Hello!
Enter your email address to receive promotions, special events and VIP exclusives!
GluR
Pomaglumetad methionil
CAS:956385-05-0
Pomaglumetad methionil is an oral methionine prodrug of the potent specific agonist of mGlu2/3 receptor …
Formula:
C12H20N2O8S2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
384.43
Estimated delivery in United States, on Monday 7 Feb 2022
Ampalex
CAS:154235-83-3
Ampalex (Ampakine CX516; CX516; BDP 12), an ampakine and nootropic, acts as an AMPA receptor …
Formula:
C14H15N3O
Purity:
98.00%
Color and Shape:
Tan Solid
Molecular weight:
241.29
Estimated delivery in United States, on Monday 7 Feb 2022
LY3020371 hydrochloride
CAS:1377615-44-5
LY3020371 hydrochloride exerts an antidepressant-like signature in vivo. LY3020371 hydrochloride is a potent, selective metabotropic …
Formula:
C15H16ClF2NO5S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
395.81
Estimated delivery in United States, on Monday 7 Feb 2022
Foliglurax
CAS:1883329-51-8
Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) …
Formula:
C23H23N3O3S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
421.51
Estimated delivery in United States, on Monday 7 Feb 2022
Memantine hydrochloride
CAS:41100-52-1
Memantine hydrochloride is an AMANTADINE derivative that has some dopaminergic effects. Memantine hydrochloride has been …
Formula:
C12H22ClN
Purity:
98.00%
Color and Shape:
Crystalline Solid
Molecular weight:
215.76
Estimated delivery in United States, on Monday 7 Feb 2022
4-oxo-1,4-dihydroquinoline-2-carboxylic acid
CAS:13593-94-7
4-oxo-1,4-dihydroquinoline-2-carboxylic acid is a GluR and NMDA inhibitor.
Formula:
C10H7NO3
Purity:
99.49%
Color and Shape:
solid
Molecular weight:
189.167
Estimated delivery in United States, on Monday 7 Feb 2022
Caroverine HCL
CAS:55750-05-5
Caroverine HCL is a potent, competitive and reversible antagonist of NMDA and AMPA glutamate receptor. …
Formula:
C22H28ClN3O2
Molecular weight:
401.9
Estimated delivery in United States, on Monday 7 Feb 2022
JNJ-40411813
CAS:1127498-03-6
JNJ-40411813 (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor (mGlu2R, …
Formula:
C20H25ClN2O
Purity:
99.57%
Color and Shape:
solid
Molecular weight:
344.88
Estimated delivery in United States, on Monday 7 Feb 2022
NBQX disodium salt
CAS:118876-58-7
Potent, selective and competitive AMPA receptor antagonist. Neuroprotective and anticonvulsant; active in vivo.
Formula:
C12H8N4O6S
Purity:
97.66%
Color and Shape:
solid
Molecular weight:
336.28
Estimated delivery in United States, on Monday 7 Feb 2022
Org-26576
CAS:1026791-61-6
Org-26576 is a positive allosteric modulator of the AMPA receptor.
Formula:
C11H12N2O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
204.23
Estimated delivery in United States, on Monday 7 Feb 2022
GET73
CAS:202402-01-5
GET73 is an negative allosteric modulator of mGluR5. GET73 is a naturally occurring neurotransmitter. GET73 …
Formula:
C13H16F3NO2
Purity:
99.54%
Molecular weight:
275.27
Estimated delivery in United States, on Monday 7 Feb 2022
(±)-trans-ACPD
CAS:67684-64-4
(±)-trans-ACPD is an equimolecular mixture of (1S, 3R)- and (1R, 3S)-ACPD. (±)-trans-ACPD is a selective …
Formula:
C7H11NO4
Purity:
99.53%
Color and Shape:
solid
Molecular weight:
173.17
Estimated delivery in United States, on Monday 7 Feb 2022
Evans blue
CAS:314-13-6
Evans blue is an azo dye, inhibits L-glutamate uptake via the membrane-bound excitatory amino acid …
Formula:
C34H24N6Na4O14S4
Purity:
98.85%
Color and Shape:
Dark Brown
Molecular weight:
960.78
Estimated delivery in United States, on Monday 7 Feb 2022
DHPG
CAS:146255-66-5
DHPG ((RS)-3,5-DHPG) is an effective antagonist of mGluR linked to phospholipase D. It is an …
Formula:
C8H9NO4
Purity:
99.55%
Color and Shape:
solid
Molecular weight:
183.16
Estimated delivery in United States, on Monday 7 Feb 2022
AZD-8529 mesylate
CAS:1314217-69-0
AZD-8529 mesylate is a highly selective, and orally bioavailable positive allosteric modulator of mGluR2 (EC50: …
Formula:
C25H28F3N5O6S
Purity:
99.50%
Color and Shape:
Solid
Molecular weight:
583.58
Estimated delivery in United States, on Monday 7 Feb 2022
IDRA-21
CAS:22503-72-6
IDRA-21 is a positive AMPA receptor modulator.
