Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
YHO-13351 free base
CAS:912288-64-3
YHO-13351 free base is the water-soluble prodrug of YHO-13177 which is an inhibitor of BCRP …
Formula:
C26H33N3O4S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
483.62
Ref: TM-T13365
| 1mg | 35.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 291.00 € | ||
| 100mg | 446.00 € | ||
| 500mg | 977.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Picrotin
CAS:21416-53-5
Picrotin is an inhibitor of glycine receptors. Picrotin blocks α2 GlyR, α1 GlyR, and α3 …
Formula:
C15H18O7
Purity:
97.11%
Color and Shape:
Solid
Molecular weight:
310.3
Ref: TM-T16533
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 74.00 € | ||
| 50mg | 93.00 € | ||
| 100mg | 140.00 € | ||
| 500mg | 343.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Pinacidil
CAS:60560-33-0
Pinacidil (P 1134) is a guanidine that opens potassium channels and directly dilates peripheral blood …
Formula:
C13H19N5
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
245.32
Ref: TM-T12478L
| 5mg | 49.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 161.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
VRT-532
CAS:38214-71-0
VRT-532 (CFpot-532) is an effective modulator of CFTR and is commonly used in studies of …
Formula:
C16H14N2O
Purity:
100% - 99.89%
Color and Shape:
Solid
Molecular weight:
250.3
Ref: TM-T29114
| 1mg | 94.00 € | ||
| 5mg | 228.00 € | ||
| 10mg | 342.00 € | ||
| 25mg | 566.00 € | ||
| 50mg | 762.00 € | ||
| 100mg | 1,003.00 € | ||
| 200mg | 1,327.00 € | ||
| 1mL*10mM (DMSO) | 204.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
CFTR corrector 8
CAS:1918142-35-4
CFTR corrector 8: potent for cystic fibrosis research, modulates CFTR protein.
Formula:
C29H27F2NO7
Purity:
99.58%
Color and Shape:
Liquid
Molecular weight:
539.52
Ref: TM-T63806
| 1mg | 80.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 258.00 € | ||
| 25mg | 522.00 € | ||
| 50mg | 820.00 € | ||
| 100mg | 1,345.00 € | ||
| 1mL*10mM (DMSO) | 216.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Mavatrep
CAS:956274-94-5
Mavatrep (JNJ-39439335) is a selective antagonist of TRPV1 with Ki of 6.5 nM and can …
Formula:
C25H21F3N2O
Purity:
98.01% - 98.38%
Color and Shape:
Solid
Molecular weight:
422.44
Ref: TM-T16014
| 1mg | 65.00 € | ||
| 5mg | 143.00 € | ||
| 10mg | 225.00 € | ||
| 25mg | 449.00 € | ||
| 50mg | 724.00 € | ||
| 100mg | 1,154.00 € | ||
| 500mg | 2,312.00 € | ||
| 1mL*10mM (DMSO) | 158.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
CyPPA
CAS:73029-73-9
CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.
Formula:
C16H23N5
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
285.39
Ref: TM-T20968
| 2mg | 43.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 277.00 € | ||
| 100mg | 458.00 € | ||
| 500mg | 1,009.00 € | ||
| 1mL*10mM (DMSO) | 70.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
MSP3
CAS:1820968-63-5
MSP3 is an agonist of TRPV1 (EC50 = 0.87 μM) and shows antinociceptive and neuroprotective …
Formula:
C16H19NO3S
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
305.39
Ref: TM-T28118
| 2mg | 34.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 164.00 € | ||
| 50mg | 247.00 € | ||
| 100mg | 364.00 € | ||
| 200mg | 515.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
TRPV4 agonist-1
CAS:2314467-60-0
TRPV4 agonist-1 is an agonist of TRPV4 (EC50: 60 nM in the hTRPV4 Ca2+ assay).
Formula:
C25H23ClF2N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
484.93
Ref: TM-T13214
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
PF 05089771 tosylate
CAS:1430806-04-4
PF-05089771 inhibits Nav1.7 channels (IC50: 11-33 nM), selective over Nav1.1-1.6/1.8, Ca+, K+ channels, TRPV1; 1000x …
Formula:
C18H12Cl2FN5O3S2·C7H8O3S
Purity:
97.76%
Color and Shape:
Solid
Molecular weight:
672.56
Ref: TM-T7502
| 1mg | 62.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 159.00 € | ||
| 25mg | 381.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
HC-070
CAS:1628291-95-1
HC-070 is a TRPC5 and TRPC4 antagonist (IC50 = 9.3 nM and 46 nM).
