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Histamine Receptor

Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.

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products per page. 203 products on this category.

BrandProduct dataPurityPrice rangeEstimated delivery
Targetmol logo
Cetirizine Impurity B dihydrochloride
REF: TM-T9084CAS: 1000690-91-4 		99.24%35.00 €~272.00 €Tue 10 Dec 24
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Hydroxyzine dihydrochloride
REF: TM-T2200CAS: 2192-20-3 		99.79% - 99.79%34.00 €~51.00 €Tue 10 Dec 24
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OXOMEMAZINE
REF: TM-T9353CAS: 3689-50-7 		99.49%To inquireTue 10 Dec 24
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Ranitidine
REF: TM-T3610CAS: 66357-35-5 		99.1%41.00 €~362.00 €Tue 10 Dec 24
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Bepotastine
REF: TM-T7893CAS: 125602-71-3 		99.96%45.00 €~917.00 €Tue 10 Dec 24
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Ciproxifan
REF: TM-T6164CAS: 184025-18-1 		98.00%43.00 €~393.00 €Tue 07 Jan 25
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Lodoxamide tromethamine
REF: TM-T15772CAS: 63610-09-3 		99.58%46.00 €~273.00 €Tue 07 Jan 25
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PF-03654764
REF: TM-T61213CAS: 935840-35-0 		100%305.00 €~2,009.00 €Tue 21 Jan 25
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CP-66948
REF: TM-T15005CAS: 101189-47-3 		99.14%654.00 €~1,672.00 €Tue 21 Jan 25
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PF-03654746
REF: TM-T16476CAS: 935840-31-6 		98.83% - 99.1%236.00 €~3,693.00 €Tue 21 Jan 25
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Bamirastine
REF: TM-T13566CAS: 215529-47-8 		96.68%651.00 €~1,678.00 €Tue 21 Jan 25
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H3 receptor-MO-1
REF: TM-T10499CAS: 1240914-03-7 		99.11%651.00 €~1,682.00 €Tue 21 Jan 25
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Rocastine
REF: TM-T16778CAS: 91833-49-7 		98.26%650.00 €~1,671.00 €Tue 21 Jan 25
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PF-03654746 Tosylate
REF: TM-T12416CAS: 1039399-17-1 		98%276.00 €~1,668.00 €Tue 21 Jan 25
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KP136
REF: TM-T15666CAS: 76239-32-2 		98.16% - 99.86%275.00 €~2,331.00 €Tue 21 Jan 25
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Iodophenpropit dihydrobromide
REF: TM-T15590CAS: 145196-87-8 		98%279.00 €~2,329.00 €Tue 21 Jan 25
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Immethridine dihydrobromide
REF: TM-T22864CAS: 699020-93-4 		97.49% - 98.16%63.00 €~2,497.00 €Tue 21 Jan 25
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(R)-(-)-α-Methylhistamine dihydrobromide
REF: TM-T12630CAS: 868698-49-1 		98%907.00 €~2,337.00 €Tue 21 Jan 25
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SUN 1334H
REF: TM-T13040CAS: 607736-84-5 		98%To inquireTue 21 Jan 25
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Toreforant
REF: TM-T17118CAS: 952494-46-1 		98%1,549.00 €~2,609.00 €Tue 21 Jan 25
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Cetirizine Impurity B dihydrochloride
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Cetirizine Impurity B dihydrochloride

CAS:1000690-91-4
Cetirizine Impurity B dihydrochloride is a Cetirizine antihistamine byproduct with anti-allergic properties.
Formula:
C19H23Cl3N2O2
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
417.76

Ref: TM-T9084

10mg35.00 €
25mg54.00 €
50mg85.00 €
100mg120.00 €
1mL*10mM (DMSO)40.00 €
Estimated delivery in United States, on Tuesday 10 Dec 2024
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Hydroxyzine dihydrochloride
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Hydroxyzine dihydrochloride

CAS:2192-20-3
Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.
Formula:
C21H27ClN2O2·2HCl
Purity:
99.79% - 99.79%
Color and Shape:
Oil Powder
Molecular weight:
447.83

Ref: TM-T2200

1g51.00 €
200mg34.00 €
500mg41.00 €
1mL*10mM (DMSO)45.00 €
Estimated delivery in United States, on Tuesday 10 Dec 2024
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OXOMEMAZINE
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OXOMEMAZINE

CAS:3689-50-7
Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in …
Formula:
C18H22N2O2S
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
330.44

Ref: TM-T9353

10mg35.00 €
25mgTo inquire
50mgTo inquire
1mL*10mM (DMSO)45.00 €
Estimated delivery in United States, on Tuesday 10 Dec 2024
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Ranitidine
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Ranitidine

CAS:66357-35-5
Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion …
Formula:
C13H22N4O3S
Purity:
99.1%
Color and Shape:
Solid Solid
Molecular weight:
314.4

Ref: TM-T3610

5mg41.00 €
10mg49.00 €
25mg89.00 €
50mg105.00 €
100mg124.00 €
200mg217.00 €
500mg362.00 €
1mL*10mM (DMSO)51.00 €
Estimated delivery in United States, on Tuesday 10 Dec 2024
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Bepotastine
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Bepotastine

CAS:125602-71-3
Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.
Formula:
C21H25ClN2O3
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
388.89

Ref: TM-T7893

2mg45.00 €
5mg66.00 €
10mg94.00 €
25mg167.00 €
50mg269.00 €
100mg402.00 €
200mg602.00 €
500mg917.00 €
1mL*10mM (DMSO)98.00 €
Estimated delivery in United States, on Tuesday 10 Dec 2024
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Ciproxifan
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Ciproxifan

