Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
U-89843A
CAS:157013-85-9
U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents …
Formula:
C16H24ClN5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
321.85
Ref: TM-T78560
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
XE991
CAS:122955-42-4
XE991 is a Kv7 (KCNQ) channel blocker.XE 991 dihydrochloride inhibits Kv7.1 (KCNQ1) and M-current and …
Formula:
C26H20N2O
Purity:
99.51%
Color and Shape:
Liquid
Molecular weight:
376.45
Ref: TM-T78570
| 1mg | 48.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 153.00 € | ||
| 25mg | 283.00 € | ||
| 50mg | 522.00 € | ||
| 100mg | 838.00 € | ||
| 500mg | 1,681.00 € | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Orphenadrine
CAS:83-98-7
Orphenadrine is a noncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist that inhibits clonal HERG channels in a …
Formula:
C18H23NO
Purity:
99.26% - 99.38%
Color and Shape:
Liquid
Molecular weight:
269.38
Ref: TM-T68599
| 5mg | 57.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 108.00 € | ||
| 50mg | 156.00 € | ||
| 100mg | 225.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
TC-I 2014
CAS:1221349-53-6
TC-I 2014 shows antiallodynic properties in pain models.
Formula:
C23H19F6N3O
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
467.41
Ref: TM-T17006
| 1mg | 60.00 € | ||
| 5mg | 127.00 € | ||
| 10mg | 202.00 € | ||
| 25mg | 406.00 € | ||
| 50mg | 655.00 € | ||
| 100mg | 1,074.00 € | ||
| 200mg | 1,454.00 € | ||
| 1mL*10mM (DMSO) | 133.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Phaclofen
CAS:114012-12-3
GABAB antagonist
Formula:
C9H13ClNO3P
Purity:
99.32%
Color and Shape:
White Solid
Molecular weight:
249.63
Ref: TM-T23147
| 1mg | 81.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 283.00 € | ||
| 25mg | 652.00 € | ||
| 50mg | 908.00 € | ||
| 100mg | 1,216.00 € | ||
| 200mg | 1,644.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
GX-674
CAS:1432913-36-4
GX-674 is a highly potent and selective voltage-gated sodium channel 1.7 (Nav1.7) antagonist with an …
Formula:
C21H13ClF2N6O3S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
534.95
Ref: TM-T22829
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
ANO1-IN-1
CAS:407587-01-3
ANO1-IN-1 blocks ANO1/2 channels (IC50: 2.56/15.43 μM) and hinders glioma cell growth.
Formula:
C18H28N2O2S
Purity:
99.66%
Color and Shape:
Liquid
Molecular weight:
336.49
Ref: TM-T61051
| 5mg | 47.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 116.00 € | ||
| 50mg | 180.00 € | ||
| 100mg | 264.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
ABCG2-IN-2
CAS:2559759-59-8
ABCG2-IN-2 is a potent inhibitor of ABCG2, exhibiting favorable oral pharmacokinetic profiles in mice, and …
Formula:
C25H34N4O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
454.56
Ref: TM-T79514
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Suriclone
CAS:53813-83-5
Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.
Formula:
C20H20ClN5O3S2
Purity:
98.17% - 98.52%
Color and Shape:
Solid
Molecular weight:
477.99
Ref: TM-T28887
| 1mg | 143.00 € | ||
| 5mg | 333.00 € | ||
| 10mg | 504.00 € | ||
| 25mg | 817.00 € | ||
| 50mg | 1,121.00 € | ||
| 100mg | 1,510.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
ZM 226600
CAS:147695-92-9
ZM 226600 is an ATP-sensitive potassium channel opener with an EC50 value of 500 nM. …
Formula:
C16H14F3NO4S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
373.35
Ref: TM-T23563
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 145.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 335.00 € | ||
| 200mg | 469.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
TWIK-1/TREK-1-IN-2
CAS:1440532-32-0
TWIK-1/TREK-1-IN-2 (Compound 2g) serves as an inhibitor of both TWIK-1 and TREK-1, targeting the TREK-1 …
Formula:
C20H29F3N2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
386.45
Ref: TM-T78869
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Leminoprazole
CAS:104340-86-5
Leminoprazole is an orally available H+,K(+)-ATPase inhibitor that protects gastric mucosal cells from various cellular …
Formula:
C19H23N3OS
Purity:
98.87% - 99.56%
Color and Shape:
Solid
Molecular weight:
341.47
Ref: TM-T27812
| 1mg | 128.00 € | ||
| 5mg | 304.00 € | ||
| 10mg | 457.00 € | ||
| 25mg | 747.00 € | ||
| 50mg | 1,026.00 € | ||
| 100mg | 1,406.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
PD-118057
CAS:313674-97-4
PD-118057, a potent hERG activator, may treat long QT syndrome and heart failure without hERG …
Formula:
C21H17Cl2NO2
Purity:
98.97% - 99.16%
Color and Shape:
Solid
Molecular weight:
386.27
Ref: TM-T16444
| 1mg | 96.00 € | ||
| 5mg | 202.00 € | ||
| 10mg | 311.00 € | ||
| 25mg | 597.00 € | ||
| 50mg | 948.00 € | ||
| 100mg | 1,510.00 € | ||
| 1mL*10mM (DMSO) | 224.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
TRAM 39
CAS:197525-99-8
TRAM 39 (2-Chloro-α,α-diphenylbenzeneacetonitrile) is a selective blocker of intermediate-conductance Ca2+-activated K+channels.
Formula:
C20H14ClN
Purity:
99.51%
Color and Shape:
Solid
Molecular weight:
303.78
Ref: TM-T23471
| 1mg | 35.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 107.00 € | ||
| 25mg | 210.00 € | ||
| 50mg | 335.00 € | ||
| 100mg | 530.00 € | ||
| 500mg | 1,121.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Tracazolate hydrochloride
CAS:1135210-68-2
Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant …
Formula:
C16H25ClN4O2
Purity:
99.07%
Color and Shape:
Solid
Molecular weight:
340.85
Ref: TM-T23470
| 10mg | 116.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 21 Apr 2025
Lupanine
CAS:550-90-3
Lupanine has a weak sedative effect on the central nervous system, interaction with specific drugs …
Formula:
C15H24N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
248.36
Ref: TM-TMA0805
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
E2730
CAS:1520073-91-9
E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying …
Formula:
C9H8F4N2O2S
Purity:
98.22% - 98.54%
Color and Shape:
Liquid
Molecular weight:
284.23
Ref: TM-T79399
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
BPDBA
CAS:312281-74-6
BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory …
Formula:
C19H20Cl2N2O
Purity:
99.24% - 99.86%
Color and Shape:
Solid
Molecular weight:
363.28
Ref: TM-T26891
| 5mg | 40.00 € | ||
| 10mg | 58.00 € | ||
| 25mg | 109.00 € | ||
| 50mg | 170.00 € | ||
| 100mg | 273.00 € | ||
| 200mg | 378.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
AGN-201904
CAS:651729-53-2
AGN-201904 is a proton pump inhibitor, an omeprazole prodrug, which delays aging and may be …
Formula:
C25H25N3O8S2
Purity:
97.32%
Color and Shape:
Solid
Molecular weight:
559.61
Ref: TM-T23667
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Ani9
CAS:356102-14-2
Ani9 selectively blocks ANO1/TMEM16A with a 77 nM IC50, useful for ANO1 research and treating …
Formula:
C17H17ClN2O3
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
332.78
Ref: TM-T26630
| 1mg | 39.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 454.00 € | ||
| 100mg | 655.00 € | ||
| 500mg | 1,406.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
