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  7. Histamine Receptor
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Histamine Receptor

Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.

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products per page. 203 products on this category.

BrandProduct dataPurityPrice rangeEstimated delivery
Targetmol logo
Irdabisant
REF: TM-T32191CAS: 1005402-19-6 		99.77%57.00 €~1,291.00 €Mon 27 Jan 25
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KSK68
REF: TM-T79499CAS: 2566715-91-9 		97.22%74.00 €~2,210.00 €Mon 27 Jan 25
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MK-0249
REF: TM-T12054CAS: 862309-06-6 		99.79%225.00 €~2,785.00 €Mon 27 Jan 25
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Impromidine hydrochloride
REF: TM-T68921CAS: 65573-02-6 		99.50%240.00 €~4,577.00 €Mon 27 Jan 25
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JNJ 10191584 maleate
REF: TM-T22879CAS: 869497-75-6 		99.82%To inquireMon 27 Jan 25
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Vapitadine dihydrochloride
REF: TM-T29096CAS: 279253-83-7 		100% - 99.92%241.00 €~1,718.00 €Mon 27 Jan 25
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Noberastine
REF: TM-T25875CAS: 110588-56-2 		100% - 99.67%141.00 €~2,005.00 €Mon 27 Jan 25
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GSK-239512
REF: TM-T27462CAS: 720691-69-0 		98.50% - 99.72%46.00 €~416.00 €Mon 27 Jan 25
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Nedocromil
REF: TM-T16280CAS: 69049-73-6 		95.00%69.00 €~508.00 €Mon 27 Jan 25
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Imetit dihydrobromide
REF: TM-T15565CAS: 32385-58-3 		98%To inquireMon 27 Jan 25
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JTE-952
REF: TM-T11729CAS: 1255303-54-8 		98%To inquireMon 10 Feb 25
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ST-1006
REF: TM-T34709CAS: 1196994-11-2 		98.31% - 99.56%186.00 €~4,568.00 €Mon 10 Feb 25
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H3 receptor antagonist 1
REF: TM-T10911CAS: 935840-13-4 		98%904.00 €~2,329.00 €Mon 10 Feb 25
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Ebrotidine
REF: TM-T15195CAS: 100981-43-9 		97.5%44.00 €~94.00 €Mon 10 Feb 25
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Dothiepin
REF: TM-T78126CAS: 113-53-1 		98%To inquireMon 10 Feb 25
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H4R antagonist 2
REF: TM-T79786CAS: 1148115-99-4 		98%To inquireMon 10 Feb 25
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Enerisant
REF: TM-T67828CAS: 1152747-82-4 		99.7%95.00 €~1,836.00 €Mon 10 Feb 25
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H3R-IN-1 Hydrochloride
REF: TM-T11531CAS: 2319790-07-1 		98%1,030.00 €~2,131.00 €Mon 10 Mar 25
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H3R antagonist 1
REF: TM-T200063CAS: 1448422-61-4 		- - -To inquireMon 10 Mar 25
Targetmol logo
TAAR1 agonist 2
REF: TM-T200140CAS: 1804128-38-8 		- - -To inquireMon 10 Mar 25
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Irdabisant
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Irdabisant

CAS:1005402-19-6
Irdabisant (CEP-26401) is an H3R antagonist/inverse agonist, BBB permeable, with cognition-enhancing effects for schizophrenia/cognitive research.
Formula:
C18H23N3O2
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
313.39

Ref: TM-T32191

1mg57.00 €
5mg131.00 €
10mg184.00 €
25mg328.00 €
50mg460.00 €
100mg647.00 €
500mg1,291.00 €
1mL*10mM (DMSO)92.00 €
Estimated delivery in United States, on Monday 27 Jan 2025
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KSK68
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KSK68

CAS:2566715-91-9
KSK68 is a sigma-1 and histamine H3 receptor antagonist with analgesic activity, inhibits H3 receptors …
Formula:
C23H28N2O2
Purity:
97.22%
Color and Shape:
Solid
Molecular weight:
364.48

