Tyrosine Kinase/Adaptors
Tyrosine kinase and adaptor inhibitors are compounds that target tyrosine kinases and their associated adaptor proteins, which play pivotal roles in cell signaling, growth, and differentiation. These inhibitors are essential tools in cancer research, as many tyrosine kinases are involved in the signaling pathways that drive tumor growth and metastasis. By inhibiting tyrosine kinases, these compounds can block critical signaling cascades, offering potential therapeutic strategies for various cancers and other diseases involving abnormal cell signaling. At CymitQuimica, we provide a comprehensive range of high-quality tyrosine kinase and adaptor inhibitors to support your research in oncology, molecular biology, and targeted therapy development.
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Subcategories of "Tyrosine Kinase/Adaptors"
ALK
CSF-1R
EGFR
Ephrin Receptor
FLT
Fibroblast Growth Factor Receptor (FGFR)
HER
Hck
IGF-1R
PDGFR
PYK2
Src
TAM Receptor
Tie-2
Trk receptor
Tyrosine Kinases
VEGFR
c-Fms
c-Kit
c-Met/HGFR
c-RET
Show 13 more subcategories
Products of "Tyrosine Kinase/Adaptors"
R1530
CAS:882531-87-5
R1530 is a multikinase inhibitor with antineoplastic and antiangiogenesis activities.
Formula:
C18H14ClFN4O
Purity:
97.96%
Color and Shape:
Solid
Molecular weight:
356.78
Ref: TM-TQ0317
| 1mg | 52.00 € | ||
| 2mg | 74.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 324.00 € | ||
| 50mg | 552.00 € | ||
| 100mg | 796.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ribociclib
CAS:1211441-98-3
Ribociclib (LEE011) is an orally available, and highly specific CDK4/6 inhibitor (IC50:10/39 nM).
Formula:
C23H30N8O
Purity:
100% - 99.96%
Color and Shape:
Solid
Molecular weight:
434.54
Ref: TM-T6199
| 2mg | 42.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 116.00 € | ||
| 100mg | 168.00 € | ||
| 500mg | 412.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
(S)-Sunvozertinib
CAS:2370013-49-1
(S)-Sunvozertinib (DZD9008) is a rationally designed selective, irreversible EGFR/HER2 inhibitor.
Formula:
C29H35ClFN7O3
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
584.08
Ref: TM-T9304
| 1mg | 62.00 € | ||
| 5mg | 134.00 € | ||
| 10mg | 207.00 € | ||
| 25mg | 415.00 € | ||
| 50mg | 612.00 € | ||
| 100mg | 878.00 € | ||
| 1mL*10mM (DMSO) | 169.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BI-4020
CAS:2664214-60-0
BI-4020 is a fourth-generation, orally active, and non-covalent inhibitor of EGFR tyrosine kinase.
Formula:
C30H38N8O2
Purity:
100.00% - 98.44%
Color and Shape:
Solid
Molecular weight:
542.68
Ref: TM-T10534
| 1mg | 164.00 € | ||
| 5mg | 383.00 € | ||
| 10mg | 547.00 € | ||
| 25mg | 817.00 € | ||
| 50mg | 1,089.00 € | ||
| 100mg | 1,455.00 € | ||
| 200mg | 1,985.00 € | ||
| 1mL*10mM (DMSO) | 455.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
WHI-P154
CAS:211555-04-3
WHI-P154 (Jak3 inhibitor ii) is a potent JAK3 inhibitor.
Formula:
C16H14BrN3O3
Purity:
98% - 99.6%
Color and Shape:
Solid
Molecular weight:
376.2
Ref: TM-T1985
| 2mg | 46.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 174.00 € | ||
| 50mg | 328.00 € | ||
| 100mg | 532.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Pyridone 6
CAS:457081-03-7
Pyridone 6, a selective JAK1/2/3 and Tyk2 inhibitor with IC50s: JAK1=15 nM, JAK2=1 nM, JAK3 …
Formula:
C18H16FN3O
Purity:
97.10% - 98.74%
Color and Shape:
Solid
Molecular weight:
309.34
Ref: TM-T3080
| 1mg | 81.00 € | ||
| 2mg | 105.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 218.00 € | ||
| 25mg | 441.00 € | ||
| 50mg | 648.00 € | ||
| 100mg | 918.00 € | ||
| 500mg | 1,838.00 € | ||
| 1mL*10mM (DMSO) | 176.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AG-1557 hydrochloride (189290-58-2(free base))
AG-1557 hydrochloride is an inhibitor of the epidermal growth factor receptor (EGFR) tyrosine kinase (pIC50: …
Formula:
C16H15ClIN3O2
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
443.66
Ref: TM-T4694
| 5mg | 35.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 149.00 € | ||
| 100mg | 260.00 € | ||
| 200mg | 381.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
SRI 31215 TFA
CAS:1832686-44-8
SRI 31215 TFA acts as a triplex inhibitor of matriptase, hepsin and HGFA and mimics …
Formula:
C27H34F3N5O3
Purity:
98.25% - 99.97%
Color and Shape:
Solid
Molecular weight:
533.6
Ref: TM-T5478
| 1mg | 42.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 254.00 € | ||
| 50mg | 381.00 € | ||
| 100mg | 542.00 € | ||
| 200mg | 733.00 € | ||
| 1mL*10mM (DMSO) | 99.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
NVP-BHG712 isomer
CAS:2245892-85-5
NVP-BHG712 isomer shows conserved non-bonded binding to EPHA2 and EPHB4.