Formula:
C22H20Cl2N4O4
Purity:
97.06%
Color and Shape:
Solid
Molecular weight:
475.32
Ref: TM-T15465
| 1mg | 90.00 € | ||
| 5mg | 173.00 € | ||
| 10mg | 263.00 € | ||
| 25mg | 435.00 € | ||
| 50mg | 612.00 € | ||
| 100mg | 825.00 € | ||
| 200mg | 1,052.00 € | ||
| 1mL*10mM (DMSO) | 171.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Abeprazan hydrochloride
CAS:1902954-87-3
Abeprazan hydrochloride (Fexuprazan hydrochloride) is an effective reversible potassium-competitive acid blocker with oral activity, inhibiting …
Formula:
C19H18ClF3N2O3S
Purity:
98.62%
Color and Shape:
Solid
Molecular weight:
446.87
Ref: TM-T10221
| 1mg | 63.00 € | ||
| 5mg | 143.00 € | ||
| 10mg | 204.00 € | ||
| 25mg | 327.00 € | ||
| 50mg | 444.00 € | ||
| 100mg | 570.00 € | ||
| 200mg | 753.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
RL648_81
CAS:1919050-87-5
RL648_81 is a selective activator of KCNQ2/3 channels (EC50 = 190 nM). RL648_81 can be …
Formula:
C17H17F4N3O2
Purity:
98.85%
Color and Shape:
Solid
Molecular weight:
371.33
Ref: TM-T28544
| 2mg | 43.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 103.00 € | ||
| 25mg | 220.00 € | ||
| 50mg | 326.00 € | ||
| 100mg | 467.00 € | ||
| 200mg | 633.00 € | ||
| 1mL*10mM (DMSO) | 75.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Lesogaberan
CAS:344413-67-8
Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity …
Formula:
C3H9FNO2P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
141.08
Ref: TM-T15737
| 25mg | 1,406.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
FR-167356
CAS:174185-16-1
FR-167356 inhibits a3 isoform H⁺-ATPase (IC50: 170-370 nM), targeting osteoclasts, kidneys, macrophages; reduces B16-F10 bone …
Formula:
C19H17Cl2NO3
Purity:
98.44% - 99.19%
Color and Shape:
Solid
Molecular weight:
378.25
Ref: TM-T27371
| 1mg | 118.00 € | ||
| 5mg | 276.00 € | ||
| 10mg | 377.00 € | ||
| 25mg | 570.00 € | ||
| 50mg | 766.00 € | ||
| 100mg | 1,008.00 € | ||
| 200mg | 1,334.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
UK 78282 hydrochloride
CAS:136647-02-4
UK-78282 hydrochloride, a Kv1.3 blocker.UK-78282 hydrochloride inhibits Kv1.3 voltage-gated potassium channels and suppresses human T …
Formula:
C29H36ClNO2
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
466.05
Ref: TM-T23497
| 1mg | 91.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 325.00 € | ||
| 25mg | 540.00 € | ||
| 50mg | 771.00 € | ||
| 100mg | 1,019.00 € | ||
| 500mg | 2,083.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Puliginurad
CAS:2013582-27-7
Puliginurad (YL-90148) is a urate transporter protein inhibitor that inhibits the reabsorption of uric acid.Puliginurad …
Formula:
C19H16N2O2S
Purity:
99.96% - 99.96%
Color and Shape:
Liquid
Molecular weight:
336.41
Ref: TM-T61048
| 1mg | 66.00 € | ||
| 5mg | 142.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
NaV1.2/1.6 channel blocker-1
CAS:1199944-04-1
NaV1.2/1.6 channel blocker-1 is a NaV1.2/1.6 channel blocker that inhibits rNaV1.6 and can be used …
Formula:
C14H14N2OS
Purity:
99.54%
Color and Shape:
Liquid
Molecular weight:
258.34
Ref: TM-T72170
| 1mg | 40.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 116.00 € | ||
| 25mg | 225.00 € | ||
| 50mg | 333.00 € | ||
| 100mg | 495.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
TC-I 2014
CAS:1221349-53-6
TC-I 2014 shows antiallodynic properties in pain models.
Formula:
C23H19F6N3O
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
467.41
Ref: TM-T17006
| 1mg | 113.00 € | ||
| 5mg | 270.00 € | ||
| 10mg | 402.00 € | ||
| 25mg | 644.00 € | ||
| 50mg | 909.00 € | ||
| 100mg | 1,201.00 € | ||
| 500mg | 2,432.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
GX-674
CAS:1432913-36-4
GX-674 is a highly potent and selective voltage-gated sodium channel 1.7 (Nav1.7) antagonist with an …
Formula:
C21H13ClF2N6O3S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
534.95
Ref: TM-T22829
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
