GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
Found 363 products for "GABA Receptor".
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Suritozole
CAS:Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptorFormula:C10H10FN3SPurity:99.25%Color and Shape:SolidMolecular weight:223.27Ref: TM-T8568
1mg58.00€1mL*10mM (DMSO)104.00€5mg116.00€10mg172.00€25mg281.00€50mg396.00€100mg537.00€200mg712.00€Cholesterol myristate
CAS:Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.Formula:C41H72O2Purity:99.65%Color and Shape:White SolidMolecular weight:597.01α-Thujone
CAS:α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.Formula:C10H16OPurity:97.02% - 98.41%Color and Shape:Transparent OilMolecular weight:152.23(2S)-6-Prenylnaringenin
CAS:(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.Formula:C20H20O5Purity:99.47%Color and Shape:SolidMolecular weight:340.37Piperazine citrate
CAS:Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.Formula:C24H46N6O14Purity:99.8%Color and Shape:Crystals IndicationMolecular weight:642.65Loreclezole hydrochloride
CAS:Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.Formula:C10H7Cl4N3Color and Shape:SolidMolecular weight:310.99Temgicoluril
CAS:Temgicoluril (mebikar) acts on GABA Receptor.Formula:C8H14N4O2Purity:99.8%Color and Shape:SolidMolecular weight:198.22Tiagabine hydrochloride hydrate
CAS:Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.Formula:C20H28ClNO3S2Color and Shape:SolidMolecular weight:430.022'MeO6MF
CAS:2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functionalFormula:C17H14O3Purity:99.28% - 99.63%Color and Shape:SolidMolecular weight:266.29Ref: TM-T8887
1mg49.00€1mL*10mM (DMSO)96.00€5mg102.00€10mg152.00€25mg243.00€50mg340.00€100mg460.00€200mg627.00€Jujuboside A
CAS:Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.Formula:C58H94O26Purity:98% - >99.99%Color and Shape:SolidMolecular weight:1207.35AZD7325
CAS:AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.Formula:C19H19FN4O2Purity:99.83%Color and Shape:SolidMolecular weight:354.38Piperazine
CAS:Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.Formula:C4H10N2Color and Shape:SolidMolecular weight:86.14ONO-8590580
CAS:ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.Formula:C21H21FN6Purity:99.43%Color and Shape:SolidMolecular weight:376.43Ref: TM-TQ0040
1mg57.00€5mg119.00€1mL*10mM (DMSO)133.00€10mg166.00€25mg356.00€50mg532.00€100mg760.00€Pikamilone
CAS:Pikamilone (Picamilon) is an intelligent medicine.Formula:C10H12N2O3Purity:99.38%Color and Shape:White Crystalline PowderMolecular weight:208.21(+)-Kavain
CAS:(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.Formula:C14H14O3Purity:97% - ≥95%Color and Shape:White Fine PowderMolecular weight:230.26Acamprosate calcium
CAS:Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.Formula:C10H20CaN2O8S2Purity:98% - 99.93%Color and Shape:White Odorless Or Nearly Odorless PowderMolecular weight:400.48Imepitoin
CAS:Imepitoin (AWD 131-138), a new low-affinity partial benzodiazepine receptor agonist, shows potent anticonvulsant and anxiolytic properties in rodent models.Formula:C13H14ClN3O2Purity:99.82%Color and Shape:SolidMolecular weight:279.72Ginkgolide A
CAS:Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.Formula:C20H24O9Purity:98.76% - 99.81%Color and Shape:White SolidMolecular weight:408.40SKF89976A hydrochloride
CAS:SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) andFormula:C22H26ClNO2Purity:98.02%Color and Shape:SolidMolecular weight:371.9Ref: TM-T12930
1mg34.00€5mg65.00€1mL*10mM (DMSO)71.00€10mg89.00€25mg167.00€50mg264.00€100mg409.00€200mg590.00€Miltirone
CAS:Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Formula:C19H22O2Purity:99.22% - 99.66%Color and Shape:SolidMolecular weight:282.38Phenibut (hydrochloride)
CAS:Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Formula:C10H14ClNO2Purity:99.93%Color and Shape:White SolidMolecular weight:215.68(-)-Securinine
CAS:(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.Formula:C13H15NO2Purity:99.58% - 99.87%Color and Shape:Yellow SolidMolecular weight:217.26NS11394
CAS:NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(Formula:C23H19N3OPurity:99.44% - 99.86%Color and Shape:SolidMolecular weight:353.42Ref: TM-T2067
2mg33.00€5mg52.00€1mL*10mM (DMSO)55.00€10mg75.00€25mg124.00€50mg200.00€100mg304.00€200mg437.00€Ginsenoside Rc
