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Bradykinin Receptor

Bradykinin Receptor

Bradykinin receptors are GPCRs that mediate the effects of bradykinin, a peptide involved in inflammatory responses, pain sensation, and blood pressure regulation. There are two main types of bradykinin receptors, B1 and B2, each playing distinct roles in pathophysiological processes. Bradykinin receptor antagonists are used in the treatment of conditions such as hereditary angioedema, chronic pain, and hypertension. At CymitQuimica, we offer a variety of high-quality bradykinin receptor modulators to support your research in inflammation, pain management, and cardiovascular biology.

Found 59 products of "Bradykinin Receptor"

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  • Anatibant 2HCl
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    Anatibant 2HCl

    CAS:
    <p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>
    Formula:C34H36Cl2N6O5S·2ClH
    Purity:99.17% - 99.58%
    Color and Shape:Soild
    Molecular weight:784.58

    Ref: TM-T26627L

  • [Des-Arg9]-Bradykinin acetate
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    [Des-Arg9]-Bradykinin acetate

    CAS:
    <p>[Des-Arg9]-Bradykinin acetate is a selective agonist of Bradykinin B1 receptor.</p>
    Formula:C46H65N11O12
    Purity:99.05%
    Color and Shape:Solid
    Molecular weight:964.07

    Ref: TM-TP1445

  • Fasitibant chloride
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    Fasitibant chloride

    CAS:
    <p>Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.</p>
    Formula:C36H49Cl3N6O6S
    Color and Shape:Solid
    Molecular weight:800.23

    Ref: TM-T38544

  • Icatibant
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    Icatibant

    CAS:
    <p>Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).</p>
    Formula:C59H89N19O13S
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:1304.52

    Ref: TM-T15547

  • [Phe8Ψ(CH-NH)-Arg9]-Bradykinin
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    [Phe8Ψ(CH-NH)-Arg9]-Bradykinin

    CAS:
    <p>Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage.</p>
    Formula:C50H75N15O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1046.23

    Ref: TM-TP2076

  • Bombinakinin M
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    Bombinakinin M

    CAS:
    <p>Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.</p>
    Formula:C100H159N31O24
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2179.55

    Ref: TM-TP2075

  • Lys-(Des-Arg9,Leu8)-Bradykinin
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    Lys-(Des-Arg9,Leu8)-Bradykinin

    CAS:
    <p>Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].</p>
    Formula:C47H75N13O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:998.18

    Ref: TM-T80117

  • (Hyp³)-Bradykinin acetate
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    (Hyp³)-Bradykinin acetate

    <p>(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in cultured human fibroblasts.</p>
    Formula:C52H77N15O14
    Purity:99.46%
    Color and Shape:Solid
    Molecular weight:1136.26

    Ref: TM-T36442L

  • Sar-[D-Phe8]-des-Arg9-Bradykinin
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    Sar-[D-Phe8]-des-Arg9-Bradykinin

    CAS:
    <p>Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.</p>
    Formula:C47H66N12O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:975.11

    Ref: TM-TP1917

  • [Des-Arg9]-Bradykinin
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    [Des-Arg9]-Bradykinin

    CAS:
    <p>[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.</p>
    Formula:C44H61N11O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:904.02

    Ref: TM-T7645

  • B-Raf IN 14
    Targetmol
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    B-Raf IN 14

    CAS:
    <p>B-Raf IN 14 is a BRAF inhibitor.</p>
    Formula:C15H14BrN5O3S
    Purity:98.32%
    Color and Shape:Solid
    Molecular weight:424.27

    Ref: TM-T72070

  • Labradimil
    Targetmol
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    Labradimil

    CAS:
    <p>Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.</p>
    Formula:C49H75N15O12S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1098.29

    Ref: TM-T27790

  • CymitQuimica logo
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    [Des-Arg10]-HOE I40 TFA

    <p>[Des-Arg10]-HOE I40 TFA is a potent antagonist of the bradykinin B1 receptor.</p>
    Formula:C53H77N15O12S·xC2HF3O2
    Color and Shape:Solid

