Tyrosine Kinase/Adaptors
Tyrosine kinase and adaptor inhibitors are compounds that target tyrosine kinases and their associated adaptor proteins, which play pivotal roles in cell signaling, growth, and differentiation. These inhibitors are essential tools in cancer research, as many tyrosine kinases are involved in the signaling pathways that drive tumor growth and metastasis. By inhibiting tyrosine kinases, these compounds can block critical signaling cascades, offering potential therapeutic strategies for various cancers and other diseases involving abnormal cell signaling. At CymitQuimica, we provide a comprehensive range of high-quality tyrosine kinase and adaptor inhibitors to support your research in oncology, molecular biology, and targeted therapy development.
Read more
Subcategories of "Tyrosine Kinase/Adaptors"
ALK
CSF-1R
EGFR
Ephrin Receptor
FLT
Fibroblast Growth Factor Receptor (FGFR)
HER
Hck
IGF-1R
PDGFR
PYK2
Src
TAM Receptor
Tie-2
Trk receptor
Tyrosine Kinases
VEGFR
c-Fms
c-Kit
c-Met/HGFR
c-RET
Show 13 more subcategories
Products of "Tyrosine Kinase/Adaptors"
OD36 hydrochloride
CAS:2387510-88-3
OD36 hydrochloride (OD-36 hydrochloride) is a potent RIPK2 inhibitor with an IC50 of 5.3 nM.OD36 …
Formula:
C16H16Cl2N4O2
Purity:
99.85%
Color and Shape:
Liquid
Molecular weight:
367.23
Ref: TM-T61424
| 25mg | 1,197.00 € | ||
| 50mg | 1,561.00 € | ||
| 100mg | 2,320.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
GTP-14564
CAS:34823-86-4
GTP-14564 is a novel tyrosine kinase inhibitor that also inhibits wt-FLT3 and ITD-FLT3.
Formula:
C15H10N2O
Purity:
99.69%
Color and Shape:
Liquid
Molecular weight:
234.25
Ref: TM-T71857
| 1mg | 46.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 340.00 € | ||
| 50mg | 540.00 € | ||
| 100mg | 777.00 € | ||
| 500mg | 1,579.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
IACS-9439
CAS:2231259-57-5
IACS-9439 is a potent, selective, and orally active inhibitor of CSF1R, exhibiting a K(i) of …
Formula:
C23H26ClN7O3S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
516.02
Ref: TM-T69759
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Larotinib
CAS:1438072-11-7
Larotinib is an orally active, potent, and broad-spectrum tyrosine kinase inhibitor (TKI) with an IC50 …
Formula:
C24H26ClFN4O4
Purity:
98.45%
Color and Shape:
Liquid
Molecular weight:
488.94
Ref: TM-T73334
| 1mg | 80.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 253.00 € | ||
| 25mg | 430.00 € | ||
| 50mg | 615.00 € | ||
| 100mg | 861.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
YK-2-69
CAS:2619846-89-6
YK-2-69 selectively blocks DYRK2 at Lys-231 and Lys-234, outperforming enzalutamide in prostate cancer treatment.
Formula:
C25H27FN8OS
Purity:
98.45% - 99.57%
Color and Shape:
Liquid
Molecular weight:
506.6
Ref: TM-T69564
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Sotuletinib dihydrochloride
CAS:2222138-40-9
Sotuletinib (BLZ945) dihydrochloride is an orally administered, blood-brain barrier-permeable inhibitor specifically targeting CSF1-R with an …
Formula:
C20H24Cl2N4O3S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
471.4
Ref: TM-T78603
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
c-Fms-IN-8
CAS:1255303-58-2
c-Fms-IN-8 is a colony-stimulating factor-1 receptor (CSF-1R, c-FMS) Type II inhibitor (IC50: 9.1 nM). It …
Formula:
C27H30N2O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
462.54
Ref: TM-T10647
| 25mg | 1,299.00 € | ||
| 50mg | 1,687.00 € | ||
| 100mg | 2,367.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Protein kinase inhibitor 5
CAS:2278204-94-5
Protein kinase inhibitor 5 is a potent inhibitor of TRK-A, demonstrating an IC50 of 1.8 …
Formula:
C29H31F2N7O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
531.6
Ref: TM-T79125
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
TRK-IN-23
CAS:2924344-29-4
TRK-IN-23 (compound 24b) is a potent, orally active inhibitor of TRK with IC50s of 0.5 …
Formula:
C20H17FN4O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
364.37
Ref: TM-T78968
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
H-9 dihydrochloride
CAS:116700-36-8
H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.
