Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
P-1075
CAS:60559-98-0
P-1075 activates SUR2-KIR6 channels at 45 nM; may open mitoKATP channels and protect the heart.
Formula:
C12H17N5
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
231.3
Ref: TM-T16420
| 1mg | 60.00 € | ||
| 2mg | 87.00 € | ||
| 5mg | 125.00 € | ||
| 10mg | 200.00 € | ||
| 25mg | 369.00 € | ||
| 50mg | 553.00 € | ||
| 100mg | 791.00 € | ||
| 200mg | 628.00 € | ||
| 500mg | 1,607.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
GSK3395879
CAS:2215852-91-6
GSK3395879 is a selective and orally bioavailable antagonist of transient receptor potential vanilloid-4 (TRPV4) (IC50: …
Formula:
C20H15F4N3O5S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
485.41
Ref: TM-T15439
| 25mg | 1,967.00 € | ||
| 50mg | 2,598.00 € | ||
| 100mg | 3,458.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Maralixibat Chloride
CAS:228113-66-4
Maralixibat Chloride (LUM001 chloride), an apical, sodium-dependent, bile acid transport inhibitor, prevents enterohepatic bile acid …
Formula:
C40H56ClN3O4S
Purity:
100.00% - 98.36%
Color and Shape:
Solid
Molecular weight:
710.41
Ref: TM-T32873
| 1mg | 244.00 € | ||
| 5mg | 461.00 € | ||
| 10mg | 692.00 € | ||
| 25mg | 1,234.00 € | ||
| 50mg | 1,744.00 € | ||
| 100mg | 2,440.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
PZ-II-029
CAS:164025-44-9
PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.
Formula:
C18H15N3O3
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
321.33
Ref: TM-T28479
| 1mg | 52.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 168.00 € | ||
| 25mg | 302.00 € | ||
| 50mg | 466.00 € | ||
| 100mg | 715.00 € | ||
| 500mg | 1,435.00 € | ||
| 1mL*10mM (DMSO) | 200.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
p-Tolylmaleimide
CAS:1631-28-3
p-Tolylmaleimide (p Tolylmaleimide) is an inhibitor of the water channel and binds to Aquaporin Z.
Formula:
C11H9NO2
Purity:
98.69%
Color and Shape:
Solid
Molecular weight:
187.19
Ref: TM-T21044
| 10mg | 45.00 € | ||
| 25mg | 84.00 € | ||
| 50mg | 116.00 € | ||
| 100mg | 169.00 € | ||
| 200mg | 248.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
A 425619
CAS:581809-67-8
A 425619 (1-(4-(TRIFLUOROMETHYL)BENZYL)-3-(ISOQUINOLIN-5-YL)UREA) is a potent TRPV1 antagonist
Formula:
C18H14F3N3O
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
345.32
Ref: TM-T8562
| 1mg | 85.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € | ||
| 1mL*10mM (DMSO) | 172.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
MCT1-IN-3
CAS:2878360-80-4
MCT1-IN-3 is a monocarboxylate transporter 1 (MCT1) inhibitor.
Formula:
C22H19N3O4
Purity:
98.87%
Color and Shape:
Soild
Molecular weight:
389.4
Ref: TM-T67727
| 1mg | 113.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 551.00 € | ||
| 50mg | 771.00 € | ||
| 100mg | 1,052.00 € | ||
| 500mg | 2,112.00 € | ||
| 1mL*10mM (DMSO) | 271.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
VU0463271
CAS:1391737-01-1
VU0463271: KCC2 antagonist, IC50 61 nM, >100x selective over NKCC1, inactive on other GPCRs, channels, …
Formula:
C19H18N4OS2
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
382.5
Ref: TM-T17243
| 5mg | 49.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 240.00 € | ||
| 100mg | 354.00 € | ||
| 200mg | 504.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
CFTR corrector 12
CAS:958941-60-1
CFTR corrector 12 is a CFTR corrector that rescues all mutant proteins except M760R ABCA3 …
Formula:
C19H21ClN4O2S2
Purity:
99.78%
Color and Shape:
Liquid
Molecular weight:
436.98
Ref: TM-T79578
| 1mg | 171.00 € | ||
| 5mg | 427.00 € | ||
| 10mg | 605.00 € | ||
| 25mg | 925.00 € | ||
| 50mg | 1,293.00 € | ||
| 100mg | 1,752.00 € | ||
| 200mg | 2,361.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
(Rac)-AMG8379
CAS:1641574-26-6
(Rac)-AMG8379 ((Rac)-AMG8380) is a racemate of AMG8379 which is an orally active and selective sulfonamide …
Formula:
C25H16ClF2N3O5S
Purity:
99.6%
Color and Shape:
Solid
Molecular weight:
543.93
Ref: TM-T12655
| 1mg | 183.00 € | ||
| 2mg | 274.00 € | ||
| 5mg | 421.00 € | ||
| 10mg | 618.00 € | ||
| 25mg | 926.00 € | ||
| 50mg | 1,295.00 € | ||
| 100mg | 1,773.00 € | ||
| 200mg | 1,404.00 € | ||
| 500mg | 3,511.00 € | ||
| 1mL*10mM (DMSO) | 533.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
BPO-27 racemate
CAS:1314873-02-3
BPO-27 racemate (BPO-27 (racemate)) is an effective CFTR inhibitor with IC50 of 8 nM.
