Tyrosine Kinase/Adaptors
Tyrosine kinase and adaptor inhibitors are compounds that target tyrosine kinases and their associated adaptor proteins, which play pivotal roles in cell signaling, growth, and differentiation. These inhibitors are essential tools in cancer research, as many tyrosine kinases are involved in the signaling pathways that drive tumor growth and metastasis. By inhibiting tyrosine kinases, these compounds can block critical signaling cascades, offering potential therapeutic strategies for various cancers and other diseases involving abnormal cell signaling. At CymitQuimica, we provide a comprehensive range of high-quality tyrosine kinase and adaptor inhibitors to support your research in oncology, molecular biology, and targeted therapy development.
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Subcategories of "Tyrosine Kinase/Adaptors"
ALK
CSF-1R
EGFR
Ephrin Receptor
FLT
Fibroblast Growth Factor Receptor (FGFR)
HER
Hck
IGF-1R
PDGFR
PYK2
Src
TAM Receptor
Tie-2
Trk receptor
Tyrosine Kinases
VEGFR
c-Fms
c-Kit
c-Met/HGFR
c-RET
Show 13 more subcategories
Products of "Tyrosine Kinase/Adaptors"
SU6656
CAS:330161-87-0
SU 6656 is a selective inhibitor of Src family kinases, with IC50 of 280 nM, …
Formula:
C19H21N3O3S
Purity:
97% - 98.21%
Color and Shape:
Solid
Molecular weight:
371.45
Ref: TM-T6997
| 1mg | 40.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 265.00 € | ||
| 50mg | 439.00 € | ||
| 100mg | 652.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Selitrectinib
CAS:2097002-61-2
Selitrectinib (LOXO-195) is a potent and selective inhibitor of the receptor tyrosine kinases(TRK).Cost-effective and quality-assured.
Formula:
C20H21FN6O
Purity:
99.55% - ≥95%
Color and Shape:
Solid
Molecular weight:
380.42
Ref: TM-T7435
| 1mg | 40.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 223.00 € | ||
| 50mg | 331.00 € | ||
| 100mg | 440.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
SB-431542
CAS:301836-41-9
SB-431542 is an inhibitor of ALK5/TGF-β type I Receptor (IC50=94 nM) and is selective.
Formula:
C22H16N4O3
Purity:
100% - 99.87%
Color and Shape:
Solid
Molecular weight:
384.39
Ref: TM-T1726
| 5mg | 55.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | 279.00 € | ||
| 100mg | 517.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ponatinib
CAS:943319-70-8
Ponatinib (AP24534) is an orally available, multitargeted kinase inhibitor (IC50s: 0.37/1.1/1.5/2.2/5.4 nM for Abl, PDGFRα, …
Formula:
C29H27F3N6O
Purity:
98% - 99.74%
Color and Shape:
Solid
Molecular weight:
532.56
Ref: TM-T2372
| 10mg | 54.00 € | ||
| 50mg | 69.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 136.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GSK1838705A
CAS:1116235-97-2
GSK1838705A: IGF-1R inhibitor (IC50=2.0nM), IR (1.6nM), ALK (0.5nM), minimal other kinase impact.
Formula:
C27H29FN8O3
Purity:
100% - 99.63%
Color and Shape:
Solid
Molecular weight:
532.57
Ref: TM-T3079
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 262.00 € | ||
| 50mg | 472.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
ZM39923 hydrochloride
CAS:1021868-92-7
ZM39923 hydrochloride (JAK3 Inhibitor IV) is an JAK1/3 inhibitor, almost no activity to JAK2 and …
Formula:
C23H25NO·HCl
Purity:
98.05%
Color and Shape:
Solid
Molecular weight:
367.91
Ref: TM-T6145
| 5mg | 58.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 304.00 € | ||
| 100mg | 455.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Alflutinib
CAS:1869057-83-9
Alflutinib (ASK120067) is an inhibitor of EGFR, and its targets including EGFR activating mutations and …
Formula:
C28H31F3N8O2
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
568.59
Ref: TM-T22254
| 1mg | 210.00 € | ||
| 5mg | 428.00 € | ||
| 10mg | 610.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,295.00 € | ||
| 100mg | 1,755.00 € | ||
| 1mL*10mM (DMSO) | 556.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Crizotinib
CAS:877399-52-5
Crizotinib (PF-02341066) is an ATP-competitive small-molecule tyrosine kinases inhibitor of c-MET (IC50: 8 nM) and …
Formula:
C21H22Cl2FN5O
Purity:
99% - 99.87%
Color and Shape:
Solid
Molecular weight:
450.34
Ref: TM-T1661
| 10mg | 55.00 € | ||
| 25mg | 64.00 € | ||
| 50mg | 73.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 100.00 € | ||
| 500mg | 158.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GNF-5837
CAS:1033769-28-6
GNF-5837 is a specific, and orally bioavailable pan-TRK inhibitor for TrkA/TrkB (IC50: 8/12 nM).