Formula:
C8H9ClN2O2S
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
232.68
Estimated delivery in United States, on Monday 7 Feb 2022
VU0652835
CAS:1848252-81-2
VU0652835 is a negative allosteric modulator of metabotropic glutamate receptor subtype 5 (mGlu5) (IC50: 81 …
Formula:
C16H19N3O3S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
333.41
Estimated delivery in United States, on Monday 7 Feb 2022
MPEP
CAS:96206-92-7
MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable …
Formula:
C14H11N
Purity:
99.31%
Color and Shape:
solid
Molecular weight:
193.24
Estimated delivery in United States, on Monday 7 Feb 2022
VU 0364439
CAS:1246086-78-1
VU 0364439 is a mGlu4 positive allosteric modulator (C50: 19.8 nM).
Formula:
C18H13Cl2N3O3S
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
422.29
Estimated delivery in United States, on Monday 7 Feb 2022
Chelidamic acid
CAS:138-60-3
Chelidamic acid is a heterocyclic organic acid with a pyran skeleton. Chelidamic acid is inhibitors …
Formula:
C7H5NO5
Purity:
98.00%
Color and Shape:
Pale Yellow Powder
Molecular weight:
183.12
Estimated delivery in United States, on Monday 7 Feb 2022
JNJ-46778212
CAS:1363281-27-9
JNJ-46778212 is an effective mGlu5 allosteric modulator (EC50: 260 nM).
Formula:
C20H17FN2O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
352.36
Estimated delivery in United States, on Monday 7 Feb 2022
gamma-DGG
CAS:6729-55-1
gamma-DGG is a competitive blocker of AMPA receptor.
Formula:
C7H12N2O5
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
204.18
Estimated delivery in United States, on Monday 7 Feb 2022
VU6001376
CAS:1968546-34-0
VU6001376 is an effective and selective positive allosteric modulator of the metabotropic glutamate receptor 4 …
Formula:
C18H14F2N6OS
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
400.41
Estimated delivery in United States, on Monday 7 Feb 2022
JNJ-46281222
CAS:1254980-38-5
JNJ-46281222 is an metabotropic glutamate (mGlu) 2-selective, highly potent PAM (positive allosteric modulator). It has …
Formula:
C23H25F3N4
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
414.47
Estimated delivery in United States, on Monday 7 Feb 2022
Lu AF21934
CAS:1445605-23-1
Lu AF21934 is a brain-penetrant and selective mGlu4 receptor positive allosteric modulator (IC50: 500 nM, …
Formula:
C14H16Cl12N2O2
Purity:
97.96%
Color and Shape:
Solid
Molecular weight:
315.2
Estimated delivery in United States, on Monday 7 Feb 2022
Decoglurant
CAS:911115-16-7
Decoglurant is a negative allosteric modulator of mGluR2 and mGluR3 and it also is developed …
Formula:
C21H11F6N5
Purity:
99.39%
Color and Shape:
solid
Molecular weight:
447.34
Estimated delivery in United States, on Monday 7 Feb 2022
D-glutamine
CAS:5959-95-5
D-glutamine, an D type stereoisomer of glutamine, is one of the 20 amino acids which …
Formula:
C5H10N2O3
Purity:
99.92%
Color and Shape:
White Or Off-White Powder
Molecular weight:
146.14
Estimated delivery in United States, on Monday 7 Feb 2022
DNQX
CAS:2379-57-9
DNQX is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for …
Formula:
C8H4N4O6
Purity:
98.00%
Color and Shape:
Off-White Powder With A Yellow Tinge
Molecular weight:
252.14
Estimated delivery in United States, on Monday 7 Feb 2022
Lithium citrate tribasic tetrahydrate
CAS:6080-58-6
Lithium Citrate, the active component of Lithium, is a medicine used in the therapy of …
Formula:
C6H13Li3O11
Purity:
98.00%
Color and Shape:
White Crystalline Powder
Molecular weight:
281.98
Estimated delivery in United States, on Monday 7 Feb 2022
JNJ42153605
CAS:1254977-87-1
JNJ-42153605 is a mGlu2 receptor positive allosteric modulator (EC50: 17 nM).
