5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
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Pimethixene
CAS:314-03-4
Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.
Formula:
C19H19NS
Purity:
97.50%
Color and Shape:
Solid
Molecular weight:
293.43
Ref: TM-T12489
| 2mg | 34.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 106.00 € | ||
| 50mg | 158.00 € | ||
| 100mg | 226.00 € | ||
| 200mg | 339.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Trimipramine maleate
CAS:521-78-8
Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.
Formula:
C24H30N2O4
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
410.51
Ref: TM-T1045
| 50mg | 39.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 74.00 € | ||
| 500mg | 110.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Granisetron hydrochloride
CAS:107007-99-8
Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used …
Formula:
C18H25ClN4O
Purity:
99.88% - 99.93%
Color and Shape:
White To Off-White Crystalline Solid
Molecular weight:
348.87
Ref: TM-T1042
| 10mg | 38.00 € | ||
| 25mg | 56.00 € | ||
| 50mg | 81.00 € | ||
| 100mg | 127.00 € | ||
| 200mg | 178.00 € | ||
| 500mg | 304.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
RS102895 hydrochloride
CAS:1173022-16-6
RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).
Formula:
C21H22ClF3N2O2
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
426.86
Ref: TM-T12773
| 2mg | 48.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 180.00 € | ||
| 50mg | 320.00 € | ||
| 100mg | 480.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
NEO 376
CAS:496921-73-4
NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing …
Formula:
C20H24ClN3O
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
357.88
Ref: TM-T12207
| 1mg | 74.00 € | ||
| 5mg | 140.00 € | ||
| 10mg | 215.00 € | ||
| 25mg | 373.00 € | ||
| 50mg | 522.00 € | ||
| 100mg | 702.00 € | ||
| 200mg | 944.00 € | ||
| 1mL*10mM (DMSO) | 156.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Alprenolol
CAS:13655-52-2
Alprenolol (Alpheprol) is a non-selective β-adrenergic receptor (β-AR) antagonist that is also an antagonist of …
Formula:
C15H23NO2
Purity:
99.73% - 99.78%
Color and Shape:
Solid
Molecular weight:
249.35
Ref: TM-T4560
| 50mg | 52.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Sertraline hydrochloride
CAS:79559-97-0
Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the …
Formula:
C17H18Cl3N
Purity:
99.12% - 99.89%
Color and Shape:
Solid Powder
Molecular weight:
342.691
Ref: TM-T0482
| 5mg | 51.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 103.00 € | ||
| 50mg | 180.00 € | ||
| 100mg | 235.00 € | ||
| 200mg | 304.00 € | ||
| 500mg | 515.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Lofepramine
CAS:23047-25-8
Lofepramine (Leo 640) is a potent tricyclic antidepressant that is extensively metabolized to desipramine.
Formula:
C26H27ClN2O
Purity:
98.38%
Color and Shape:
Crystals From Methanol Or Acetone Solid
Molecular weight:
418.96
Ref: TM-T15773
| 2mg | 48.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 178.00 € | ||
| 50mg | 266.00 € | ||
| 100mg | 400.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Iloperidone
CAS:133454-47-4
Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.
Formula:
C24H27FN2O4
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
426.48
Ref: TM-T1539
| 25mg | 48.00 € | ||
| 50mg | 62.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 140.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Alverine citrate
CAS:5560-59-8
Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.
Formula:
C26H35NO7
Purity:
98.53% - 99.43%
Color and Shape:
Coa
Molecular weight:
473.57
Ref: TM-T0428
| 1g | 81.00 € | ||
| 500mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Sumatriptan succinate
CAS:103628-48-4
Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment …
Formula:
C18H27N3O6S
Purity:
97.53% - 99.51%
Color and Shape:
White Powder
Molecular weight:
413.49
Ref: TM-T0203
| 25mg | 37.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 74.00 € | ||
| 500mg | 169.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Spiperone
CAS:749-02-0
Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.
Formula:
C23H26FN3O2
Purity:
99.34% - 99.89%
Color and Shape:
Solid
Molecular weight:
395.47
Ref: TM-T0280
| 5mg | 47.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Fluoxetine
CAS:54910-89-3
Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.
Formula:
C17H18F3NO
Purity:
99.07% - 99.28%
Color and Shape:
Solid
Molecular weight:
309.33
Ref: TM-T0450
| 10mg | 35.00 € | ||
| 25mg | 48.00 € | ||
| 50mg | 63.00 € | ||
| 100mg | 81.00 € | ||
| 200mg | 120.00 € | ||
| 500mg | 213.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Pheniramine maleate
CAS:132-20-7
Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 …
Formula:
C16H20N2·C4H4O4
Purity:
99.85%
Color and Shape:
Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°C
Molecular weight:
356.42
Ref: TM-T0370
| 25mg | 35.00 € | ||
| 50mg | 46.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 66.00 € | ||
| 500mg | 92.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Quetiapine hemifumarate
CAS:111974-72-2
Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, …
Formula:
C46H54N6O8S2
Purity:
100% - 99.59%
Color and Shape:
White Crystalline Solid
Molecular weight:
883.09
Ref: TM-T6241
| 1g | 52.00 € | ||
| 200mg | 35.00 € | ||
| 500mg | 50.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Pizotifen Malate
CAS:5189-11-7
Pizotifen Malate (BC-105 malate), a highly selective 5-HT receptor blocking agent, is a drug based …
Formula:
C19H21NS·C4H6O5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
429.53
Ref: TM-T0225
| 50mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Eletriptan hydrobromide
CAS:177834-92-3
Eletriptan hydrobromide (Eletriptan HBr) is an orally active agonist with specific affinity for the 5-hydroxytriptamine1B/1D …
Formula:
C22H27BrN2O2S
Purity:
100% - 99.69%
Color and Shape:
Tan Solid
Molecular weight:
463.43
Ref: TM-T0216
| 2mg | 39.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 134.00 € | ||
| 50mg | 235.00 € | ||
| 100mg | 427.00 € | ||
| 200mg | 555.00 € | ||
| 500mg | 890.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Clozapine
CAS:5786-21-0
Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.
Formula:
C18H19ClN4
Purity:
99.91% - 99.93%
Color and Shape:
Yellow Crystals From Acetone-Petroleum Ether Solid
Molecular weight:
326.82
Ref: TM-T0455
| 1g | 449.00 € | ||
| 10mg | 35.00 € | ||
| 25mg | 52.00 € | ||
| 50mg | 70.00 € | ||
| 100mg | 96.00 € | ||
| 200mg | 170.00 € | ||
| 500mg | 303.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Zolmitriptan
CAS:139264-17-8
Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, …
Formula:
C16H21N3O2
Purity:
99.69% - 99.91%
Color and Shape:
White Or Kind Of White Powder
Molecular weight:
287.36
Ref: TM-T1092
| 10mg | 58.00 € | ||
| 25mg | 99.00 € | ||
| 50mg | 141.00 € | ||
| 100mg | 216.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
PF-04995274
CAS:1331782-27-4
PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive …
Formula:
C23H32N2O6
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
432.51
Ref: TM-T16481
| 1mg | 35.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 197.00 € | ||
| 50mg | 350.00 € | ||
| 100mg | 505.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
