Tyrosine Kinase/Adaptors
Tyrosine kinase and adaptor inhibitors are compounds that target tyrosine kinases and their associated adaptor proteins, which play pivotal roles in cell signaling, growth, and differentiation. These inhibitors are essential tools in cancer research, as many tyrosine kinases are involved in the signaling pathways that drive tumor growth and metastasis. By inhibiting tyrosine kinases, these compounds can block critical signaling cascades, offering potential therapeutic strategies for various cancers and other diseases involving abnormal cell signaling. At CymitQuimica, we provide a comprehensive range of high-quality tyrosine kinase and adaptor inhibitors to support your research in oncology, molecular biology, and targeted therapy development.
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Subcategories of "Tyrosine Kinase/Adaptors"
ALK
CSF-1R
EGFR
Ephrin Receptor
FLT
Fibroblast Growth Factor Receptor (FGFR)
HER
Hck
IGF-1R
PDGFR
PYK2
Src
TAM Receptor
Tie-2
Trk receptor
Tyrosine Kinases
VEGFR
c-Fms
c-Kit
c-Met/HGFR
c-RET
Show 13 more subcategories
Products of "Tyrosine Kinase/Adaptors"
CEP-40783
CAS:1437321-24-8
CEP-40783 (RXDX-106) is an effective, specific and orally active AXL/c-Met inhibitor (IC50: 7/12 nM). It …
Formula:
C31H26F2N4O6
Purity:
99.45% - 99.64%
Color and Shape:
Solid
Molecular weight:
588.56
Ref: TM-T4426
| 5mg | 50.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 164.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 293.00 € | ||
| 200mg | 423.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
JNJ-38158471
CAS:951151-97-6
JNJ-38158471 (CS-2660), a highly selective, orally available, well tolerated VEGFR2 inhibitor, inhibits closely related tyrosine …
Formula:
C15H17ClN6O3
Purity:
97.08%
Color and Shape:
Solid
Molecular weight:
364.79
Ref: TM-T22349
| 1mg | 51.00 € | ||
| 2mg | 72.00 € | ||
| 5mg | 102.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 364.00 € | ||
| 100mg | 490.00 € | ||
| 200mg | 673.00 € | ||
| 1mL*10mM (DMSO) | 109.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Tucatinib
CAS:937263-43-9
Tucatinib (ONT-380) is a potent and selective HER2 inhibitor (IC50: 8 nM).
Formula:
C26H24N8O2
Purity:
99.05% - 99.96%
Color and Shape:
Solid
Molecular weight:
480.52
Ref: TM-T2364
| 1g | 1,110.00 € | ||
| 2mg | 40.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 127.00 € | ||
| 50mg | 189.00 € | ||
| 100mg | 343.00 € | ||
| 500mg | 812.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Golvatinib
CAS:928037-13-2
Golvatinib (E-7050) is an orally bioavailable dual kinase inhibitor of c-Met (hepatocyte growth factor receptor) …
Formula:
C33H37F2N7O4
Purity:
98.24% - ≥95%
Color and Shape:
Solid
Molecular weight:
633.69
Ref: TM-T6517
| 2mg | 45.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 155.00 € | ||
| 50mg | 195.00 € | ||
| 100mg | 347.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
FIIN-3
CAS:1637735-84-2
FIIN-3 is an irreversible inhibitor of FGFR.
Formula:
C34H36Cl2N8O4
Purity:
97.63% - 98.92%
Color and Shape:
Solid
Molecular weight:
691.61
Ref: TM-T3466
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 244.00 € | ||
| 50mg | 360.00 € | ||
| 100mg | 513.00 € | ||
| 200mg | 699.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ningetinib Tosylate
CAS:1394820-77-9
Ningetinib Tosylate is an orally bioavailable tyrosine kinase inhibitor with IC50s of <1.0, 1.9 and …
Formula:
C38H37FN4O8S
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
728.79
Ref: TM-TQ0041
| 5mg | 47.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 107.00 € | ||
| 50mg | 191.00 € | ||
| 100mg | 350.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Gandotinib
CAS:1229236-86-5
LY2784544(Gandotinib (LY2784544)) is a potent JAK2 inhibitor (IC50: 3 nM), effective in JAK2V617F(Ki: 0.245 nM).
Formula:
C23H25ClFN7O
Purity:
99.16% - 99.86%
Color and Shape:
Solid
Molecular weight:
469.94
Ref: TM-T2638
| 5mg | 51.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 290.00 € | ||
| 100mg | 460.00 € | ||
| 500mg | 1,012.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Insulin(cattle)
CAS:11070-73-8
Insulin(cattle) is a peptide hormone that promotes glycogen synthesis. Insulin) has hypoglycemic activity. Cost-effective and …
Formula:
C254H377N65O75S6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
5733.49
Ref: TM-TP1125
| 10mg | 52.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 127.00 € | ||
| 100mg | 185.00 € | ||
| 200mg | 292.00 € | ||
| 500mg | 519.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
WZ8040
CAS:1214265-57-2
WZ8040 is a novel mutant-selective irreversible EGFRT790M inhibitor, does not inhibit ERBB2 phosphorylation (T798I).