CAS:Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.Formula:C53H90O22Purity:98.83% - 99.86%Color and Shape:White SolidMolecular weight:1079.27Fluralaner
CAS:Fluralaner (A1443) is an isoxazoline ectoparasiticide.Formula:C22H17Cl2F6N3O3Purity:99.72% - 99.99%Color and Shape:White SolidMolecular weight:556.29U93631
CAS:GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.Formula:C17H21N3O2Purity:99.65% - 99.76%Color and Shape:SolidMolecular weight:299.37Isonipecotic acid
CAS:Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA receptor partial agonist.Formula:C6H11NO2Purity:99.82%Color and Shape:White To Faint Pink-Beige PowderMolecular weight:129.16Darigabat
CAS:Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.Formula:C22H21FN4O3SPurity:98.42% - 99.29%Color and Shape:SolidMolecular weight:440.49Riluzole
CAS:Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.Formula:C8H5F3N2OSPurity:99.71% - 99.88%Color and Shape:SolidMolecular weight:234.2Nitrazolam
CAS:Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.Formula:C17H13N5O2Color and Shape:SolidMolecular weight:319.32Pyrazolam
CAS:Pyrazolam is a psychoactive benzodiazepine compound serving as a central nervous system depressant. [Pyrazolam] can lead to psychomotor impairment.Formula:C16H12BrN5Color and Shape:SolidMolecular weight:354.2CGP36216 hydrochloride
CAS:CGP36216 hydrochloride acts as a selective antagonist at the presynaptic GABA receptor, specifically binding to the GABAB receptor with a Ki value of 0.3 μM. This compound is leveraged in research focused on anxiety and trauma-related disorders [1] [2].Formula:C5H15ClNO2PColor and Shape:SolidMolecular weight:187.6TB 21007
CAS:GABAA receptor inverse agonistFormula:C15H17NO2S3Purity:98%Color and Shape:SolidMolecular weight:339.5β-CCB
CAS:benzodiazepine receptor ligandFormula:C16H16N2O2Purity:98%Color and Shape:SolidMolecular weight:268.31NO 711
CAS:NO 711（NNC-711 free acid） is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.Formula:C21H22N2O3Purity:99.70%Color and Shape:White SolidMolecular weight:350.41(±)-Homoproline Hydrochloride
CAS:(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can TrustFormula:C6H12ClNO2Purity:99.69%Color and Shape:SolidMolecular weight:165.62CP-457920
CAS:CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.Formula:C18H17N3O3Purity:99.06% - 99.74%Color and Shape:White SolidMolecular weight:323.35Ro 41-3290
CAS:Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is an agonist of nonbenzodiazepine partial at the benzodiazepine receptor.Formula:C24H21ClN2O3Purity:98%Color and Shape:SolidMolecular weight:420.89PF-0713
CAS:PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.Formula:C14H22OPurity:98%Color and Shape:SolidMolecular weight:206.32HZ166
CAS:HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.Formula:C21H16N4O2Purity:98%Color and Shape:SolidMolecular weight:356.38Pregabalin arenacarbil
CAS:Pregabalin arenacarbil is a gabamimetic.Formula:C15H27NO6Color and Shape:SolidMolecular weight:317.38NCS-382
CAS:γ-Hydroxybutyric acid antagonistFormula:C13H14O3Purity:98%Color and Shape:SolidMolecular weight:218.25Ro 19-4603
CAS:Benzodiazepine inverse agonistFormula:C15H17N3O3SPurity:98%Color and Shape:SolidMolecular weight:319.38GABAA receptor agent 4
CAS:Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.Formula:C17H24N2OColor and Shape:SolidMolecular weight:272.39mGAT3/4-IN-1
CAS:mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.Formula:C26H31ClN2O2S2Color and Shape:SolidMolecular weight:503.12CGP11952
CAS:CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.Formula:C21H21Cl2N5O2Purity:98%Color and Shape:SolidMolecular weight:446.3317-PA
CAS:17-PA is a GABAA receptor antagonist.Formula:C25H34OPurity:98%Color and Shape:SolidMolecular weight:350.54MK-0343
CAS:MK0343 is an orally bioavailable GABAA receptor subtype-selective partial agonist and is a non-sedating anxiolytic.Formula:C19H17F2N7OPurity:98%Color and Shape:White SolidMolecular weight:397.38DS2
CAS:Positive allosteric modulator of δ-subunit containing GABAA receptorsFormula:C18H12ClN3OSPurity:98%Color and Shape:SolidMolecular weight:353.83CGS8216
CAS:CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.Formula:C16H11N3OPurity:98.53%Color and Shape:Yellow SolidMolecular weight:261.28
