Tyrosine Kinase/Adaptors
Tyrosine kinase and adaptor inhibitors are compounds that target tyrosine kinases and their associated adaptor proteins, which play pivotal roles in cell signaling, growth, and differentiation. These inhibitors are essential tools in cancer research, as many tyrosine kinases are involved in the signaling pathways that drive tumor growth and metastasis. By inhibiting tyrosine kinases, these compounds can block critical signaling cascades, offering potential therapeutic strategies for various cancers and other diseases involving abnormal cell signaling. At CymitQuimica, we provide a comprehensive range of high-quality tyrosine kinase and adaptor inhibitors to support your research in oncology, molecular biology, and targeted therapy development.
Read more
Subcategories of "Tyrosine Kinase/Adaptors"
ALK
CSF-1R
EGFR
Ephrin Receptor
FLT
Fibroblast Growth Factor Receptor (FGFR)
HER
Hck
IGF-1R
PDGFR
PYK2
Src
TAM Receptor
Tie-2
Trk receptor
Tyrosine Kinases
VEGFR
c-Fms
c-Kit
c-Met/HGFR
c-RET
Show 13 more subcategories
Products of "Tyrosine Kinase/Adaptors"
DBPR112
CAS:1226549-49-0
DBPR112: oral furanopyrimidine EGFR inhibitor; IC50: 15 nM (EGFRWT), 48 nM (L858R/T790M); blocks ATP site, …
Formula:
C32H31N5O3
Purity:
98.29%
Color and Shape:
Solid
Molecular weight:
533.62
Ref: TM-T10965
| 1mg | 75.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 300.00 € | ||
| 25mg | 484.00 € | ||
| 50mg | 645.00 € | ||
| 100mg | 888.00 € | ||
| 1mL*10mM (DMSO) | 187.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Chiauranib
CAS:1256349-48-0
Chiauranib, a potent anticancer agent, inhibits angiogenesis kinases (VEGFR1-3, PDGFRα, c-Kit), Aurora B, and CSF1R …
Formula:
C27H21N3O3
Purity:
96.25%
Color and Shape:
Solid
Molecular weight:
435.47
Ref: TM-T35570
| 1mg | 89.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 300.00 € | ||
| 25mg | 508.00 € | ||
| 50mg | 732.00 € | ||
| 100mg | 1,003.00 € | ||
| 1mL*10mM (DMSO) | 213.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
SDZ281-977
CAS:150779-71-8
SDZ 281-977 is a derivative of Lavendustin A which is the EGF receptor tyrosine kinase …
Formula:
C18H20O5
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
316.35
Ref: TM-T16866
| 1mg | 97.00 € | ||
| 5mg | 231.00 € | ||
| 10mg | 369.00 € | ||
| 25mg | 739.00 € | ||
| 50mg | 1,146.00 € | ||
| 1mL*10mM (DMSO) | 257.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
TRK II-IN-1
CAS:2904690-41-9
TRK II-IN-1: potent type II TRK inhibitor; IC50s: TRKA (3.3 nM), TRKB (6.4 nM), TRKC …
Formula:
C29H31F3N8O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
564.6
Ref: TM-T73033
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
ACP-5862
CAS:2230757-47-6
ACP-5862, active metabolite of Acalabrutinib, is a BTK inhibitor with an IC50 of 5.0 nM.
Formula:
C26H23N7O3
Color and Shape:
Solid
Molecular weight:
481.51
Ref: TM-T10240
| 25mg | 1,410.00 € | ||
| 50mg | 1,854.00 € | ||
| 100mg | 2,340.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Nuvenzepine
CAS:96487-37-5
Nuvenzepine is an antagonist of mAChR. It has the potential for gastrospasm treatment.
Formula:
C19H20N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
336.39
Ref: TM-T16362
| 25mg | 1,410.00 € | ||
| 50mg | 1,875.00 € | ||
| 100mg | 2,317.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
TG 100801 Hydrochloride
CAS:1018069-81-2
TG 100801: prodrug for macular degeneration. TG 100572: inhibits kinases (VEGFRs, FGFRs, PDGFRβ, Src family), …
Formula:
C33H31Cl2N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
616.54
Ref: TM-T13157L
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
CP-547632 hydrochloride
CAS:252003-71-7
CP-547632 hydrochloride: oral VEGFR-2/FGF inhibitor (IC50: 11/9 nM), well-tolerated, antitumor.
Formula:
C20H25BrClF2N5O3S
Color and Shape:
Solid
Molecular weight:
568.86
Ref: TM-T10870
| 2mg | 51.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
SB-633825
CAS:956613-01-7
SB-633825 can inhibit cancer cell growth and angiogenesis.