Formula:
C22H23F3N4
Purity:
97.25%
Color and Shape:
solid
Molecular weight:
400.45
Estimated delivery in United States, on Monday 7 Feb 2022
JNJ16259685
CAS:409345-29-5
JNJ16259685 is a selective mGluR1 antagonist, and inhibits the synaptic activation of mGluR1 in a …
Formula:
C20H23NO3
Purity:
99.39%
Molecular weight:
325.4
Estimated delivery in United States, on Monday 7 Feb 2022
FPTQ
CAS:1025802-62-3
FPTQ is an antagonist of mGluR1.
Formula:
C17H12FN5
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
305.32
Estimated delivery in United States, on Monday 7 Feb 2022
gamma-DGG acetate(6729-55-1 free base)
gamma-DGG acetate is a competitive blocker of AMPA receptor.
Formula:
C9H16N2O7
Purity:
99.81%
Molecular weight:
264.23
Estimated delivery in United States, on Monday 7 Feb 2022
Decanoic Acid
CAS:334-48-5
Decanoic Acid acts as a non-competitive AMPA receptor antagonist.
Formula:
C10H20O2
Purity:
99.87%
Color and Shape:
Crystalline Solid Solid
Molecular weight:
172.26
Estimated delivery in United States, on Monday 7 Feb 2022
Ro 67-7476
CAS:298690-60-5
Ro 67-7476 is a positive allosteric modulator of mGlu1 receptors. No activity at human mGlu1 …
Formula:
C17H18FNO2S
Purity:
99.48%
Color and Shape:
solid
Molecular weight:
319.39
Estimated delivery in United States, on Monday 7 Feb 2022
LYPLAL1-IN-1
CAS:1966129-74-7
LYPLAL1-IN-1 is a selective covalent small-molecule inhibitor of Lysophospholipase-like 1 (IC50: 0.006 μM). LYPLAL1-IN-1 also …
Formula:
C29H29N7O4
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
539.59
Estimated delivery in United States, on Monday 7 Feb 2022
BMT-145027
CAS:2018282-44-3
BMT-145027 is a positive allosteric modulator of mGluR5 without inherent agonist activity (EC50: 47 nM).
Formula:
C23H14ClF3N4
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
438.83
Estimated delivery in United States, on Monday 7 Feb 2022
CDPPB
CAS:781652-57-1
CDPPB is a modulator of mGluR5 positive allosteric(with an EC50 of 27 nM in Chinese …
Formula:
C23H16N4O
Purity:
99.39%
Color and Shape:
solid
Molecular weight:
364.4
Estimated delivery in United States, on Monday 7 Feb 2022
NPS2390
CAS:226878-01-9
NPS2390 is a first generation quinoxaline derivative that acts as a noncompetitive antagonist of mGluR1 …
Formula:
C19H21N3O
Purity:
99.24%
Color and Shape:
solid
Molecular weight:
307.4
Estimated delivery in United States, on Monday 7 Feb 2022
Ro0711401
CAS:714971-87-6
Ro0711401 is an agonist of mGlu1 receptor.
Formula:
C18H11F3N2O3
Purity:
98.54%
Molecular weight:
360.29
Estimated delivery in United States, on Monday 7 Feb 2022
SIB-1757
CAS:31993-01-8
SIB-1757 is a selective antagonist of mGlu5 metabotropic glutamate receptor subtype (hmGlu5, IC50 : 0.4 …
Formula:
C12H11N3O
Purity:
98.49%
Color and Shape:
solid
Molecular weight:
213.24
Estimated delivery in United States, on Monday 7 Feb 2022
ADX88178
CAS:1235318-89-4
ADX88178 is a potent positive allosteric modulator for metabotropic glutamate receptor 4 (mGluR4) with EC50 …
Formula:
C12H12N6S
Molecular weight:
272.33
Estimated delivery in United States, on Monday 7 Feb 2022
AZD 9272
CAS:327056-26-8
AZD 9272 is a antagonist of brain penetrant mGluR5.