CAS:184025-18-1
Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).
Formula:
C16H18N2O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
270.33

Ref: TM-T6164

1mg43.00 €
2mg54.00 €
5mg80.00 €
10mg109.00 €
25mg220.00 €
50mg393.00 €
Estimated delivery in United States, on Tuesday 7 Jan 2025
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Lodoxamide tromethamine
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Lodoxamide tromethamine

CAS:63610-09-3
Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in …
Formula:
C19H28ClN5O12
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
553.91

Ref: TM-T15772

5mg46.00 €
10mg59.00 €
25mg93.00 €
50mg109.00 €
100mg183.00 €
200mg273.00 €
1mL*10mM (DMSO)53.00 €
Estimated delivery in United States, on Tuesday 7 Jan 2025
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PF-03654764
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PF-03654764

CAS:935840-35-0
PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with …
Formula:
C20H28F2N2O
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
350.45

Ref: TM-T61213

1mg305.00 €
5mg736.00 €
25mg1,483.00 €
50mg2,009.00 €
Estimated delivery in United States, on Tuesday 21 Jan 2025
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CP-66948
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CP-66948

CAS:101189-47-3
CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion …
Formula:
C13H20N6S
Purity:
99.14%
Color and Shape:
Solid
Molecular weight:
292.4

Ref: TM-T15005

1mg654.00 €
5mg1,672.00 €
Estimated delivery in United States, on Tuesday 21 Jan 2025
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PF-03654746
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PF-03654746

CAS:935840-31-6
PF-03654746: selective H3 antagonist, boosts cognition in Alzheimer's, may treat allergic rhinitis.
Formula:
C18H24F2N2O
Purity:
98.83% - 99.1%
Color and Shape:
Solid
Molecular weight:
322.39

Ref: TM-T16476

1mg236.00 €
5mg590.00 €
10mg822.00 €
25mg1,262.00 €
50mg1,641.00 €
100mg2,470.00 €
Estimated delivery in United States, on Tuesday 21 Jan 2025
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Bamirastine
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Bamirastine

CAS:215529-47-8
Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value …
Formula:
C31H37N5O3
Purity:
96.68%
Color and Shape:
Solid
Molecular weight:
527.66

Ref: TM-T13566

1mg651.00 €
5mg1,678.00 €
Estimated delivery in United States, on Tuesday 21 Jan 2025
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discount label
H3 receptor-MO-1
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H3 receptor-MO-1

CAS:1240914-03-7
H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can …
Formula:
C20H27N3O2
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
341.45

Ref: TM-T10499

1mg651.00 €
5mg1,682.00 €
Estimated delivery in United States, on Tuesday 21 Jan 2025
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Rocastine
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Rocastine

CAS:91833-49-7
Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.
Formula:
C13H19N3OS
Purity:
98.26%
Color and Shape:
Solid
Molecular weight:
265.37

Ref: TM-T16778

1mg650.00 €
Estimated delivery in United States, on Tuesday 21 Jan 2025
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PF-03654746 Tosylate
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PF-03654746 Tosylate

CAS:1039399-17-1
PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
Formula:
C25H32F2N2O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
494.6

Ref: TM-T12416

25mg854.00 €
50mg1,096.00 €
100mg1,668.00 €
Estimated delivery in United States, on Tuesday 21 Jan 2025
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KP136
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KP136

CAS:76239-32-2
KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 …
Formula:
C16H18N4O3
Purity:
98.16% - 99.86%
Color and Shape:
Solid
Molecular weight:
314.34

Ref: TM-T15666

1mg275.00 €
5mg676.00 €
10mg924.00 €
25mg1,410.00 €
50mg1,847.00 €
100mg2,331.00 €
Estimated delivery in United States, on Tuesday 21 Jan 2025
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Iodophenpropit dihydrobromide
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Iodophenpropit dihydrobromide

CAS:145196-87-8
Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).
Formula:
C15H20BrIN4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
495.22

Ref: TM-T15590

5mg279.00 €
10mg418.00 €
Estimated delivery in United States, on Tuesday 21 Jan 2025
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Immethridine dihydrobromide
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Immethridine dihydrobromide

CAS:699020-93-4
Immethridine dihydrobromide is a histamine H3 receptor agonist.
Formula:
C9H11Br2N3
Purity:
97.49% - 98.16%
Color and Shape:
Solid
Molecular weight:
321.01

Ref: TM-T22864

1mg63.00 €
5mg183.00 €
10mg245.00 €
25mg549.00 €
50mg915.00 €
100mg1,258.00 €
500mg2,497.00 €
Estimated delivery in United States, on Tuesday 21 Jan 2025
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(R)-(-)-α-Methylhistamine dihydrobromide
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(R)-(-)-α-Methylhistamine dihydrobromide

CAS:868698-49-1
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 …
Formula:
C6H13Br2N3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
287

Ref: TM-T12630

50mg1,783.00 €
Estimated delivery in United States, on Tuesday 21 Jan 2025
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SUN 1334H
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SUN 1334H

CAS:607736-84-5
SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 …
Formula:
C23H28Cl2F2N2O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
489.38

Ref: TM-T13040

25mgTo inquire
50mgTo inquire
100mgTo inquire
Estimated delivery in United States, on Tuesday 21 Jan 2025
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Toreforant
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Toreforant

CAS:952494-46-1
Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: …
Formula:
C23H32N6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
392.54

Ref: TM-T17118

25mg1,549.00 €
50mg2,031.00 €
100mg2,609.00 €
Estimated delivery in United States, on Tuesday 21 Jan 2025
+ info
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