00 € | ||
| 5mg | 299.00 € | ||
| 10mg | 449.00 € | ||
| 25mg | 735.00 € | ||
| 50mg | 1,009.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
AM12
CAS:2387510-84-9
AM12 inhibits Lanthanide-evoked TRPC5 activity (IC50: 0.28 μM).
Formula:
C15H9BrO5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
349.13
Ref: TM-T13546
| 10mg | 448.00 € | ||
| 50mg | 1,874.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Dimethindene
CAS:5636-83-9
Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits …
Formula:
C20H24N2
Purity:
99% - 99.44%
Color and Shape:
Solid
Molecular weight:
292.42
Ref: TM-T31488
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 251.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 551.00 € | ||
| 50mg | 776.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Thursday 16 Jan 2025
(5R)-BW-4030W92
CAS:189013-61-4
(5R)-BW-4030W92 is the R-type of BW-4030W92, the active enantiomer.
Formula:
C11H9Cl2FN4
Purity:
98.27%
Color and Shape:
Solid
Molecular weight:
287.12
Ref: TM-T13428
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
SM-6586
CAS:103898-38-0
SM-6586 is a potent calcium channel antagonist with inhibitory effects on Na+/H+ and Na+/Ca2+ exchange …
Formula:
C26H27N5O5
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
489.52
Ref: TM-T16897
| 1mg | 652.00 € | ||
| 5mg | 1,677.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
GS 39783
CAS:39069-52-8
GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties …
Formula:
C15H23N5O2S
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
337.44
Ref: TM-T22813
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 134.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 399.00 € | ||
| 100mg | 579.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
GSK1702934A
CAS:924377-85-5
GSK1702934A is a TRPC3 agonist with pro-arrhythmic and positive inotropic effects and is used in …
Formula:
C22H25N3O2S
Purity:
98.15%
Color and Shape:
Solid
Molecular weight:
395.52
Ref: TM-T15425
| 1mg | 76.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Dicirenone
CAS:41020-79-5
Dicirenone (SC26304) inhibits the Mineralocorticoid receptor (MR), aldosterone regulation of the urinary K+:Na+ ratio, and …
Formula:
C26H36O5
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
428.56
Ref: TM-T13881
| 1mg | 650.00 € | ||
| 5mg | 1,672.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Nisoxetine hydrochloride
CAS:57754-86-6
Nisoxetine hydrochloride is a noradrenaline transporter (NET) inhibitor
Formula:
C17H21NO2·HCl
Purity:
98.52%
Color and Shape:
White Solid
Molecular weight:
307.82
Ref: TM-T23070
| 5mg | 69.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 171.00 € | ||
| 50mg | 268.00 € | ||
| 100mg | 426.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
AVE-0118
CAS:498577-53-0
AVE-0118 is a potassium channel blocker and suppresses persistent atrial fibrillation.
Formula:
C30H29N3O3
Purity:
98.89% - 99.52%
Color and Shape:
Solid
Molecular weight:
479.57
Ref: TM-T26689
| 1mg | 74.00 € | ||
| 5mg | 140.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 320.00 € | ||
| 50mg | 473.00 € | ||
| 100mg | 688.00 € | ||
| 200mg | 569.00 € | ||
| 500mg | 1,412.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
3α,21-Dihydroxy-5α-pregnan-20-one
CAS:567-02-2
3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like …
Formula:
C21H34O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
334.49
Ref: TM-T26390
| 1mg | 141.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Thursday 16 Jan 2025
Anxiolytic/nonsedative agent-1
CAS:355022-97-8
TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy …
Formula:
C18H15N3O4
Purity:
97.05%
Color and Shape:
Solid
Molecular weight:
337.33
Ref: TM-T23445
| 1mg | 63.00 € | ||
| 2mg | 95.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 148.00 € | ||
| 25mg | 325.00 € | ||
| 50mg | 463.00 € | ||
| 100mg | 643.00 € | ||
| 500mg | 1,267.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
GW 542573X
CAS:660846-41-3
GW 542573X is a potent and selective small molecule Ca2+-activated K+ 2 (SK2) channel activator.GW …
Formula:
C19H28N2O5
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
364.44
Ref: TM-T22826
| 1mg | 58.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 207.00 € | ||
| 25mg | 430.00 € | ||
| 50mg | 722.00 € | ||
| 100mg | 979.00 € | ||
| 500mg | 1,940.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Divaplon
CAS:90808-12-1
Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics …
Formula:
C17H17N3O2
Purity:
96.90% - 97.49%
Color and Shape:
Solid
Molecular weight:
295.34
Ref: TM-T27186
| 1mg | 141.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 797.00 € | ||
| 50mg | 1,100.00 € | ||
| 100mg | 1,476.00 € | ||
| 500mg | 2,980.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
DPI 201-106
CAS:97730-95-5
DPI 201-106: cardioselective h1 Na channel inhibitor, enhances heart contraction, blocks potassium and calcium currents.
Formula:
C29H30N4O2
Purity:
97.26%
Color and Shape:
Solid
Molecular weight:
466.57
Ref: TM-T27205
| 5mg | 41.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 119.00 € | ||
| 50mg | 176.00 € | ||
| 1mL*10mM (DMSO) | 42.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Tiludronate disodium
CAS:149845-07-8
Tiludronate disodium: osteoclast inhibitor for metabolic bone disorder research.
Formula:
C7H7ClNa2O6P2S
Purity:
100% - 100%
Color and Shape:
Fine White To Off-White Crystalline Powder
Molecular weight:
362.57
Ref: TM-T13159
| 5mg | 79.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 277.00 € | ||
| 100mg | 411.00 € | ||
| 500mg | 827.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