Formula:
C14H6F2N4O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
284.22
Estimated delivery in United States, on Monday 7 Feb 2022
TAT-GluA2 3Y acetate(1404188-93-7 free base)
TAT-GluA2 3Y acetate is an inhibitor of AMPA receptor endocytosis. Induces increased hind paw withdrawal …
Formula:
C115H185N43O29
Molecular weight:
2634.02
Estimated delivery in United States, on Monday 7 Feb 2022
GYKI53655 hydrochloride
CAS:143692-48-2
GYKI53655 hydrochloride is an antagonist of -amino-3-hydroxy-5-methylisoxazole-4-propionic acid (AMPA).
Formula:
C19H21ClN4O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
388.85
Estimated delivery in United States, on Monday 7 Feb 2022
DL-AP3
CAS:20263-06-3
DL-AP3 is a competitive group I metabotropic glutamate receptor antagonist and inhibitor of phosphoserine phosphatase.
Formula:
C3H8NO5P
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
169.07
Estimated delivery in United States, on Monday 7 Feb 2022
VU 29
CAS:890764-36-0
VU-29 is a positive allosteric mGlu5 receptor modulator with EC50=9 nM and Ki=244 nM for …
Formula:
C22H16N4O3
Purity:
99.47%
Color and Shape:
solid
Molecular weight:
384.39
Estimated delivery in United States, on Monday 7 Feb 2022
MPEP hydrochloride
CAS:219911-35-0
MPEP hydrochloride is an effective and highly specific non-competitive antagonist at the mGlu5 receptor subtype …
Formula:
C14H12ClN
Purity:
99.75%
Color and Shape:
solid
Molecular weight:
229.7
Estimated delivery in United States, on Monday 7 Feb 2022
CNQX
CAS:115066-14-3
CNQX is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM for …
Formula:
C9H4N4O4
Purity:
98.00%
Color and Shape:
Pale Yellow Solid
Molecular weight:
232.15
Estimated delivery in United States, on Monday 7 Feb 2022
LY377604
CAS:204592-94-9
LY377604 is a human 3-adrenergic receptor agonist (EC50: 2.4 nM). It also a 1- and …
Formula:
C31H32N4O4
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
524.61
Estimated delivery in United States, on Monday 7 Feb 2022
L-Glutamic acid monosodium salt
CAS:142-47-2
L-Glutamic acid monosodium salt (Monosodium glutamate) is an activator of mGlu1 receptor.
Formula:
C5H8NO4·Na
Purity:
99.45%
Color and Shape:
White Solid Crystalline
Molecular weight:
169.11
Estimated delivery in United States, on Monday 7 Feb 2022
MTEP hydrochloride
CAS:1186195-60-7
MTEP hydrochloride is non-competitive mGlu5 antagonist (IC50 and Ki of 5 nM and 16 nM, …
Formula:
C11H9ClN2S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
236.72
Estimated delivery in United States, on Monday 7 Feb 2022
M77976
CAS:394237-61-7
M77976 is the potential for the research of obesity and diabetes. M77976 is a specific …
Formula:
C17H16N2O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
296.32
Estimated delivery in United States, on Monday 7 Feb 2022
MSOP
CAS:66515-29-5
MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM …
Formula:
C4H10NO6P
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
199.1
Estimated delivery in United States, on Monday 7 Feb 2022
ML 254
CAS:1428630-86-7
ML254 competitively interacts with the MPEP allosteric binding site. ML254 is highly selective for mGlu5 …
Formula:
C18H15FN2O2
Molecular weight:
310.32
Estimated delivery in United States, on Monday 7 Feb 2022
L-Cysteic acid monohydrate
CAS:23537-25-9
L-Cysteic acid is an oxidation product of L-cysteine that may be used as a competitive …
Formula:
C3H9NO6S
Purity:
99.28%
Color and Shape:
White Powder
Molecular weight:
187.17
Estimated delivery in United States, on Monday 7 Feb 2022
FTIDC
CAS:873551-53-2
FTIDC is a highly potent and selective allosteric antagonist of mGluR1 receptors and shows very …
Formula:
C18H23FN6O
Purity:
94.58%
Color and Shape:
Solid
Molecular weight:
358.42
Estimated delivery in United States, on Monday 7 Feb 2022
LY2140023
CAS:635318-55-7
LY2140023 has the potential for schizophrenia.LY2140023 is an orally active prodrug of LY404039. LY404039 is …
Formula:
C12H18N2O7S2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
366.41
Estimated delivery in United States, on Monday 7 Feb 2022
VU0650786
CAS:1809085-30-0
VU0650786 is a selective and potent CNS penetrant negative allosteric modulator of metabotropic glutamate receptor …
Formula:
C18H15ClFN5O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
387.8
Estimated delivery in United States, on Monday 7 Feb 2022
AMN 082 dihydrochloride
CAS:97075-46-2
AMN 082 dihydrochloride is a selective metabotropic glutamate mGlu7 receptor agonist reported to exhibit antidepressant …
Formula:
C28H30Cl2N2
Molecular weight:
465.46
Estimated delivery in United States, on Monday 7 Feb 2022
1-BCP
CAS:34023-62-6
1-BCP is a centrally active drug that modulates AMPA receptor gated currents.
