Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
L-822179
CAS:215874-86-5
L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with …
Formula:
C17H14N8O2
Purity:
98.34% - 98.74%
Color and Shape:
Solid
Molecular weight:
362.35
Ref: TM-T24381
| 1mg | 44.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 180.00 € | ||
| 50mg | 268.00 € | ||
| 100mg | 383.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
A 425619
CAS:581809-67-8
A 425619 (1-(4-(TRIFLUOROMETHYL)BENZYL)-3-(ISOQUINOLIN-5-YL)UREA) is a potent TRPV1 antagonist
Formula:
C18H14F3N3O
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
345.32
Ref: TM-T8562
| 1mg | 85.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € | ||
| 1mL*10mM (DMSO) | 172.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
VU0463271
CAS:1391737-01-1
VU0463271: KCC2 antagonist, IC50 61 nM, >100x selective over NKCC1, inactive on other GPCRs, channels, …
Formula:
C19H18N4OS2
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
382.5
Ref: TM-T17243
| 5mg | 49.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 240.00 € | ||
| 100mg | 354.00 € | ||
| 200mg | 504.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
BPO-27 racemate
CAS:1314873-02-3
BPO-27 racemate (BPO-27 (racemate)) is an effective CFTR inhibitor with IC50 of 8 nM.
Formula:
C26H18BrN3O6
Purity:
98.19%
Color and Shape:
Solid
Molecular weight:
548.34
Ref: TM-T10591
| 1mg | 45.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 169.00 € | ||
| 25mg | 271.00 € | ||
| 50mg | 395.00 € | ||
| 100mg | 545.00 € | ||
| 200mg | 731.00 € | ||
| 1mL*10mM (DMSO) | 130.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
CLP257
CAS:1181081-71-9
CLP257 is a selective K+-Cl− cotransporter KCC2 activator (EC50: 616 nM) and it is inactive …
Formula:
C14H14FN3O2S
Purity:
98.13%
Color and Shape:
Solid
Molecular weight:
307.34
Ref: TM-T14984
| 1mg | 45.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 279.00 € | ||
| 50mg | 456.00 € | ||
| 100mg | 672.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
SCS
CAS:3232-36-8
SCS is a GABAA receptor antagonist.
Formula:
C14H12N2O3
Purity:
98.89%
Color and Shape:
Solid
Molecular weight:
256.26
Ref: TM-T23339
| 10mg | 42.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | 89.00 € | ||
| 100mg | 130.00 € | ||
| 200mg | 182.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
PF-05105679
CAS:1398583-31-7
PF-05105679 is a selective TRPM8 antagonist (IC50 = 103 nM). PF-05105679 can be used in …
Formula:
C26H21FN2O3
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
428.45
Ref: TM-T16483
| 1mg | 48.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 159.00 € | ||
| 25mg | 302.00 € | ||
| 50mg | 467.00 € | ||
| 100mg | 701.00 € | ||
| 200mg | 926.00 € | ||
| 500mg | 1,412.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
TPA 023
CAS:252977-51-8
TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 …
Formula:
C20H22FN7O
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
395.43
Ref: TM-T17144
| 1mg | 222.00 € | ||
| 5mg | 538.00 € | ||
| 10mg | 806.00 € | ||
| 25mg | 1,188.00 € | ||
| 50mg | 1,605.00 € | ||
| 100mg | 2,162.00 € | ||
| 1mL*10mM (DMSO) | 591.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
DNDS
CAS:3709-43-1
DNDS is a channel blocker of voltage-dependent cystic fibrosis transmembrane conductance regulator (CFTR).
Formula:
C14H8N2Na2O10S2
Purity:
99.88%
Color and Shape:
Physical Description White Powder (Ntp 1992)
Molecular weight:
474.33
Ref: TM-T20341
| 1g | 34.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
(+)-Bicuculline methiodide
CAS:40709-69-1
(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in …
Formula:
C21H20INO6
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
509.29
Ref: TM-T22604
| 1mg | 38.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
JT010
CAS:917562-33-5
JT010 is an effective agonist of TRPA1 (EC50 = 0.65 nM).
Formula:
C16H19ClN2O3S
Purity:
98.5%
Color and Shape:
Solid
Molecular weight:
354.85
Ref: TM-T15628
| 2mg | 34.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 150.00 € | ||
| 50mg | 232.00 € | ||
| 100mg | 346.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Clobutinol hydrochloride
CAS:1215-83-4
Clobutinol hydrochloride, an antitussive agent, influences heart rate and blood pressure, and is utilized in …
Formula:
C14H23Cl2NO
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
292.25
Ref: TM-T78523
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Aneratrigine hydrochloride
CAS:2097163-75-0
Aneratrigine hydrochloride is a Nav 1.9 blocker that may be used to prevent or treat …
Formula:
C19H21Cl2F2N5O2S2
Purity:
99.33% - 99.39%
Color and Shape:
Liquid
Molecular weight:
524.43
Ref: TM-T79835
| 1mg | 182.00 € | ||
| 5mg | 451.00 € | ||
| 10mg | 646.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,390.00 € | ||
| 100mg | 1,837.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
6-Iodoamiloride
CAS:60398-23-4
6-Iodoamiloride is a potent inhibitor of acid-sensing ion channel 1 (ASIC1), exhibiting an IC50 value …
Formula:
C6H8IN7O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
321.08
Ref: TM-T79246
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 4 Mar 2025
COR659
CAS:544450-68-2
COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.
Formula:
C16H16ClNO3S
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
337.82
Ref: TM-T36520
| 1mg | 51.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 112.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 313.00 € | ||
| 50mg | 436.00 € | ||
| 100mg | 598.00 € | ||
| 200mg | 814.00 € | ||
| 1mL*10mM (DMSO) | 124.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Soraprazan
CAS:261944-46-1
BS3 Crosslinker (Bis(sulfosuccinimidyl)suberate) is an ADC linker that can be used to synthesize antibody-coupled active …
Formula:
C21H25N3O3
Purity:
97.69% - 99.84%
Color and Shape:
Solid
Molecular weight:
367.44
Ref: TM-T12977
| 5mg | 419.00 € | ||
| 25mg | 1,419.00 € | ||
| 50mg | 1,884.00 € | ||
| 100mg | 3,048.00 € | ||
| 1mL*10mM (DMSO) | 406.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
CP-409092
CAS:194098-25-4
CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.
Formula:
C17H19N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
297.35
Ref: TM-T10869L
| 25mg | 1,688.00 € | ||
| 50mg | 2,225.00 € | ||
| 100mg | 2,897.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Co 102862
CAS:181144-66-1
Co 102862 is a voltage-gated sodium channel blocker. Co 102862 can be used for anticonvulsant …
Formula:
C14H12FN3O2
Purity:
99.54%
Color and Shape:
Solid
Molecular weight:
273.26
Ref: TM-T22675
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 140.00 € | ||
| 50mg | 209.00 € | ||
| 100mg | 341.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
C 101248
CAS:361368-24-3
C 101248 (KCNK13-IN-1) is a selective and potent tandem pore halogen inhibitor of K+ channel …
Formula:
C15H12N6O
Purity:
99.25% - 99.31%
Color and Shape:
Liquid
Molecular weight:
292.3
Ref: TM-T83962
| 10mg | 329.00 € | ||
| 50mg | 1,381.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
CRF1 receptor antagonist-1
CAS:2635364-30-4
CRF1 Receptor Antagonist-1 (Compound 2), a CRF1 receptor antagonist, is utilized in research pertaining to …
Formula:
C27H28ClFN2O2S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
499.04
Ref: TM-T79793
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 4 Mar 2025
