Tyrosine Kinase/Adaptors
Tyrosine kinase and adaptor inhibitors are compounds that target tyrosine kinases and their associated adaptor proteins, which play pivotal roles in cell signaling, growth, and differentiation. These inhibitors are essential tools in cancer research, as many tyrosine kinases are involved in the signaling pathways that drive tumor growth and metastasis. By inhibiting tyrosine kinases, these compounds can block critical signaling cascades, offering potential therapeutic strategies for various cancers and other diseases involving abnormal cell signaling. At CymitQuimica, we provide a comprehensive range of high-quality tyrosine kinase and adaptor inhibitors to support your research in oncology, molecular biology, and targeted therapy development.
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Subcategories of "Tyrosine Kinase/Adaptors"
ALK
CSF-1R
EGFR
Ephrin Receptor
FLT
Fibroblast Growth Factor Receptor (FGFR)
HER
Hck
IGF-1R
PDGFR
PYK2
Src
TAM Receptor
Tie-2
Trk receptor
Tyrosine Kinases
VEGFR
c-Fms
c-Kit
c-Met/HGFR
c-RET
Show 13 more subcategories
Products of "Tyrosine Kinase/Adaptors"
Neratinib
CAS:698387-09-6
Neratinib (HKI-272) (HKI-272) is an orally available, irreversible tyrosine kinase inhibitor for HER2 and EGFR …
Formula:
C30H29ClN6O3
Purity:
100% - 98.55%
Color and Shape:
Solid
Molecular weight:
557.04
Ref: TM-T2325
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 92.00 € | ||
| 100mg | 122.00 € | ||
| 200mg | 184.00 € | ||
| 500mg | 307.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Osimertinib mesylate
CAS:1421373-66-1
Osimertinib mesylate (AZD-9291 mesylate) is an EGFR third-generation inhibitor. Osimertinib mesylate has antitumor activity. Cost-effective …
Formula:
C29H37N7O5S
Purity:
100% - 99.53%
Color and Shape:
Solid
Molecular weight:
595.71
Ref: TM-T3634
| 1g | 149.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 60.00 € | ||
| 50mg | 86.00 € | ||
| 100mg | 94.00 € | ||
| 200mg | 111.00 € | ||
| 500mg | 129.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PF-6274484
CAS:1035638-91-5
PF-6274484 is an EGFR inhibitor with Ki values of 0.14 and 0.18 nM for EGFR-L858R/T790M …
Formula:
C18H14ClFN4O2
Purity:
97.71%
Color and Shape:
Solid
Molecular weight:
372.78
Ref: TM-T22396
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | 510.00 € | ||
| 500mg | 1,112.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
RG13022
CAS:136831-48-6
RG13022 (Tyrphostin RG13022) is a tyrosine kinase inhibitor; inhibits the autophosphorylation reaction of the EGF …
Formula:
C16H14N2O2
Purity:
98.38%
Color and Shape:
Solid
Molecular weight:
266.29
Ref: TM-T3545
| 2mg | 46.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 177.00 € | ||
| 50mg | 298.00 € | ||
| 100mg | 470.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Scutellarein
CAS:529-53-3
Scutellarein (6-Hydroxyapigenin) reduces inflammatory responses by inhibiting Src kinase activity.
Formula:
C15H10O6
Purity:
98.32% - 99.63%
Color and Shape:
Solid
Molecular weight:
286.24
Ref: TM-T3319
| 20mg | 107.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PRT-060318
CAS:1194961-19-7
PRT-060318 (P142-76) is a novel selective inhibitor of the Syk tyrosine kinase, as an approach …
Formula:
C18H24N6O
Purity:
98.82%
Color and Shape:
Solid
Molecular weight:
340.42
Ref: TM-T6957
| 1mg | 41.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 133.00 € | ||
| 25mg | 270.00 € | ||
| 50mg | 455.00 € | ||
| 100mg | 664.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
LDN-192960
CAS:184582-62-5
LDN-192960 is a potent inhibitor of Haspin and DYRK2 (IC50s: 10 nM and 48 nM).
Formula:
C18H20N2O2S
Purity:
98.01% - 99.51%
Color and Shape:
Solid
Molecular weight:
328.43
Ref: TM-TQ0111
| 1mg | 130.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 247.00 € | ||
| 25mg | 496.00 € | ||
| 50mg | 722.00 € | ||
| 100mg | 1,013.00 € | ||
| 200mg | 807.00 € | ||
| 500mg | 2,018.00 € | ||
| 1mL*10mM (DMSO) | 167.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
SU14813
CAS:627908-92-3
SU14813: inhibits multiple kinases (VEGFR2, VEGFR1, PDGFRβ, KIT) with IC50s of 50, 2, 4, 15 …
Formula:
C23H27FN4O4
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
442.48
Ref: TM-T7945
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 142.00 € | ||
| 100mg | 220.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AIM-100
CAS:873305-35-2
AIM-100 is a Ack1 inhibitor (IC50: 24 nM).
