Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
NS11394
CAS:951650-22-9
NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile …
Formula:
C23H19N3O
Purity:
99.44% - 99.86%
Color and Shape:
Solid
Molecular weight:
353.42
Ref: TM-T2067
| 2mg | 33.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 308.00 € | ||
| 200mg | 442.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
M084
CAS:51314-51-3
M084 (N-Butyl-1H-benzimidazol-2-amine) is a blocker of TRPC4/5 channel, with antidepressant and anxiolytic effects.
Formula:
C11H15N3
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
189.26
Ref: TM-T8607
| 1mg | 85.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € | ||
| 1mL*10mM (DMSO) | 141.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
GsMTx4 TFA (1209500-46-8 free base)
GsMTx4 TFA is a spider venom peptide that selectively inhibits cationic permeable mechanically-sensitive channels (MSCs). …
Formula:
C185H273N49O45S6·C2F3HO2
Purity:
98% - 99.81%
Color and Shape:
Solid
Molecular weight:
4209.84
Ref: TM-TP1300
| 1mg | 435.00 € | ||
| 5mg | 1,003.00 € | ||
| 10mg | 1,352.00 € | ||
| 25mg | 2,033.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
(E)-3,4,5-Trimethoxycinnamic acid
CAS:20329-98-0
(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium …
Formula:
C12H14O5
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
238.24
Ref: TM-TN2865
| 1g | 128.00 € | ||
| 100mg | 46.00 € | ||
| 500mg | 87.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
Dofetilide
CAS:115256-11-6
Dofetilide (UK 68789), a class III antiarrhythmic sulfonamide, blocks Ikr cardiac channels, prolongs action potential, …
Formula:
C19H27N3O5S2
Purity:
97.85% - 99.06%
Color and Shape:
Off-White Or Yellowish Crystalline Powder
Molecular weight:
441.56
Ref: TM-T6476
| 5mg | 54.00 € | ||
| 10mg | 68.00 € | ||
| 25mg | 115.00 € | ||
| 50mg | 174.00 € | ||
| 100mg | 245.00 € | ||
| 200mg | 472.00 € | ||
| 500mg | 764.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
Basmisanil
CAS:1159600-41-5
Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in …
Formula:
C21H20FN3O5S
Purity:
99.21% - ≥98%
Color and Shape:
Solid
Molecular weight:
445.46
Ref: TM-T7165
| 2mg | 38.00 € | ||
| 5mg | 55.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 121.00 € | ||
| 50mg | 193.00 € | ||
| 100mg | 375.00 € | ||
| 500mg | 844.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
ONO-8590580
CAS:1802661-73-9
ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.
Formula:
C21H21FN6
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
376.43
Ref: TM-TQ0040
| 1mg | 65.00 € | ||
| 2mg | 92.00 € | ||
| 5mg | 125.00 € | ||
| 10mg | 167.00 € | ||
| 25mg | 372.00 € | ||
| 50mg | 556.00 € | ||
| 100mg | 793.00 € | ||
| 1mL*10mM (DMSO) | 139.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
Acetoxyvalerensre
CAS:81397-67-3
Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a …
Formula:
C17H24O4
Purity:
98.22%
Color and Shape:
Solid
Molecular weight:
292.37
Ref: TM-TN6773
| 1mg | 128.00 € | ||
| 2mg | 185.00 € | ||
| 5mg | 278.00 € | ||
| 10mg | 421.00 € | ||
| 25mg | 694.00 € | ||
| 50mg | 979.00 € | ||
| 1mL*10mM (DMSO) | 281.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
AZD7325
CAS:942437-37-8
AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.
Formula:
C19H19FN4O2
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
354.38
Ref: TM-T7699
| 5mg | 69.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 276.00 € | ||
| 100mg | 418.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
AUT1
CAS:1311136-84-1
AUT1 (AUT-1) is a novel specific modulator of Kv3 channels (EC50: 4.7 and 4.9 uM …
Formula:
C18H19N3O4
Purity:
99.80%
Color and Shape:
Solid
Molecular weight:
341.36
Ref: TM-T5183
| 1mg | 35.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 314.00 € | ||
| 100mg | 458.00 € | ||
| 1mL*10mM (DMSO) | 82.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
Temgicoluril
CAS:10095-06-4
Temgicoluril (mebikar) acts on GABA Receptor.