Formula:
C26H18BrN3O6
Purity:
98.19%
Color and Shape:
Solid
Molecular weight:
548.34
Ref: TM-T10591
| 1mg | 45.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 169.00 € | ||
| 25mg | 271.00 € | ||
| 50mg | 395.00 € | ||
| 100mg | 545.00 € | ||
| 200mg | 731.00 € | ||
| 1mL*10mM (DMSO) | 130.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
AMG-0347
CAS:946615-43-6
AMG-0347 inhibits TRPA1 ion channels in sensory neurons, blocking pain perception.
Formula:
C24H26F3N3O2
Purity:
99.7%
Color and Shape:
Solid
Molecular weight:
445.48
Ref: TM-T29968
| 1mg | 369.00 € | ||
| 5mg | 901.00 € | ||
| 10mg | 1,205.00 € | ||
| 25mg | 1,818.00 € | ||
| 50mg | 2,443.00 € | ||
| 100mg | 3,291.00 € | ||
| 1mL*10mM (DMSO) | 939.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
CLP257
CAS:1181081-71-9
CLP257 is a selective K+-Cl− cotransporter KCC2 activator (EC50: 616 nM) and it is inactive …
Formula:
C14H14FN3O2S
Purity:
98.13%
Color and Shape:
Solid
Molecular weight:
307.34
Ref: TM-T14984
| 1mg | 45.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 279.00 € | ||
| 50mg | 456.00 € | ||
| 100mg | 672.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
LFS-1107
CAS:1799330-91-8
LFS-1107, a reversible CRM1 inhibitor (Kd: 12.5 pM), selectively targets and eliminates ENKTL cells, offering …
Formula:
C12H11N5OS2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
305.38
Ref: TM-T81936
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 29 Jan 2025
SCS
CAS:3232-36-8
SCS is a GABAA receptor antagonist.
Formula:
C14H12N2O3
Purity:
98.89%
Color and Shape:
Solid
Molecular weight:
256.26
Ref: TM-T23339
| 10mg | 42.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | 89.00 € | ||
| 100mg | 130.00 € | ||
| 200mg | 182.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
PF-05105679
CAS:1398583-31-7
PF-05105679 is a selective TRPM8 antagonist (IC50 = 103 nM). PF-05105679 can be used in …
Formula:
C26H21FN2O3
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
428.45
Ref: TM-T16483
| 1mg | 48.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 159.00 € | ||
| 25mg | 302.00 € | ||
| 50mg | 467.00 € | ||
| 100mg | 701.00 € | ||
| 200mg | 926.00 € | ||
| 500mg | 1,412.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Linaprazan
CAS:248919-64-4
Linaprazan (AZD0865) inhibits gastric H+,K+-ATPase by K+-competitive binding with an IC50 of 1.0 μM.
Formula:
C21H26N4O2
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
366.46
Ref: TM-T10435
| 5mg | 50.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 204.00 € | ||
| 100mg | 344.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
TPA 023
CAS:252977-51-8
TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 …
Formula:
C20H22FN7O
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
395.43
Ref: TM-T17144
| 1mg | 222.00 € | ||
| 5mg | 538.00 € | ||
| 10mg | 806.00 € | ||
| 25mg | 1,188.00 € | ||
| 50mg | 1,605.00 € | ||
| 100mg | 2,162.00 € | ||
| 1mL*10mM (DMSO) | 591.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
DNDS
CAS:3709-43-1
DNDS is a channel blocker of voltage-dependent cystic fibrosis transmembrane conductance regulator (CFTR).
Formula:
C14H8N2Na2O10S2
Purity:
99.88%
Color and Shape:
Physical Description White Powder (Ntp 1992)
Molecular weight:
474.33
Ref: TM-T20341
| 1g | 34.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
(+)-Bicuculline methiodide
CAS:40709-69-1
(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in …
Formula:
C21H20INO6
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
509.29
Ref: TM-T22604
| 1mg | 38.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