Ref: TM-T79499

1mg74.00 €
5mg159.00 €
10mg224.00 €
25mg372.00 €
50mg558.00 €
100mg796.00 €
500mg2,210.00 €
Estimated delivery in United States, on Monday 27 Jan 2025
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MK-0249
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MK-0249

CAS:862309-06-6
MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).
Formula:
C23H24F3N3O2
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
431.45

Ref: TM-T12054

1mg225.00 €
5mg555.00 €
10mg804.00 €
25mg1,191.00 €
50mg1,585.00 €
100mg2,147.00 €
200mg2,785.00 €
Estimated delivery in United States, on Monday 27 Jan 2025
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Impromidine hydrochloride
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Impromidine hydrochloride

CAS:65573-02-6
Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular …
Formula:
C14H26Cl3N7S
Purity:
99.50%
Color and Shape:
Liquid
Molecular weight:
430.83

Ref: TM-T68921

1mg240.00 €
5mg599.00 €
10mg853.00 €
25mg1,280.00 €
50mg1,729.00 €
100mg2,331.00 €
500mg4,577.00 €
Estimated delivery in United States, on Monday 27 Jan 2025
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JNJ 10191584 maleate
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JNJ 10191584 maleate

CAS:869497-75-6
JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor …
Formula:
C17H19ClN4O5
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
394.81

Ref: TM-T22879

1mg53.00 €
2mg81.00 €
5mg105.00 €
10mg130.00 €
25mg278.00 €
50mg403.00 €
100mgTo inquire
Estimated delivery in United States, on Monday 27 Jan 2025
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Vapitadine dihydrochloride
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Vapitadine dihydrochloride

CAS:279253-83-7
Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on …
Formula:
C17H22Cl2N4O
Purity:
100% - 99.92%
Color and Shape:
Solid
Molecular weight:
369.29

Ref: TM-T29096

1mg241.00 €
5mg600.00 €
10mg852.00 €
25mg1,280.00 €
50mg1,718.00 €
Estimated delivery in United States, on Monday 27 Jan 2025
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Noberastine
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Noberastine

CAS:110588-56-2
Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine …
Formula:
C17H21N5O
Purity:
100% - 99.67%
Color and Shape:
Solid
Molecular weight:
311.38

Ref: TM-T25875

1mg141.00 €
5mg327.00 €
10mg495.00 €
25mg958.00 €
50mg1,299.00 €
100mg2,005.00 €
Estimated delivery in United States, on Monday 27 Jan 2025
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GSK-239512
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GSK-239512

CAS:720691-69-0
GSK-239512 is an antagonist of H3 receptor and can be used in studies about the …
Formula:
C23H27N3O2
Purity:
98.50% - 99.72%
Color and Shape:
Solid
Molecular weight:
377.48

Ref: TM-T27462

1mg46.00 €
5mg94.00 €
10mg111.00 €
25mg184.00 €
50mg276.00 €
100mg416.00 €
Estimated delivery in United States, on Monday 27 Jan 2025
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Nedocromil
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Nedocromil

CAS:69049-73-6
Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene …
Formula:
C19H17NO7
Purity:
95.00%
Color and Shape:
Solid
Molecular weight:
371.34

Ref: TM-T16280

5mg69.00 €
10mg94.00 €
25mg198.00 €
50mg325.00 €
100mg508.00 €
Estimated delivery in United States, on Monday 27 Jan 2025
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Imetit dihydrobromide
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Imetit dihydrobromide

CAS:32385-58-3
Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors …
Formula:
C6H12Br2N4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
332.06

Ref: TM-T15565

50mgTo inquire
100mgTo inquire
Estimated delivery in United States, on Monday 27 Jan 2025
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JTE-952
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JTE-952

CAS:1255303-54-8
JTE-952: oral, selective Type II CSF-1R inhibitor, IC50 = 13 nM for CSF1R, 261 nM …
Formula:
C30H34N2O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
518.6

Ref: TM-T11729

25mg1,559.00 €
50mg2,040.00 €
100mg2,888.00 €
Estimated delivery in United States, on Monday 10 Feb 2025
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ST-1006
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ST-1006

