Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
Xilmenolone
CAS:2368807-26-3
Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].
Formula:
C26H37N3O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
423.59
Ref: TM-T78670
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
VMAT2-IN-2 tosylate
CAS:2608770-12-1
VMAT2-IN-2 tosylate is a potent inhibitor of VMAT2 and is applicable in the research of …
Formula:
C27H36F3NO6S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
559.64
Ref: TM-T79061
| 25mg | 1,827.00 € | ||
| 50mg | 2,412.00 € | ||
| 100mg | 3,178.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
Soraprazan
CAS:261944-46-1
Soraprazan (BYK61359) is a potassium channel inhibitor that inhibits gastric acid secretion and may ameliorate …
Formula:
C21H25N3O3
Purity:
97.69%
Color and Shape:
Solid
Molecular weight:
367.44
Ref: TM-T12977
| 5mg | 419.00 € | ||
| 25mg | 1,419.00 € | ||
| 50mg | 1,884.00 € | ||
| 100mg | 3,048.00 € | ||
| 1mL*10mM (DMSO) | 406.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
DPO-1
CAS:43077-30-1
DPO-1 is a blocker of IKur ultrarapid delayed rectifier potassium current and KV1.5 channels
Formula:
C22H29OP
Purity:
97.52%
Color and Shape:
Solid
Molecular weight:
340.44
Ref: TM-T22745
| 2mg | 42.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 200.00 € | ||
| 50mg | 299.00 € | ||
| 100mg | 430.00 € | ||
| 200mg | 602.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
(-)-Bicuculline methochloride
CAS:53552-05-9
(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.
Formula:
C21H20ClNO6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
417.84
Ref: TM-T12044
| 5mg | 157.00 € | ||
| 10mg | 274.00 € | ||
| 25mg | 598.00 € | ||
| 50mg | 936.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
CP-409092
CAS:194098-25-4
CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.
Formula:
C17H19N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
297.35
Ref: TM-T10869L
| 25mg | 1,688.00 € | ||
| 50mg | 2,225.00 € | ||
| 100mg | 2,897.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
L-822179
CAS:215874-86-5
L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with …
Formula:
C17H14N8O2
Purity:
98.34% - 98.74%
Color and Shape:
Solid
Molecular weight:
362.35
Ref: TM-T24381
| 1mg | 44.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 180.00 € | ||
| 50mg | 268.00 € | ||
| 100mg | 383.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
Co 102862
CAS:181144-66-1
Co 102862 is a voltage-gated sodium channel blocker. Co 102862 can be used for anticonvulsant …
Formula:
C14H12FN3O2
Purity:
99.54%
Color and Shape:
Solid
Molecular weight:
273.26
Ref: TM-T22675
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 140.00 € | ||
| 50mg | 209.00 € | ||
| 100mg | 341.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
CRF1 receptor antagonist-1
CAS:2635364-30-4
CRF1 Receptor Antagonist-1 (Compound 2), a CRF1 receptor antagonist, is utilized in research pertaining to …
Formula:
C27H28ClFN2O2S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
499.04
Ref: TM-T79793
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 10 Feb 2025
Mesendogen
CAS:864716-85-8
Mesendogen is an inhibitor of transient receptor potential cation channel, subfamily M, member 6 (TRPM6) …
Formula:
C18H16ClF3N2OS
Purity:
98.90%
Color and Shape:
Solid
Molecular weight:
400.85
Ref: TM-T28020
| 1mg | 42.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 300.00 € | ||
| 50mg | 523.00 € | ||
| 100mg | 736.00 € | ||
| 1mL*10mM (DMSO) | 103.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
AMG2850
CAS:1470018-52-0
AMG2850 is a potent, orally bioavailable, and selective antagonist of transient receptor potential melastatin 8 …
Formula:
C19H17F6N3O
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
417.35
Ref: TM-T10300
| 1mg | 72.00 € | ||
| 5mg | 164.00 € | ||
| 10mg | 239.00 € | ||
| 25mg | 430.00 € | ||
| 50mg | 638.00 € | ||
| 100mg | 818.00 € | ||
| 1mL*10mM (DMSO) | 175.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
CFTR corrector 16
CAS:1210305-23-9
CFTRcorrector 16 (Compound 39) is a corrector of the cystic fibrosis transmembrane conductance regulator (CFTR), …
Formula:
C27H26ClN5O2S
Color and Shape:
Liquid
Molecular weight:
520.05
Ref: TM-T200113
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 10 Mar 2025
(+)-Tetrabenazine
CAS:1026016-83-0
(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 …
Formula:
C19H27NO3
Purity:
98.31%
Color and Shape:
Solid
Molecular weight:
317.42
Ref: TM-T13134
| 5mg | 51.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 142.00 € | ||
| 100mg | 221.00 € | ||
| 500mg | 547.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
TRPA1 Antagonist 1
CAS:1984825-08-2
TRPA1 Antagonist 1 is an antagonist of TRPA1(IC50: 8 nM) and is a methylene phosphate …
Formula:
C24H22F6N5Na2O7PS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
715.47
Ref: TM-T13212
| 25mg | 3,079.00 € | ||
| 50mg | 4,094.00 € | ||
| 100mg | 5,701.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
SP100030 analogue 1
CAS:154934-68-6
SP100030 analogue 1 (compound 11) is a selective transcription activation (SITA) inhibitor within the SP100030 …
Formula:
C13H5ClF7N3O
Color and Shape:
Liquid
Molecular weight:
387.64
Ref: TM-T89990
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 10 Mar 2025
CFTR corrector 15
CAS:1170387-92-4
CFTR Corrector 15 (Compound 4172) serves as a corrector for cystic fibrosis transmembrane conductance regulator …
Formula:
C24H22ClN5O2S
Color and Shape:
Liquid
Molecular weight:
479.98
Ref: TM-T89966
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 10 Mar 2025
Picrotoxinin
CAS:17617-45-7
Picrotoxinin blocks chloride channels, antagonizes GABAA noncompetitively (IC50: 1.15 μM, α1β2γ2L), and induces convulsions.
Formula:
C15H16O6
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
292.28
Ref: TM-T16535
| 10mg | 47.00 € | ||
| 25mg | 67.00 € | ||
| 50mg | 89.00 € | ||
| 100mg | 133.00 € | ||
| 500mg | 314.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Lubeluzole dihydrochloride
CAS:144665-09-8
Lubeluzole (dihydrochloride) acts as a neuroprotective agent by blocking neuronal voltage-gated sodium channels and also …
Formula:
C22H27Cl2F2N3O2S
Color and Shape:
Liquid
Molecular weight:
506.44
Ref: TM-T200178
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 10 Mar 2025
GSK2798745
CAS:1419609-94-1
GSK2798745 is an orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker (IC50s: …
Formula:
C25H28N6O3
Color and Shape:
Solid
Molecular weight:
460.53
Ref: TM-T15434
| 25mg | 2,106.00 € | ||
| 50mg | 2,789.00 € | ||
| 100mg | 3,744.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Valbenazine tosylate
CAS:1639208-54-0
Valbenazine tosylate, the tosylate salt of valbenazine, is a vesicular monoamine transporter 2 (VMAT2) inhibitor …
Formula:
C38H54N2O10S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
762.97
Ref: TM-T22452
| 25mg | 2,662.00 € | ||
| 50mg | 3,533.00 € | ||
| 100mg | 4,860.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