Formula:
C13H15NO3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
233.26
Estimated delivery in United States, on Monday 7 Feb 2022
LY404187
CAS:211311-95-4
LY404187 is a positive allosteric modulator of AMPA receptors
Formula:
C19H22N2O2S
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
342.46
Estimated delivery in United States, on Monday 7 Feb 2022
TCN 238
CAS:125404-04-8
TCN 238 is an orally bioavailable positive allosteric modulator of the metabotropic glutamate receptor 4 …
Formula:
C12H11N3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
197.24
Estimated delivery in United States, on Monday 7 Feb 2022
YM90K hydrochloride
CAS:154164-30-4
YM90K hydrochloride is an antagonist of AMPA receptor.
Formula:
C11H8ClN5O4
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
309.66
Estimated delivery in United States, on Monday 7 Feb 2022
M-110
CAS:1395048-49-3
M-110 inhibits PIM-1 and PIM-2 with similar (IC50s: 2.5 μM) and it also inhibits the …
Formula:
C22H28ClN5O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
445.94
Estimated delivery in United States, on Monday 7 Feb 2022
LY 541850
CAS:852679-76-6
LY541850 is a selective orthosteric mGlu2 agonist and mGlu3 antagonist with IC50 values of 0.161 …
Formula:
C9H13NO4
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
199.2
Estimated delivery in United States, on Monday 7 Feb 2022
ADX 47273
CAS:851881-60-2
ADX-47273 is a positive and selective allosteric modulator for the metabotropic glutamate receptor subtype mGluR5(EC50=170 …
Formula:
C20H17F2N3O2
Purity:
97.00%
Color and Shape:
solid
Molecular weight:
369.36
Estimated delivery in United States, on Monday 7 Feb 2022
FITM
CAS:932737-65-0
FITM is a potent negative allosteric modulator of mGlu1 receptor(Ki : 2.5 nM).
Formula:
C18H18FN5OS
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
371.43
Estimated delivery in United States, on Monday 7 Feb 2022
L-APB
CAS:23052-81-5
L-APB is an effective and specific agonist for the group III mGluRs (EC50s: 0.13, 0.29, …
Formula:
C4H10NO5P
Purity:
98.00%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
183.1
Estimated delivery in United States, on Monday 7 Feb 2022
L-Glutamine
CAS:56-85-9
L-glutamine, a non-essential amino acid, is synthesized from glutamic acid and ammonia.
Formula:
C5H10N2O3
Purity:
99.36%
Color and Shape:
Solid Crystalline
Molecular weight:
146.14
Estimated delivery in United States, on Monday 7 Feb 2022
Basimglurant
CAS:802906-73-6
Basimglurant is a potent, selective and orally available modulator of mGlu5 negative allosteric(Kd of 1.1 …
Formula:
C18H13ClFN3
Purity:
99.38%
Color and Shape:
solid
Molecular weight:
325.77
Estimated delivery in United States, on Monday 7 Feb 2022
MFZ 10-7 hydrochloride
CAS:1779796-36-9
MFZ 10-7 hydrochloride is a highly potent and selective negative allosteric modulator of mGluR5 NAM
Formula:
C15H10ClFN2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
272.7
Estimated delivery in United States, on Monday 7 Feb 2022
ATPO
CAS:252930-37-3
ATPO is Competitive antagonist at GluR1-4 (AMPA-preferring) receptors.
