VEGFR
VEGFR (Vascular Endothelial Growth Factor Receptor) inhibitors are compounds that block the signaling of VEGFR, a key receptor in the VEGF pathway, which is crucial for angiogenesis. VEGFR inhibitors prevent the formation of new blood vessels that supply nutrients and oxygen to tumors, thereby inhibiting tumor growth. These inhibitors are widely used in cancer therapy and research to study the mechanisms of angiogenesis and develop anti-cancer treatments. At CymitQuimica, we provide a comprehensive range of high-quality VEGFR inhibitors to support your research in oncology, vascular biology, and angiogenesis.
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AST 487
CAS:630124-46-8
AST 487 (NVP-AST 487) is a RET kinase inhibitor, inhibiting RET autophosphorylation and activation of …
Formula:
C26H30F3N7O2
Purity:
98.17% - 99.56%
Color and Shape:
Solid
Molecular weight:
529.56
Ref: TM-T4053
| 1mg | 36.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 349.00 € | ||
| 100mg | 522.00 € | ||
| 500mg | 1,133.00 € | ||
| 1mL*10mM (DMSO) | 91.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MAZ51
CAS:163655-37-6
MAZ51 is a VEGFR-3 (Flt-4) tyrosine kinase inhibitor.
Formula:
C21H18N2O
Purity:
98.53%
Color and Shape:
Solid
Molecular weight:
314.38
Ref: TM-T8496
| 1mg | 40.00 € | ||
| 2mg | 56.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 242.00 € | ||
| 50mg | 403.00 € | ||
| 100mg | 599.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Regorafenib
CAS:755037-03-7
Regorafenib (BAY 73-4506) is a multi-targeted receptor tyrosine kinase inhibitor that inhibits RET, C-RAF, VEGFR2, …
Formula:
C21H15ClF4N4O3
Purity:
98% - 99.95%
Color and Shape:
Solid
Molecular weight:
482.82
Ref: TM-T1792
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 142.00 € | ||
| 200mg | 181.00 € | ||
| 500mg | 304.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
JNJ-38158471
CAS:951151-97-6
JNJ-38158471 (CS-2660), a highly selective, orally available, well tolerated VEGFR2 inhibitor, inhibits closely related tyrosine …
Formula:
C15H17ClN6O3
Purity:
97.08%
Color and Shape:
Solid
Molecular weight:
364.79
Ref: TM-T22349
| 1mg | 51.00 € | ||
| 2mg | 72.00 € | ||
| 5mg | 102.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 364.00 € | ||
| 100mg | 490.00 € | ||
| 200mg | 673.00 € | ||
| 1mL*10mM (DMSO) | 109.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
VEGFR-2-IN-5
CAS:1430089-64-7
VEGFR-2-IN-5 (UNC0064-12), multikinase inhibitor and has a -NH2 terminal linker for further synthesis.
Formula:
C19H24N8
Purity:
98.13%
Color and Shape:
Solid
Molecular weight:
364.45
Ref: TM-T2056
| 1mg | 94.00 € | ||
| 5mg | 230.00 € | ||
| 10mg | 345.00 € | ||
| 25mg | 578.00 € | ||
| 50mg | 827.00 € | ||
| 100mg | 1,112.00 € | ||
| 1mL*10mM (DMSO) | 235.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BMS-794833
CAS:1174046-72-0
BMS-794833 is a potent ATP competitive inhibitor of Met/VEGFR2; a prodrug of BMS-817378.
Formula:
C23H15ClF2N4O3
Purity:
98% - 99.69%
Color and Shape:
Solid
Molecular weight:
468.84
Ref: TM-T2419
| 1mg | 41.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 152.00 € | ||
| 25mg | 296.00 € | ||
| 50mg | 533.00 € | ||
| 100mg | 754.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Gandotinib
CAS:1229236-86-5
LY2784544(Gandotinib (LY2784544)) is a potent JAK2 inhibitor (IC50: 3 nM), effective in JAK2V617F(Ki: 0.245 nM).
Formula:
C23H25ClFN7O
Purity:
99.16% - 99.86%
Color and Shape:
Solid
Molecular weight:
469.94
Ref: TM-T2638
| 5mg | 51.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 290.00 € | ||
| 100mg | 460.00 € | ||
| 500mg | 1,012.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ZD-4190
CAS:413599-62-9
ZD-4190 blocks VEGFR2 and EGFR, aiding cancer treatment.
Formula:
C19H16BrFN6O2
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
459.27
Ref: TM-T5475
| 1mg | 82.00 € | ||
| 5mg | 177.00 € | ||
| 10mg | 266.00 € | ||
| 25mg | 422.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € | ||
| 1mL*10mM (DMSO) | 179.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
SKLB1002
CAS:1225451-84-2
SKLB1002 is a potent and ATP-competitive VEGFR2 inhibitor with IC50 of 32 nM.
