Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
R 56865
CAS:104606-13-5
R 56865 is a weak potential-operated channel inhibitor that inhibits the late sodium current in …
Formula:
C23H28FN3OS
Purity:
99.08%
Color and Shape:
Solid
Molecular weight:
413.55
Ref: TM-T26016
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
GAL-021 sulfate
CAS:1380342-00-6
GAL-021 sulfate is a BKCa channel blocker that inhibits the analgesic effects of opioids and …
Formula:
C11H24N6O5S
Purity:
99.68%
Color and Shape:
Liquid
Molecular weight:
352.41
Ref: TM-T61239
| 1mg | 74.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 225.00 € | ||
| 25mg | 379.00 € | ||
| 50mg | 563.00 € | ||
| 100mg | 803.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Istaroxime hydrochloride
CAS:374559-48-5
Istaroxime hydrochloride (PST2744 hydrochloride) is a Na+/K+-ATPase inhibitor and SERCA 2 activator, and is a …
Formula:
C21H33ClN2O3
Color and Shape:
Solid
Molecular weight:
396.95
Ref: TM-T15599
| 2mg | 132.00 € | ||
| 5mg | 217.00 € | ||
| 10mg | 358.00 € | ||
| 50mg | 750.00 € | ||
| 100mg | 1,121.00 € | ||
| 1mL*10mM (DMSO) | 240.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Bamocaftor
CAS:2204245-48-5
Bamocaftor corrects CFTR in CF, restoring F508del-CFTR function, used with tezacaftor and VX-561 for F508del/MF …
Formula:
C28H32F3N5O4S
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
591.65
Ref: TM-T30293
| 1mg | 354.00 € | ||
| 5mg | 847.00 € | ||
| 10mg | 1,159.00 € | ||
| 25mg | 1,700.00 € | ||
| 50mg | 2,308.00 € | ||
| 100mg | 3,117.00 € | ||
| 1mL*10mM (DMSO) | 1,225.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
ZTZ240
CAS:325457-98-5
ZTZ240 is a KCNQ2 channel activator used in the study of epilepsy.
Formula:
C12H8ClFN2O
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
250.66
Ref: TM-T29236
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
ABCG2-IN-1
CAS:2559759-40-7
ABCG2-IN-1 (compound K2), an analog of Ko143, constitutes an orally active inhibitor targeting ABCG2 with …
Formula:
C26H36N4O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
468.59
Ref: TM-T79513
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Sarmazenil
CAS:78771-13-8
Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used …
Formula:
C15H14ClN3O3
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
319.74
Ref: TM-T16844
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
CBS9106
CAS:1076235-04-5
CBS9106 (SL-801) is a CRM1 inhibitor with CRM1-degrading and anti-tumor activity that inhibits CRM1-dependent nuclear …
Formula:
C18H21ClF3N3O3
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
419.83
Ref: TM-T14885
| 1mg | 250.00 € | ||
| 5mg | 612.00 € | ||
| 10mg | 847.00 € | ||
| 25mg | 1,311.00 € | ||
| 50mg | 1,786.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
(E)-GABAB receptor antagonist 1
CAS:1611483-29-4
(E)-GABAB antagonist 1 inhibits GABA IP3 production, with an IC50 of 37.9 μM and acts …
Formula:
C18H24O4
Purity:
95.26%
Color and Shape:
Solid
Molecular weight:
304.38
Ref: TM-T11137
| 1mg | 115.00 € | ||
| 5mg | 255.00 € | ||
| 10mg | 375.00 € | ||
| 25mg | 562.00 € | ||
| 50mg | 787.00 € | ||
| 100mg | 1,074.00 € | ||
| 200mg | 1,454.00 € | ||
| 1mL*10mM (DMSO) | 246.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
UK 66914
CAS:113049-11-9
UK 66914 is a K(+) channel blocker for the study of cardiac arrhythmias.
Formula:
C18H24N4O3S
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
376.47
Ref: TM-T29050
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
NC-1300-B
CAS:104340-52-5
NC-1300-B inhibits H(+)-K(+)-ATPase and is used in the study of gastric ulcers.
Formula:
C17H19N3OS
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
313.42
Ref: TM-T28136
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Riluzole hydrochloride
CAS:850608-87-6
Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).
Formula:
C8H6ClF3N2OS
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
270.66
Ref: TM-T41265
| 25mg | 37.00 € | ||
| 50mg | 52.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
GX-585
CAS:2098540-08-8
GX-585 is a novel potent inhibitor of NaV1.7 and highly selective against NaV1.5, having limited …
Formula:
C24H25Cl2FN4O3S
Purity:
100% - 99.18%
Color and Shape:
Liquid
Molecular weight:
539.45
Ref: TM-T69915
| 1mg | 279.00 € | ||
| 5mg | 683.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,415.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,612.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
PG01
CAS:853138-65-5
PG01 is a potent CFTR Cl-channel potentiator, effective against ΔF508 (Ka 0.3 μM), and also …
Formula:
C28H29N3O2
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
439.55
Ref: TM-T16516
| 1mg | 84.00 € | ||
| 5mg | 215.00 € | ||
| 10mg | 324.00 € | ||
| 25mg | 520.00 € | ||
| 50mg | 702.00 € | ||
| 100mg | 950.00 € | ||
| 200mg | 1,283.00 € | ||
| 500mg | 3,192.00 € | ||
| 1mL*10mM (DMSO) | 210.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
SCH 50911
CAS:733717-87-8
SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow …
Formula:
C8H15NO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
173.21
Ref: TM-T12867L
| 50mg | 2,480.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Amsacrine
CAS:51264-14-3
Amsacrine (AMSA) (mAMSA) an antineoplastic agent which can intercalate into the DNA of tumor cells.
Formula:
C21H19N3O3S
Purity:
98.59%
Color and Shape:
Yellow Crystalline Powder Solid
Molecular weight:
393.46
Ref: TM-T1206
| 10mg | 47.00 € | ||
| 25mg | 60.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
TRPM4-IN-2
CAS:667411-04-3
NBA, or TRPM4-IN-2, is a potent TRPM4 inhibitor with IC50 of 0.16 μM, used in …
Formula:
C19H14ClNO4
Purity:
99.21%
Color and Shape:
Liquid
Molecular weight:
355.77
Ref: TM-T61275
| 2mg | To inquire |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Vernakalant
CAS:794466-70-9
Vernakalant (RSD-1235) is a mixed ion channel blocker.
Formula:
C20H31NO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
349.46
Ref: TM-TQ0307
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Lirequinil
CAS:143943-73-1
Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.
Formula:
C26H25ClN2O3
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
448.94
Ref: TM-T27838
| 1mg | 158.00 € | ||
| 5mg | 380.00 € | ||
| 10mg | 570.00 € | ||
| 25mg | 912.00 € | ||
| 50mg | 1,216.00 € | ||
| 100mg | 1,663.00 € | ||
| 500mg | 3,315.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
RO 4938581
CAS:883093-10-5
RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, …
Formula:
C13H8BrF2N5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
352.14
Ref: TM-T16794
| 25mg | 1,169.00 € | ||
| 50mg | 1,529.00 € | ||
| 100mg | 2,517.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
