PPAR
Peroxisome Proliferator-Activated Receptors (PPARs) are a group of nuclear receptor proteins that function as transcription factors regulating the expression of genes involved in metabolism, particularly fatty acid storage and glucose metabolism. PPAR inhibitors are important tools for studying metabolic disorders such as diabetes, obesity, and cardiovascular diseases. These inhibitors can modulate lipid metabolism, insulin sensitivity, and inflammation, making them valuable in therapeutic research. At CymitQuimica, we offer a range of PPAR inhibitors to support your research in metabolic diseases, endocrinology, and drug development.
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Clofibrate
CAS:637-07-0
Clofibrate (Clofibrato) is an aryloxyisobutyric acid derivate with antihyperlipidemic activity.
Formula:
C12H15ClO3
Purity:
99.87%
Color and Shape:
Oil Liquid
Molecular weight:
242.7
Ref: TM-T1298
| 1g | 62.00 € | ||
| 5g | 81.00 € | ||
| 200mg | 36.00 € | ||
| 500mg | 52.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
DG172 dihydrochloride
CAS:1361504-77-9
DG172 dihydrochloride (DG-172 dihydrochloride) is an antagonist of PPARβ/δ(IC50 : 27 nM).
Formula:
C20H22BrCl2N3
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
455.2
Ref: TM-T7821
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 299.00 € | ||
| 100mg | 488.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
L-165041
CAS:79558-09-1
L-165041 is a potent and selective agonist of the nuclear receptor PPARβ and PPARδ(Ki = …
Formula:
C22H26O7
Purity:
97.97%
Color and Shape:
Solid
Molecular weight:
402.44
Ref: TM-T7159
| 5mg | 47.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 206.00 € | ||
| 100mg | 329.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
GSK3787
CAS:188591-46-0
GSK3787 is a specific and irreversible PPARδ inhibitor(pIC50= 6.6).
Formula:
C15H12ClF3N2O3S
Purity:
98% - 98.53%
Color and Shape:
Solid
Molecular weight:
392.78
Ref: TM-T1941
| 5mg | 54.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 304.00 € | ||
| 100mg | 509.00 € | ||
| 500mg | 1,091.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Oroxin A
CAS:57396-78-8
Oroxin A (Baicalein 7-O-glucoside) has antitussive and expectorant effects.
Formula:
C21H20O10
Purity:
98.05% - 99.74%
Color and Shape:
Solid
Molecular weight:
432.38
Ref: TM-T5S0788
| 1mg | 43.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 132.00 € | ||
| 25mg | 219.00 € | ||
| 50mg | 363.00 € | ||
| 100mg | 497.00 € | ||
| 500mg | 1,068.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
AMG131
CAS:315224-26-1
AMG131 (CHS 131) , is a novel, non-thiazolidinedione (TZD), selective peroxisome proliferator-activated receptor (PPAR)gamma modulator, …
Formula:
C21H12Cl4N2O3S
Purity:
98.01%
Color and Shape:
Solid
Molecular weight:
514.21
Ref: TM-T8780
| 1mg | 41.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 247.00 € | ||
| 50mg | 402.00 € | ||
| 100mg | 600.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Gypenoside XLIX
CAS:94987-08-3
Extracted from whole herb of Gynostemsma pentaphyllum(Thunb.)Mak.;Store the product in sealed, cool and dry condition
Formula:
C52H86O21
Purity:
99.59% - 99.78%
Color and Shape:
Solid
Molecular weight:
1047.23
Ref: TM-T2985
| 5mg | 58.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 160.00 € | ||
| 50mg | 262.00 € | ||
| 100mg | 442.00 € | ||
| 500mg | 920.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Elafibranor
CAS:923978-27-2
Elafibranor (GFT505) is an agonist of the peroxisome proliferator-activated receptor-α (PPAR-α) and peroxisome proliferator-activated receptor-δ …
Formula:
C22H24O4S
Purity:
99.5% - 99.55%
Color and Shape:
Solid
Molecular weight:
384.49
Ref: TM-T4408
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 133.00 € | ||
| 50mg | 211.00 € | ||
| 100mg | 346.00 € | ||
| 500mg | 807.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Cinnamyl alcohol
CAS:104-54-1
Cinnamyl alcohol (Styryl Carbinol) readily autoxidizes upon air exposure, and forms strong sensitizers as determined …
Formula:
C9H10O
Purity:
98.77%
Color and Shape:
Colourless Liquid
Molecular weight:
134.18
Ref: TM-T5S1550
| 1g | 37.00 € | ||
| 5g | 76.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Tesaglitazar
CAS:251565-85-2
Tesaglitazar is a potent and selective peroxide PPARα / γ receptor dual agonist with a …
Formula:
C20H24O7S
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
408.47
Ref: TM-T17044
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 249.00 € | ||
| 50mg | 465.00 € | ||
| 100mg | 674.00 € | ||
| 500mg | 1,411.00 € | ||
| 1mL*10mM (DMSO) | 106.00 € |
Estimated delivery in United States, on Wednesday 15 Jan 2025
13-Oxo-9E,11E-octadecadienoic acid
CAS:29623-29-8
13-Oxo-9E,11E-octadecadienoic acid from tomato juice, an isomer of 9-oxo-ODA, activates PPARα and lowers triglycerides in …
Formula:
C18H30O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
294.43
Ref: TM-T10044
| 25mg | 1,406.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Saroglitazar
CAS:495399-09-2
Saroglitazar (Lipaglyn) is an agonist of PPAR with EC50 values of 0.65 pM and 3 …
Formula:
C25H29NO4S
Purity:
98.49%
Color and Shape:
Solid
Molecular weight:
439.57
Ref: TM-T12835
| 1mg | 147.00 € | ||
| 5mg | 304.00 € | ||
| 10mg | 460.00 € | ||
| 1mL*10mM (DMSO) | 328.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Peliglitazar racemate
CAS:331744-72-0
Peliglitazar racemate(BMS 426707-01 racemate) is the racemate of Peliglitazar.Peliglitazar racemate may be used as a …
Formula:
C30H30N2O7
Purity:
97.75%
Color and Shape:
Solid
Molecular weight:
530.57
Ref: TM-T12400
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
PPARγ-IN-2
CAS:2682078-97-1
"PPARγ-IN-2 (Compound 5a), a PPARγ inhibitor, exhibits an EC50 of 0.106 μM in inhibiting TG …
Formula:
C19H21N5O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
335.4
Ref: TM-T79678
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Farglitazar
CAS:196808-45-4
Farglitazar (GI-262570) is a PPAR-γ agonist and insulin sensitizer used in the study of diabetes.
Formula:
C34H30N2O5
Purity:
99.40% - 99.65%
Color and Shape:
Solid
Molecular weight:
546.61
Ref: TM-T27303
| 1mg | 276.00 € | ||
| 5mg | 679.00 € | ||
| 10mg | 928.00 € | ||
| 25mg | 1,430.00 € | ||
| 50mg | 1,862.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
THR-0921
CAS:606932-81-4
THR-0921 (CLX-0921) is a peroxisome proliferator-activated receptor (PPAR) agonist that can be used to study …
Formula:
C28H25NO7S
Purity:
98.53%
Color and Shape:
Liquid
Molecular weight:
519.57
Ref: TM-T69015
| 1mg | 266.00 € | ||
| 5mg | 656.00 € | ||
| 10mg | 896.00 € | ||
| 25mg | 1,418.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Suksdorfin
CAS:53023-17-9
Suksdorfin has hypoglycemic effects and activates PPARγ, which promotes insulin-dependent glucose uptake by adipocytes and …
Formula:
C21H24O7
Purity:
98.43%
Color and Shape:
Liquid
Molecular weight:
388.41
Ref: TM-T69146
| 1mg | 272.00 € | ||
| 2mg | 405.00 € | ||
| 5mg | 671.00 € | ||
| 10mg | 917.00 € | ||
| 25mg | 1,442.00 € | ||
| 50mg | 1,878.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Indeglitazar
CAS:835619-41-5
Indeglitazar (PPM 204) is orally available pan-agonist of PPAR (PPAR subtypes alpha (α), delta (δ), …
Formula:
C19H19NO6S
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
389.42
Ref: TM-T15575
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 185.00 € | ||
| 100mg | 279.00 € | ||
| 200mg | 427.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
PPARα-MO-1
CAS:810677-36-2
PPARα-MO-1 is a potent modulator of PPARα.
Formula:
C27H37NO5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
455.59
Ref: TM-T10505
| 25mg | 1,549.00 € | ||
| 50mg | 2,033.00 € | ||
| 100mg | 2,611.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
LG100754
CAS:180713-37-5
LG100754 (UVI 2112) is an insulin sensitizer and RXR modulator, antagonizing RXR homodimers while agonizing …
Formula:
C26H36O3
Color and Shape:
Solid
Molecular weight:
396.56
Ref: TM-T15748
| 25mg | 921.00 € | ||
| 50mg | 1,208.00 € | ||
| 100mg | 1,844.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