Formula:
C26H20F3N7O
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
503.48
Ref: TM-T19487
| 1mg | 43.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 147.00 € | ||
| 25mg | 255.00 € | ||
| 50mg | 368.00 € | ||
| 100mg | 547.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Milciclib
CAS:802539-81-7
Milciclib (PHA-848125) is a potent CDK2 inhibitor with a 45 nM IC50, selective over CDK1/2/4/5/7. …
Formula:
C25H32N8O
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
460.57
Ref: TM-T6081
| 1mg | 91.00 € | ||
| 5mg | 188.00 € | ||
| 10mg | 307.00 € | ||
| 25mg | 519.00 € | ||
| 50mg | 748.00 € | ||
| 100mg | 1,025.00 € | ||
| 200mg | 807.00 € | ||
| 1mL*10mM (DMSO) | 188.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Avitinib maleate
CAS:1557268-88-8
Avitinib maleate is a pyrrolopyrimidine-based irreversible epidermal growth factor receptor (EGFR) inhibitor.
Formula:
C30H30FN7O6
Purity:
98% - 99.77%
Color and Shape:
Solid
Molecular weight:
603.61
Ref: TM-T3721
| 5mg | 72.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 205.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 557.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
RN486
CAS:1242156-23-5
RN486 is an effective and specific BTK inhibitor (IC50: 4 nM).
Formula:
C35H35FN6O3
Purity:
99.38%
Color and Shape:
Solid
Molecular weight:
606.69
Ref: TM-T1976
| 1mg | 83.00 € | ||
| 5mg | 101.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 325.00 € | ||
| 50mg | 510.00 € | ||
| 100mg | 769.00 € | ||
| 1mL*10mM (DMSO) | 139.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
SKLB4771
CAS:1370256-78-2
SKLB4771 (FLT3-IN-1) is a novel potent and selective Flt3 inhibitor.
Formula:
C25H27N7O3S2
Purity:
100% - 98.27%
Color and Shape:
Solid
Molecular weight:
537.66
Ref: TM-T2051
| 1mg | 66.00 € | ||
| 2mg | 96.00 € | ||
| 5mg | 129.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 386.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 817.00 € | ||
| 500mg | 1,661.00 € | ||
| 1mL*10mM (DMSO) | 156.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Daphnetin
CAS:486-35-1
Daphnetin (7,8-Dihydroxycoumarin), a natural coumarin derivative, is a protein kinase inhibitor with inhibitory for EGFR …
Formula:
C9H6O4
Purity:
98.33% - 99.82%
Color and Shape:
Solid
Molecular weight:
178.14
Ref: TM-T2851
| 10mg | 50.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | 239.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
H-89 dihydrochloride
CAS:130964-39-5
H-89 dihydrochloride (5-Isoquinolinesulfonamide) is a potent inhibitor of protein kinase A (PKA; IC50: 0.14 μM, …
Formula:
C20H20BrN3O2S·2HCl
Purity:
100% - 99.4%
Color and Shape:
Solid
Molecular weight:
519.28
Ref: TM-T6250
| 5mg | 39.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 105.00 € | ||
| 50mg | 198.00 € | ||
| 100mg | 339.00 € | ||
| 200mg | 503.00 € | ||
| 500mg | 796.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Spebrutinib
CAS:1202757-89-8
Spebrutinib (LMK-435) is an orally bioavailable, selective inhibitor of Bruton's agammaglobulinemia tyrosine kinase (BTK), with …
Formula:
C22H22FN5O3
Purity:
100% - 97.02%
Color and Shape:
Solid
Molecular weight:
423.44
Ref: TM-T2603
| 2mg | 41.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 122.00 € | ||
| 100mg | 194.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Alflutinib mesylate
CAS:2130958-55-1
Alflutinib mesylate (AST2818 mesylate) ,is an irreversible tyrosine kinase inhibitor that selectively inhibits EGFR mutations, …
Formula:
C29H35F3N8O5S
Purity:
97.94% - 99.81%
Color and Shape:
Solid
Molecular weight:
664.7
Ref: TM-T7175
| 1mg | 77.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 230.00 € | ||
| 25mg | 388.00 € | ||
| 50mg | 576.00 € | ||
| 100mg | 816.00 € | ||
| 500mg | 1,662.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
SU4984
CAS:186610-89-9
SU4984 is a cell-permeable, ATP-competitive and reversible inhibitor of the fibroblast growth factor receptor 1 …
Formula:
C20H19N3O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
333.38
Ref: TM-T9030
| 5mg | 38.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 113.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 302.00 € | ||
| 200mg | 435.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
7BIO
CAS:916440-85-2
7BIO triggers nonapoptotic death, blocks FLT3, DYRK1A/2, Aurora B/C kinases.
Formula:
C16H10BrN3O2
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
356.17
Ref: TM-T22012
| 5mg | 44.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 112.00 € | ||
| 50mg | 172.00 € | ||
| 100mg | 273.00 € | ||
| 200mg | 387.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
KRN-633
CAS:286370-15-8
KRN-633 is an effective VEGFR inhibitor. The IC50s of KRN-633(KRN633) for VEGFR1, VEGFR2, and VEGFR3 …
Formula:
C20H21ClN4O4
Purity:
99.22% - 99.65%
Color and Shape:
Solid
Molecular weight:
416.86
Ref: TM-T6137
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 302.00 € | ||
| 200mg | 430.00 € | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
