Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
Amsacrine
CAS:51264-14-3
Amsacrine (AMSA) (mAMSA) an antineoplastic agent which can intercalate into the DNA of tumor cells.
Formula:
C21H19N3O3S
Purity:
98.59%
Color and Shape:
Yellow Crystalline Powder Solid
Molecular weight:
393.46
Ref: TM-T1206
| 10mg | 51.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
SCH 50911
CAS:733717-87-8
SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow …
Formula:
C8H15NO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
173.21
Ref: TM-T12867L
| 50mg | 2,475.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
PG01
CAS:853138-65-5
PG01 is a potent CFTR Cl-channel potentiator, effective against ΔF508 (Ka 0.3 μM), and also …
Formula:
C28H29N3O2
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
439.55
Ref: TM-T16516
| 1mg | 121.00 € | ||
| 5mg | 351.00 € | ||
| 10mg | 527.00 € | ||
| 25mg | 852.00 € | ||
| 50mg | 1,143.00 € | ||
| 100mg | 1,559.00 € | ||
| 500mg | 3,121.00 € | ||
| 1mL*10mM (DMSO) | 348.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
(E)-GABAB receptor antagonist 1
CAS:1611483-29-4
(E)-GABAB antagonist 1 inhibits GABA IP3 production, with an IC50 of 37.9 μM and acts …
Formula:
C18H24O4
Purity:
95.26%
Color and Shape:
Solid
Molecular weight:
304.38
Ref: TM-T11137
| 1mg | 112.00 € | ||
| 5mg | 248.00 € | ||
| 10mg | 365.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 765.00 € | ||
| 100mg | 1,044.00 € | ||
| 200mg | 1,413.00 € | ||
| 1mL*10mM (DMSO) | 240.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
CBS9106
CAS:1076235-04-5
CBS9106 (SL-801) is a CRM1 inhibitor with CRM1-degrading and anti-tumor activity that inhibits CRM1-dependent nuclear …
Formula:
C18H21ClF3N3O3
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
419.83
Ref: TM-T14885
| 1mg | 247.00 € | ||
| 5mg | 605.00 € | ||
| 10mg | 836.00 € | ||
| 25mg | 1,293.00 € | ||
| 50mg | 1,761.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
ABCG2-IN-1
CAS:2559759-40-7
ABCG2-IN-1 (compound K2), an analog of Ko143, constitutes an orally active inhibitor targeting ABCG2 with …
Formula:
C26H36N4O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
468.59
Ref: TM-T79513
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
E2730
CAS:1520073-91-9
E2730 is a selective and noncompetitive inhibitor of the gamma-aminobutyric acid (GABA) transporter 1 (GAT1) …
Formula:
C9H8F4N2O2S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
284.23
Ref: TM-T79399
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
TWIK-1/TREK-1-IN-2
CAS:1440532-32-0
TWIK-1/TREK-1-IN-2 (Compound 2g) serves as an inhibitor of both TWIK-1 and TREK-1, targeting the TREK-1 …
Formula:
C20H29F3N2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
386.45
Ref: TM-T78869
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
ABCG2-IN-2
CAS:2559759-59-8
ABCG2-IN-2 is a potent inhibitor of ABCG2, exhibiting favorable oral pharmacokinetic profiles in mice, and …
Formula:
C25H34N4O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
454.56
Ref: TM-T79514
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
XE991
CAS:122955-42-4
XE991 is a Kv7 (KCNQ) channel blocker.XE 991 dihydrochloride inhibits Kv7.1 (KCNQ1) and M-current and …
Formula:
C26H20N2O
Purity:
99.51%
Color and Shape:
Liquid
Molecular weight:
376.45
Ref: TM-T78570
| 1mg | 48.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 277.00 € | ||
| 50mg | 512.00 € | ||
| 100mg | 824.00 € | ||
| 500mg | 1,651.00 € | ||
| 1mL*10mM (DMSO) | 104.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
U-89843A
CAS:157013-85-9
U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents …
Formula:
C16H24ClN5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
321.85
Ref: TM-T78560
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
TWIK-1/TREK-1-IN-3
CAS:1440532-33-1
TWIK-1/TREK-1-IN-3 is a potassium channel TREK-1 inhibitor TWIK-1/TREK-1-IN-3 has antidepressant activity and can be used …
Formula:
C19H27F3N2O2
Purity:
99.04%
Color and Shape:
Liquid
Molecular weight:
372.43
Ref: TM-T78870
| 1mg | 86.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 305.00 € | ||
| 25mg | 509.00 € | ||
| 50mg | 727.00 € | ||
| 100mg | 984.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
TWIK-1/TREK-1-IN-1
CAS:1440532-30-8
Compound 2a, identified as TWIK-1/TREK-1-IN-1, acts as an inhibitor of the TREK-1, a two-pore domain …
Formula:
C21H24F3NO3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
395.42
Ref: TM-T78868
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
DMCM hydrochloride
CAS:1215833-62-7
DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.
Formula:
C17H19ClN2O4
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
350.8
Ref: TM-T11061
| 1mg | 37.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 248.00 € | ||
| 50mg | 461.00 € | ||
| 100mg | 650.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
UCCF-853
CAS:625458-06-2
UCCF-853 is a small-molecule CFTR modulator that can be used to study cystic fibrosis.
Formula:
C14H8ClF3N2O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
312.67
Ref: TM-T29041
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 179.00 € | ||
| 50mg | 267.00 € | ||
| 100mg | 396.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
ABT-239
CAS:460746-46-7
ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 …
Formula:
C22H22N2O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
330.42
Ref: TM-T14087
| 1mg | 47.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 348.00 € | ||
| 50mg | 518.00 € | ||
| 100mg | 732.00 € | ||
| 500mg | 1,537.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
D-3263 hydrochloride
CAS:1008763-54-9
D-3263 hydrochloride (D3263 HCl salt) is enteric-coated, orally bioavailable transient receptor potential melatonin member 8 …
Formula:
C21H32ClN3O3
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
409.95
Ref: TM-T10929L
| 1mg | 50.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 103.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Vernakalant Hydrochloride
CAS:748810-28-8
Vernakalant Hydrochloride (RSD1235 hydrochloride) is a mixed voltage- and frequency-dependent Na+ and atria-preferred K+ channel …
Formula:
C20H32ClNO4
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
385.93
Ref: TM-T17227
| 1mg | 74.00 € | ||
| 2mg | 95.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 269.00 € | ||
| 25mg | 512.00 € | ||
| 50mg | 740.00 € | ||
| 100mg | 1,016.00 € | ||
| 1mL*10mM (DMSO) | 185.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
R(+)-IAA-94
CAS:54197-31-8
R(+)-IAA-94 (Methylindazone) blocks epithelial chloride channels; inhibits Nef-sdAb19 binding.
Formula:
C17H18Cl2O4
Purity:
98.95% - 99.22%
Color and Shape:
Solid
Molecular weight:
357.23
Ref: TM-T12788
| 2mg | 36.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 163.00 € | ||
| 50mg | 276.00 € | ||
| 100mg | 399.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
TC-N 1752
CAS:1211866-85-1
TC-N 1752 is an orally active inhibitor of Nav1.7 channel with IC50 of 0.17 μM. …
Formula:
C25H27F3N6O3
Purity:
97.87%
Color and Shape:
Solid
Molecular weight:
516.52
Ref: TM-T23439
| 1mg | 36.00 € | ||
| 5mg | 81.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 262.00 € | ||
| 50mg | 387.00 € | ||
| 100mg | 550.00 € | ||
| 200mg | 714.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