Formula:
C24H25ClN6OS
Purity:
97.42%
Color and Shape:
Solid
Molecular weight:
481.01
Ref: TM-T6734
| 1mg | 47.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 147.00 € | ||
| 25mg | 241.00 € | ||
| 50mg | 358.00 € | ||
| 100mg | 527.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
ZD-4190
CAS:413599-62-9
ZD-4190 blocks VEGFR2 and EGFR, aiding cancer treatment.
Formula:
C19H16BrFN6O2
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
459.27
Ref: TM-T5475
| 1mg | 82.00 € | ||
| 5mg | 177.00 € | ||
| 10mg | 266.00 € | ||
| 25mg | 422.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € | ||
| 1mL*10mM (DMSO) | 179.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
MCB-613
CAS:1162656-22-5
MCB-613 is an effective steroid receptor coactivator (SRC) stimulator.
Formula:
C20H20N2O
Purity:
98.17% - 99.48%
Color and Shape:
Solid
Molecular weight:
304.39
Ref: TM-T6886
| 1mg | 45.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 256.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 560.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
X-376
CAS:1365267-27-1
X-376 (Ensartinib) is an orally available small molecule inhibitor of the receptor tyrosine kinase ALK …
Formula:
C25H25Cl2FN6O3
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
547.41
Ref: TM-T3550
| 1mg | 35.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 255.00 € | ||
| 50mg | 422.00 € | ||
| 100mg | 574.00 € | ||
| 1mL*10mM (DMSO) | 104.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
SKLB1002
CAS:1225451-84-2
SKLB1002 is a potent and ATP-competitive VEGFR2 inhibitor with IC50 of 32 nM.
Formula:
C13H12N4O2S2
Purity:
100% - 99.15%
Color and Shape:
Solid
Molecular weight:
320.39
Ref: TM-T2421
| 1mg | 44.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 81.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 201.00 € | ||
| 50mg | 340.00 € | ||
| 100mg | 551.00 € | ||
| 500mg | 1,187.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Mutant EGFR inhibitor
CAS:1421373-62-7
Selective, potent inhibitor for mutated EGFR: L858R, Exon19 deletion, T790M resistance mutants.
Formula:
C27H30ClN7O2
Purity:
96.21% - 98%
Color and Shape:
Solid
Molecular weight:
520.03
Ref: TM-T2705
| 1mg | 36.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 258.00 € | ||
| 100mg | 371.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 104.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PF 477736
CAS:952021-60-2
PF 477736 (PF-736,PF-00477736) is a specifc, effective and ATP-competitive Chk1 inhibitor (Ki: 0.49 nM ) …
Formula:
C22H25N7O2
Purity:
98% - 98.34%
Color and Shape:
Solid
Molecular weight:
419.48
Ref: TM-T6028
| 2mg | 49.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PD153035 hydrochloride
CAS:183322-45-4
PD153035 hydrochloride (ZM 252868) is a effective and selective inhibitor of EGFR; few influence against …
Formula:
C16H15BrClN3O2
Purity:
100% - ≥95%
Color and Shape:
Solid
Molecular weight:
396.67
Ref: TM-T1761
| 5mg | 35.00 € | ||
| 10mg | 44.00 € | ||
| 25mg | 81.00 € | ||
| 50mg | 142.00 € | ||
| 100mg | 233.00 € | ||
| 500mg | 530.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BMS817378
CAS:1174161-69-3
BMS817378 is a potent and selective inhibitor of MET(IC50 : 1.7 nM).
Formula:
C24H18ClF2N4O7P
Purity:
100%
Color and Shape:
Solid
Molecular weight:
578.85
Ref: TM-T7787
| 1mg | 91.00 € | ||
| 2mg | 114.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 241.00 € | ||
| 25mg | 438.00 € | ||
| 50mg | 642.00 € | ||
| 100mg | 915.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Filgotinib
CAS:1206161-97-8
Filgotinib (GLPG0634) is a selective JAK1 inhibitor. The IC50 values against JAK1, JAK2, JAK3, and …
Formula:
C21H23N5O3S
Purity:
98.03% - ≥95%
Color and Shape:
Solid
Molecular weight:
425.5
Ref: TM-T1929
| 1mg | 38.00 € | ||
| 5mg | 77.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 161.00 € | ||
| 50mg | 241.00 € | ||
| 100mg | 318.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
VU6015929
CAS:2442597-56-8
VU6015929 is an inhibitor of active dual discoidin domain receptor 1/2 (DDR1/2)( IC50s of 4.67 …
Formula:
C24H19F4N5O2
Purity:
97.07% - 99.63%
Color and Shape:
Solid
Molecular weight:
485.43
Ref: TM-T7862
| 1mg | 68.00 € | ||
| 5mg | 136.00 € | ||
| 10mg | 205.00 € | ||
| 25mg | 338.00 € | ||
| 50mg | 478.00 € | ||
| 100mg | 643.00 € | ||
| 200mg | 867.00 € | ||
| 1mL*10mM (DMSO) | 145.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Masitinib
CAS:790299-79-5
Masitinib (AB1010) is a tyrosine-kinase inhibitor used in the treatment of mast cell tumors in …
Formula:
C28H30N6OS
Purity:
100% - 99.91%
Color and Shape:
Solid
Molecular weight:
498.64
Ref: TM-T2609
| 5mg | 36.00 € | ||
| 10mg | 52.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 156.00 € | ||
| 200mg | 236.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