Formula:
C11H19N2O7P
Purity:
99.41%
Color and Shape:
solid
Molecular weight:
322.25
Estimated delivery in United States, on Monday 7 Feb 2022
UV0155041
CAS:1093757-42-6
UV0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, …
Formula:
C14H15Cl2NO3
Purity:
99.56%
Color and Shape:
solid
Molecular weight:
316.18
Estimated delivery in United States, on Monday 7 Feb 2022
VU6012962
CAS:2313526-86-0
VU6012962 is an orally bioavailable negative allosteric modulator of CNS-penetrant metabotropic glutamate receptor 7(mGlu7; IC50: …
Formula:
C21H19F3N4O4
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
448.4
Estimated delivery in United States, on Monday 7 Feb 2022
Philanthotoxin 74 dihydrochloride
CAS:1227301-51-0
Philanthotoxin 74 dihydrochloride is an AMPAR antagonist. Philanthotoxin 74 dihydrochloride inhibits GluR3 and GluR1 (IC50s: …
Formula:
C24H44Cl2N4O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
507.54
Estimated delivery in United States, on Monday 7 Feb 2022
Fenobam
CAS:57653-26-6
Fenobam shows inverse agonist activity which blocks the mGlu5 receptor basal activity(IC50: 84 nM). Fenobam …
Formula:
C11H11ClN4O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
266.68
Estimated delivery in United States, on Monday 7 Feb 2022
CTEP
CAS:871362-31-1
CTEP (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 …
Formula:
C19H13ClF3N3O
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
391.77
Estimated delivery in United States, on Monday 7 Feb 2022
Biphenylindanone A
CAS:866823-73-6
Biphenylindanone A is a selective potentiator of human mGluR2 (hmGluR2),and for the treatment of neurological …
Formula:
C30H30O4
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
454.56
Estimated delivery in United States, on Monday 7 Feb 2022
Cyclothiazide
CAS:2259-96-3
Cyclothiazide is a benzothiadiazide that acts as a potentiator of AMPA receptorsthat potently inhibits AMPA …
Formula:
C14H16ClN3O4S2
Purity:
100.00%
Color and Shape:
Crystals From Dilute Alcohol Solid
Molecular weight:
389.9
Estimated delivery in United States, on Monday 7 Feb 2022
HBT1
CAS:489408-02-8
HBT1 is an AMPA receptor potentiator that induces production of brain-derived neurotrophic factor (BDNF) and …
Formula:
C16H17F3N4O2S
Color and Shape:
Solid
Molecular weight:
386.39
Estimated delivery in United States, on Monday 7 Feb 2022
(RS)-MCPG
CAS:146669-29-6
(RS)-MCPG is a non-selective group I/II metabotropic glutamate receptor antagonist.
Formula:
C10H11NO4
Purity:
99.96%
Color and Shape:
solid
Molecular weight:
209.2
Estimated delivery in United States, on Monday 7 Feb 2022
Piracetam
CAS:7491-74-9
Piracetam, a cyclic derivative of the neurotransmitter gamma-aminobutyric acid (GABA), is used in therapy of …
Formula:
C6H10N2O2
Purity:
99.72%
Color and Shape:
Crystals From Isopropanol
Molecular weight:
142.16
Estimated delivery in United States, on Monday 7 Feb 2022
VU 0364770
CAS:61350-00-3
VU 0364770(EC50=1.1 μM), a positive allosteric modulator(PAM) of mGlu4, shows insignificant activity at 68 other …
Formula:
C12H9ClN2O
Purity:
99.92%
Color and Shape:
solid
Molecular weight:
232.67
Estimated delivery in United States, on Monday 7 Feb 2022
Harmine hydrochloride
CAS:343-27-1
Harmine hydrochloride is extracted from Peganum Harmala Genus.
Formula:
C13H13ClN2O
Purity:
99.45%
Color and Shape:
Yellow To Slightly Green Crystalline Powder
Molecular weight:
248.71
Estimated delivery in United States, on Monday 7 Feb 2022
PHCCC
CAS:179068-02-1
PHCCC is a Group I metabotropic glutamate receptor antagonist and a positive allosteric modulator of …
Formula:
C17H14N2O3
Purity:
99.31%
Color and Shape:
Solid
Molecular weight:
294.31
Estimated delivery in United States, on Monday 7 Feb 2022
VU 0361737
CAS:1161205-04-4
VU 0361737 is a specific positive allosteric modulator (PAM) of mGlu4 receptor.The EC50 of VU …
Formula:
C13H11ClN2O2
Purity:
99.86%
Color and Shape:
solid
Molecular weight:
262.69
Estimated delivery in United States, on Monday 7 Feb 2022
LY450108
CAS:376594-67-1
LY450108 is a potentiator of the AMPA receptor.