    Ref: TM-T207446

  • Des-Arg9-[Leu8]-Bradykinin acetate
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    Des-Arg9-[Leu8]-Bradykinin acetate

    CAS:
    <p>Des-Arg9-[Leu8]-Bradykinin acetate is a potent antagonist of the bradykinin receptor 1 (B1R), utilized in renal fibrosis research [1].</p>
    Formula:C43H67N11O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:930.06

    Ref: TM-T80072

  • Bombinakinin M acetate
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    Bombinakinin M acetate

    <p>Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and is</p>
    Formula:C102H163N31O26
    Purity:99.80%
    Color and Shape:Solid
    Molecular weight:2239.58

    Ref: TM-TP2075L

  • NPC 567 acetate
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    NPC 567 acetate

    <p>NPC 567 acetate is a bradykinin B2 antagonist and can be used in studies about the treatment of allergic airway disease.</p>
    Formula:C62H91N19O15
    Purity:97.72%
    Color and Shape:Solid
    Molecular weight:1342.5

    Ref: TM-T21060L

  • FR190997
    Targetmol
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    FR190997

    CAS:
    <p>FR190997 is an agonist of bradykinin B2 receptor.</p>
    Formula:C37H33Cl2N5O5
    Color and Shape:Solid
    Molecular weight:698.59

    Ref: TM-T27377

  • Fasitibant chloride hydrochloride
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    Fasitibant chloride hydrochloride

    CAS:
    <p>Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.</p>
    Formula:C36H50Cl4N6O6S
    Color and Shape:Solid
    Molecular weight:836.7

    Ref: TM-T31747

  • Lys-Bradykinin
    Targetmol
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    Lys-Bradykinin

    CAS:
    <p>Endogenous bradykinin receptor agonist</p>
    Formula:C56H85N17O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1188.38

    Ref: TM-TP2268

  • Zoliprofen
    Targetmol
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    Zoliprofen

    CAS:
    <p>Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.</p>
    Formula:C12H11NO3S
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:249.29

    Ref: TM-T68025

  • NPC 567
    Targetmol
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    NPC 567

    CAS:
    <p>NPC 567 is an antagonist of the bradykinin receptor.</p>
    Formula:C60H87N19O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1282.48

    Ref: TM-T21060

  • L 366811
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    L 366811

    CAS:
    <p>L 366811 is a potent oxytocin antagonist.</p>
    Formula:C43H56N8O6
    Color and Shape:Solid
    Molecular weight:780.95

    Ref: TM-T24291

  • FR167344 free base
    Targetmol
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    FR167344 free base

    CAS:
    <p>FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.</p>
    Formula:C30H28BrCl2N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:673.38

    Ref: TM-T15347

  • Bradykinin (1-3)
    Targetmol
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    Bradykinin (1-3)

    CAS:
    <p>Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.</p>
    Formula:C16H28N6O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:368.43

    Ref: TM-TP1780

  • JMV-1645
    Targetmol
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    JMV-1645

    CAS:
    <p>JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.</p>
    Formula:C49H69N13O12S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1064.23

    Ref: TM-T25555

  • Lys-[Des-Arg9]Bradykinin TFA
    Targetmol
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    Lys-[Des-Arg9]Bradykinin TFA

    CAS:
    <p>Lys-[Des-Arg9]Bradykinin TFA: natural kinin, selective B1 agonist; Ki: 0.12 nM (human), 1.7 nM (mouse), 0.23 nM (rabbit); weak on B2 receptors.</p>
    Formula:C54H75F6N13O15
    Color and Shape:Solid
    Molecular weight:1260.24

    Ref: TM-T73646

  • MEN 11270
    Targetmol
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    MEN 11270

    CAS:
    <p>B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.</p>
    Formula:C60H90N20O11S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1299.56

    Ref: TM-TP1999

  • Methionyl-Lysyl-Bradykinin
    Targetmol
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    Methionyl-Lysyl-Bradykinin