Formula:
C11H15Cl2N3O2S
Purity:
96.57%
Color and Shape:
Solid
Molecular weight:
324.23
Ref: TM-T22833
| 1mg | 35.00 € | ||
| 5mg | 71.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 152.00 € | ||
| 50mg | 219.00 € | ||
| 100mg | 324.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
SI-2 hydrochloride
CAS:1992052-49-9
SI-2 hydrochloride, an SRC-3 inhibitor, induces breast cancer cell death (IC50: 3-20 nM) with good …
Formula:
C15H16ClN5
Purity:
98.18%
Color and Shape:
Solid
Molecular weight:
301.77
Ref: TM-T12906
| 5mg | 35.00 € | ||
| 10mg | 46.00 € | ||
| 25mg | 63.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Tyrphostin A25
CAS:118409-58-8
Tyrphostin A25 (Tyrphostin AG 82) is a specific EGFR tyrosine kinase inhibitor and GPR35 agonist …
Formula:
C10H6N2O3
Purity:
98.76%
Color and Shape:
Yellow Green Powder /Off-White Solid
Molecular weight:
202.17
Ref: TM-T21622
| 2mg | 38.00 € | ||
| 5mg | 55.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 117.00 € | ||
| 50mg | 173.00 € | ||
| 100mg | 246.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
EGFR-IN-73
CAS:2857033-34-0
EGFR-IN-73 (Compound 3f) effectively inhibits the prevalent EGFR mutation, EGFR Del19, exhibiting an IC50 value …
Formula:
C19H17ClFN3O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
405.81
Ref: TM-T73165
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Glesatinib
CAS:936694-12-1
Glesatinib is an orally active and potent dual inhibitor of MET/SMO.
Formula:
C31H27F2N5O3S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
619.7
Ref: TM-T15384
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Epertinib
CAS:908305-13-5
Epertinib is a reversible and selective tyrosine kinase inhibitor of EGFR, HER2, and HER4 (IC50s: …
Formula:
C30H27ClFN5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
560.02
Ref: TM-T11213L
| 25mg | 1,262.00 € | ||
| 50mg | 1,644.00 € | ||
| 100mg | 2,336.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
VEGFR-2-IN-6
CAS:444731-47-9
VEGFR-2-IN-6 (WO 02/059110, example 64) is a potent inhibitor of VEGFR2, a crucial receptor involved …
Formula:
C20H21N7O2S
Purity:
99.01%
Color and Shape:
Liquid
Molecular weight:
423.49
Ref: TM-T37078
| 1mg | 95.00 € | ||
| 5mg | 222.00 € | ||
| 10mg | 346.00 € | ||
| 25mg | To inquire | ||
| 1mL*10mM (DMSO) | 244.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
EGFR-IN-82
CAS:2568086-81-5
EGFR-IN-82 (Compound 8a) is a potent, orally active inhibitor of EGFR, exhibiting IC50 values of …
Formula:
C32H41BrN9O2P
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
694.6
Ref: TM-T78788
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
FN-1501
CAS:1429515-59-2
FN-1501 is a potent FLT3 and CDK inhibitor (IC50s: 2.47, 0.85, 1.96, and 0.28 nM …
Formula:
C22H25N9O
Purity:
96.35%
Color and Shape:
Solid
Molecular weight:
431.49
Ref: TM-T15335
| 1mg | 90.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 300.00 € | ||
| 25mg | 545.00 € | ||
| 50mg | 832.00 € | ||
| 100mg | 1,133.00 € | ||
| 1mL*10mM (DMSO) | 214.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
AC710 Mesylate
CAS:1351522-05-8
AC710 Mesylate is a potent PDGFR inhibitor (Kds: 0.6, 1.57, 1, 1.3, 1.0 nM for …
Formula:
C32H46N6O7S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
658.81
Ref: TM-T10228
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
DDR-TRK-1
CAS:1934246-19-1
DDR-TRK-1 is a selective discoid domain receptor 1 (DDR1) inhibitor with IC50 value of 9.4 …
Formula:
C26H23F3N6O
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
492.5
Ref: TM-T10984
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 551.00 € | ||
| 50mg | 771.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 305.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