Formula:
C8H14N4O2
Purity:
99.80%
Color and Shape:
Solid
Molecular weight:
198.22
Ref: TM-T9424
| 25mg | 39.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 8 Jan 2025
Iptakalim Hydrochloride
CAS:642407-63-4
Iptakalim, a lipophilic para-amino compound, is a novel ATP-sensitive potassium channel (KATP) opener, as well …
Formula:
C9H22ClN
Purity:
95%
Color and Shape:
Solid
Molecular weight:
179.731
Ref: TM-T27624
| 5mg | 52.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 224.00 € | ||
| 100mg | 337.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
GSK369796 Dihydrochloride
CAS:1010411-21-8
GSK369796 Dihydrochloride (N-tert-butylisoquine),is an anti-malaria drug candidate.
Formula:
C20H24Cl3N3O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
428.78
Ref: TM-T7195
| 1mg | 78.00 € | ||
| 2mg | 99.00 € | ||
| 5mg | 148.00 € | ||
| 10mg | 193.00 € | ||
| 25mg | 368.00 € | ||
| 50mg | 556.00 € | ||
| 100mg | 793.00 € | ||
| 1mL*10mM (DMSO) | 144.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
Rosuvastatin
CAS:287714-41-4
Rosuvastatin (ZD4522) is an inhibitor of HMG-CoA reductase (HMGCR). Rosuvastatin has hypolipidemic and antiatherosclerotic effects. …
Formula:
C22H28FN3O6S
Purity:
95.24% - 99.8%
Color and Shape:
Solid
Molecular weight:
481.54
Ref: TM-T1676
| 5mg | 49.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 121.00 € | ||
| 50mg | 163.00 € | ||
| 100mg | 259.00 € | ||
| 200mg | 363.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
Rimtuzalcap
CAS:2167246-24-2
Rimtuzalcap (CAD-1883), a selective modulator for SK channels, may treat movement disorders like SCA and …
Formula:
C18H24F2N6O
Purity:
99.54%
Color and Shape:
Solid
Molecular weight:
378.42
Ref: TM-T9522
| 1mg | 35.00 € | ||
| 5mg | 76.00 € | ||
| 10mg | 108.00 € | ||
| 25mg | 210.00 € | ||
| 50mg | 312.00 € | ||
| 100mg | 440.00 € | ||
| 200mg | 616.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
SB-705498
CAS:501951-42-4
SB705498 is a TRPV1 antagonist for hTRPV1. SB-705498 has been investigated for the treatment of …
Formula:
C17H16BrF3N4O
Purity:
98% - ≥95%
Color and Shape:
Solid
Molecular weight:
429.23
Ref: TM-T6660
| 5mg | 47.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 293.00 € | ||
| 100mg | 423.00 € | ||
| 200mg | 589.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
Imidazenil
CAS:151271-08-8
Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion …
Formula:
C18H12BrFN4O
Purity:
98.4%
Color and Shape:
Solid
Molecular weight:
399.22
Ref: TM-T8971
| 1mg | 98.00 € | ||
| 5mg | 203.00 € | ||
| 10mg | 335.00 € | ||
| 25mg | 553.00 € | ||
| 50mg | 807.00 € | ||
| 1mL*10mM (DMSO) | 248.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
L-DABA
CAS:1758-80-1
L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 >500 μM).
Formula:
C4H10N2O2
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
118.13
Ref: TM-T7595
| 25mg | 34.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
RQ-00203078
CAS:1254205-52-1
RQ-00203078 is a highly selective, potent and orally available TRPM8 antagonist.
Formula:
C21H13ClF6N2O5S
Purity:
98% - 99.17%
Color and Shape:
Solid
Molecular weight:
554.85
Ref: TM-T2007
| 5mg | 50.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 121.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 345.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
ICA-069673
CAS:582323-16-8
ICA-069673 is an activator of KCNQ2/Q3 potassium channel (IC50: 0.69 μM).
Formula:
C11H6ClF2N3O
Purity:
98.97% - 99.66%
Color and Shape:
Solid
Molecular weight:
269.63
Ref: TM-T3959
| 5mg | 45.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 249.00 € | ||
| 100mg | 362.00 € | ||
| 200mg | 525.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
