Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
Progabide
CAS:62666-20-0
Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.
Formula:
C17H16ClFN2O2
Purity:
99.7%
Color and Shape:
Solid
Molecular weight:
334.77
Ref: TM-T16581
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 151.00 € | ||
| 100mg | 230.00 € | ||
| 200mg | 326.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Radequinil
CAS:219846-31-8
Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) …
Formula:
C18H14N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
334.33
Ref: TM-T16717
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
FR183998 free base
CAS:239440-20-1
FR183998 free base is an inhibitor of Na+/Ca2+ Exchanger.
Formula:
C17H19Cl2N5O2S
Purity:
97.66%
Color and Shape:
Solid
Molecular weight:
428.34
Ref: TM-T11319
| 1mg | 102.00 € | ||
| 5mg | 243.00 € | ||
| 10mg | 372.00 € | ||
| 25mg | 682.00 € | ||
| 50mg | 916.00 € | ||
| 100mg | 1,237.00 € | ||
| 200mg | 1,668.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
EIPA hydrochloride
CAS:1345839-28-2
EIPA hydrochloride also inhibits Na+/H+-exchanger (NHE) and macropinocytosisEIPA hydrochloride (L593754 hydrochloride) is a TRPP3 channel …
Formula:
C11H19Cl2N7O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
336.22
Ref: TM-T11172
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Thursday 16 Jan 2025
Besipirdine
CAS:119257-34-0
Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular …
Formula:
C16H17N3
Purity:
97% - 98.59%
Color and Shape:
Solid
Molecular weight:
251.33
Ref: TM-T26778
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,434.00 € | ||
| 50mg | 1,867.00 € | ||
| 100mg | 2,357.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Muscimol HBr
CAS:18174-72-6
Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.
Formula:
C4H7BrN2O2
Purity:
100%
Color and Shape:
Off-White Powder
Molecular weight:
195.01
Ref: TM-T20657
| 1mg | 118.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 247.00 € | ||
| 10mg | 398.00 € | ||
| 25mg | 642.00 € | ||
| 50mg | 929.00 € | ||
| 100mg | 1,243.00 € | ||
| 500mg | 2,513.00 € | ||
| 1mL*10mM (DMSO) | 214.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
FEMA-4809
CAS:1374760-95-8
FEMA-4809 activates TRPM8, the ion channel for cold sensation, and is used as a cooling …
Formula:
C17H17N3O2S
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
327.4
Ref: TM-T27308
| 1mg | 53.00 € | ||
| 5mg | 114.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 311.00 € | ||
| 50mg | 440.00 € | ||
| 100mg | 626.00 € | ||
| 500mg | 1,238.00 € | ||
| 1mL*10mM (DMSO) | 132.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Olvanil
CAS:58493-49-5
Olvanil (N-Vannilyloleoylamide) is a vanilloid receptor agonist with EC50 of 0.7nM.
Formula:
C26H43NO3
Purity:
95.06%
Color and Shape:
Solid
Molecular weight:
417.62
Ref: TM-T23106
| 1mg | 49.00 € | ||
| 2mg | 72.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 159.00 € | ||
| 25mg | 261.00 € | ||
| 50mg | 364.00 € | ||
| 100mg | 521.00 € | ||
| 200mg | 703.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
VU 0240551
CAS:893990-34-6
VU 0240551 is a selective antagonist of neuronal K-Cl cotransporter KCC2 inhibitor with an IC50 …
Formula:
C16H14N4OS2
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
342.44
Ref: TM-TQ0139
| 1mg | 36.00 € | ||
| 5mg | 77.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 253.00 € | ||
| 50mg | 435.00 € | ||
| 100mg | 696.00 € | ||
| 200mg | 926.00 € | ||
| 500mg | 1,383.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Almokalant
CAS:123955-10-2
Almokalant: Class III antiarrhythmic, K+ channel blocker, inhibits Ikr current.
Formula:
C18H28N2O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
352.49
Ref: TM-T14189
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
(+)-KCC2 blocker 1
CAS:1228439-71-1
(+)-KCC2 blocker 1 is a selective blocker of KCC2 (IC50 = 0.4 μM).