Formula:
C28H25N3O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
483.58
Ref: TM-T16853
| 2mg | 182.00 € | ||
| 5mg | 368.00 € | ||
| 25mg | 1,113.00 € | ||
| 50mg | 1,502.00 € | ||
| 100mg | 2,367.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
PDGFRα kinase inhibitor 1
CAS:2209053-93-8
PDGFRα kinase inhibitor 1 is a type II PDGFRα kinase inhibitor that inhibits both PDGFRα …
Formula:
C34H34N8O2
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
586.69
Ref: TM-T12396
| 2mg | 372.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
TrkA-IN-1
CAS:1680179-43-4
TrkA-IN-1 is a potent and selective inhibitor of Tropomyosin-related kinase A (TrkA) (IC50: 99 nM …
Formula:
C25H20N4O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
392.45
Ref: TM-T13208
| 25mg | 1,021.00 € | ||
| 50mg | 1,354.00 € | ||
| 100mg | 2,055.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
CLK-IN-T3
CAS:2109805-56-1
CLK-IN-T3 is an inhibitor of CLK1, CLK2, and CLK3 with IC50s of 0.67, 15, and …
Formula:
C28H30N6O2
Purity:
98.37%
Color and Shape:
Solid
Molecular weight:
482.58
Ref: TM-T14980
| 1mg | 58.00 € | ||
| 2mg | 82.00 € | ||
| 5mg | 123.00 € | ||
| 10mg | 205.00 € | ||
| 25mg | 435.00 € | ||
| 50mg | 640.00 € | ||
| 100mg | 909.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
TL02-59 dihydrochloride
CAS:2415263-06-6
TL02-59 dihydrochloride is an orally active inhibitor of Src-family kinase Fgr (IC50: 0.03 nM).
Formula:
C32H36Cl2F3N5O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
682.56
Ref: TM-T13186L
| 10mg | 734.00 € | ||
| 50mg | 3,073.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
SU16f
CAS:251356-45-3
SU16f, a 3-substituted indolin-2-one, is a selective PDGFRβ inhibitor; IC50: 10 nM (PDGFRβ), 140 nM …
Formula:
C24H22N2O3
Purity:
98.38%
Color and Shape:
Solid
Molecular weight:
386.44
Ref: TM-T16947
| 1mg | 46.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 199.00 € | ||
| 50mg | 296.00 € | ||
| 100mg | 427.00 € | ||
| 1mL*10mM (DMSO) | 97.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
BKI-1369
CAS:1951431-22-3
BKI-1369 is a bumped kinase inhibitor. BKI-1369 increases hERG-inhibitory activity (IC50:1.52 μM).
Formula:
C23H27N7O
Color and Shape:
Solid
Molecular weight:
417.51
Ref: TM-T10556
| 5mg | 444.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,854.00 € | ||
| 100mg | 2,340.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
RO9021
CAS:1446790-62-0
RO9021 is an orally bioavailable, novel ATP-competitive SYK inhibitor (average IC50: 5.6 nM).
Formula:
C18H25N7O
Purity:
97.19%
Color and Shape:
Solid
Molecular weight:
355.44
Ref: TM-T16776
| 1mg | 87.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 282.00 € | ||
| 25mg | 468.00 € | ||
| 50mg | 681.00 € | ||
| 100mg | 927.00 € | ||
| 200mg | 729.00 € | ||
| 500mg | 1,813.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Tavilermide
CAS:263251-78-1
Tavilermide (MIM-D3) is a selective TrkA agonist, a cyclic mimetic, which can be used to …
Formula:
C24H32N6O11
Purity:
98.98%
Color and Shape:
Solid
Molecular weight:
580.54
Ref: TM-T17000
| 5mg | 419.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,865.00 € | ||
| 100mg | 2,367.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
DUN73423
CAS:2414373-42-3
DUN73423 (RET-IN-21) is a potent tyrosine kinase (RET) inhibitor with antitumour activity for the study …
Formula:
C19H16N6O
Color and Shape:
Liquid
Molecular weight:
344.37
Ref: TM-T69644
| 1mg | 52.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 299.00 € | ||
| 50mg | 445.00 € | ||
| 100mg | 638.00 € | ||
| 500mg | 1,290.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Cloperastine fendizoate
CAS:85187-37-7
Cloperastine fendizoate (Hustazol) inhibits the hERG K+ currents in a concentration-dependent manner (IC50: 27 nM).
Formula:
C40H38ClNO5
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
648.19
Ref: TM-T13619
| 500mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Antiproliferative agent-34
CAS:2910858-34-1
Antiproliferative Agent-34 (Compound A14), a multitarget kinase inhibitor, demonstrates IC50 values of 177 nM for …
Formula:
C27H27N7O5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
529.55
Ref: TM-T79368
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