CAS:1196994-11-2
ST-1006: histamine H4 agonist, pKi 7.94, anti-inflammatory, anti-pruritic, promotes basophil migration.
Formula:
C16H20Cl2N6
Purity:
98.31% - 99.56%
Color and Shape:
Solid
Molecular weight:
367.28

Ref: TM-T34709

1mg186.00 €
2mg277.00 €
5mg468.00 €
10mg750.00 €
25mg1,217.00 €
50mg1,500.00 €
100mg1,867.00 €
Estimated delivery in United States, on Monday 10 Feb 2025
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H3 receptor antagonist 1
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H3 receptor antagonist 1

CAS:935840-13-4
H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor …
Formula:
C20H28F2N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
350.45

Ref: TM-T10911

25mg1,410.00 €
50mg1,845.00 €
100mg2,329.00 €
Estimated delivery in United States, on Monday 10 Feb 2025
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Ebrotidine
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Ebrotidine

CAS:100981-43-9
Ebrotidine (FI3542) is a competitive H2-receptor antagonist with Ki of 127.5 nM. Ebrotidine has a …
Formula:
C14H17BrN6O2S3
Purity:
97.5%
Color and Shape:
Solid
Molecular weight:
477.42

Ref: TM-T15195

2mg44.00 €
5mg64.00 €
10mg94.00 €
1mL*10mM (DMSO)71.00 €
Estimated delivery in United States, on Monday 10 Feb 2025
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discount label
Dothiepin
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Dothiepin

CAS:113-53-1
Dothiepin (Dosulepin; Dothep), an antidepressant with sedative/anxiolytic properties, preferentially inhibits noradrenaline over serotonin uptake, enhancing
Formula:
C19H21NS
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
295.44

Ref: TM-T78126

5mgTo inquire
50mgTo inquire
Estimated delivery in United States, on Monday 10 Feb 2025
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H4R antagonist 2
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H4R antagonist 2

CAS:1148115-99-4
H4R Antagonist 2, a potent Furo[3,2-d]pyrimidine derivative, serves as a histamine H4 receptor antagonist and …
Formula:
C13H17N5O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
259.31

Ref: TM-T79786

5mgTo inquire
50mgTo inquire
Estimated delivery in United States, on Monday 10 Feb 2025
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Enerisant
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Enerisant

CAS:1152747-82-4
Enerisant (TS-091) is a histamine H3 receptor antagonist that promotes pro-cognitive effects and reverses scopolamine-induced …
Formula:
C22H30N4O3
Purity:
99.7%
Color and Shape:
Soild
Molecular weight:
398.50

Ref: TM-T67828

1mg95.00 €
5mg212.00 €
10mg340.00 €
25mg717.00 €
50mg1,146.00 €
100mg1,836.00 €
1mL*10mM (DMSO)187.00 €
Estimated delivery in United States, on Monday 10 Feb 2025
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H3R-IN-1 Hydrochloride
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H3R-IN-1 Hydrochloride

CAS:2319790-07-1
H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .
Formula:
C19H24ClN3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
377.87

Ref: TM-T11531

25mg1,030.00 €
50mg1,356.00 €
100mg2,131.00 €
Estimated delivery in United States, on Monday 10 Mar 2025
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discount label
H3R antagonist 1
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H3R antagonist 1

CAS:1448422-61-4
H3R-IN-1 is an effective inverse agonist of the histamine receptor 3 (H3R).
Formula:
C19H23N3O3
Color and Shape:
Liquid
Molecular weight:
341.4

Ref: TM-T200063

10mgTo inquire
50mgTo inquire
Estimated delivery in United States, on Monday 10 Mar 2025
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TAAR1 agonist 2
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TAAR1 agonist 2

CAS:1804128-38-8
TAAR1 agonist 2 (compound 30), a full agonist at trace amine-associated receptor 1 (TAAR1) (pEC50=7.5), …
Formula:
C9H11NO
Color and Shape:
Liquid
Molecular weight:
149.19

Ref: TM-T200140

10mgTo inquire
50mgTo inquire
Estimated delivery in United States, on Monday 10 Mar 2025
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