Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(97 products)
- Adiponectin receptor(5 products)
- CFTR(66 products)
- CGRP Receptor(53 products)
- Calcium Channel(573 products)
- Chloride channel(54 products)
- GABA Receptor(373 products)
- Monoamine Transporter(30 products)
- Monocarboxylate transporter(18 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(10 products)
- OAT(32 products)
- OCT(7 products)
- P-gp(55 products)
- Potassium Channel(304 products)
- Proton pump(42 products)
- SGLT(31 products)
- Sodium Channel(260 products)
- TRP/TRPV Channel(95 products)
Show 13 more subcategories
Found 2734 products of "Membrane Transporter/Ion Channel"
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Nerispirdine
CAS:Nerispirdine is a biochemical that inhibits batrachotoxin binding to voltage-dependent sodium channels.Formula:C17H18FN3Color and Shape:SolidMolecular weight:283.34Ro 18-3981
CAS:Ro 18-3981 inhibits myocardial Ca2+ channels; KD is 1.0 nM, close to IC50 for ICa block (2.3 nM).Formula:C24H33N3O8SColor and Shape:SolidMolecular weight:523.6Azelnidipine, (R)-
CAS:Azelnidipine is an L-type CCB that improves HF severity and cardiac nerve activity in HT and HFpEF compared to cilnidipine.Formula:C33H34N4O6Color and Shape:SolidMolecular weight:582.65SR-33805
CAS:SR-33805: calcium channel blocker for atherosclerosis/heart failure, enhances myocyte function, modulates myofilament phosphorylation.Formula:C32H40N2O5SColor and Shape:SolidMolecular weight:564.74TG41
CAS:TG41 is a GABAA receptors positive modulator.Formula:C18H13BrCl2N2O2Purity:98%Color and Shape:SolidMolecular weight:440.12Caldaret
CAS:Caldaret is an intracellular Ca2+ handling modulator that acts through reverse mode Na+/Ca2+ exchanger inhibition.Formula:C11H16N2O3SColor and Shape:SolidMolecular weight:256.32CAY10719
CAS:CAY10719 selectively inhibits ABCG2 (IC50 = 0.23 μM), reverses SN 38 resistance, and inhibits ATPase, with low ABCG1 activity.Formula:C25H20Cl2N2O2Color and Shape:SolidMolecular weight:451.34PBI-51
CAS:PBI-51 is a competitive inhibitor of abscisic acid-regulated gene expression.Formula:C15H22O3Color and Shape:SolidMolecular weight:250.33Corrector C4
CAS:Corrector C4, a corrector commonly used to study cystic fibrosis mutants, works by alleviating the interaction between CFTR transmembrane domain mutants andFormula:C21H17ClN4O2S2Purity:99.98%Color and Shape:SolidMolecular weight:456.97ORM-10962
CAS:ORM-10962 is a potent, highly selective inhibitor of sodium-calcium exchanger (NCX) (for the reverse and forward mode inhibition with IC50 values of 67 and 55Formula:C27H29N3O4Purity:98%Color and Shape:SolidMolecular weight:459.54Zatebradine hydrochloride
CAS:Zatebradine hydrochloride (UL-FS-49CL) inhibits HCN channels (IC50: ~1.9 µM) blocking human HCN1-4 currents effectively.Formula:C26H37ClN2O5Purity:98.61%Color and Shape:SolidMolecular weight:493.04Ref: TM-T13387L
500mgTo inquire5mg50.00€1mL*10mM (DMSO)51.00€10mg73.00€25mg146.00€50mg268.00€100mg411.00€NMDA receptor modulator 3
CAS:NMDA receptor modulator 3 (Compound 99) is a potent modulator of NMDA receptor that can be used in the research of neurological disorder [1].Formula:C12H9F3N2O2SColor and Shape:SolidMolecular weight:302.27Topiramate lithium
CAS:Topiramate lithium: antiepileptic, GluR5 antagonist, enhances GABA, inhibits kainate/AMPA, Na+/Ca2+ channels; ↑ K+ conductance; ↓ carbonic anhydrase.Formula:C12H20LiNO8SColor and Shape:SolidMolecular weight:345.29AMG9678
CAS:AMG9678 is a selective, potent, orally active TRPM8 antagonist (IC50: 31.2 nM).Formula:C20H18F6N2OColor and Shape:SolidMolecular weight:416.36Lidoflazine
CAS:Lidoflazine: antianginal, blocks HERG K+ & Ca channels, risks QT prolongation & arrhythmia.Formula:C30H35F2N3OPurity:98%Color and Shape:SolidMolecular weight:491.62PF-0713
CAS:PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.Formula:C14H22OPurity:98%Color and Shape:SolidMolecular weight:206.32P-gp inhibitor 1
CAS:P-gp inhibitor 1 inhibits reversing P-glycoprotein-mediated multidrug resistance with an EC50 of 57.9 nM (K562/A02 cells).Formula:C32H31N5O2Purity:98.65%Color and Shape:SolidMolecular weight:517.62Ref: TM-T12341
5mg50.00€1mL*10mM (DMSO)58.00€10mg84.00€25mg150.00€50mg219.00€100mg304.00€200mg419.00€(2R,3S)-Chlorpheg
CAS:(2R,3S)-Chlorpheg is a NMDA receptor antagonist.Formula:C11H12ClNO4Purity:98%Color and Shape:SolidMolecular weight:257.67Cyclic ADP-ribose
CAS:cADPR, made from NAD+, boosts calcium in cells via Ryanodine receptors and TRPM2 channels.Formula:C15H21N5O13P2Purity:98%Color and Shape:Lyophilized PowderMolecular weight:541.3PF05020182
CAS:PF05020182, a Kv7.2/4 opener, prevents convulsions in MES tests, supporting its potential use in refractory epilepsy treatment.Formula:C18H30N4O4Color and Shape:SolidMolecular weight:366.46
