Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
ZM 226600
CAS:147695-92-9
ZM 226600 is an ATP-sensitive potassium channel opener with an EC50 value of 500 nM. …
Formula:
C16H14F3NO4S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
373.35
Ref: TM-T23563
| 1mg | 39.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 231.00 € | ||
| 50mg | 374.00 € | ||
| 100mg | 547.00 € | ||
| 500mg | 1,189.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Leminoprazole
CAS:104340-86-5
Leminoprazole is an orally available H+,K(+)-ATPase inhibitor that protects gastric mucosal cells from various cellular …
Formula:
C19H23N3OS
Purity:
98.87% - 99.56%
Color and Shape:
Solid
Molecular weight:
341.47
Ref: TM-T27812
| 1mg | 125.00 € | ||
| 5mg | 298.00 € | ||
| 10mg | 446.00 € | ||
| 25mg | 735.00 € | ||
| 50mg | 1,003.00 € | ||
| 100mg | 1,380.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
PD-118057
CAS:313674-97-4
PD-118057, a potent hERG activator, may treat long QT syndrome and heart failure without hERG …
Formula:
C21H17Cl2NO2
Purity:
98.97% - 99.16%
Color and Shape:
Solid
Molecular weight:
386.27
Ref: TM-T16444
| 1mg | 94.00 € | ||
| 5mg | 199.00 € | ||
| 10mg | 306.00 € | ||
| 25mg | 584.00 € | ||
| 50mg | 926.00 € | ||
| 100mg | 1,481.00 € | ||
| 1mL*10mM (DMSO) | 222.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
TRAM 39
CAS:197525-99-8
TRAM 39 (2-Chloro-α,α-diphenylbenzeneacetonitrile) is a selective blocker of intermediate-conductance Ca2+-activated K+channels.
Formula:
C20H14ClN
Purity:
99.51%
Color and Shape:
Solid
Molecular weight:
303.78
Ref: TM-T23471
| 1mg | 36.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 106.00 € | ||
| 25mg | 209.00 € | ||
| 50mg | 332.00 € | ||
| 100mg | 524.00 € | ||
| 500mg | 1,095.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Tracazolate hydrochloride
CAS:1135210-68-2
Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant …
Formula:
C16H25ClN4O2
Purity:
99.07%
Color and Shape:
Solid
Molecular weight:
340.85
Ref: TM-T23470
| 10mg | 43.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 18 Feb 2025
BPDBA
CAS:312281-74-6
BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory …
Formula:
C19H20Cl2N2O
Purity:
99.24% - 99.86%
Color and Shape:
Solid
Molecular weight:
363.28
Ref: TM-T26891
| 5mg | 41.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 111.00 € | ||
| 50mg | 171.00 € | ||
| 100mg | 276.00 € | ||
| 200mg | 381.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Ani9
CAS:356102-14-2
Ani9 selectively blocks ANO1/TMEM16A with a 77 nM IC50, useful for ANO1 research and treating …
Formula:
C17H17ClN2O3
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
332.78
Ref: TM-T26630
| 1mg | 39.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 264.00 € | ||
| 50mg | 444.00 € | ||
| 100mg | 644.00 € | ||
| 500mg | 1,375.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
TRPM4-IN-2
CAS:667411-04-3
NBA, or TRPM4-IN-2, is a potent TRPM4 inhibitor with IC50 of 0.16 μM, used in …
Formula:
C19H14ClNO4
Purity:
99.21%
Color and Shape:
Liquid
Molecular weight:
355.77
Ref: TM-T61275
| 2mg | To inquire |
Estimated delivery in United States, on Tuesday 18 Feb 2025
RO 4938581
CAS:883093-10-5
RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, …
Formula:
C13H8BrF2N5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
352.14
Ref: TM-T16794
| 25mg | 1,141.00 € | ||
| 50mg | 1,499.00 € | ||
| 100mg | 2,468.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
KT-362 fumarate
CAS:105394-80-7
KT-362 fumarate, a novel antagonist of Ca, K, and Na channels, induces vasodilation and relaxes …
Formula:
C26H32N2O7S
Purity:
100% - 99.87%
Color and Shape:
Solid
Molecular weight:
516.61
Ref: TM-T27753
| 1mg | 300.00 € | ||
| 5mg | 694.00 € | ||
| 10mg | 981.00 € | ||
| 25mg | 1,449.00 € | ||
| 50mg | 1,930.00 € | ||
| 100mg | 2,627.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
JYL 1421
CAS:401907-26-4
JYL 1421 (SC 0030) is an antagonist of TRPV1 receptor (IC50 = 8 nM).