Formula:
C19H22F2N2O3S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
396.45
Estimated delivery in United States, on Monday 7 Feb 2022
E4CPG
CAS:170846-89-6
E4CPG is a novel group I/II metabotropic glutamate receptor antagonist, more potent than (RS)-MCPG.
Formula:
C11H13NO4
Color and Shape:
Solid
Molecular weight:
223.23
Estimated delivery in United States, on Monday 7 Feb 2022
Xanthurenic Acid
CAS:59-00-7
Xanthurenic acid, a molecule arising from tryptophan metabolism by transamination of 3-hydroxykynurenine, activates mGlu2/3 Metabotropic …
Formula:
C10H7NO4
Purity:
93.54%
Color and Shape:
Solid
Molecular weight:
205.17
Estimated delivery in United States, on Monday 7 Feb 2022
CFMTI
CAS:864864-17-5
CFMTI is a potent and selective metabotropic glutamate receptor (mGluR) 1 allosteric antagonist (IC50: 2.6 …
Formula:
C19H16FN5O
Purity:
98.61%
Color and Shape:
Solid
Molecular weight:
349.37
Estimated delivery in United States, on Monday 7 Feb 2022
IEM 1754 2HBr
CAS:162831-31-4
IEM 1754 2HBr is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 …
Formula:
C16H30N2·2HBr
Purity:
98.0%
Molecular weight:
412.25
Estimated delivery in United States, on Monday 7 Feb 2022
CMPDA
CAS:380607-77-2
CMPDA is a positive allosteric modulator of AMPA receptors (EC50s: 45.4 nM/63.4 nM for GluA2i/GluA2o …
Formula:
C16H28N2O4S2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
376.53
Estimated delivery in United States, on Monday 7 Feb 2022
3-MATIDA
CAS:518357-51-2
3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a). Displays 40-fold selectivity over …
Formula:
C8H9NO4S
Purity:
98.41%
Color and Shape:
solid
Molecular weight:
215.22
Estimated delivery in United States, on Monday 7 Feb 2022
Chicago Sky Blue 6B
CAS:2610-05-1
Chicago sky blue 6B, a vesicular glutamate transporters inhibitor, attenuates methamphetamine-induced hyperactivity and behavioral sensitization …
Formula:
C34H24N6Na4O16S4
Purity:
91.79%
Color and Shape:
Greenish Blue Powder
Molecular weight:
992.8
Estimated delivery in United States, on Monday 7 Feb 2022
VU 0357121
CAS:433967-28-3
VU0357121, a positive allosteric modulator of mGlu5 (EC50: 33 nM), is inactive or very weakly …
Formula:
C17H17F2NO2
Color and Shape:
solid
Molecular weight:
305.32
Estimated delivery in United States, on Monday 7 Feb 2022
Farampator
CAS:211735-76-1
Farampator (CX-691;Org24448) is an AMPA receptor positive modulator.
Formula:
C12H13N3O2
Purity:
99.83%
Color and Shape:
solid
Molecular weight:
231.26
Estimated delivery in United States, on Monday 7 Feb 2022
pep2-EVKI acetate(1315378-67-6 free base)
Pep2-EVKI acetate is a cell-permeable peptide. Pep2-EVKI acetate interferes the interaction between protein interacting with …
Formula:
C64H99N13O21
Molecular weight:
1386.55
Estimated delivery in United States, on Monday 7 Feb 2022
AMN082
CAS:83027-13-8
AMN082 is a metabotropic glutamate receptor 7 allosteric agonist.
Formula:
C28H28N2
Molecular weight:
392.54
Estimated delivery in United States, on Monday 7 Feb 2022
(R)-ADX-47273
CAS:851881-59-9
(R)-ADX-47273 is a potent mGluR5 positive allosteric modulator(EC50 of 168 nM for potentiation ).
Formula:
C20H17F2N3O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
369.36
Estimated delivery in United States, on Monday 7 Feb 2022