Formula:
C22H25NO5S
Purity:
98.12%
Color and Shape:
Solid
Molecular weight:
415.5
Ref: TM-T12504
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 249.00 € | ||
| 10mg | 366.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 769.00 € | ||
| 100mg | 1,049.00 € | ||
| 500mg | 2,098.00 € | ||
| 1mL*10mM (DMSO) | 282.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
SCH28080
CAS:76081-98-6
SCH28080 is a reversible and K+-competitive inhibitor of gastric H+/K+-ATPase with an IC50 value of …
Formula:
C17H15N3O
Purity:
97.12%
Color and Shape:
Solid
Molecular weight:
277.32
Ref: TM-T16865
| 1mg | 37.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 136.00 € | ||
| 25mg | 261.00 € | ||
| 50mg | 387.00 € | ||
| 100mg | 551.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
SKA-111
CAS:1369170-24-0
SKA-111 activates KCa3.1 potassium channels, modulates membrane potential in endothelial cells, and dilates rat coronary …
Formula:
C12H10N2S
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
214.29
Ref: TM-T24799
| 1mg | 69.00 € | ||
| 5mg | 149.00 € | ||
| 10mg | 245.00 € | ||
| 25mg | 496.00 € | ||
| 50mg | 711.00 € | ||
| 100mg | 993.00 € | ||
| 500mg | 1,997.00 € | ||
| 1mL*10mM (DMSO) | 166.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Bamaluzole
CAS:87034-87-5
Bamaluzole is an agonist of GABA receptor.
Formula:
C14H12ClN3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
273.72
Ref: TM-T10456
| 25mg | 1,406.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Saviprazole
CAS:121617-11-6
Saviprazole (Hoe-731), a proton pump inhibitor, is used potentially for treatment of gastric ulcer.
Formula:
C15H10F7N3O2S2
Purity:
97.73% - 99.20%
Color and Shape:
Solid
Molecular weight:
461.38
Ref: TM-T28665
| 1mg | 139.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 496.00 € | ||
| 25mg | 803.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,483.00 € | ||
| 500mg | 2,980.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
TC-AQP1-1
CAS:37710-81-9
TC-AQP1-1 blocks aquaporin 1; found via virtual screening; hinders water flux in Xenopus oocytes at …
Formula:
C12H10O4
Purity:
97.26%
Color and Shape:
Solid
Molecular weight:
218.21
Ref: TM-T24859
| 5mg | 41.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 112.00 € | ||
| 50mg | 174.00 € | ||
| 100mg | 273.00 € | ||
| 200mg | 388.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
SET 2
CAS:2313525-20-9
SET 2 is an antagonist of transient receptor potential vanilloid type 2(TRPV2) with an IC50 …
Formula:
C17H21F3N4O2S
Purity:
98.43%
Color and Shape:
Liquid
Molecular weight:
402.43
Ref: TM-T37097
| 5mg | 57.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 174.00 € | ||
| 50mg | 294.00 € | ||
| 100mg | 429.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Cilobradine hydrochloride
CAS:186097-54-1
Cilobradine hydrochloride (DK-AH 269) is an HCN Channel blocker and an open channel blocker of …
Formula:
C28H39ClN2O5
Purity:
97.46%
Color and Shape:
Solid
Molecular weight:
519.07
Ref: TM-T10813
| 1mg | 63.00 € | ||
| 5mg | 137.00 € | ||
| 10mg | 200.00 € | ||
| 25mg | 331.00 € | ||
| 50mg | 463.00 € | ||
| 100mg | 631.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
RWJ-51204
CAS:205701-85-5
RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.
Formula:
C21H19F2N3O3
Purity:
100% - 99.57%
Color and Shape:
Solid
Molecular weight:
399.39
Ref: TM-T16811
| 1mg | 327.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,850.00 € | ||
| 100mg | 2,322.00 € | ||
| 500mg | 4,549.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
GABAB receptor antagonist 1
CAS:797-17-1
(E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM.GABAB …
Formula:
C18H24O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
304.38
Ref: TM-T11350
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