Formula:
C20H26FN3O2S2
Color and Shape:
Solid
Molecular weight:
423.57
Ref: TM-T15634
| 25mg | 710.00 € | ||
| 50mg | 934.00 € | ||
| 100mg | 1,470.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Elismetrep
CAS:1400699-64-0
Elismetrep (MT-8554) is an orally available TRPM8 inhibitor with potential analgesic activity for the study …
Formula:
C27H21F3N2O5S
Purity:
99.57% - 99.86%
Color and Shape:
Solid
Molecular weight:
542.53
Ref: TM-T27253
| 1mg | 123.00 € | ||
| 5mg | 294.00 € | ||
| 10mg | 459.00 € | ||
| 25mg | 916.00 € | ||
| 50mg | 1,368.00 € | ||
| 100mg | 1,846.00 € | ||
| 200mg | 2,492.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
SKF96067
CAS:115607-61-9
SKF96067 is a reversible gastric H+/K+-ATPase inhibitor that can induce relaxation of human airway smooth …
Formula:
C21H22N2O2
Purity:
99.14%
Color and Shape:
Solid
Molecular weight:
334.41
Ref: TM-T16894
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
TASK-1-IN-1
CAS:600125-11-9
TASK-1-IN-1: Potent, selective TASK-1 blocker (IC50: 148 nM), weaker on TASK-3 (IC50: 1750 nM), anticancer …
Formula:
C22H20N2O2
Purity:
100%
Color and Shape:
Soild
Molecular weight:
344.41
Ref: TM-T72064
| 1mg | 40.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 270.00 € | ||
| 50mg | 423.00 € | ||
| 100mg | 625.00 € | ||
| 500mg | 1,327.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Nerisopam
CAS:102771-12-0
Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.
Formula:
C18H19N3O2
Purity:
97.27%
Color and Shape:
Solid
Molecular weight:
309.36
Ref: TM-T28159
| 1mg | 138.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 496.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,477.00 € | ||
| 500mg | 2,960.00 € | ||
| 1mL*10mM (DMSO) | 449.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Fengabine
CAS:80018-06-0
Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat …
Formula:
C17H17Cl2NO
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
322.23
Ref: TM-T27310
| 1mg | 82.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 242.00 € | ||
| 25mg | 470.00 € | ||
| 50mg | 643.00 € | ||
| 100mg | 912.00 € | ||
| 500mg | 1,829.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Pazinaclone
CAS:103255-66-9
Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.
Formula:
C25H23ClN4O4
Purity:
98.12% - 99%
Color and Shape:
Solid
Molecular weight:
478.93
Ref: TM-T28303
| 1mg | 138.00 € | ||
| 5mg | 325.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 797.00 € | ||
| 50mg | 1,100.00 € | ||
| 100mg | 1,476.00 € | ||
| 500mg | 2,980.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Transcainide
CAS:88296-62-2
Transcainide (R 54718), an oral lidocaine-like antiarrhythmic, blocks BTX-activated Na+ channels in heart/muscle.
Formula:
C22H35N3O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
373.53
Ref: TM-T26287
| 1mg | 250.00 € | ||
| 5mg | 616.00 € | ||
| 10mg | 879.00 € | ||
| 25mg | 1,299.00 € | ||
| 50mg | 1,746.00 € | ||
| 100mg | 2,378.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
RN9893
CAS:1803003-68-0
RN9893 is a selective and potent TRPV4 receptor antagonist with IC50 values of 320, 420 …
Formula:
C21H23F3N4O5S
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
500.49
Ref: TM-T28548
| 1mg | 46.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 141.00 € | ||
| 25mg | 268.00 € | ||
| 50mg | 397.00 € | ||
| 100mg | 578.00 € | ||
| 500mg | 1,187.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Elpetrigine
CAS:212778-82-0
Elpetrigine (GW273293) is a potential sodium channel blocker with antiepileptic activity that can be used …
Formula:
C10H7Cl3N4
Purity:
98.77% - 99.78%
Color and Shape:
Solid
Molecular weight:
289.55
Ref: TM-T31614
| 1mg | 273.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,416.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