Formula:
C23H21N3O2
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
371.43
Ref: TM-T5092
| 2mg | 49.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 203.00 € | ||
| 50mg | 353.00 € | ||
| 100mg | 558.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Baricitinib
CAS:1187594-09-7
Baricitinib (INCB028050) is an orally JAK1 and JAK2 inhibitor. Baricitinib has anti-inflammatory and anti-tumor activity. …
Formula:
C16H17N7O2S
Purity:
100% - 99.79%
Color and Shape:
Solid
Molecular weight:
371.42
Ref: TM-T2485
| 5mg | 50.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 89.00 € | ||
| 50mg | 113.00 € | ||
| 100mg | 142.00 € | ||
| 200mg | 184.00 € | ||
| 500mg | 306.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Src Inhibitor 1
CAS:179248-59-0
Src Inhibitor 1 (Src Kinase Inhibitor 1) is a potent and selective dual site Src …
Formula:
C22H19N3O3
Purity:
100% - 99.38%
Color and Shape:
Solid
Molecular weight:
373.4
Ref: TM-T3593
| 1mg | 39.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 77.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 372.00 € | ||
| 100mg | 541.00 € | ||
| 500mg | 1,133.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Vimseltinib
CAS:1628606-05-2
Vimseltinib (DCC-3014) is a c-FMS (CSF-IR) and c-Kit dual inhibitor (IC50s: <0.01 μM and 0.1-1 …
Formula:
C23H25N7O2
Purity:
98.98% - 99.57%
Color and Shape:
Solid
Molecular weight:
431.49
Ref: TM-T10652
| 1mg | 91.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 308.00 € | ||
| 25mg | 527.00 € | ||
| 50mg | 719.00 € | ||
| 100mg | 926.00 € | ||
| 1mL*10mM (DMSO) | 212.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
WS3
CAS:1421227-52-2
WS3, a β cell proliferation inducer, regulates Erb3 binding protein-1 (EBP1) and the IκB kinase …
Formula:
C28H30F3N7O3
Purity:
97.93% - 98.81%
Color and Shape:
Solid
Molecular weight:
569.58
Ref: TM-T2055
| 5mg | 52.00 € | ||
| 10mg | 75.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 209.00 € | ||
| 100mg | 386.00 € | ||
| 1mL*10mM (DMSO) | 70.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CL-387785
CAS:194423-06-8
CL-387785 is an irreversible EGFR inhibitor with IC50 of 370 pM; overcomes T790M mutation resistance.
Formula:
C18H13BrN4O
Purity:
96.68% - 98.09%
Color and Shape:
Solid
Molecular weight:
381.23
Ref: TM-T2245
| 5mg | 38.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 163.00 € | ||
| 100mg | 255.00 € | ||
| 200mg | 359.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Zoligratinib
CAS:1265229-25-1
Zoligratinib (CH5183284) is a selective and orally available FGFR inhibitor, which is for FGFR1, FGFR2, …
Formula:
C20H16N6O
Purity:
95.28% - 98.94%
Color and Shape:
Solid
Molecular weight:
356.38
Ref: TM-T6024
| 5mg | 46.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 121.00 € | ||
| 50mg | 184.00 € | ||
| 100mg | 343.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Remibrutinib
CAS:1787294-07-8
Remibrutinib inhibits BTK activity with an IC50 value of 0.023 μM in blood.
Formula:
C27H27F2N5O3
Purity:
99.21%
Color and Shape:
Solid
Molecular weight:
507.53
Ref: TM-T16730
| 1mg | 95.00 € | ||
| 5mg | 217.00 € | ||
| 10mg | 352.00 € | ||
| 25mg | 594.00 € | ||
| 50mg | 744.00 € | ||
| 100mg | 1,144.00 € | ||
| 200mg | 1,547.00 € | ||
| 1mL*10mM (DMSO) | 247.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Savolitinib
CAS:1313725-88-0
Savolitinib (Volitinib) (AZD-6094) is an effective, selective, and orally bioavailable c-Met inhibitor (IC50s: 5 nM/3 …
Formula:
C17H15N9
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
345.36
Ref: TM-TQ0210
| 1mg | 49.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 366.00 € | ||
| 100mg | 555.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
UNC2881
CAS:1493764-08-1
UNC2881 is a specific Mer tyrosine kinase inhibitor (IC50: 4.3 nM). It is about 83- …
Formula:
C25H33N7O2
Purity:
98.97% - 99.74%
Color and Shape:
Solid
Molecular weight:
463.58
Ref: TM-T2629
| 5mg | 45.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 116.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 302.00 € | ||
| 200mg | 435.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
ON123300
CAS:1357470-29-1
ON123300 is a potent and multi-targeted kinase inhibitor for CDK4/Ark5/PDGFRβ/FGFR1/RET/Fyn (IC50: 3.9/5/26/26/9.2/11 nM).
Formula:
C24H27N7O
Purity:
99.22% - 99.53%
Color and Shape:
Solid
Molecular weight:
429.52
Ref: TM-T6920
| 1mg | 46.00 € | ||
| 2mg | 61.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 146.00 € | ||
| 25mg | 268.00 € | ||
| 50mg | 437.00 € | ||
| 100mg | 635.00 € | ||
| 200mg | 515.00 € | ||
| 500mg | 1,291.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Capmatinib xHCl
CAS:1029714-89-3
Capmatinib xHCl (INCB28060) is a potent, orally active, selective, and ATP competitive c-Met kinase inhibitor, …
Formula:
C23H18ClFN6O
Purity:
99.12% - 99.24%
Color and Shape:
Solid
Molecular weight:
448.89
Ref: TM-T8416
| 1mg | 43.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 77.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 180.00 € | ||
| 50mg | 271.00 € | ||
| 100mg | 406.00 € | ||
| 500mg | 917.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