Formula:
C28H21F4N5O2
Purity:
96.17% - 99.29%
Color and Shape:
Solid
Molecular weight:
535.49
Ref: TM-T6097
| 5mg | 50.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 185.00 € | ||
| 100mg | 305.00 € | ||
| 200mg | 398.00 € | ||
| 500mg | 643.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
TAK-659 hydrochloride
CAS:1952251-28-3
TAK-659 hydrochloride (TAK-659) is a potent and selective inhibitor of spleen tyrosine kinase (SYK) with …
Formula:
C17H22ClFN6O
Purity:
99.28% - 99.63%
Color and Shape:
Solid
Molecular weight:
380.85
Ref: TM-T4209
| 1mg | 39.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 500.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Insulin (human)
CAS:11061-68-0
Insulin (human) is a peptide hormone that promotes glycogen synthesis and regulates glucose levels in …
Formula:
C257H383N65O77S6
Purity:
97.32% - 99.99%
Color and Shape:
Solid
Molecular weight:
5807.57
Ref: TM-T8221
| 5mg | 35.00 € | ||
| 10mg | 46.00 € | ||
| 25mg | 65.00 € | ||
| 50mg | 82.00 € | ||
| 100mg | 92.00 € | ||
| 200mg | 130.00 € | ||
| 500mg | 212.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
NVP-AEW541
CAS:475489-16-8
NVP-AEW541 (AEW541), a potent inhibitor of IGF-1R(IC50=150 nM) and InsR(IC50=140 nM), exhibits excellent efficiency and …
Formula:
C27H29N5O
Purity:
96.03% - 99.55%
Color and Shape:
Solid
Molecular weight:
439.55
Ref: TM-T6080
| 1mg | 48.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 149.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BLU-263
CAS:2505078-08-8
BLU-263 is an investigational, potent, and selective oral small molecule inhibitor of KIT with sub-nanomolar …
Formula:
C27H29FN10O
Purity:
99.67%
Color and Shape:
Solid
Molecular weight:
528.58
Ref: TM-T9295
| 1mg | 64.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 220.00 € | ||
| 25mg | 423.00 € | ||
| 50mg | 553.00 € | ||
| 100mg | 793.00 € | ||
| 200mg | 1,063.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CP-673451
CAS:343787-29-1
CP-673451 is a specific inhibitor of PDGFRα/β (IC50: 10/1 nM) with antiangiogenic and antitumor activity …
Formula:
C24H27N5O2
Purity:
99.88% - 99.93%
Color and Shape:
Solid
Molecular weight:
417.5
Ref: TM-T6091
| 1mg | 52.00 € | ||
| 2mg | 65.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 346.00 € | ||
| 50mg | 529.00 € | ||
| 100mg | 761.00 € | ||
| 500mg | 1,576.00 € | ||
| 1mL*10mM (DMSO) | 114.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Hepln-13
CAS:64369-13-7
Hepln-13 is a hepsin inhibitor that acts by hindering prostate cancer bone metastasis.
Formula:
C17H13BrN2
Purity:
97.67%
Color and Shape:
Solid
Molecular weight:
325.2
Ref: TM-T25492
| 1mg | 37.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 351.00 € | ||
| 100mg | 488.00 € | ||
| 200mg | 675.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BMS-986142
CAS:1643368-58-4
BMS-986142 is a potent and highly selective reversible BTK inhibitor (IC50: 0.5 nM).
Formula:
C32H30F2N4O4
Purity:
98.7% - 99.76%
Color and Shape:
Solid
Molecular weight:
572.6
Ref: TM-T5138
| 1mg | 138.00 € | ||
| 5mg | 369.00 € | ||
| 10mg | 587.00 € | ||
| 25mg | 919.00 € | ||
| 50mg | 1,234.00 € | ||
| 100mg | 1,653.00 € | ||
| 200mg | 2,256.00 € | ||
| 500mg | 3,333.00 € | ||
| 1mL*10mM (DMSO) | 485.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Roblitinib
CAS:1708971-55-4
Roblitinib (FGF-401), an FGFR4 inhibitor, potentially blocks tumor growth by halting cell proliferation and survival.
Formula:
C25H30N8O4
Purity:
97.27% - 99%
Color and Shape:
Solid
Molecular weight:
506.56
Ref: TM-T4235
| 1mg | 58.00 € | ||
| 2mg | 82.00 € | ||
| 5mg | 101.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 302.00 € | ||
| 50mg | 523.00 € | ||
| 100mg | 735.00 € | ||
| 500mg | 1,550.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
WS6
CAS:1421227-53-3
WS6, a β cell proliferation inducer, regulates Erb3 binding protein-1 (EBP1) and the IκB kinase …
Formula:
C29H31F3N6O3
Purity:
97.23% - 99.83%
Color and Shape:
Solid
Molecular weight:
568.59
Ref: TM-T2106
| 1mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 220.00 € | ||
| 100mg | 327.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
SU5214
CAS:186611-04-1
SU5214 is a modulator of tyrosine kinase signal transduction.
Formula:
C16H13NO2
Purity:
99.52% - 99.55%
Color and Shape:
Solid
Molecular weight:
251.28
Ref: TM-T3569
| 5mg | 38.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 107.00 € | ||
| 50mg | 169.00 € | ||
| 100mg | 269.00 € | ||
| 200mg | 391.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BPR1J-097 hydrochloride (1327167-19-0(free base))
BPR1J-097, a new-type small molecule FLT-3 inhibitor(IC50=11±7 nM), is with great anti-tumor activities in vivo.
Formula:
C27H29ClN6O3S
Purity:
98% - 98.73%
Color and Shape:
Solid
Molecular weight:
553.07
Ref: TM-T4261
| 1mg | 50.00 € | ||
| 2mg | 65.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 152.00 € | ||
| 25mg | 265.00 € | ||
| 50mg | 448.00 € | ||
| 100mg | 644.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
