Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
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KSK94
CAS:2566716-07-0
KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value …
Formula:
C25H26N4O
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
398.5
Ref: TM-T79500
| 1mg | 59.00 € | ||
| 5mg | 122.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 277.00 € | ||
| 50mg | 428.00 € | ||
| 100mg | 623.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Wy 49051
CAS:113418-56-7
Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).
Formula:
C28H33N5O3
Purity:
97.9%
Color and Shape:
Solid
Molecular weight:
487.59
Ref: TM-T13352
| 1mg | 144.00 € | ||
| 5mg | 273.00 € | ||
| 10mg | 397.00 € | ||
| 25mg | 621.00 € | ||
| 50mg | 835.00 € | ||
| 100mg | 1,080.00 € | ||
| 200mg | 1,446.00 € | ||
| 1mL*10mM (DMSO) | 362.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
FRG8701
CAS:108498-50-6
FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to …
Formula:
C22H30N2O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
418.55
Ref: TM-T11324
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
H4R antagonist 1
CAS:1429375-54-1
H4R antagonist 1: selective histamine H4R inhibitor, IC50 27 nM, no affinity for H1R, H2R, …
Formula:
C11H11BrN8
Color and Shape:
Solid
Molecular weight:
335.16
Ref: TM-T11532
| 25mg | 1,410.00 € | ||
| 50mg | 1,854.00 € | ||
| 100mg | 2,340.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
(±)-Tazifylline
CAS:79712-55-3
(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.
Formula:
C23H32N6O3S
Purity:
98.97%
Color and Shape:
Solid
Molecular weight:
472.6
Ref: TM-T10000
| 1mg | 146.00 € | ||
| 5mg | 278.00 € | ||
| 10mg | 403.00 € | ||
| 25mg | 631.00 € | ||
| 50mg | 849.00 € | ||
| 100mg | 1,098.00 € | ||
| 1mL*10mM (DMSO) | 368.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
ReN-1869
CAS:170149-99-2
ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity …
Formula:
C24H27NO2
Purity:
99.87% - 99.89%
Color and Shape:
Solid
Molecular weight:
361.48
Ref: TM-T28516
| 1mg | 201.00 € | ||
| 5mg | 502.00 € | ||
| 10mg | 725.00 € | ||
| 25mg | 1,117.00 € | ||
| 50mg | 1,852.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Mianserin
CAS:24219-97-4
Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) …
Formula:
C18H20N2
Purity:
99.39%
Color and Shape:
Solid
Molecular weight:
264.36
Ref: TM-T21428
| 1mg | 369.00 € | ||
| 5mg | 900.00 € | ||
| 10mg | 1,198.00 € | ||
| 25mg | 1,811.00 € | ||
| 50mg | 2,448.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
BMY-25271
CAS:78441-82-4
BMY-25271 is an antagonist of histamine H2 receptor.
Formula:
C12H19N5O2S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
329.44
Ref: TM-T10575
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Azelastine
CAS:58581-89-8
Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.
Formula:
C22H24ClN3O
Purity:
99.35%
Color and Shape:
White Crystal Powder
Molecular weight:
381.9
Ref: TM-T0211
| 100mg | 59.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
ReN-1869 hydrochloride
CAS:170149-76-5
ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
Formula:
C24H28ClNO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
397.94
Ref: TM-T12703
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
ROS 234 dioxalate
CAS:1781941-93-2
ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)
Formula:
C17H19N5O8
Purity:
98%
Color and Shape:
Solid
Molecular weight:
421.37
Ref: TM-T12756
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Lavoltidine
CAS:76956-02-0
Lavoltidine, an irreversible oral H2-receptor antagonist, reduces stomach acid and increases gastrin.
Formula:
C19H29N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
359.47
Ref: TM-T15722
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Clemastine
CAS:15686-51-8
Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.
Formula:
C21H26ClNO
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
343.89
Ref: TM-T19966
| 10mg | 66.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 151.00 € | ||
| 100mg | 220.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Bavisant
CAS:929622-08-2
Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.
Formula:
C19H27N3O2
Purity:
96.06% - 98%
Color and Shape:
Solid
Molecular weight:
329.44
Ref: TM-TQ0046
| 1mg | 42.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 320.00 € | ||
| 100mg | 455.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Dimethindene maleate
CAS:3614-69-5
Dimethindene maleate (SU 6518) is a histamine H1 antagonist and can be used in studies …
Formula:
C24H28N2O4
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
408.49
Ref: TM-T21472
| 1mg | 36.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 110.00 € | ||
| 25mg | 246.00 € | ||
| 50mg | 325.00 € | ||
| 100mg | 425.00 € | ||
| 500mg | 922.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Pitolisant
CAS:362665-56-3
Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human …
Formula:
C17H26ClNO
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
295.85
Ref: TM-T60636
| 5mg | 47.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 119.00 € | ||
| 50mg | 185.00 € | ||
| 100mg | 306.00 € | ||
| 500mg | 734.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Niperotidine
CAS:84845-75-0
Niperotidine is an antagonist of histamine H2-receptor.
Formula:
C20H26N4O5S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
434.51
Ref: TM-T12228
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
JNJ-39220675
CAS:959740-39-7
JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats.
Formula:
C21H24FN3O2
Purity:
97.95% - 99.78%
Color and Shape:
Solid
Molecular weight:
369.43
Ref: TM-T27678
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,417.00 € | ||
| 50mg | 1,846.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
N-Acetylhistamine
CAS:673-49-4
N-Acetylhistamine (N-Omega-acetylhistamine) is a metabolite of histamine.
Formula:
C7H11N3O
Purity:
97.72%
Color and Shape:
Solid
Molecular weight:
153.18
Ref: TM-T19443
| 10mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Abt-288
CAS:948845-91-8
ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate …
Formula:
C23H24N4O
Purity:
98% - 98.84%
Color and Shape:
Solid
Molecular weight:
372.46
Ref: TM-T26526
| 1mg | 183.00 € | ||
| 5mg | 452.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,009.00 € | ||
| 50mg | 1,383.00 € | ||
| 100mg | 1,828.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