    CAS:
    <p>Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin [1] [2] .</p>
    Formula:C61H94N18O13S
    Color and Shape:Solid
    Molecular weight:1319.58

    Ref: TM-T76384

  • Bradykinin (1-7)
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    Bradykinin (1-7)

    CAS:
    <p>Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.</p>
    Formula:C35H52N10O9
    Purity:98%
    Color and Shape:White Lyophilized Powder
    Molecular weight:756.85

    Ref: TM-TP1210

  • Bradykinin (1-6)
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    Bradykinin (1-6)

    CAS:
    <p>Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.</p>
    Formula:C30H45N9O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:659.73

    Ref: TM-TP1747

  • Lys-[Des-Arg9]Bradykinin
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    Lys-[Des-Arg9]Bradykinin

    CAS:
    <p>Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (&gt;30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.</p>
    Formula:C50H73N13O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1032.21

    Ref: TM-TP1918

  • Retrobradykinin
    Targetmol
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    Retrobradykinin

    CAS:
    <p>Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.</p>
    Formula:C50H73N15O11
    Color and Shape:Solid
    Molecular weight:1060.228

    Ref: TM-T37795

  • Lys-[Hyp3]-Bradykinin
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    Lys-[Hyp3]-Bradykinin

    CAS:
    <p>Lys-[Hyp3]-Bradykinin, a human urine-derived kinin and bradykinin agonist, is used for inflammation research.</p>
    Formula:C56H85N17O13
    Color and Shape:Solid
    Molecular weight:1204.38

    Ref: TM-T76293

  • Bradykinin (1-5)
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    Bradykinin (1-5)

    CAS:
    <p>Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.</p>
    Formula:C27H40N8O6
    Color and Shape:Solid
    Molecular weight:572.66

    Ref: TM-TP1725

  • Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
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    Sar-[D-Phe8]-des-Arg9-Bradykinin acetate

    <p>Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to</p>
    Formula:C49H70N12O13
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:1035.15

    Ref: TM-TP1917L1

  • Icatibant Acetate
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    Icatibant Acetate

    CAS:
    <p>Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.</p>
    Formula:C61H93N19O15S
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:1364.57

    Ref: TM-T22344

  • 5-Hydroxy-1-methylhydantoin
    Targetmol
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    5-Hydroxy-1-methylhydantoin

    CAS:
    <p>5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.</p>
    Formula:C4H6N2O3
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:130.1

    Ref: TM-T28222

  • Bradykinin
    Targetmol
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    Bradykinin

    CAS:
    <p>Bradykinin is an inflammatory mediator.</p>
    Formula:C50H73N15O11
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:1060.21

    Ref: TM-TP1277

  • Emorfazone
    Targetmol
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    Emorfazone

    CAS:
    <p>Emorfazone (PH011085) has an anti-nociceptive effect.</p>
    Formula:C11H17N3O3
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:239.27

    Ref: TM-T9132

  • ELN-441958
    Targetmol
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    ELN-441958

    CAS:
    <p>ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.</p>
    Formula:C29H29ClN4O2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:501.02

    Ref: TM-T2086

  • SSR240612
    Targetmol
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    SSR240612

    CAS:
    <p>SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,</p>
    Formula:C42H53ClN4O7S
    Purity:98.59% - 99.16%
    Color and Shape:Solid
    Molecular weight:793.41

    Ref: TM-T5048

  • Bradykinin (acetate)
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    Bradykinin (acetate)

    CAS:
    <p>Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.</p>
    Formula:C52H77N15O13
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1120.26

    Ref: TM-T21610

  • Lys-[Des-Arg9]Bradykinin,TFA
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    Lys-[Des-Arg9]Bradykinin,TFA

    <p>Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and &gt; 30000 nM at human B1 and B2</p>
    Formula:C54H75F6N13O15
    Purity:97.35%
    Color and Shape:Solid
    Molecular weight:1260.24

