Bradykinin Receptor
Bradykinin receptors are GPCRs that mediate the effects of bradykinin, a peptide involved in inflammatory responses, pain sensation, and blood pressure regulation. There are two main types of bradykinin receptors, B1 and B2, each playing distinct roles in pathophysiological processes. Bradykinin receptor antagonists are used in the treatment of conditions such as hereditary angioedema, chronic pain, and hypertension. At CymitQuimica, we offer a variety of high-quality bradykinin receptor modulators to support your research in inflammation, pain management, and cardiovascular biology.
Found 61 products of "Bradykinin Receptor"
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Anatibant 2HCl
CAS:Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.
Formula:C34H36Cl2N6O5S·2ClHPurity:99.17% - 99.58%Color and Shape:SoildMolecular weight:784.58Fasitibant chloride
CAS:Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.
Formula:C36H49Cl3N6O6SColor and Shape:SolidMolecular weight:800.23Methionyl-Lysyl-Bradykinin
CAS:Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin [1] [2] .Formula:C61H94N18O13SColor and Shape:SolidMolecular weight:1319.58Lys-[Des-Arg9]Bradykinin TFA
CAS:Lys-[Des-Arg9]Bradykinin TFA: natural kinin, selective B1 agonist; Ki: 0.12 nM (human), 1.7 nM (mouse), 0.23 nM (rabbit); weak on B2 receptors.Formula:C54H75F6N13O15Color and Shape:SolidMolecular weight:1260.24Icatibant
CAS:Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).Formula:C59H89N19O13SPurity:98%Color and Shape:White SolidMolecular weight:1304.52[Phe8Ψ(CH-NH)-Arg9]-Bradykinin
CAS:Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage.Formula:C50H75N15O10Purity:98%Color and Shape:SolidMolecular weight:1046.23Bombinakinin M
CAS:Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.Formula:C100H159N31O24Purity:98%Color and Shape:SolidMolecular weight:2179.55Lys-(Des-Arg9,Leu8)-Bradykinin
CAS:Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].Formula:C47H75N13O11Purity:98%Color and Shape:SolidMolecular weight:998.18(Hyp³)-Bradykinin acetate
(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in cultured human fibroblasts.Formula:C52H77N15O14Purity:99.46%Color and Shape:SolidMolecular weight:1136.26Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS:Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.Formula:C47H66N12O11Purity:98%Color and Shape:SolidMolecular weight:975.11Labradimil
CAS:Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.Formula:C49H75N15O12SPurity:98%Color and Shape:SolidMolecular weight:1098.29[Des-Arg10]-HOE I40 TFA
[Des-Arg10]-HOE I40 TFA is a potent antagonist of the bradykinin B1 receptor.
Formula:C53H77N15O12S·xC2HF3O2Color and Shape:SolidDes-Arg9-[Leu8]-Bradykinin acetate
CAS:Des-Arg9-[Leu8]-Bradykinin acetate is a potent antagonist of the bradykinin receptor 1 (B1R), utilized in renal fibrosis research [1].Formula:C43H67N11O12Purity:98%Color and Shape:SolidMolecular weight:930.06Bombinakinin M acetate
Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and is
Formula:C102H163N31O26Purity:99.80%Color and Shape:SolidMolecular weight:2239.58NPC 567 acetate
NPC 567 acetate is a bradykinin B2 antagonist and can be used in studies about the treatment of allergic airway disease.Formula:C62H91N19O15Purity:97.72%Color and Shape:SolidMolecular weight:1342.5T-kinin
CAS:T-kinin (Ile-Ser-bradykinin) is a bradykinin-containing peptide utilized in inflammation research [1] [2].Formula:C59H89N17O14Molecular weight:1260.44Fasitibant chloride hydrochloride
CAS:Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.Formula:C36H50Cl4N6O6SColor and Shape:SolidMolecular weight:836.7Lys-Bradykinin
CAS:Endogenous bradykinin receptor agonistFormula:C56H85N17O12Purity:98%Color and Shape:SolidMolecular weight:1188.38Zoliprofen
CAS:Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.Formula:C12H11NO3SPurity:99.62%Color and Shape:SolidMolecular weight:249.29Ref: TM-T68025
1mg85.00€5mg170.00€10mg256.00€25mg480.00€50mg655.00€100mg933.00€500mg1,872.00€1mL*10mM (DMSO)168.00€NPC 567
CAS:NPC 567 is an antagonist of the bradykinin receptor.Formula:C60H87N19O13Purity:98%Color and Shape:SolidMolecular weight:1282.48Thrombostatin cont-1
CAS:Thrombostatin cont-1, an analogue of the bradykinin metabolite thrombostatin, has been shown to reduce platelet activation in the canine carotid arteryFormula:C87H142N34O29S2Molecular weight:2192.4FR167344 free base
CAS:FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.Formula:C30H28BrCl2N5O4Purity:98%Color and Shape:SolidMolecular weight:673.38Bradykinin (1-3)
CAS:Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.