Formula:
C13H12N4O2S2
Purity:
100% - 99.15%
Color and Shape:
Solid
Molecular weight:
320.39
Ref: TM-T2421
| 1mg | 44.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 81.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 201.00 € | ||
| 50mg | 340.00 € | ||
| 100mg | 551.00 € | ||
| 500mg | 1,187.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Lenvatinib mesylate
CAS:857890-39-2
Lenvatinib mesylate (E7080 (mesylate)) is an oral and multi-targeted inhibitor of VEGFR1-3, FGFR1-4, PDGFR, KIT, …
Formula:
C22H23ClN4O7S
Purity:
99.03% - 99.79%
Color and Shape:
Solid
Molecular weight:
522.96
Ref: TM-T8541
| 10mg | 40.00 € | ||
| 25mg | 59.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 109.00 € | ||
| 200mg | 162.00 € | ||
| 500mg | 263.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PF 477736
CAS:952021-60-2
PF 477736 (PF-736,PF-00477736) is a specifc, effective and ATP-competitive Chk1 inhibitor (Ki: 0.49 nM ) …
Formula:
C22H25N7O2
Purity:
98% - 98.34%
Color and Shape:
Solid
Molecular weight:
419.48
Ref: TM-T6028
| 2mg | 49.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
OSI-930
CAS:728033-96-3
OSI-930 is an oral c-Kit/VEGFR-2 inhibitor targeting tumor growth and angiogenesis.
Formula:
C22H16F3N3O2S
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
443.44
Ref: TM-T2624
| 1mg | 51.00 € | ||
| 5mg | 100.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 259.00 € | ||
| 50mg | 419.00 € | ||
| 100mg | 605.00 € | ||
| 1mL*10mM (DMSO) | 100.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Regorafenib monohydrate
CAS:1019206-88-2
Regorafenib Monohydrate is a novel oral multikinase inhibitor with IC50 values of 13, 4.2, 46, …
Formula:
C21H17ClF4N4O4
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
500.83
Ref: TM-T1792L
| 5mg | 36.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 138.00 € | ||
| 200mg | 204.00 € | ||
| 500mg | 348.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
VEGFR2-IN-2
CAS:737818-56-3
VEGFR2-IN-2 has anti-inflammatory and analgesic activities.
Formula:
C15H11BrN2O
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
315.16
Ref: TM-T9724
| 1mg | 37.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 107.00 € | ||
| 25mg | 198.00 € | ||
| 50mg | 317.00 € | ||
| 100mg | 453.00 € | ||
| 200mg | 627.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ripretinib
CAS:1442472-39-0
Ripretinib (DCC-2618) is an orally bioavailable inhibitor of KIT and PDGFRA.
Formula:
C24H21BrFN5O2
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
510.36
Ref: TM-T8482
| 1mg | 391.00 € | ||
| 2mg | 585.00 € | ||
| 5mg | 930.00 € | ||
| 10mg | 1,274.00 € | ||
| 25mg | 1,722.00 € | ||
| 50mg | 2,401.00 € | ||
| 100mg | 3,353.00 € | ||
| 500mg | 5,402.00 € | ||
| 1mL*10mM (DMSO) | 427.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
XL092
CAS:2367004-54-2
XL092 (JUN04542) is an Axl Mer cMet KDR inhibitor for the treatment of Axl and …
Formula:
C29H25FN4O5
Purity:
99.51%
Color and Shape:
Solid
Molecular weight:
528.53
Ref: TM-T9052
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 132.00 € | ||
| 50mg | 208.00 € | ||
| 100mg | 346.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TAK-659 hydrochloride
CAS:1952251-28-3
TAK-659 hydrochloride (TAK-659) is a potent and selective inhibitor of spleen tyrosine kinase (SYK) with …
Formula:
C17H22ClFN6O
Purity:
99.28% - 99.63%
Color and Shape:
Solid
Molecular weight:
380.85
Ref: TM-T4209
| 1mg | 39.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 500.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
CP-673451
CAS:343787-29-1
CP-673451 is a specific inhibitor of PDGFRα/β (IC50: 10/1 nM) with antiangiogenic and antitumor activity …
Formula:
C24H27N5O2
Purity:
99.88% - 99.93%
Color and Shape:
Solid
Molecular weight:
417.5
Ref: TM-T6091
| 1mg | 52.00 € | ||
| 2mg | 65.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 346.00 € | ||
| 50mg | 529.00 € | ||
| 100mg | 761.00 € | ||
| 500mg | 1,576.00 € | ||
| 1mL*10mM (DMSO) | 114.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Sakuranetin
CAS:2957-21-3
Sakuranetin, a flavanone phytoalexin from ultraviolet-irradiated rice leaves, it has antifungal, antimutagenic, anti-inflammatory and antioxidant …
Formula:
C16H14O5
Purity:
99% - 99.65%
Color and Shape:
Solid
Molecular weight:
286.28
Ref: TM-TN1126
| 1mg | 47.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 321.00 € | ||
| 100mg | 462.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
(Z)-Guggulsterone
CAS:39025-23-5
(Z)-Guggulsterone triggers apoptosis in prostate cancer cells and blocks angiogenesis by inhibiting VEGF pathways.
Formula:
C21H28O2
Purity:
98.47% - 99.72%
Color and Shape:
Solid
Molecular weight:
312.45
Ref: TM-T17280
| 5mg | 88.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 243.00 € | ||
| 50mg | 365.00 € | ||
| 100mg | 548.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