    Ref: TM-TP1918L

  • [Des-Arg9]-Bradykinin TFA
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    [Des-Arg9]-Bradykinin TFA

    CAS:
    <p>[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.</p>
    Formula:C46H62F3N11O12
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1018.05

    Ref: TM-T8809

  • Bradykinin (2-9)
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    Bradykinin (2-9)

    CAS:
    <p>Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.</p>
    Formula:C44H61N11O10
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:904.02

    Ref: TM-TP1181

  • R715 TFA(185052-09-9 free base)
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    R715 TFA(185052-09-9 free base)

    <p>R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49).</p>
    Formula:C59H82F3N13O14
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1254.36

    Ref: TM-TP1933

  • Lys-Bradykinin acetate(342-10-9 free base)
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    Lys-Bradykinin acetate(342-10-9 free base)

    CAS:
    <p>Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.</p>
    Formula:C58H89N17O14
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:1248.43

    Ref: TM-TP2268L

  • Lys-[Des-Arg9]Bradykinin acetate
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    Lys-[Des-Arg9]Bradykinin acetate

    <p>Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and &gt; 30000 nM at human B1 and</p>
    Formula:C52H77N13O13
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:1092.27

    Ref: TM-TP1918L1

  • BKM-570
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    BKM-570

    CAS:
    <p>BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.</p>
    Formula:C34H34Cl2F5N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:698.55

    Ref: TM-T26833

  • Anatibant
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    Anatibant

    CAS:
    <p>Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.</p>
    Formula:C34H36Cl2N6O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:711.66

    Ref: TM-T26627

  • Fulimetibant
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    Fulimetibant

    CAS:
    <p>Fulimetibant is a bradykinin receptor antagonist.</p>
    Formula:C25H21F4N3O3
    Color and Shape:Solid
    Molecular weight:487.45

    Ref: TM-T63241

  • B 4148
    Targetmol
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    B 4148

    CAS:
    <p>B 4148 is a bradykinin inhibitor.</p>
    Formula:C62H95N19O14S2
    Color and Shape:Solid
    Molecular weight:1394.67

    Ref: TM-T71571

  • NPC 17731
    Targetmol
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    NPC 17731

    CAS:
    <p>NPC 17731 is a bradykinin receptor antagonist.</p>
    Formula:C59H95N19O14
    Color and Shape:Solid
    Molecular weight:1294.5

    Ref: TM-T70576

  • MK-0686
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    MK-0686

    CAS:
    <p>MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.</p>
    Formula:C22H19ClF4N2O4
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:486.84

    Ref: TM-T33421

  • Safotibant
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    Safotibant

    CAS:
    <p>Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edema</p>
    Formula:C25H34N4O5S
    Purity:99.62% - 99.67%
    Color and Shape:Solid
    Molecular weight:502.63

    Ref: TM-T34485

  • NVP-SAA164
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    NVP-SAA164

    CAS:
    <p>NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.</p>
    Formula:C36H45N5O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:659.84

    Ref: TM-T25895

  • FK-3657
    Targetmol
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    FK-3657

    CAS:
    <p>FK-3657 is a non-peptide antagonist of bradykinin (BK)-B2 receptor.</p>
    Formula:C30H27Cl2N5O4
    Color and Shape:Solid
    Molecular weight:592.47

    Ref: TM-T24065

  • Fasitibant
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    Fasitibant

    CAS:
    <p>Fasitibant is a potent and selective nonpeptide kinin B2 receptor antagonist.</p>
    Formula:C36H49Cl2N6O6S
    Color and Shape:Solid
    Molecular weight:764.78

    Ref: TM-T68486

  • BI-113823
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    BI-113823

    CAS:
    <p>BI-113823 is an orally active and selective bradykinin B1 receptor antagonist. It alleviates mechanical hyperalgesia induced by complete Freund's adjuvant in rats. BI-113823 is applicable for research on chronic inflammatory pain.</p>
    Formula:C26H44N4O5S
    Color and Shape:Solid
    Molecular weight:524.716

    Ref: TM-T205108