Formula:C16H28N6O4Purity:98%Color and Shape:SolidMolecular weight:368.43FR190997
CAS:FR190997 is an agonist of bradykinin B2 receptor.Formula:C37H33Cl2N5O5Color and Shape:SolidMolecular weight:698.59L 366811
CAS:L 366811 is a potent oxytocin antagonist.Formula:C43H56N8O6Color and Shape:SolidMolecular weight:780.95MEN 11270
CAS:B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.Formula:C60H90N20O11SPurity:98%Color and Shape:SolidMolecular weight:1299.56JMV-1645
CAS:JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.Formula:C49H69N13O12SPurity:98%Color and Shape:SolidMolecular weight:1064.23Bradykinin (1-7)
CAS:Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.Formula:C35H52N10O9Purity:98%Color and Shape:White Lyophilized PowderMolecular weight:756.85Bradykinin (1-6)
CAS:Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.Formula:C30H45N9O8Purity:98%Color and Shape:SolidMolecular weight:659.73Lys-[Des-Arg9]Bradykinin
CAS:Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.Formula:C50H73N13O11Purity:98%Color and Shape:SolidMolecular weight:1032.21Retrobradykinin
CAS:Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.Formula:C50H73N15O11Color and Shape:SolidMolecular weight:1060.228Lys-[Hyp3]-Bradykinin
CAS:Lys-[Hyp3]-Bradykinin, a human urine-derived kinin and bradykinin agonist, is used for inflammation research.Formula:C56H85N17O13Color and Shape:SolidMolecular weight:1204.38[Des-Arg9]-Bradykinin
CAS:[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.
Formula:C44H61N11O10Purity:98%Color and Shape:SolidMolecular weight:904.02B-Raf IN 14
CAS:B-Raf IN 14 is a BRAF inhibitor.Formula:C15H14BrN5O3SPurity:98.38%Color and Shape:SolidMolecular weight:424.27[Des-Arg9]-Bradykinin acetate
CAS:[Des-Arg9]-Bradykinin acetate is a selective agonist of Bradykinin B1 receptor.Formula:C46H65N11O12Purity:99.05%Color and Shape:SolidMolecular weight:964.07Bradykinin (1-5)
CAS:Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.Formula:C27H40N8O6Color and Shape:SolidMolecular weight:572.66Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant toFormula:C49H70N12O13Purity:99.93%Color and Shape:SolidMolecular weight:1035.15Icatibant Acetate
CAS:Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.Formula:C61H93N19O15SPurity:99.68% - 99.90%Color and Shape:SolidMolecular weight:1364.57Ref: TM-T22344
1mg66.00€2mg92.00€5mg177.00€10mg281.00€25mg475.00€50mg677.00€100mg888.00€1mL*10mM (DMSO)355.00€5-Hydroxy-1-methylhydantoin
CAS:5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.Formula:C4H6N2O3Purity:99.99%Color and Shape:SolidMolecular weight:130.1Bradykinin
CAS:Bradykinin is an inflammatory mediator.Formula:C50H73N15O11Purity:99.68%Color and Shape:SolidMolecular weight:1060.21Emorfazone
CAS:Emorfazone (PH011085) has an anti-nociceptive effect.Formula:C11H17N3O3Purity:99.89%Color and Shape:SolidMolecular weight:239.27Ref: TM-T9132
1mg84.00€5mg168.00€10mg245.00€25mg404.00€50mg567.00€100mg767.00€200mg1,018.00€1mL*10mM (DMSO)152.00€ELN-441958
CAS:ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.Formula:C29H29ClN4O2Purity:99.88%Color and Shape:SolidMolecular weight:501.02Ref: TM-T2086
1mg58.00€5mg128.00€10mg200.00€25mg339.00€50mg485.00€100mg658.00€200mg889.00€1mL*10mM (DMSO)141.00€SSR240612
CAS:SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,Formula:C42H53ClN4O7SPurity:98.59% - 99.16%Color and Shape:SolidMolecular weight:793.41Ref: TM-T5048
1mg222.00€5mg512.00€10mg700.00€25mg982.00€50mg1,333.00€100mg1,783.00€1mL*10mM (DMSO)612.00€Bradykinin (acetate)
CAS:Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.Formula:C52H77N15O13Purity:>99.99%Color and Shape:SolidMolecular weight:1120.26Lys-[Des-Arg9]Bradykinin,TFA
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2Formula:C54H75F6N13O15Purity:97.35%Color and Shape:SolidMolecular weight:1260.24[Des-Arg9]-Bradykinin TFA
CAS:[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.Formula:C46H62F3N11O12Purity:>99.99%Color and Shape:SolidMolecular weight:1018.05Bradykinin (2-9)
CAS:Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.Formula:C44H61N11O10Purity:>99.99%Color and Shape:SolidMolecular weight:904.02Ref: TM-TP1181
1mg42.00€5mg93.00€10mg137.00€25mg221.00€50mg329.00€100mg490.00€200mg697.00€1mL*10mM (DMSO)153.00€R715 TFA(185052-09-9 free base)
R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49).Formula:C59H82F3N13O14Purity:>99.99%Color and Shape:SolidMolecular weight:1254.36Lys-Bradykinin acetate(342-10-9 free base)
CAS:Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.Formula:C58H89N17O14Purity:99.86%Color and Shape:SolidMolecular weight:1248.43Lys-[Des-Arg9]Bradykinin acetate
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and
Formula:C52H77N13O13Purity:99.93%Color and Shape:SolidMolecular weight:1092.27B 4148
CAS:B 4148 is a bradykinin inhibitor.Formula:C62H95N19O14S2Color and Shape:SolidMolecular weight:1394.67NPC 17731
CAS:NPC 17731 is a bradykinin receptor antagonist.Formula:C59H95N19O14Color and Shape:SolidMolecular weight:1294.5BKM-570
CAS:BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.Formula:C34H34Cl2F5N3O3Purity:98%Color and Shape:SolidMolecular weight:698.55Anatibant
CAS:Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.Formula:C34H36Cl2N6O5SPurity:98%Color and Shape:SolidMolecular weight:711.66Fulimetibant
CAS:Fulimetibant is a bradykinin receptor antagonist.Formula:C25H21F4N3O3Color and Shape:SolidMolecular weight:487.45MK-0686
CAS:MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.Formula:C22H19ClF4N2O4Purity:99.88%Color and Shape:SolidMolecular weight:486.84Safotibant
CAS:Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edemaFormula:C25H34N4O5SPurity:99.62% - 99.67%Color and Shape:SolidMolecular weight:502.63NVP-SAA164
CAS:NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.Formula:C36H45N5O5SPurity:98%Color and Shape:SolidMolecular weight:659.84FK-3657
CAS:FK-3657 is a non-peptide antagonist of bradykinin (BK)-B2 receptor.Formula:C30H27Cl2N5O4Color and Shape:SolidMolecular weight:592.47BI-113823
CAS:BI-113823 is an orally active and selective bradykinin B1 receptor antagonist. It alleviates mechanical hyperalgesia induced by complete Freund's adjuvant in rats. BI-113823 is applicable for research on chronic inflammatory pain.Formula:C26H44N4O5SColor and Shape:SolidMolecular weight:524.716Fasitibant
CAS:Fasitibant is a potent and selective nonpeptide kinin B2 receptor antagonist.Formula:C36H49Cl2N6O6SColor and Shape:SolidMolecular weight:764.78
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